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1. 发明授权

US4054668A N-substituted amino acid derivatives 失效
标题翻译： N-取代氨基酸衍生物
公开(公告)号：US4054668A
公开(公告)日：1977-10-18
申请号：US619125
申请日：1975-10-02
申请人： Osamu Kirino , Tadashi Ooishi , Nobuyuki Kameda , Toshiro Kato , Akira Fujinami , Toshiaki Ozaki
发明人： Osamu Kirino , Tadashi Ooishi , Nobuyuki Kameda , Toshiro Kato , Akira Fujinami , Toshiaki Ozaki
IPC分类号： A01N37/44 , C07C101/28 , A01N9/24 , A01N9/30 , C07C103/48
CPC分类号： A01N37/44
摘要： Novel N-substituted amino acid derivatives of the formula: ##STR1## wherein R.sub.1 is an alkenyl group having 2 to 5 carbon atoms, a halogen-substituted alkenyl group having 2 to 5 carbon atoms or an alkynyl group having 2 to 5 carbon atoms, R.sub.2 is a methyl or ##STR2## group in which R.sub.2 ' is an alkyl group having 1 to 4 carbon atoms or a halogen-substituted alkyl group having 1 to 4 carbon atoms; and R.sub.3 is a hydrogen atom, an alkyl having 1 to 20 carbon atoms, cycloalkyl having 3 to 6 carbon atoms, benzyl, hydroxyethyl or methoxyethyl group, and inorganic or organic acid addition salts thereof, which possess useful soil fungicidal activities and can be produced by reacting a sarcosine derivative of the formula:CH.sub.3 HNCH.sub.2 COOR.sub.3 (II)wherein R.sub.3 is as defined above, with a halogen compound of the formula:R.sub.1 -- X (III)wherein R.sub.1 is as defined above and X is a halogen atom, or by reacting an N-substituted glycine derivative of the formula: ##STR3## wherein R.sub.1 and R.sub.3 are as defined above, with an acyl compound of the formula: ##STR4## wherein R.sub.2 ' is as defined above and X is a halogen atom.
摘要翻译：式（I）的新型N-取代氨基酸衍生物：其中R 1是具有2至5个碳原子的烯基，具有2至5个碳原子的卤素取代的烯基或具有2至5个炔基的新的N-取代的氨基酸衍生物碳原子，R2是甲基或者基团，其中R2'是具有1至4个碳原子的烷基或具有1至4个碳原子的卤素取代的烷基; R3为氢原子，碳原子数1〜20的烷基，碳原子数为3〜6的环烷基，苄基，羟乙基或甲氧基乙基，以及无机或有机酸加成盐，具有有效的土壤杀真菌活性，通过使下式的肌氨酸衍生物：

2. 发明授权

US4025651A N-substituted-aminoacetamides used as fungicides 失效
标题翻译：用作杀真菌剂的N-取代 - 氨基乙酰胺
公开(公告)号：US4025651A
公开(公告)日：1977-05-24
申请号：US558604
申请日：1975-03-14
申请人： Osamu Kirino , Tadashi Ooishi , Nobuyuki Kameda , Toshiro Kato , Toshiaki Ozaki , Akira Fujinami
发明人： Osamu Kirino , Tadashi Ooishi , Nobuyuki Kameda , Toshiro Kato , Toshiaki Ozaki , Akira Fujinami
IPC分类号： C08K5/00 , A01N37/44 , A61K8/00 , A61K8/42 , A61Q17/00 , B27K3/36 , C07C67/00 , C07C231/00 , C07C231/02 , C07C231/06 , C07C237/06 , C08K5/20 , C08L1/00 , C08L7/00 , C08L21/00 , C08L27/00 , C08L77/00 , C09D7/00 , C09D7/12 , A01N9/20
CPC分类号： A01N37/44
摘要： N-substituted-aminoacetamide compounds having the formula (I) ##STR1## wherein R.sub.1 represents a lower alkenyl group having up to 5 carbon atoms, a halogen-substituted lower alkenyl group having up to 5 carbon atoms or a lower alkynyl group having up to 5 carbon atoms, R.sub.2 and R.sub.3, which may be the same or different, each represents a hydrogen atom or a lower akyl group having up to 4 carbon atoms, and the inorganic and organic acid addition salts thereof, which are useful as fungicidal agents, processesfor preparing N-substituted-aminoacetamide compounds and fungicidal compositions containing at least one compound of the formula (I) as an active inredient.
摘要翻译：具有式（I）的N-取代 - 氨基乙酰胺化合物其中R 1表示具有至多5个碳原子的低级烯基，具有至多5个碳原子的卤素取代的低级链烯基或低级炔基具有至多5个碳原子，可以相同或不同的R 2和R 3各自表示氢原子或具有至多4个碳原子的低级烷基，及其无机和有机酸加成盐，其可用作杀真菌剂，制备N-取代 - 氨基乙酰胺化合物的方法和含有至少一种式（I）化合物作为活性成分的杀真菌组合物。

