专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明授权

US5707930A 4-cycloalkyl-5-substituted pyrimidine compounds useful as crop protection agents 失效
标题翻译：用作作物保护剂的4-环烷基-5-取代的嘧啶化合物
公开(公告)号：US5707930A
公开(公告)日：1998-01-13
申请号：US715293
申请日：1996-09-16
申请人： Raymond A. Felix , Hsiao-Ling M. Chin , Frank X. Woolard , David L. Lee , David B. Kanne
发明人： Raymond A. Felix , Hsiao-Ling M. Chin , Frank X. Woolard , David L. Lee , David B. Kanne
IPC分类号： A01N43/54 , A01N47/12 , A01N47/16 , A01N47/20 , A01N47/24 , C07D239/26 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , A01N43/40
CPC分类号： C07D239/26 , A01N43/54 , A01N47/12 , A01N47/16 , A01N47/20 , A01N47/24 , C07D401/06 , C07D401/12 , C07D401/14
摘要： Herbicidal 4-cycloalkyl-5-substituted pyrimidine compounds of the formula ##STR1## are described. Herbicidal compositions containing such substituted-pyrimidinyl compounds and methods of controlling undesirable vegetation employing these compounds are also disclosed. The compounds in which XR, is hydroxyl are also useful as intermediates for producing the disclosed substituted-pyrimidinyl derivatives.
摘要翻译：描述了式（I）的除草4-环烷基-5-取代的嘧啶化合物。还公开了含有这种取代的嘧啶基化合物的除草组合物和使用这些化合物控制不期望的植物的方法。其中XR是羟基的化合物也可用作产生所公开的取代的 - 嘧啶基衍生物的中间体。

2. 发明授权

US5925795A Processes for the preparation of aryl-.beta.-diketones, arylpyrimidine ketones and crop protection intermediates 失效
标题翻译：制备芳基-β-二酮，芳基嘧啶酮和作物保护中间体的方法
公开(公告)号：US5925795A
公开(公告)日：1999-07-20
申请号：US715292
申请日：1996-09-16
申请人： Raymond A. Felix , Hsiao-Ling M. Chin , Frank X. Woolard , David L. Lee
发明人： Raymond A. Felix , Hsiao-Ling M. Chin , Frank X. Woolard , David L. Lee
IPC分类号： B01J23/44 , B01J31/04 , C07B61/00 , C07C45/67 , C07C49/76 , C07C49/80 , C07C49/807 , C07C49/813 , C07C69/738 , C07C205/45 , C07C225/14 , C07D213/50 , C07D239/00 , C07D239/26 , C07D401/06 , C07C45/00 , C07C65/00
CPC分类号： C07D239/26 , C07C201/12 , C07C221/00 , C07C45/676 , C07C49/80 , C07C49/807 , C07C49/813 , C07C67/00 , C07D213/50 , C07D401/06 , C07B2200/07 , C07C2101/02
摘要： This invention relates to processes for the preparation of aryl-.beta.-diketones and aryl-pyrimidine ketones. In addition, this invention relates to the preparation of aryl-.beta.-triketones and dimethyl aminomethylene .beta.-diketones, which are useful as crop protection intermediates.
摘要翻译：本发明涉及制备芳基-β-二酮和芳基 - 嘧啶酮的方法。此外，本发明涉及芳基-β-三酮和二甲基氨基亚甲基β-二酮的制备，其可用作作物保护中间体。

3. 发明授权

US4913722A Iminophenylthiazolidines, process of preparation and method of use 失效
标题翻译：咪嗪基噻唑烷，其制备方法和使用方法
公开(公告)号：US4913722A
公开(公告)日：1990-04-03
申请号：US269819
申请日：1988-11-15
申请人： Raymond A. Felix , Jeffery T. Springer , Eugene G. Teach , Frank X. Woolard
发明人： Raymond A. Felix , Jeffery T. Springer , Eugene G. Teach , Frank X. Woolard
IPC分类号： A01N43/78 , A01N47/02 , C07D277/18
CPC分类号： A01N47/02 , A01N43/78 , C07D277/18
摘要： A 2-iminophenyl thiazolidine having the formula ##STR1## wherein R is hydrogen or methyl; R.sub.1 is halo, nitro, cyano, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, perhalomethyl, difluoromethyl, pentafluoroethyl, trifluoromethylthhio, difluoromethoxy, trifluoromethoxy, tetrafluoroethoxy, methylsulfonyl, C.sub.1 -C.sub.4 alkyloxyiminomethyl, benzyloxyiminomethyl, 1-(C.sub.1 -C.sub.4 alkyl)-oxyiminoethyl or 1-benzyloxyiminoethyl; R.sub.2 is hydrogen or halo; R.sub.3 and R.sub.4 are independently hydrogen, halo, nitro, cyano, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 fluoroalkoxy, C.sub.1 -C.sub.4 alkoxy or C.sub.1 -C.sub.4 alkylthio; and X is hydrogen or halogen.Also disclosed is a process for making the compounds and a method of use which comprises applying the compound or composition to the locus where control is desired.

