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1. 发明授权

US5783580A .alpha.-pyrimidinyl acrylic acid derivatives 失效
标题翻译： α-嘧啶基丙烯酸衍生物
公开(公告)号：US5783580A
公开(公告)日：1998-07-21
申请号：US652865
申请日：1996-05-23
申请人： Martin Eberle , Fritz Schaub , Gerald Wayne Craig
发明人： Martin Eberle , Fritz Schaub , Gerald Wayne Craig
IPC分类号： A01N43/54 , A01N43/78 , A01N43/80 , C07D239/46 , C07D239/52 , C07D405/12 , C07D413/12 , C07D417/12 , C07D521/00 , C07D239/47
CPC分类号： C07D239/47 , A01N43/54 , A01N43/78 , A01N43/80 , C07D231/12 , C07D233/56 , C07D239/52 , C07D249/08 , C07D405/12 , C07D413/12 , C07D417/12
摘要： This invention relates to compounds of formula I ##STR1## wherein R.sup.1 is C.sub.1-4 alkoxy or --NR.sup.8 R.sup.9 ; R.sup.2 is heteroaryl, heteroaryloxy or a group ##STR2## R.sup.3 is hydrogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, cyano, nitro or halogen; R.sup.4 is hydrogen, halogen, C.sub.1-4 alkoxy or C.sub.1-4 alkyl; R.sup.5 is hydrogen or methyl; R.sup.7 is hydrogen or methyl; R.sup.8 and R.sup.9 are independently C.sub.1-4 alkyl or together C.sub.3-6 alkylene; E is C.sub.1-3 alkylene; X is CH or nitrogen; and Y is OCH.sub.3, NH.sub.2, NHCH.sub.3 or N(CH.sub.3).sub.2.
摘要翻译：本发明涉及式Ⅰ化合物其中R 1是C 1-4烷氧基或-NR 8 R 9; R 2是杂芳基，杂芳氧基或基团R 3是氢，C 1-4烷基，C 1-4烷氧基，氰基，硝基或卤素; R4是氢，卤素，C1-4烷氧基或C1-4烷基; R5是氢或甲基; R7是氢或甲基; R 8和R 9独立地为C 1-4烷基或C 3-6亚烷基; E为C1-3亚烷基; X是CH或氮; Y是OCH 3，NH 2，NHCH 3或N（CH 3）2。

2. 发明授权

US5776941A 4-alkylthio-pyrimidin-5-ylacetic acid derivates 失效
标题翻译： 4-烷硫基 - 嘧啶-5-基乙酸衍生物
公开(公告)号：US5776941A
公开(公告)日：1998-07-07
申请号：US606911
申请日：1996-02-26
申请人： Gerald Wayne Craig , Martin Eberle , Fritz Schaub
发明人： Gerald Wayne Craig , Martin Eberle , Fritz Schaub
IPC分类号： A01N43/54 , A01N43/56 , A01N43/78 , A01N43/80 , C07D239/38 , C07D239/56 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/12 , C07D239/46
CPC分类号： C07D239/56 , A01N43/54 , A01N43/80 , C07D239/38 , C07D413/12
摘要： This invention relates to 2-(4-alkylthio-pyrimidin-5-yl)-acetic acid derivatives; fungicidal compositions comprising such compounds and a method of combating phytopathogenic fungi comprising applying such compounds to the fungi or their habitat.
摘要翻译：本发明涉及2-（4-烷硫基 - 嘧啶-5-基） - 乙酸衍生物; 包含这种化合物的杀真菌组合物和防治植物病原真菌的方法包括将这些化合物施用于真菌或其栖息地。