3. 发明授权

US3966789A N-substituted aminonitrile derivatives 失效
标题翻译： N-取代氨基腈衍生物
公开(公告)号：US3966789A
公开(公告)日：1976-06-29
申请号：US503425
申请日：1974-09-05
申请人： Tadashi Oishi , Nobuyuki Kameda , Toshiro Kato , Akira Fujinami , Toshiaki Ozaki , Eiyashi Itooka
发明人： Tadashi Oishi , Nobuyuki Kameda , Toshiro Kato , Akira Fujinami , Toshiaki Ozaki , Eiyashi Itooka
IPC分类号： A01N37/34 , A01N20060101 , C02F1/50 , C07C20060101 , C07C67/00 , C07C253/00 , C07C255/29 , C07C121/417
摘要： N-substituted aminonitrile derivatives of the formula (I) ##EQU1## wherein R.sub.1, R.sub.2, R.sub.3 and R.sub.4 are as hereinafter defined, useful as fungicides, method for their preparation, and fungicidal compositions containing the N-substituted aminonitrile derivatives of the formula (I).
摘要翻译：式（I）的N-取代的氨基腈衍生物OR2R3 PARALLEL || R1-CNC-CN（I）| R4其中R1，R2，R3和R4如下文所定义，可用作杀真菌剂，其制备方法和杀真菌组合物含有式（I）的N-取代的氨基腈衍生物。

4. 发明授权

US4151290A Fungicidal 1-cycloalkylcarbonyl-3-(3,5-dihalophenyl)imidazolidine-2,4-diones 失效
标题翻译：杀真菌剂1-环烷基羰基-3-（3,5-二卤苯基）咪唑烷-2,4-二酮
公开(公告)号：US4151290A
公开(公告)日：1979-04-24
申请号：US851899
申请日：1977-11-16
申请人： Chiyozo Takayama , Toshiro Kato , Shigeo Yamamoto , Yoshio Hisada , Nobuyuki Kameda , Akira Fujinami
发明人： Chiyozo Takayama , Toshiro Kato , Shigeo Yamamoto , Yoshio Hisada , Nobuyuki Kameda , Akira Fujinami
IPC分类号： A01N47/38 , A01N43/50 , A01N53/00 , A01N53/04 , A01P3/00 , C07D233/80 , A61K31/415
CPC分类号： C07D233/80 , A01N43/50 , A01N53/00
摘要： 1-Cycloalkylcarbonyl-3-(3,5-dihalophenyl)imidazolidine-2,4-diones of the formula: ##STR1## wherein X is a chlorine or bromine atom, R.sub.1 is a C.sub.3 -C.sub.6 cycloalkyl, tetramethylcyclopropyl, 2,2-dimethyl-3-isobutenylcyclopropyl or 2,2-dimethyl-3-dichlorovinylcyclopropyl group and R.sub.2 and R.sub.3 are individually a hydrogen atom or a methyl group, which show high fungicidal activities without any material toxicity to mammals and plants and which can be produced by reacting the corresponding 1-unsubstituted compound with a cycloalkanecarboxylic acid or a reactive derivative thereof.
摘要翻译：下式的1-环烷基羰基-3-（3,5-二卤苯基）咪唑烷-2,4-二酮其中X是氯或溴原子，R 1是C 3 -C 6环烷基，四甲基环丙基，二甲基-3-异丁烯基环丙基或2,2-二甲基-3-二氯乙烯基环丙基，R2和R3分别为氢原子或甲基，它们对哺乳动物和植物没有任何物质毒性，具有高杀真菌活性，可以通过使相应的1-未取代的化合物与环烷烃羧酸或其活性衍生物。