4. 发明授权

US5234895A Arylpyridone herbicides 失效
标题翻译：芳基吡啶酮除草剂
公开(公告)号：US5234895A
公开(公告)日：1993-08-10
申请号：US901008
申请日：1992-06-19
申请人： Raymond A. Felix
发明人： Raymond A. Felix
IPC分类号： A01N43/40 , C07D211/76 , C07D211/86 , C07D213/64
CPC分类号： C07D213/64 , A01N43/40 , C07D211/76 , C07D211/86
摘要： Compounds having the formula ##STR1## in which: R.sub.1 is hydrogen or fluoro;R.sub.2 is halo, trihalomethyl, pentahaloethyl, mono- or difluoromethyl, di-, tri- or tetrafluoroethyl, C.sub.1 -C.sub.2 fluoroalkylthio, C.sub.1 -C.sub.2 fluoroalkoxy, methylthio, methylsulfonyl, halomethylsulfonyl, C.sub.1 -C.sub.2 alkyl or methoxy;R.sub.3 is hydrogen or halo;R.sub.4 is hydrogen, C.sub.1 -C.sub.4 alkyl; C.sub.2 -C.sub.4 alkenyl; C.sub.2 -C.sub.4 alkynyl; C.sub.1 -C.sub.4 haloalkyl; C.sub.2 -C.sub.4 haloalkenyl; C.sub.1 -C.sub.4 alkoxy; C.sub.2 -C.sub.4 alkoxyalkyl, 3-trifluoromethylphenyl, or --(CH.sub.2).sub.n Y;R.sub.5 and R.sub.6 are hydrogen, or R.sub.5 and R.sub.6 together form a bond;R.sub.7 is C.sub.1 -C.sub.4 alkyl;R.sub.8 and R.sub.9 are hydrogen, or R.sub.8 and R.sub.9 together form a bond;Y is cyano; 4-chlorophenyl; C.sub.3 -C.sub.6 cycloalkyl, furyl or tetrahydrofuryl optionally substituted by halo or C.sub.1 -C.sub.4 alkyl; or COR.sub.10 in which R.sub.10 is hydroxy, C.sub.1 -C.sub.5 alkoxy, C.sub.1 -C.sub.5 alkylthio, --OCH.sub.2 COO(C.sub.1 -C.sub.4 alkyl) or NR.sub.11 R.sub.12 in which R.sub.11 and R.sub.12 are independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.6 alkoxy, or C.sub.2 -C.sub.4 alkoxyalkyl; andn is 1 or 2 are herbicides.
摘要翻译：具有式“IMAGE”的化合物，其中：R 1是氢或氟; R2是卤素，三卤甲基，五卤代乙基，一或二氟甲基，二或三氟或四氟乙基，C 1 -C 2氟代烷硫基，C 1 -C 2氟烷氧基，甲硫基，甲基磺酰基，卤甲基磺酰基，C 1 -C 2烷基或甲氧基; R3是氢或卤素; R4是氢，C1-C4烷基; C 2 -C 4烯基; C2-C4炔基; C 1 -C 4卤代烷基; C 2 -C 4卤代烯基; C1-C4烷氧基; C 2 -C 4烷氧基烷基，3-三氟甲基苯基或 - （CH 2）n Y; R5和R6是氢，或R5和R6一起形成键; R7是C1-C4烷基; R8和R9是氢，或R8和R9一起形成键; Y是氰基; 4-氯苯基; 任选被卤素或C 1 -C 4烷基取代的C 3 -C 6环烷基，呋喃基或四氢呋喃基; 或其中R 10是羟基，C 1 -C 5烷氧基，C 1 -C 5烷硫基，-OCH 2 COO（C 1 -C 4烷基）或NR 11 R 12的COR 10，其中R 11和R 12独立地是氢，C 1 -C 4烷基，C 1 -C 6烷氧基或C 2 -C 6烷氧基， C4烷氧基烷基; n为1或2为除草剂。

