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1. 发明授权

US4634465A Fused N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N'triazinylureas 失效
标题翻译：熔融的N-苯基磺酰基-N'-嘧啶基脲和N-苯基磺酰基-N'-三嗪基脲
公开(公告)号：US4634465A
公开(公告)日：1987-01-06
申请号：US512091
申请日：1983-07-08
申请人： Josef Ehrenfreund , Werner Fory , Willy Meyer , Werner Topfl
发明人： Josef Ehrenfreund , Werner Fory , Willy Meyer , Werner Topfl
IPC分类号： A01N47/36 , C07D209/08 , C07D215/00 , C07D215/36 , C07D239/00 , C07D251/00 , C07D307/00 , C07D307/79 , C07D307/82 , C07D307/83 , C07D307/88 , C07D311/00 , C07D311/18 , C07D311/20 , C07D311/22 , C07D311/58 , C07D311/70 , C07D311/76 , C07D317/00 , C07D317/46 , C07D317/62 , C07D319/00 , C07D319/18 , C07D327/00 , C07D327/04 , C07D327/06 , C07D333/00 , C07D333/54 , C07D333/62 , C07D335/00 , C07D335/06 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D411/12 , C07D417/12 , C07D521/00
CPC分类号： C07D307/79 , A01N47/36 , C07D209/08 , C07D215/36 , C07D307/83 , C07D307/88 , C07D311/18 , C07D311/22 , C07D311/58 , C07D311/70 , C07D311/76 , C07D317/46 , C07D317/62 , C07D319/18 , C07D327/06 , C07D333/54 , C07D335/06 , C07D521/00
摘要： The invention relates to N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N-triazinylureas of the general formula ##STR1## wherein Z is oxygen or sulfur,E is nitrogen or .dbd.CH--,R.sub.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 alkoxycarbonyl, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkylsulfinyl, C.sub.1 -C.sub.4 alkylsulfonyl or C.sub.2 -C.sub.5 alkoxyalkoxy,R.sub.2 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.3 alkoxy,R.sub.3 and R.sub.4, each independently of the other, are hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 haloalkylthio, C.sub.1 -C.sub.4 alkylthio, halogen, C.sub.2 -C.sub.5 alkoxyalkyl, C.sub.2 -C.sub.5 alkoxyalkoxy or --NR.sub.5 R.sub.6, wherein R.sub.5 and R.sub.6 are hydrogen or C.sub.1 -C.sub.4 alkyl, andA is an unsubstituted or substituted bridge of 3 or 4 atoms which contains 1 or 2 oxygen, sulfur or nitrogen atoms and, together with the linking carbon atom, forms a non-aromatic 5- or 6-membered heterocyclic ring system, with the proviso that two oxygen atoms are separated by at least one carbon atom and that oxygen and sulfur atoms are only linked to each other if the sulfur atom takes the form of the --SO-- or --SO.sub.2 -- group;and to the salts of these compounds with amines, alkali metal bases or alkaline earth metal bases or with quaternary ammonium bases. These compounds have good pre- and postemergence selective herbicidal and growth regulating properties.
摘要翻译：本发明涉及通式为（I）的N-苯基磺酰基-N'-嘧啶基脲和N-苯基磺酰基-N-三嗪基脲，其中Z是氧或硫，E是氮或= CH-，R 1是氢，卤素，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4烷氧基羰基，C1-C4烷硫基，C1-C4烷基亚磺酰基，C1-C4烷基磺酰基或C2-C5烷氧基烷氧基，R2是氢，C 1 -C 4烷基或C 1 -C 3烷氧基，R 3和R 4各自独立地是氢，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基，C 1 -C 4卤代烷硫基，C 1 -C 4烷硫基，卤素，C 2 -C 5烷氧基烷基，C 2 -C 5烷氧基烷氧基或-NR 5 R 6，其中R 5和R 6是氢或C 1 -C 4烷基，A是3或4个原子的未取代或取代的桥，其含有1或2个氧，硫或氮原子，并与连接碳原子一起形成非芳族的5或6元杂环系，条件是两个氧原子被至少一个碳原子隔开，而氧如果硫原子是-SO-或-SO 2 - 基团的形式，则硫原子彼此相连; 以及这些化合物与胺，碱金属碱或碱土金属碱或季铵碱的盐。这些化合物具有良好的芽前和芽后选择性除草和生长调节性质。