3. 发明授权

US5635508A Pyrimidinyl acrylic acid derivatives 失效
标题翻译：嘧啶丙烯酸衍生物
公开(公告)号：US5635508A
公开(公告)日：1997-06-03
申请号：US435053
申请日：1995-05-08
申请人： Martin Eberle , Fritz Schaub , Gerald W. Craig
发明人： Martin Eberle , Fritz Schaub , Gerald W. Craig
IPC分类号： A01N43/54 , C07D239/34 , C07D239/56 , C07D401/12 , C07D239/46
CPC分类号： C07D401/12 , A01N43/54 , C07D239/34 , C07D239/56
摘要： The invention discloses compounds of formula I It has now been found that compounds of formula I ##STR1## wherein R.sub.1 is hydrogen, methyl, ethyl or trifluoromethyl, andR.sub.2 is hydrogen, methyl, ethyl, C.sub.1-4 alkylthio, C.sub.1-4 alkoxy, or di-C.sub.1-4 alkylamino, andR.sub.3 is C.sub.1-10 alkyl, C.sub.1-10 haloalkyl, aryl, heteroaryl, aryl-C.sub.1-4 alkyl, heteroaryl-C.sub.1-4 alkyl, aryloxy-C.sub.1-4 alkyl, aryloxyaryl, arylaryl, heteroaryl, aryl-C.sub.1-4 alkoxyaryl, aryl-C.sub.1-4 alkoxy-C.sub.1-4 alkyl, heteroaryloxyaryl, aryloxy-C.sub.1-4 alkylaryl or aryl substituted by a group selected from --C(CH.sub.3).dbd.N--O--CH.sub.2 --aryl, --C(CH.sub.3).dbd.N--O--CH(CH.sub.3)--aryl, --C(CH.sub.3).dbd.N--C.sub.1-4 alkoxy, --C(CH.sub.3).dbd.N--C.sub.3-4 alkenyloxy, --C(CH.sub.3).dbd.N--C.sub.3-4 alkynyloxy, or --CH.sub.2 --O--N.dbd.C(CH.sub.3)--aryl, wherein each of the aromatic rings may be optionally substituted;the use of such compounds for the control of phytopathogens, compositions for facilitating such use, and the preparation of the compounds of fomula I.
摘要翻译：本发明公开了式I的化合物现已发现式Ⅰ化合物其中R1是氢，甲基，乙基或三氟甲基，R2是氢，甲基，乙基，C1-4烷硫基，C1-4烷氧基，或二-C 1-4烷基氨基，R 3为C 1-10烷基，C 1-10卤代烷基，芳基，杂芳基，芳基-C 1-4烷基，杂芳基-C 1-4烷基，芳氧基-C 1-4烷基，芳氧基芳基，芳基芳基，杂芳基，芳基-C 烷氧基芳基，芳基-C 1-4烷氧基-C 1-4烷基，杂芳氧基芳基，芳氧基-C 1-4烷基芳基或被选自-C（CH 3）= NO-CH 2 - 芳基，-C（CH 3）= NO-CH （CH 3）= N-C 3-4烷氧基，-C（CH 3）= N-C 3-4炔基氧基或-CH 2 -ON = C（CH 3）） - 芳基，其中每个芳环可以任选被取代; 使用这种化合物来控制植物病原体，促进这种用途的组合物和制备化合物I.

4. 发明授权

US5547919A .alpha.-pyrimidinyl acrylic acid derivatives 失效
标题翻译： α-嘧啶基丙烯酸衍生物
公开(公告)号：US5547919A
公开(公告)日：1996-08-20
申请号：US370992
申请日：1995-01-10
申请人： Martin Eberle , Fritz Schaub , Gerald W. Craig
发明人： Martin Eberle , Fritz Schaub , Gerald W. Craig
IPC分类号： C07D239/47 , A01N43/28 , A01N43/54 , A01N43/56 , A01N43/76 , A01N43/78 , A01N43/80 , C07D239/34 , C07D239/46 , C07D239/52 , C07D317/10 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12 , C07D239/02
CPC分类号： C07D239/47 , A01N43/54 , A01N43/56 , A01N43/76 , A01N43/78 , A01N43/80 , C07D239/52 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12
摘要： The invention discloses compounds of formula I ##STR1## the use of such compounds for the control of phytopathogens, composition for facilitating such use, and the preparation of the compounds of formula I.
摘要翻译：本发明公开了式I的化合物（I）使用这些化合物来控制植物病原体，促进这种用途的组合物和式I化合物的制备。