5. 发明授权

US4123549A N-(3,5-dihalophenyl)-.alpha.-spirocycloalkanesuccinimides, and their preparation and use 失效
标题翻译： N-（3,5-二卤代苯基） - {60-螺环烷基琥珀酰亚胺及其制备和用途
公开(公告)号：US4123549A
公开(公告)日：1978-10-31
申请号：US859756
申请日：1977-12-12
申请人： Nobuyuki Kameda , Yoshio Hisada , Chiyozo Takayama , Toshiro Kato , Akira Fujinami
发明人： Nobuyuki Kameda , Yoshio Hisada , Chiyozo Takayama , Toshiro Kato , Akira Fujinami
IPC分类号： A01N37/32 , A01P3/00 , C07D207/40 , C07D209/54 , A61K31/40
CPC分类号： C07D209/54 , A01N37/32
摘要： N-(3,5-Dihalophenyl)-.alpha.-spirocycloalkanesuccinimides of the formula: ##STR1## wherein X is a chlorine or bromine atom and R is a C.sub.3 -C.sub.6 alkylene group, which show high fungicidal activities without any material toxicity to mammals and plants and which can be produced by reacting the corresponding .alpha.-spirocycloalkanesuccinic acid or its anhydride with 3,5-dichloroaniline or 3,5-dibromoaniline.
摘要翻译： N-（3,5-二卤代苯基）-α-螺环烷基琥珀酰亚胺，其结构式如下：其中X为氯或溴原子，R为C3-C6亚烷基，对哺乳动物没有任何物质毒性，具有高杀真菌活性，植物，并且可以通过使相应的α-螺环烷基琥珀酸或其酸酐与3,5-二氯苯胺或3,5-二溴苯胺反应来制备。

6. 发明授权

US4082849A Halogenated N-(3,5-dihalophenyl)cyclopropanedicarboximides 失效
标题翻译：羟基化N-（3,5-二羟基苯基）环丙烷二羧酸
公开(公告)号：US4082849A
公开(公告)日：1978-04-04
申请号：US730984
申请日：1976-10-08
申请人： Nobuyuki Kameda , Yoshio Hisada , Toshiro Kato , Akira Fujinami
发明人： Nobuyuki Kameda , Yoshio Hisada , Toshiro Kato , Akira Fujinami
IPC分类号： A01N53/00 , A01N37/32 , A01N53/12 , A01P1/00 , A01P3/00 , C07D209/52 , A61K31/40
CPC分类号： C07D209/52
摘要： Novel N-(3,5-dihalophenyl)cyclopropanedicarboximides of the formula: ##STR1## wherein X and Y are each a chlorine atom or a bromine atom and R.sub.1, R.sub.2 and R.sub.3 are individually a hydrogen atom or a methyl group, which show high microbicidal activities against various fungi and bacteria without any material toxicity to mammals and plants and which can be produced by reacting the corresponding cyclopropanedicarboxylic acid or its anhydride with a 3,5-dihaloaniline.