2. 发明授权

US4677212A Intermediate 1,2-benzoxathiin derivatives 失效
标题翻译：中间体1,2-苯并恶嗪衍生物
公开(公告)号：US4677212A
公开(公告)日：1987-06-30
申请号：US658003
申请日：1984-10-04
申请人： Josef Ehrenfreund , Werner Fory , Willy Meyer , Werner Topfl
发明人： Josef Ehrenfreund , Werner Fory , Willy Meyer , Werner Topfl
IPC分类号： A01N47/36 , C07D209/08 , C07D215/00 , C07D215/36 , C07D239/00 , C07D251/00 , C07D307/00 , C07D307/79 , C07D307/82 , C07D307/83 , C07D307/88 , C07D311/00 , C07D311/18 , C07D311/20 , C07D311/22 , C07D311/58 , C07D311/70 , C07D311/76 , C07D317/00 , C07D317/46 , C07D317/62 , C07D319/00 , C07D319/18 , C07D327/00 , C07D327/04 , C07D327/06 , C07D333/00 , C07D333/54 , C07D333/62 , C07D335/00 , C07D335/06 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D411/12 , C07D417/12 , C07D521/00
CPC分类号： C07D307/79 , A01N47/36 , C07D209/08 , C07D215/36 , C07D307/83 , C07D307/88 , C07D311/18 , C07D311/22 , C07D311/58 , C07D311/70 , C07D311/76 , C07D317/46 , C07D317/62 , C07D319/18 , C07D327/06 , C07D333/54 , C07D335/06 , C07D521/00
摘要： The invention relates to N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N-triazinylureas of the general formula ##STR1## wherein Q is selected from a radical ##STR2## Z is oxygen or sulfur, E is nitrogen or .dbd.CH--,R.sub.2 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.3 alkoxy, andR.sub.3 and R.sub.4, each independently of the other, are hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 haloalkylthio, C.sub.1 -C.sub.4 alkylthio, halogen, C.sub.2 -C.sub.5 alkoxyalkyl, C.sub.2 -C.sub.5 alkoxyalkoxy or --NR.sub.5 R.sub.6, wherein R.sub.5 and R.sub.6 are hydrogen or C.sub.1 -C.sub.4 alkyl,and to the salts of these compounds with amines, alkali metal bases or alkaline earth metal bases or with quaternary ammonium bases. These compounds have good pre- and postemergence selective herbicidal and growth regulating properties.
摘要翻译：本发明涉及通式为（I）的N-苯基磺酰基-N'-嘧啶基脲和N-苯基磺酰基-N-三嗪基脲，其中Q选自基团Z是氧或硫，E是氮或= CH-，R 2是氢，C 1 -C 4烷基或C 1 -C 3烷氧基，R 3和R 4各自独立地是氢，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4 卤代烷氧基，C 1 -C 4卤代烷硫基，C 1 -C 4烷硫基，卤素，C 2 -C 5烷氧基烷基，C 2 -C 5烷氧基烷氧基或-NR 5 R 6，其中R 5和R 6是氢或C 1 -C 4烷基，以及这些化合物与胺，碱金属碱或碱土金属碱或季铵碱。这些化合物具有良好的芽前和芽后选择性除草和生长调节性质。