5. 发明授权

US5453427A Pyrimidinyl acrylic acid derivatives 失效
标题翻译：嘧啶丙烯酸衍生物
公开(公告)号：US5453427A
公开(公告)日：1995-09-26
申请号：US273033
申请日：1994-07-08
申请人： Martin Eberle , Fritz Schaub , Gerald W. Craig
发明人： Martin Eberle , Fritz Schaub , Gerald W. Craig
IPC分类号： A01N43/54 , C07D239/34 , C07D239/56 , C07D401/12 , C07D239/42 , C07D239/52
CPC分类号： C07D401/12 , A01N43/54 , C07D239/34 , C07D239/56
摘要： The invention discloses compounds of formula I It has now been found that compounds of formula I ##STR1## wherein R.sub.1 is hydrogen, methyl, ethyl or trifluoromethyl, andR.sub.2 is hydrogen, methyl, ethyl, C.sub.1-4 alkylthio, C.sub.1-4 alkoxy, or di-C.sub.1-4 alkylamino, andR.sub.3 is C.sub.1-10 alkyl, C.sub.1-10 haloalkyl, aryl, heteroaryl, aryl-C.sub.1-4 alkyl, heteroaryl-C.sub.1-4 alkyl, aryloxy-C.sub.1-4 alkyl, aryloxyaryl, arylaryl, heteroaryl, aryl-C.sub.1-4 alkoxyaryl, aryl-C.sub.1-4 alkoxy-C.sub.1-4 alkyl, heteroaryloxyaryl, aryloxy-C.sub.1-4 alkylaryl or aryl substituted by a group selected from --C(CH.sub.3).dbd.N--O--CH.sub.2 --aryl, --C(CH.sub.3).dbd.N--O--CH(CH.sub.3)--aryl, --C(CH.sub.3).dbd.N--C.sub.1-4 alkoxy, --C(CH.sub.3).dbd.N--C.sub.3-4 alkenyloxy,--C(CH.sub.3).dbd.N--C.sub.3-4 alkynyloxy, or --CH.sub.2 --O--N.dbd.C(CH.sub.3)--aryl, wherein each of the aromatic rings may be optionally substituted;the use of such compounds for the control of phytopathogens, compositions for facilitating such use, and the preparation of the compounds of fomula I.
摘要翻译：本发明公开了式I的化合物现已发现式Ⅰ化合物其中R1是氢，甲基，乙基或三氟甲基，R2是氢，甲基，乙基，C1-4烷硫基，C1-4烷氧基，或二-C 1-4烷基氨基，R 3为C 1-10烷基，C 1-10卤代烷基，芳基，杂芳基，芳基-C 1-4烷基，杂芳基-C 1-4烷基，芳氧基-C 1-4烷基，芳氧基芳基，芳基芳基，杂芳基，芳基-C 烷氧基芳基，芳基-C 1-4烷氧基-C 1-4烷基，杂芳氧基芳基，芳氧基-C 1-4烷基芳基或被选自-C（CH 3）= NO-CH 2 - 芳基，-C（CH 3）= NO-CH （CH 3）= N-C 3-4烷氧基，-C（CH 3）= N-C 3-4炔基氧基或-CH 2 -ON = C（CH 3）） - 芳基，其中每个芳环可以任选被取代; 使用这种化合物来控制植物病原体，促进这种用途的组合物和制备化合物I.

