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1. 发明授权

US06673820B2 Aminoheterocyclylamides as pesticides and antiparasitic agents 失效
标题翻译：氨基杂环酰胺作为农药和抗寄生虫剂
公开(公告)号：US06673820B2
公开(公告)日：2004-01-06
申请号：US10148644
申请日：2002-05-31
申请人： Pierre Ducray , Jacques Bouvier , Maurizio Schwarzenbach
发明人： Pierre Ducray , Jacques Bouvier , Maurizio Schwarzenbach
IPC分类号： C07D41712
CPC分类号： C07D275/03 , C07D277/46 , C07D285/08 , C07D333/36 , C07D409/12 , C07D417/12
摘要： The invention relates to novel compounds of the general formula: in which R1 is hydrogen, halogen, C1-C6alkyl, C1-C6alkoxy, C1-C6haloalkyl or unsubstituted or mono- to pentasubstituted phenyl, where the substituents are selected from the group consisting of C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, aryloxy, halogen, cyano and nitro, where, if the number of substituents exceeds 1, the substituents can be identical or different; R2 is hydrogen, C1-C6alkyl, (C1-C6alkylene)phenyl, pyridyl, COOR6, CONR7R8, COR6, allyl or CH2—O—R6; R3 is unsubstituted or substituted heterocyclyl, where the substituents are in each case selected from the group consisting of unsubstituted or substituted phenyl, where the substituents are selected from the group consisting of C1-C6alkyl, C1-C6alkoxy, halogen, cyano and nitro, where, if the number of substituents exceeds 1, the substituents can be identical or different, benzyl, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, aryloxy, halogen, cyano, hydroxyl, amino and nitro, where, if the number of substituents exceeds 1, the substituents can be identical or different; R6 is C1-C6alkyl, phenyl or benzyl; R7 and R8 independently of one another are hydrogen or C1-C6alkyl; X1 and X2 are each N; and X3 is O or S. The novel compounds have advantageous pesticidal properties and are particularly suitable for controlling pests in domestic and useful animals.
摘要翻译：本发明涉及以下通式的新化合物：其中R 1是氢，卤素，C 1 -C 6烷基，C 1 -C 6烷氧基，C 1 -C 6卤代烷基或未被取代的或一至五取代的苯基，其中取代基选自C1 C 1-6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基，芳氧基，卤素，氰基和硝基，其中如果取代数超过1，则取代基可以相同或不同; R2是氢，C1-C6烷基，（C1-C6亚烷基）苯基，吡啶基，COOR6，CONR7R8，COR6，烯丙基或CH2-O-R6; R3是未取代或取代的杂环基，其中取代基各自选自未取代或取代的苯基，其中取代基选自C 1 -C 6烷基，C 1 -C 6烷氧基，卤素，氰基和硝基，其中如果取代基数目超过1，则取代基可以相同或不同，苄基，C1-C6烷基，C1-C6卤代烷基，C1-C6烷氧基，芳氧基，卤素，氰基，羟基，氨基和硝基，其中如果取代基数目超过1，取代基可以相同或不同; R6是C1-C6烷基，苯基或苄基; R 7和R 8彼此独立地是氢或C 1 -C 6烷基; X1和X2分别为N; X3是O或S.新化合物具有有利的杀虫特性，特别适用于控制家畜和有用动物的害虫。

2. 发明授权

US07271184B2 Acyclic and cyclic guanidine- and acetamidine derivatives, their preparation and their use as pesticides, esp. as parasiticides 失效
标题翻译：非环状和环状胍和乙脒衍生物，其制备及其作为农药的用途，作为杀寄生虫剂
公开(公告)号：US07271184B2
公开(公告)日：2007-09-18
申请号：US10779932
申请日：2004-02-17
申请人： Thomas Goebel , Eliane Humbert-Droz , Maurizio Schwarzenbach
发明人： Thomas Goebel , Eliane Humbert-Droz , Maurizio Schwarzenbach
IPC分类号： A61K31/44 , A61K31/425 , C07D277/04 , C07D277/08 , C07D277/20 , C07D275/02 , C07D417/00 , C07D513/00 , A01N43/78 , A01N43/80
CPC分类号： C07D277/32 , A01N47/12 , A01N47/16 , A01N47/44 , C07D213/61 , C07D417/06
摘要： Novel pesticides of formula (I) wherein the substituents, R, R1, R2, R2′, T, U, X and Y are as defined in claim 1, are described. Also described are compositions suitable for use as parasiticides comprising those compounds as active ingredient and to methods of controlling parasites that are based on the administration of those compounds or compositions, and to the use of the said compounds and compositions in a method of controlling parasites and in the manufacture of pesticides for use against parasites. Also described are intermediates of formula (XX) wherein R1, R2, R2′, T, U, X and Y are as defined in claim 1; and Hal is halogen. The latter also exhibit parasiticidal activity and are suitable for the preparation of the compounds of formula (I).
摘要翻译：式（I）的新型农药，其中取代基R 1，R 1，R 2，R 2'，T，U，X和 Y如权利要求1中所定义。还描述了适合用作包含那些化合物作为活性成分的杀寄生虫剂的组合物和控制基于这些化合物或组合物的施用的寄生虫的方法，以及所述化合物和组合物在控制寄生虫和在制造杀虫剂用于对抗寄生虫。还描述了式（XX）的中间体，其中R 1，R 2，R 2'，T，U，X和Y分别为如权利要求1所述; 而Hal是卤素。后者还具有杀寄生虫活性，适用于制备式（I）化合物。