7. 发明授权

US4394379A Amide phosphorothiolate derivatives and their use as pesticides 失效
标题翻译：酰胺二硫代磷酸衍生物及其作为农药的用途
公开(公告)号：US4394379A
公开(公告)日：1983-07-19
申请号：US113133
申请日：1980-01-17
申请人： Osamu Kirino , Masachika Hirano , Hisami Takeda , Toshiro Kato
发明人： Osamu Kirino , Masachika Hirano , Hisami Takeda , Toshiro Kato
IPC分类号： A01N57/14 , A01N57/30 , C07F9/165 , C07F9/24 , C07F9/40
CPC分类号： C07F9/1651 , A01N57/14 , A01N57/30 , C07F9/2408
摘要： Amide phosphorothiolate derivatives of the formula, ##STR1## wherein X is an oxygen or sulfur atom, Y is an oxygen or sulfur atom or imino group, R.sub.1 and R.sub.2, which may be the same or different, are each a C.sub.1 -C.sub.3 alkyl group, R.sub.3 is a C.sub.1 -C.sub.4 alkyl group, R.sub.4 is a hydrogen atom or methyl group, R.sub.5 is a C.sub.1 -C.sub.3 alkyl, methoxy or ethoxy group, Z is a hydrogen atom, a methyl group or chlorine atom and n is 1 or 2, a process for producing said derivatives characterized by reacting the salt of thiophosphoric ester represented by the formula, ##STR2## wherein X, Y, R.sub.1 and R.sub.2 are as defined above and M is a sodium or potassium atom or ammonium group, with a haloacetamide derivative of the formula, ##STR3## wherein R.sub.3, R.sub.4, R.sub.5, Z and n are as defined above and W is a halogen atom, and a combined insecticide, acaricide, nematocide and/or fungicide containing said derivatives as an active ingredient.
摘要翻译：下式的酰亚胺硫代衍生物，其中X是氧或硫原子，Y是氧或硫原子或亚氨基，可以相同或不同的R 1和R 2各自为C 1 -C 3烷基 R3为C1-C4烷基，R4为氢原子或甲基，R5为C1-C3烷基，甲氧基或乙氧基，Z为氢原子，甲基或氯原子，n为1或2 制备所述衍生物的方法，其特征在于使由下式表示的硫代磷酸酯的盐，其中X，Y，R 1和R 2如上所定义，M是钠或钾原子或铵基，与卤代乙酰胺衍生物，其中R3，R4，R5，Z和n如上所定义，W是卤素原子，以及含有所述衍生物作为活性成分的杀虫剂，杀螨剂，杀线虫剂和/或杀真菌剂的组合物。

8. 发明授权

US4235925A N-Benzoylanthranilate derivatives as phytopathogenic fungicidal agents 失效
标题翻译： N-苯甲酰基邻氨基苯甲酸酯衍生物作为植物病原性杀真菌剂
公开(公告)号：US4235925A
公开(公告)日：1980-11-25
申请号：US862527
申请日：1977-12-20
申请人： Osamu Kirino , Toshiro Kato , Shigeo Yamamoto
发明人： Osamu Kirino , Toshiro Kato , Shigeo Yamamoto
IPC分类号： A01N37/22 , A01N37/46 , A01N43/30 , A01P3/00 , C07C233/81 , C07D317/68 , A01N43/16 , A01N37/10
CPC分类号： C07D317/68 , A01N37/46 , A01N43/30
摘要： A fungicidal composition which comprises as an active ingredient a N-benzoylanthranilate compound of the formula, ##STR1## wherein X is a hydrogen or 3-halogen atom or a 3-methoxy, 4-methoxy, 2,4-dimethoxy, 3,4-dimethoxy, 3-halo-4-methoxy, 3,4-methylenedioxy or 3,5-dimethoxy group and R is a hydrogen atom or a C.sub.1 -C.sub.7 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.4 alkenyl, halo-C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.4 alkoxy C.sub.1 -C.sub.4 alkyl or N,N-di-C.sub.1 -C.sub.2 alkylamino C.sub.1 -C.sub.4 alkyl group and an inert carrier, and their preparation and use as a fungicide.
摘要翻译：一种杀真菌组合物，其包含下式的N-苯甲酰基邻氨基苯甲酸酯化合物作为活性成分，其中X是氢或3-卤素原子或3-甲氧基，4-甲氧基，2,4-二甲氧基，3,4 二甲氧基，3-卤代-4-甲氧基，3,4-亚甲二氧基或3,5-二甲氧基，R为氢原子或C 1 -C 7烷基，C 3 -C 6环烷基，C 2 -C 4烯基，卤代C1- C 3烷基，C 1 -C 4烷氧基C 1 -C 4烷基或N，N-二-C 1 -C 2烷基氨基C 1 -C 4烷基和惰性载体，及其制备和用作杀真菌剂。