6. 发明授权

US5807863A 2-(4-pyrazolyloxy-pyrimidin-5-yl) acetic acid derivatives 失效
标题翻译： 2-（4-吡唑氧基 - 嘧啶-5-基）乙酸衍生物
公开(公告)号：US5807863A
公开(公告)日：1998-09-15
申请号：US715980
申请日：1996-09-19
申请人： Martin Eberle , Clemens Lamberth , Fritz Schaub
发明人： Martin Eberle , Clemens Lamberth , Fritz Schaub
IPC分类号： C07D239/34 , A01N43/54 , A01N43/56 , A01N43/76 , A01N43/78 , C07D231/02 , C07D231/08 , C07D231/10 , C07D231/22 , C07D239/24 , C07D401/14 , C07D403/12 , C07D409/14 , C07D413/14 , C07D417/14
CPC分类号： C07D401/14 , A01N43/56 , A01N43/76 , A01N43/78 , C07D231/08 , C07D231/22 , C07D403/12 , C07D409/14 , C07D413/14 , C07D417/14
摘要： This invention relates to novel 2-(4-pyrazolyloxy-pyrimidin-5-yl) acetic acid derivatives of formula I ##STR1## wherein R.sub.1 is hydrogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-4 alkylthio, C.sub.3-6 cycloalkyl, or di-C.sub.1-4 alkylamino, R.sub.2 is hydrogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-4 alkylthio, or di-C.sub.1-4 alkyl-amino, R.sub.3 is hydrogen or methyl, R.sub.4 is aryl, aryl-C.sub.1-4 alkyl, heteroaryl, or heteroaryl-C.sub.1-4 alkyl, wherein each of the aromatic rings may be optionally substituted; and X is CH or nitrogen; the use of such compounds for the control of phytopathogens, compositions for facilitating such use, and the preparation of the compounds of formula I.
摘要翻译：本发明涉及式I（I）的新的2-（4-吡唑氧基 - 嘧啶-5-基）乙酸衍生物，其中R 1是氢，C 1-4烷基，C 1-4烷氧基，C 1-4烷硫基，C 3-6环烷基，或二-C 1-4烷基氨基，R 2是氢，C 1-4烷基，C 1-4烷氧基，C 1-4烷硫基或二-C 1-4烷基 - 氨基，R 3是氢或甲基，R 4是芳基，芳基-C 1-4烷基，杂芳基或杂芳基-C 1-4烷基，其中每个芳环可以任选被取代; X为CH或氮; 使用这些化合物来控制植物病原体，促进这种用途的组合物和式I化合物的制备。

7. 发明授权

US5300521A Pyrazoles, fungicidal compositions and use 失效
标题翻译：吡唑类，杀真菌剂和用途
公开(公告)号：US5300521A
公开(公告)日：1994-04-05
申请号：US116234
申请日：1993-09-01
申请人： Martin Eberle , Fritz Schaub
发明人： Martin Eberle , Fritz Schaub
IPC分类号： C07D231/18 , A01N43/56 , A01N43/78 , C07D231/12 , C07D409/06 , C07D417/06
CPC分类号： C07D231/12 , A01N43/56
摘要： The invention compounds of formula I ##STR1## wherein R is H, C.sub.1-4 alkyl; optionally substituted aryl or CF.sub.3 ;Y is C.sub.1-4 alkyl or optionally substituted aryl;A is nitrogen or CH; andZ is optionally substituted hydrocarbyl or optionally substituted heteroaryl;the use of such compounds for the control of phytopathogens, compositions for facilitating such use, and the preparation of compounds of formula I.
摘要翻译：本发明的式I化合物（I）其中R是H，C 1-4烷基; 任选取代的芳基或CF 3; Y为C 1-4烷基或任选取代的芳基; A是氮或CH; Z是任选取代的烃基或任选取代的杂芳基; 使用这些化合物来控制植物病原体，促进这种用途的组合物和式I化合物的制备。

8. 发明授权

US4036980A Ether substituted benzodioxan derivatives 失效
标题翻译：醚取代的苯并二恶烷衍生物
公开(公告)号：US4036980A
公开(公告)日：1977-07-19
申请号：US581509
申请日：1975-05-28
申请人： Fritz Schaub , Hanspeter Schelling
发明人： Fritz Schaub , Hanspeter Schelling
IPC分类号： A01N43/32 , A01N49/00 , C07C43/12 , C07D319/18 , C07D319/20 , C07D319/08 , A01N9/28
CPC分类号： C07D319/20 , C07C323/00 , C07C43/12
摘要： Benzodioxan derivatives of formula, ##STR1## in which R is a group of formula A ##STR2## or of formula B,--(CH.sub.2).sub.p --CR.sub.6 =CR.sub.5 --(CH.sub.2).sub.n --O--R.sub.2 BwhereinR.sub.2 is a hydrocarbon radical, e.g. alkyl or cycloalkyl,R.sub.3 and R.sub.4, independently, are hydrogen or alkyl,R.sub.5 and R.sub.6, independently, are hydrogen or methyl,m, n and p are integers,R.sub.1 is hydrogen or alkyl,X is oxygen or sulphurAndZ is hydrogen or a substituent, e.g. alkyl, are useful as insect and acarid growth inhibiting agents.
摘要翻译：其中R为式A A或式B的基团的苯并二恶烷衍生物，其中R 2为烃基， - （CH 2）p -CR 6 = CR 5 - （CH 2）n O-R 2 B，例如烷基或环烷基，R3和R4独立地是氢或烷基，R5和R6独立地是氢或甲基，M，N和P是整数，R1是氢或烷基，X是氧或硫，Z是氢或取代基，例如烷基，可用作昆虫和螨类生长抑制剂。