3. 发明授权

US4675417A Fused phenylsulfonamides 失效
标题翻译：稠油苯磺酰胺
公开(公告)号：US4675417A
公开(公告)日：1987-06-23
申请号：US825282
申请日：1986-02-03
申请人： Josef Ehrenfreund , Werner Fory
发明人： Josef Ehrenfreund , Werner Fory
IPC分类号： A01N47/36 , C07D217/24 , C07D279/02 , C07D311/18 , C07D311/76 , C07D327/06 , C07D335/06 , C07D339/08 , C07D401/12 , C07D411/12 , C07D521/00
CPC分类号： C07D521/00 , A01N47/36 , C07D217/24 , C07D327/06
摘要： Fused N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N'-triazinylureas of the general formula ##STR1## wherein Z is oxygen or sulfur,E is nitrogen or .dbd.CH--,R.sup.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, cyano, or a --X--R.sup.5, --CO--X--R.sup.6, --CO--NR.sup.7 R.sup.8, --SO--R.sup.9 or --SO.sub.2 --R.sup.10 group,R.sup.2 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkoxy,R.sup.3 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or C.sub.3 -C.sub.6 cycloalkyl,R.sup.4 is hydrogen, halogen, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.2 -C.sub.4 alkoxyalkoxy, C.sub.3 -C.sub.6 cycloalkyl or --NR.sup.11 R.sup.12,R.sup.5 is C.sub.3 -C.sub.5 alkynyl or C.sub.1 -C.sub.4 alkyl which is unsubstituted or substituted by halogen or C.sub.1 -C.sub.4 alkoxy, or is C.sub.3 -C.sub.5 alkenyl, which is unsubstituted or is substituted by halogen or C.sub.1 -C.sub.4 -alkoxy,R.sup.6 and R.sup.9 are each independently C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkylalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.7 and R.sup.8 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.5 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.10 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or --NR.sup.13 R.sup.14,R.sup.11 and R.sup.12 are each independently hydrogen or C.sub.1 -C.sub.4 alkyl,R.sup.13 and R.sup.14 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,X is oxygen or sulfur, andA is an unsubstituted or substituted unsaturated bridge of 4 atoms, of the formula --CH.dbd.CH--Y--, wherein Y is a bridge member of 2 atoms which is selected from the series consisting of --NH--CO--, --NH--SO.sub.2 --, --S--CO--, --S--SO.sub.2 --, --O--CO-- or --O--SO.sub.2 --,and the salts thereof with amines, alkali metal or alkaline earth metal bases or with quaternary ammonium bases, have good pre- and postemergence selective herbicidal and growth regulating properties.
摘要翻译：熔融的N-苯基磺酰基-N'-嘧啶基脲和通式为（I）的N-苯基磺酰基-N'-三嗪基脲其中Z是氧或硫，E是氮或= CH-，R 1是氢，卤素，硝基，C1-C4烷基，C1-C4卤代烷基，氰基或-X-R5，-CO-X-R6，-CO-NR7R8，-SO-R9或-SO2-R10基团，R2是氢，C1-C4烷基或C1 -C4烷氧基，R3是C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C3-C6环烷基，R4是氢，卤素，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C2-C4烷氧基烷氧基，C3-C6环烷基或-NR 11 R 12，R 5为未被取代或被卤素或C 1 -C 4烷氧基取代的C 3 -C 5炔基或C 1 -C 4烷基，或未被取代或被卤素或C 1 -C 4 - 烷氧基取代的C 3 -C 5烯基，R 6和R 9为 C 1 -C 4烷基，C 3 -C 5链烯基，C 3 -C 5炔基，苯基或苄基，R 7和R 8各自独立地为氢，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基， C5-C5炔基，苯基或苄基，R10是C1-C4 烷基，C1-C4烷氧基，C1-C4卤代烷氧基或-NR13R14，R11和R12各自独立地为氢或C1-C4烷基，R13和R14各自独立地为氢，C1-C4烷基，C1-C4卤代烷基，C2-C4烷氧基烷基，C3-C5烯基，C3 C 5炔基，苯基或苄基，X是氧或硫，A是4个原子的未取代或取代的不饱和桥，其具有式-CH = CH-Y-，其中Y是2个原子的桥连，由-NH-CO-，-NH-SO2-，-S-CO-，-S-SO2-，-O-CO-或-O-SO2-组成的系列及其与胺，碱金属或碱土金属碱基或季铵碱，具有良好的芽前和芽后选择性除草和生长调节性质。

4. 发明授权

US4675046A Fused N-phenylsulfonyl-N'-pyrimidinylureas 失效
标题翻译：熔融的N-苯基磺酰基-N'-嘧啶基脲
公开(公告)号：US4675046A
公开(公告)日：1987-06-23
申请号：US825283
申请日：1986-02-03
申请人： Josef Ehrenfreund , Werner Fory
发明人： Josef Ehrenfreund , Werner Fory
IPC分类号： A01N47/36 , C07D217/24 , C07D279/02 , C07D311/18 , C07D311/76 , C07D327/06 , C07D335/06 , C07D339/08 , C07D401/12 , C07D411/12 , C07D521/00 , C07D239/69 , A01N43/54
CPC分类号： C07D521/00 , A01N47/36 , C07D217/24 , C07D327/06
摘要： N-phenylsulfonyl-N'-pyrimidinylureas of the formula ##STR1## wherein Z is oxygen or sulfur,R.sup.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, cyano, or a --X--R.sup.5, --CO--X--R.sup.6, --CO--NR.sup.7 R.sup.8, --SO--R.sup.9 or --SO.sub.2 --R.sup.10 group,R.sup.2 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkoxy,R.sup.3 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or C.sub.3 -C.sub.6 cycloalkyl,R.sup.4 is hydrogen, halogen, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.2 -C.sub.4 alkoxyalkoxy, C.sub.3 -C.sub.6 cycloalkyl or --NR.sup.11 R.sup.12,R.sup.5 is C.sub.3 -C.sub.5 alkynyl or C.sub.1 -C.sub.4 alkyl which is unsubstituted or substituted by halogen or C.sub.1 -C.sub.4 -alkoxy, or is C.sub.3 -C.sub.5 alkenyl, which is unsubstituted or is substituted by halogen or C.sub.1 -C.sub.4 -alkoxy,R.sup.6 and R.sup.9 are each independently C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.7 and R.sup.8 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.10 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or --NR.sup.13 R.sup.14,R.sup.11 and R.sup.12 are each independently hydrogen or C.sub.1 -C.sub.4 alkyl,R.sup.13 and R.sup.14 are each independently hydrogen C.sub.1 -C.sub.4 alkyl C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl, andX is oxygen or sulfur,or a salt thereof have good pre and post-emergence selective herbicidal and growth regulating properties.
摘要翻译： N-苯基磺酰基-N'-嘧啶基脲，其中Z是氧或硫，R 1是氢，卤素，硝基，C 1 -C 4烷基，C 1 -C 4卤代烷基，氰基或-X-R 5，-CO-X -R6，-CO-NR7R8，-SO-R9或-SO2-R10基团，R2是氢，C1-C4烷基或C1-C4烷氧基，R3是C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C3 -C 6环烷基，R 4是氢，卤素，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基，C 2 -C 4烷氧基烷氧基，C 3 -C 6环烷基或-NR 11 R 12，R 5是未被取代或被卤素或C1取代的C 3 -C 5炔基或C 1 -C 4烷基 C 4 - 烷氧基，或者是未被取代或被卤素或C 1 -C 4烷氧基取代的C 3 -C 5烯基，R 6和R 9各自独立地为C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基， C 3 -C 5炔基，苯基或苄基，R 7和R 8各自独立地为氢，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基，C 3 -C 5炔基，苯基或苄基，R 10为C 1 -C 4烷基，C 1 -C 4烷氧基， C1-C4卤代烷氧基或-NR13R14，R11和R12各自独立地表示 R 13和R 14各自独立地为C 1 -C 4烷基C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基，C 3 -C 5炔基，苯基或苄基，X为氧或硫或其盐具有良好的前期和后期选择性除草和生长调节性质。