5. 发明授权

US4724261A Cyclic ureas 失效
标题翻译：循环脲
公开(公告)号：US4724261A
公开(公告)日：1988-02-09
申请号：US933833
申请日：1986-11-24
申请人： Raymond A. Felix
发明人： Raymond A. Felix
IPC分类号： C07D233/70
CPC分类号： C07D233/70
摘要： A process for the preparation of cyclic urea compounds in which a substituted anilino alkanone is reacted with an arylsubstituted isocyanate to form an intermediate imidazoline compound, and said imidazoline compound is hydrogenated in the presence of suitable catalyst to form an imidazolidine of the formula ##STR1## wherein X, X', Y and Y' are the same or different and are selected from the group consisting of trifluoromethyl, chloro, bromo, fluoro, hydrogen, cyano, nitro, alkyl, thioalkyl, halothioalkyl, alkoxy and sulfonylalkyl wherein the alkyl groups have from 1 to 4 carbon atoms; and R is selected from the group consisting of hydrogen and alkyl having from 1 to about 4 carbon atoms. Also included are intermediate anilino alkanones and the process of making them.
摘要翻译：一种制备环状脲化合物的方法，其中取代的苯胺基烷酮与芳基取代的异氰酸酯反应以形成中间体咪唑啉化合物，并且所述咪唑啉化合物在合适的催化剂存在下氢化以形成下式的咪唑烷：其中X，X'，Y和Y'相同或不同，并且选自三氟甲基，氯，溴，氟，氢，氰基，硝基，烷基，硫代烷基，卤代烷基，烷氧基和磺酰基烷基，其中烷基具有1至4个碳原子; 并且R选自氢和具有1至约4个碳原子的烷基。还包括中间苯胺基链烷酮和制备它们的过程。

6. 发明授权

US4535181A N-carboalkoxymethyl-N-halomethyl amides 失效
标题翻译： N-烷氧基甲基-N-卤代甲基酰胺
公开(公告)号：US4535181A
公开(公告)日：1985-08-13
申请号：US609921
申请日：1984-05-14
申请人： Raymond A. Felix
发明人： Raymond A. Felix
IPC分类号： C07C233/47 , C07F9/38 , C07F9/40 , C07C103/48
CPC分类号： C07F9/4006 , C07C233/47 , C07F9/3813
摘要： A method of preparing N-phosphonomethylglycine comprising (a) reacting a substituted triazine with an acyl halide to form the N-carboalkoxymethyl-N-halomethyl amide of the acyl halide; reacting the said amide with a phosphite to form a phosphonate compound; and hydrolyzing said phosphonate to yield N-phosphonomethylglycine.
摘要翻译：一种制备N-膦酰基甲基甘氨酸的方法，包括（a）使取代的三嗪与酰基卤反应形成酰卤的N-烷氧基甲基-N-卤甲基酰胺; 使所述酰胺与亚磷酸酯反应以形成膦酸酯化合物; 并水解所述膦酸酯以产生N-膦酰基甲基甘氨酸。

7. 发明授权

US4534902A Method for preparation of N-phosphonomethylglycine 失效
标题翻译： N-膦酰基甲基甘氨酸的制备方法
公开(公告)号：US4534902A
公开(公告)日：1985-08-13
申请号：US630156
申请日：1984-07-12
申请人： Raymond A. Felix
发明人： Raymond A. Felix
IPC分类号： C07F9/38 , C07F9/40 , C07C121/417
CPC分类号： C07F9/4006 , C07C255/00 , C07F9/3813
摘要： A method of preparing N-phosphonomethylglycine comprising (a) reacting a triazine with an acyl halide to form the N-cyanomethyl-N-halomethyl amide of the acyl halide; reacting the said amide with a phosphite to form a phosphonate compound; and hydrolyzing said phosphonate to yield N-phosphonomethylglycine.
摘要翻译：一种制备N-膦酰基甲基甘氨酸的方法，包括（a）使三嗪与酰卤反应形成酰卤的N-氰甲基-N-卤甲基酰胺; 使所述酰胺与亚磷酸酯反应以形成膦酸酯化合物; 并水解所述膦酸酯以产生N-膦酰基甲基甘氨酸。

8. 发明授权

US4476063A N-Acylaminomethyl-N-cyanomethyl phosphonates 失效
标题翻译： N-酰氨基甲基-N-氰甲基膦酸酯
公开(公告)号：US4476063A
公开(公告)日：1984-10-09
申请号：US540254
申请日：1983-10-11
申请人： Raymond A. Felix
发明人： Raymond A. Felix
IPC分类号： C07F9/38 , C07F9/40
CPC分类号： C07F9/4006 , C07C255/00 , C07F9/3808
摘要： A method of preparing N-phosphonomethylglycine comprising (a) reacting a triazine with an acyl halide to form the N-cyanomethyl-N-halomethyl amide of the acyl halide; reacting the said amide with a phosphite to form a phosphonate compound; and hydrolyzing said phosphonate to yield N-phosphonomethylglycine.
摘要翻译：一种制备N-膦酰基甲基甘氨酸的方法，包括（a）使三嗪与酰卤反应形成酰卤的N-氰甲基-N-卤甲基酰胺; 使所述酰胺与亚磷酸酯反应以形成膦酸酯化合物; 并水解所述膦酸酯以产生N-膦酰基甲基甘氨酸。