9. 发明授权

US3978097A Ether and thioether substituted 3,4-alkylenedioxybenzenes 失效
标题翻译：醚和硫醚取代的3,4-亚烷基二氧基苯
公开(公告)号：US3978097A
公开(公告)日：1976-08-31
申请号：US385738
申请日：1973-08-06
申请人： Fritz Schaub , Hans-Peter Schelling
发明人： Fritz Schaub , Hans-Peter Schelling
IPC分类号： A01N31/04 , A01N33/22 , A01N35/04 , A01N37/10 , A01N37/34 , A01N43/30 , A01N43/32 , A01N49/00 , C07C43/12 , C07C43/13 , C07C45/30 , C07D317/54 , C07D317/06 , C07D317/44 , C07D323/02
CPC分类号： C07D317/54 , C07C43/12 , C07C43/13 , C07C45/30 , Y02P20/55 , Y10S424/12
摘要： The present invention concerns novel aromatic long chain alkenyl ethers and thioethers of the formula: ##EQU1## wherein R.sub.1 is a hydrocarbon group,R.sub.2, r.sub.3 and R.sub.4 are each H or alkyl,R.sub.6 is an aromatic radical,Z is a divalent hydrocarbon group,Y is o or s, andw and n are zero or integers.The compounds are useful insecticides and acaricides.
摘要翻译：本发明涉及下式的新型芳族长链烯基醚和硫醚：R2R4 || R1-YC-（CH2）wZ-CH-（CH2）nCH = CH-R6 | R3其中R1是烃基，R2，R3 和R 4各自为H或烷基，R 6为芳族基团，Z为二价烃基，Y为o或s，W和N为零或整数。

10. 发明授权

US3933804A Insecticidal 1,3-benzodioxol derivatives 失效
标题翻译：杀虫剂1,3-苯并间二氧杂环戊烯衍生物
公开(公告)号：US3933804A
公开(公告)日：1976-01-20
申请号：US472013
申请日：1974-05-21
申请人： Hans-Peter Schelling , Fritz Schaub
发明人： Hans-Peter Schelling , Fritz Schaub
IPC分类号： C07C45/70 , C07C45/71 , C07C47/277 , C07C47/54 , C07C47/575 , C07C49/84 , C07C205/37 , C07D317/52 , C07D317/54 , C07D317/56 , C07D317/62 , C07D317/64
CPC分类号： C07D317/64 , C07C205/37 , C07C321/00 , C07C323/00 , C07C45/513 , C07C45/71 , C07D317/52 , C07D317/54 , C07D317/56 , C07D317/62
摘要： The present invention concerns novel compounds of the formula: ##EQU1## wherein R.sub.2 to R.sub.9 have various significances including e.g. alkyl, X and Y include O and S and s, v, w and z are 0 or whole numbers, Ar.sub.1 is ##SPC1##And R.sub.1 is cycloalkyl or ##SPC2##The compounds possess insecticidal properties.
摘要翻译：本发明涉及下式的新化合物：R4R6R8 || R1（CH2）s-Y-C-C-CR2C = C-（CH2）zX-Ar1 ||| R5R7vR9wR3其中R2至R9具有各种含义，烷基，X和Y包括O和S和s，v，w和z是0或整数，Ar1是AND R1是环烷基或该化合物具有杀虫性质。

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