3. 发明授权

US06759407B2 Acyclic and cyclic guanidine- and acetamidine derivatives, their preparation and their use as pesticides, ESP as parasiticides 失效
标题翻译：无环和环胍和脒衍生物，它们的制备及其作为农药的用途，作为杀寄生物的ESP
公开(公告)号：US06759407B2
公开(公告)日：2004-07-06
申请号：US10348574
申请日：2003-01-21
申请人： Thomas Goebel , Eliane Humbert-Droz , Maurizio Schwarzenbach
发明人： Thomas Goebel , Eliane Humbert-Droz , Maurizio Schwarzenbach
IPC分类号： C07D21300
CPC分类号： C07D277/32 , A01N47/12 , A01N47/16 , A01N47/44 , C07D213/61 , C07D417/06
摘要： Novel pesticides of formula (I) wherein the substituents, R, R1, R2, R2′, T, U, X and Y are as defined in claim 1, are described. Also described are compositions suitable for use as parasiticides comprising those compounds as active ingredient and to methods of controlling parasites that are based on the administration of those compounds or compositions, and to the use of the said compounds and compositions in a method of controlling parasites and in the manufacture of pesticides for use against parasites. Also described are intermediates of formula (XX) wherein R1, R2, R2′, T, U, X and Y are as defined in claim 1; and Hal is halogen. The latter also exhibit parasiticidal activity and are suitable for the preparation of the compounds of formula (I).
摘要翻译：描述了式（I）的新型农药，其中取代基R 1，R 2，R 2，R 2'，T，U，X和Y如权利要求1中所定义。还描述了适合用作包含那些化合物作为活性成分的杀寄生虫剂的组合物和控制基于这些化合物或组合物的施用的寄生虫的方法，以及所述化合物和组合物在控制寄生虫和在制造杀虫剂用于对抗寄生虫。还描述了式（XX）的中间体，其中R 1，R 2，R 2'，T，U，X和Y如权利要求1中所定义; 并且Hal是卤素，后者还具有杀寄生虫活性，并且适于制备式（I）化合物。

4. 发明授权

US06538013B2 Acyclic and cyclic guanidine-and acetamidine derivatives, their preparation and their use as pesticides, esp. as parasiticides 失效
标题翻译：非环和环胍和乙脒衍生物，它们的制备及其作为农药的用途，作为杀寄生虫剂
公开(公告)号：US06538013B2
公开(公告)日：2003-03-25
申请号：US09850378
申请日：2001-05-07
申请人： Thomas Goebel , Eliane Humbert-Droz , Maurizio Schwarzenbach
发明人： Thomas Goebel , Eliane Humbert-Droz , Maurizio Schwarzenbach
IPC分类号： C07D21300
CPC分类号： C07D277/32 , A01N47/12 , A01N47/16 , A01N47/44 , C07D213/61 , C07D417/06
摘要： Novel pesticides of formula (I) wherein the substituents R, R1, R2, R2′, T, U, X and Y are as defined in claim 1, are described. Also described are compositions suitable for use as parasiticides comprising those compounds as active ingredient and to methods of controlling parasites that are based on the administration of those compounds or compositions, and to the use of the said compounds and compositions in a method of controlling parasites and in the manufacture of pesticides for use against parasites. Also described are intermediates of formula (XX) wherein R1, R2, R2′, T, U, X and Y are as defined in claim 1 and Hal is halogen. The latter also exhibit parasiticidal activity and are suitable for the preparation of the compounds of formula (I).
摘要翻译：描述了式（I）的新型农药，其中取代基R，R 1，R 2，R 2'，T，U，X和Y如权利要求1中所定义。还描述了适合用作包含那些化合物作为活性成分的杀寄生虫剂的组合物和控制基于这些化合物或组合物的施用的寄生虫的方法，以及所述化合物和组合物在控制寄生虫和在制造杀虫剂用于对抗寄生虫。还描述了式（XX）的中间体，其中R 1，R 2，R 2'，T，U，X和Y如权利要求1中所定义，Hal是卤素。后者还具有杀寄生虫活性，适用于制备式（I）化合物。

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