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1. 发明授权

US5198587A Phenethylamine derivatives 失效
标题翻译：苯乙胺衍生物
公开(公告)号：US5198587A
公开(公告)日：1993-03-30
申请号：US737976
申请日：1991-07-30
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka , Kazuo Honda
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka , Kazuo Honda
IPC分类号： C07C217/60
CPC分类号： C07C217/60
摘要： Phenethylamine derivatives shown by the general formula ##STR1## wherein Ro represents a lower alkyl group; R.sub.1 represents a lower alkyl group or a lower alkoxy group; R.sub.2 represents hydrogen atom or a hydroxyl group; R.sub.3 and R.sub.4 each represents hydrogen atom or a lower alkyl group; R.sub.5 represents hydrogen atom or a lower alkoxy group; X represents oxygen atom or a methylene group; m is an integer of 1-3; and n is an integer of 0-2 and the acid addition salts thereof.These compounds exhibit a strong .alpha.-adrenergic blocking action and are useful as an antihypertensive agent.
摘要翻译：苯乙胺衍生物，其通式为：其中R a代表低级烷基; R1表示低级烷基或低级烷氧基; R2表示氢原子或羟基; R3和R4各自表示氢原子或低级烷基; R5表示氢原子或低级烷氧基; X表示氧原子或亚甲基; m为1-3的整数; n为0-2的整数，及其酸加成盐。这些化合物表现出强的α-肾上腺素能阻断作用，可用作抗高血压药。

2. 发明授权

US4880841A Process of producing phenethylamine derivatives 失效
标题翻译：生产苯乙胺衍生物的方法
公开(公告)号：US4880841A
公开(公告)日：1989-11-14
申请号：US307200
申请日：1989-02-03
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka , Kazuo Honda
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka , Kazuo Honda
IPC分类号： A61K20060101 , A61K31/135 , A61K31/255
CPC分类号： A61K31/135 , A61K31/255
摘要： Phenethylamine derivatives shown by the general formula ##STR1## wherein Ro represents a lower alkyl group; R.sub.1 represents a lower alkyl group or a lower alkoxy group; R.sub.2 represents hydrogen atom or a hydroxyl group; R.sub.3 and R.sub.4 each represents hydrogen atom or a lower alkyl group; R.sub.5 represents hydrogen atom or a lower alkoxy group; X represents oxygen atom or a methylene group; m is an integer of 1 -3; and n is an integer of 0-2 and the acid addition salts thereof.These compounds exhibit a strong .alpha.-adreneregic blocking action and are useful as an antihypertensive agent.
摘要翻译：苯乙胺衍生物，其通式为：其中R a代表低级烷基; R1表示低级烷基或低级烷氧基; R2表示氢原子或羟基; R3和R4各自表示氢原子或低级烷基; R5表示氢原子或低级烷氧基; X表示氧原子或亚甲基; m为1-3的整数; n为0-2的整数，及其酸加成盐。这些化合物表现出强烈的α肾上腺素能阻断作用，可用作抗高血压药。

3. 发明授权

US5063246A Phenethylamine derivative compositions and use 失效
标题翻译：苯乙烯衍生物组合物和用途
公开(公告)号：US5063246A
公开(公告)日：1991-11-05
申请号：US569780
申请日：1990-08-21
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka , Kazuo Honda
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka , Kazuo Honda
IPC分类号： A61K20060101 , A61K31/135 , A61K31/255
CPC分类号： A61K31/135 , A61K31/255
摘要： Phenethylamine derivatives shown by the general formula ##STR1## wherein Ro represents a lower alkyl group; R.sub.1 represents a lower alkyl group or a lower alkoxy group, R.sub.2 represents hydrogen atom or a hydroxyl group; R.sub.3 and R.sub.4 each represents hydrogen atom or a lower alkyl group; R.sub.5 represents hydrogen atom or a lower alkoxy group; X represents oxygen atom or a methylene group; m is an integer of 1-3; and n is an integer of 0-2and the acid addition salts thereof.These compounds exhibit a strong .alpha.-adrenergic blocking action and are useful as an antihypertensive agent.