9. 发明授权

US4347188A N-Benzoylanthranilate derivatives 失效
标题翻译： N-苯甲酰基邻氨基苯甲酸酯衍生物
公开(公告)号：US4347188A
公开(公告)日：1982-08-31
申请号：US164886
申请日：1980-06-30
申请人： Osamu Kirino , Toshiro Kato , Shigeo Yamamoto
发明人： Osamu Kirino , Toshiro Kato , Shigeo Yamamoto
IPC分类号： A01N37/46 , A01N43/30 , C07D317/68 , C07D317/44
CPC分类号： A01N37/46 , A01N43/30 , C07D317/68
摘要： A fungicidal composition which comprises as an active ingredient a N-benzoylanthranilate compound of the formula, ##STR1## wherein X is a hydrogen or 3-halogen atom or a 3-methoxy, 4-methoxy, 2,4-dimethoxy, 3,4-dimethoxy, 3-halo-4-methoxy, 3,4-methylenedioxy or 3,5-dimethoxy group and R is a hydrogen atom or a C.sub.1 -C.sub.7 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.4 alkenyl, halo-C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.4 alkoxy C.sub.1 -C.sub.4 alkyl or N,N-di-C.sub.1 -C.sub.2 alkylamino C.sub.1 -C.sub.4 alkyl group and an inert carrier, and their preparation and use as a fungicide.
摘要翻译：一种杀真菌组合物，其包含下式的N-苯甲酰基邻氨基苯甲酸酯化合物作为活性成分，其中X是氢或3-卤素原子或3-甲氧基，4-甲氧基，2,4-二甲氧基，3,4 二甲氧基，3-卤代-4-甲氧基，3,4-亚甲二氧基或3,5-二甲氧基，R为氢原子或C 1 -C 7烷基，C 3 -C 6环烷基，C 2 -C 4烯基，卤代C1- C 3烷基，C 1 -C 4烷氧基C 1 -C 4烷基或N，N-二-C 1 -C 2烷基氨基C 1 -C 4烷基和惰性载体，及其制备和用作杀真菌剂。

10. 发明授权

US4039635A Soil fungicidal phosphorothioate 失效
标题翻译：土壤杀真菌硫代磷酸酯
公开(公告)号：US4039635A
公开(公告)日：1977-08-02
申请号：US642716
申请日：1975-12-22
申请人： Toshiro Kato , Mitsuru Sasaki , Tadashi Ooishi , Kunio Mujai
发明人： Toshiro Kato , Mitsuru Sasaki , Tadashi Ooishi , Kunio Mujai
IPC分类号： A01N57/14 , C07F9/18 , C07F9/36 , C07F9/165 , A01N9/36
CPC分类号： C07F9/18 , A01N57/14
摘要： Novel phosphorothioates represented by the formula, ##STR1## wherein R.sub.1 is a chlorine or bromine atom, R.sub.2 is methyl or ethyl group and R.sub.3 is a chlorine or bromine atom or nitro group, which have a low toxicity to men and beasts as well as fishes, no phytotoxicity to crops, excellent fungicidal effect on injurious epidemic soil fungi in agriculture, horticulture and the like, and a wide range of uses for prevention of soil epidemics to effect the growth promotion of crops.
摘要翻译：由式表示的新型硫代磷酸酯，其中R1是氯或溴原子，R2是甲基或乙基，R3是氯或溴原子或硝基，对人类和野兽以及鱼类具有低毒性对作物没有植物毒性，对农业，园艺等有害流行性土壤真菌具有极好的杀真菌作用，广泛用于预防土壤流行病，促进作物生长发育。

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