9. 发明授权

US4336062A Herbicidal cyclohexenone derivatives 失效
标题翻译：除草环己烯酮衍生物
公开(公告)号：US4336062A
公开(公告)日：1982-06-22
申请号：US906495
申请日：1978-05-16
申请人： Raymond A. Felix
发明人： Raymond A. Felix
IPC分类号： C07C271/28 , A01N25/08 , A01N37/24 , A01N47/20 , A01N47/30 , A01N53/00 , A01N53/12 , C07C67/00 , C07C231/00 , C07C231/02 , C07C231/12 , C07C233/25 , C07C233/27 , C07C233/60 , C07C239/00 , C07C275/34 , C07C313/00 , C07C319/14 , C07C323/42 , C07C323/43 , C07C325/00 , C07C333/08 , A01N31/00 , A01N37/00 , A01N37/18 , A01N37/44 , C07C83/10 , C07C103/127 , C07C103/133 , C07C103/19 , C07C125/06 , C07C127/19 , C07C149/40 , C07C155/03
CPC分类号： A01N47/30 , A01N37/24 , A01N47/20 , A01N53/00
摘要： Novel compounds having the formula ##STR1## in which X is (H).sub.2 or (CH.sub.3).sub.2 ; Y is oxygen or sulfur; R.sub.1 is alkyl, lower alkenyl, cyclopropyl, lower alkoxy, thio-lower alkyl or ##STR2## R.sub.2 and R.sub.3 are independently hydrogen, lower alkyl, lower alkenyl, or lower alkoxy and n is 0 or 1. The compounds have been found to possess herbicidal activity.
摘要翻译：具有式（IMA）的新化合物，其中X是（H）2或（CH 3）2; Y是氧或硫; R 1是烷基，低级烯基，环丙基，低级烷氧基，硫代低级烷基或者R 2独立地是氢，低级烷基，低级烯基或低级烷氧基，n是0或1.已经发现这些化合物具有除草活性。

10. 发明授权

US4336058A 2-Methyl-4-(chloroacetamido)methyl-4-(2-chlorophenyl)-1,3-dioxane herbicide antidote 失效
标题翻译： 2-甲基-4-（氯代乙酰氨基）甲基-4-（2-氯苯基）-1,3-二恶烷除草剂解毒剂
公开(公告)号：US4336058A
公开(公告)日：1982-06-22
申请号：US232069
申请日：1981-02-06
申请人： Raymond A. Felix
发明人： Raymond A. Felix
IPC分类号： A01N25/32 , C07D319/06 , A01N43/00 , C07D319/04
CPC分类号： A01N25/32 , C07D319/06
摘要： An herbicide antidote compound having the formula ##STR1## and herbicide antidote compositions comprising (a) an herbicidally effective amount of a thiocarbamate compound of the formula: ##STR2## in which R.sub.1 is alkyl having 1-6 carbon atoms, inclusive; R.sub.2 is selected from the group consisting of alkyl having 1-6 carbon atoms, inclusive; and cyclohexyl; or R.sub.1 and R.sub.2 form indistinguishable parts of a single alkylene ring having 4-10 carbon atoms, inclusive; and R.sub.3 is selected from the group consisting of alkyl having 1-6 carbon atoms, inclusive; haloalkyl wherein halo is selected from the group consisting of chlorine, bromine and iodine and alkyl has 1-6 carbon atoms, inclusive; alkenyl having 2-6 carbon atoms, inclusive; halo alkenyl wherein halo is selected from the group consisting of chlorine, bromine and iodine and alkenyl has 2-6 carbon atoms, inclusive; benzyl; and halo-substituted benzyl, wherein halo is selected from the group consisting of chlorine, bromine and iodine; and(b) an non-phytotoxic antidotally effective amount of a compound of the formula ##STR3##
摘要翻译：具有式“除草剂”的除草剂解毒剂化合物和除草剂解毒剂组合物，其包含（a）除草有效量的下式的硫代氨基甲酸酯化合物：其中R 1是具有1-6个碳原子的烷基; R2选自具有1-6个碳原子的烷基，包括端基; 和环己基; 或R 1和R 2形成具有4-10个碳原子的单个亚烷基环的不可区分的部分，包括端值; 并且R 3选自具有1-6个碳原子的烷基; 卤代烷基，其中卤素选自氯，溴和碘，并且具有1-6个碳原子的烷基; 具有2-6个碳原子的烯基; 卤素烯基，其中卤素选自氯，溴和碘，烯基具有2-6个碳原子; 苄基; 和卤素取代的苄基，其中卤素选自氯，溴和碘; 和（b）非植物毒性解毒有效量的式“IMAGE”化合物

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式