4. 发明授权

US4558156A Sulfamoyl-substituted phenethylamine derivatives 失效
标题翻译：磺酰基取代的苯乙胺衍生物
公开(公告)号：US4558156A
公开(公告)日：1985-12-10
申请号：US632258
申请日：1984-07-18
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
IPC分类号： A61K31/18 , C07C311/15 , C07D203/10 , C07C143/78
CPC分类号： C07D203/10 , C07C309/00
摘要： Novel sulfamoyl-substituted phenethylamine derivatives which exhibit .alpha.-adrenergic blocking action and are useful as an antihypertensive agent and an agent for the treatment of congestive heart failure.
摘要翻译：新的氨磺酰取代的苯乙胺衍生物，其表现出α-肾上腺素能阻断作用并且可用作抗高血压剂和用于治疗充血性心力衰竭的药剂。

5. 发明授权

US4373106A Sulfamoyl-substituted phenethylamine derivatives and process of producing them 失效
标题翻译：磺酰基取代的苯乙胺衍生物及其制备方法
公开(公告)号：US4373106A
公开(公告)日：1983-02-08
申请号：US231421
申请日：1981-02-04
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
IPC分类号： A61K31/18 , A61K31/205 , A61K31/255 , A61P9/04 , A61P9/12 , C07C67/00 , C07C301/00 , C07C303/40 , C07C311/15 , C07C311/16 , C07C311/29 , C07C311/37 , C07C317/00 , C07D203/10 , C07C143/80
CPC分类号： C07D203/10 , C07C309/00
摘要： Novel sulfamoyl-substituted phenethylamine derivatives which exhibit .alpha.-adrenergic blocking action and are useful as an antihypertensive agent and an agent for the treatment of congestive heart failure.
摘要翻译：新的氨磺酰取代的苯乙胺衍生物，其表现出α-肾上腺素能阻断作用并且可用作抗高血压剂和用于治疗充血性心力衰竭的药剂。

6. 发明授权

US4703063A Sulfamoyl substituted phenethylamine derivatives and process of producing them 失效
标题翻译：磺酰胺取代的苯乙胺衍生物及其制备方法
公开(公告)号：US4703063A
公开(公告)日：1987-10-27
申请号：US756790
申请日：1985-07-18
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
IPC分类号： A61K31/18 , A61K31/205 , A61K31/255 , A61P9/04 , A61P9/12 , C07C67/00 , C07C301/00 , C07C303/40 , C07C311/15 , C07C311/16 , C07C311/29 , C07C311/37 , C07C317/00 , C07D203/10 , C07C143/78 , C07C143/80
CPC分类号： C07D203/10 , C07C309/00
摘要： Novel sulfamoyl-substituted phenethylamine derivatives which exhibit .alpha.-adrenergic blocking action and are useful as an antihypertensive agent and an agent for the treatment of congestive heart failure.

7. 发明授权

US4217305A Phenylethanolamine derivatives 失效
标题翻译：苯乙醇胺衍生物
公开(公告)号：US4217305A
公开(公告)日：1980-08-12
申请号：US946192
申请日：1978-09-27
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
IPC分类号： C07C311/37 , A61K31/137 , A61P9/12 , C07C43/23 , C07C317/32 , C07C323/67 , C07D303/34 , C07D317/64 , C07D319/20 , C07C143/78 , A61K31/18 , A61K31/335 , C07D319/18
CPC分类号： C07D317/64 , C07C43/23 , C07D303/34 , C07D319/20
摘要： Novel phenylethanolamine derivatives represented by the formula ##STR1## wherein R represents a hydrogen atom, a halogen atom, a hydroxyl group, a lower alkyl group, a lower alkoxy group, a lower alkylthio group, an amino group, a lower acylamino group, a lower alkylsulfonyl group, or a lower alkylsulfonylamino group; R.sub.1, R.sub.2, R.sub.3 and R.sub.4, which may be the same or different, each represents hydrogen or a lower alkyl group; R.sub.5 represents an aryl group which may have a substituent, a benzodioxane ring group which may have a substituent, an aryloxy group which may have a substituent, or an arylthio group which may have a substituent; said R.sub.5 being, however, a benzodioxane ring group which may have a substituent, an aryloxy group which may have a substituent, or an arylthio group which may have a substituent when R is a hydroxyl group; and n represents 0 or an integer of 1-3 and the acid addition salts thereof.The compounds of this invention exhibit .alpha.- and .beta.-adrenergic blocking actions and are useful as antihypertensive agents.
摘要翻译：其中R表示氢原子，卤素原子，羟基，低级烷基，低级烷氧基，低级烷硫基，氨基，低级酰氨基，低级烷基氨基，低级烷基磺酰基或低级烷基磺酰基氨基; R 1，R 2，R 3和R 4可以相同或不同，各自表示氢或低级烷基; R5表示可以具有取代基的芳基，可以具有取代基的苯并二恶烷环基，可以具有取代基的芳氧基或可以具有取代基的芳硫基; 然而，R 5表示可以具有取代基的苯并二恶烷环基，可以具有取代基的芳氧基或当R为羟基时可具有取代基的芳硫基; n表示0或1-3的整数，以及其酸加成盐。本发明的化合物显示出α-和β-肾上腺素能阻断作用并且可用作抗高血压药。

8. 发明授权

US4868216A Sulfamoyl-substituted phenethylamine derivatives and process of producing them 失效
标题翻译：磺酰基取代的苯乙胺衍生物及其制备方法
公开(公告)号：US4868216A
公开(公告)日：1989-09-19
申请号：US311366
申请日：1989-02-14
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto , Toichi Takenaka
IPC分类号： A61K31/18 , A61K31/205 , A61K31/255 , A61P9/04 , A61P9/12 , C07C67/00 , C07C301/00 , C07C303/40 , C07C311/15 , C07C311/16 , C07C311/29 , C07C311/37 , C07C317/00 , C07D203/10
CPC分类号： C07D203/10 , C07C309/00
摘要： Novel sulfamoyl-substituted phenethylamine derivatives which exhibit .alpha.-adrenergic blocking action and are useful as an antihypertensive agent and an agent for the treatment of congestive heart failure.

9. 发明授权

US4987152A Use of sulfamoyl-substituted phenethylamine derivatives in treatment of lower urinary tract dysfunction 失效
标题翻译：使用氨磺酰取代的苯乙胺衍生物治疗下尿路功能障碍
公开(公告)号：US4987152A
公开(公告)日：1991-01-22
申请号：US436125
申请日：1989-11-13
申请人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto
发明人： Kazuo Imai , Kunihiro Niigata , Takashi Fujikura , Shinichi Hashimoto
IPC分类号： A61K31/18 , A61K31/205 , A61K31/255 , A61P9/04 , A61P9/12 , C07C67/00 , C07C301/00 , C07C303/40 , C07C311/15 , C07C311/16 , C07C311/29 , C07C311/37 , C07C317/00 , C07D203/10
CPC分类号： C07D203/10 , C07C309/00
摘要： Novel sulfamoyl-substituted phenethylamine derivatives which exhibit .alpha.-adrenergic blocking action and are useful as an antihypertensive agent and an agent for the treatment of congestive heart failure.

10. 发明申请

US20050174336A1 Tablet apparatus 有权
标题翻译：平板电脑
公开(公告)号：US20050174336A1
公开(公告)日：2005-08-11
申请号：US11051289
申请日：2005-02-04
申请人： Naomi Nakayama , Kazuo Imai , Yoshiaki Yamaguchi , Isamu Saito
发明人： Naomi Nakayama , Kazuo Imai , Yoshiaki Yamaguchi , Isamu Saito
IPC分类号： G06F3/045 , G06F3/00 , G06F3/01 , G09G5/00
CPC分类号： G06F3/016 , G06F3/045
摘要： A pair of piezoelectric substrates, the length of which is shorter than the length of one side in the longitudinal direction of the operation panel or the supporting board, is respectively fixed to one side from the diagonal position along the longitudinal direction. At the time of detecting an inputting operation, a drive voltage is applied and the entire operation panel or the supporting board is vibrated. Even when the four corners of the operation panel or the supporting board are supported by the housing for accommodating the tablet apparatus or supported by the display device so that the vibration of the four corners is restricted, since either of the pair of piezoelectric substrates, which becomes a vibration source, a feeling of inputting operation can be transmitted to an operator by the vibration, the amplitude of which is not less than a predetermined value, irrespective of the inputting operation position.
摘要翻译：长度比操作面板或支撑板的长度方向上的一侧的长度短的一对压电基板分别从纵向的对角线位置固定在一侧。在检测到输入操作时，施加驱动电压，整个操作面板或支撑板振动。即使当操作面板或支撑板的四个角由用于容纳平板设备的壳体或由显示装置支撑的壳体支撑，使得四个角的振动受到限制时，由于一对压电基板中的任一个成为振动源，不管输入操作位置如何，可以通过振幅不小于预定值的振动将操作感觉发送给操作者。

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