5. 发明授权

US4589911A Fused N-phenylsulfonyl-N-triazinylureas 失效
标题翻译：熔融的N-苯基磺酰基-N-三嗪基脲
公开(公告)号：US4589911A
公开(公告)日：1986-05-20
申请号：US606076
申请日：1984-05-01
申请人： Josef Ehrenfreund , Werner Fory
发明人： Josef Ehrenfreund , Werner Fory
IPC分类号： A01N47/36 , C07D217/24 , C07D279/02 , C07D311/18 , C07D311/76 , C07D327/06 , C07D335/06 , C07D339/08 , C07D401/12 , C07D411/12 , C07D521/00 , A01N43/68 , A01N43/70
CPC分类号： C07D521/00 , A01N47/36 , C07D217/24 , C07D327/06
摘要： Fused N-phenylsulfonyl-N'-triazinylurea of formula I ##STR1## wherein Z is oxygen or sulfur,R.sup.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, cyano, or a --X--R.sup.5, --CO--X--R.sup.6, --CO--NR.sup.7 R.sup.8, --SO--R.sup.9 or --SO.sub.2 --R.sup.10 group,R.sup.2 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkoxy,R.sup.3 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or C.sub.3 -C.sub.6 cycloalkyl,R.sup.4 is hydrogen, halogen, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.2 -C.sub.4 alkoxyalkoxy, C.sub.3 -C.sub.6 cycloalkyl or --NR.sup.11 R.sup.12,R.sup.5 is C.sub.3 -C.sub.5 alkynyl or C.sub.1 -C.sub.4 alkyl which is unsubstituted or substituted by halogen or C.sub.1 -C.sub.4 -alkoxy, or is C.sub.3 -C.sub.5 alkenyl, which is unsubstituted or is substituted by halogen or C.sub.1 -C.sub.4 -alkoxy,R.sup.6 and R.sup.9 are each independently C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.7 and R.sup.8 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.10 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or --NR.sup.13 R.sup.14,R.sup.11 and R.sup.12 are each independently hydrogen or C.sub.1 -C.sub.4 alkyl,R.sup.13 and R.sup.14 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl, andX is oxygen or sulfur,or a salt thereof have good pre and post-emergence selective herbicidal and growth regulating properties.
摘要翻译：熔融的式I的N-苯基磺酰基-N'-三嗪基脲其中Z是氧或硫，R 1是氢，卤素，硝基，C 1 -C 4烷基，C 1 -C 4卤代烷基，氰基或-X-R 5， -CO-X-R6，-CO-NR7R8，-SO-R9或-SO2-R10基，R2是氢，C1-C4烷基或C1-C4烷氧基，R3是C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1 C 4卤代烷氧基或C 3 -C 6环烷基，R 4是氢，卤素，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基，C 2 -C 4烷氧基烷氧基，C 3 -C 6环烷基或-NR 11 R 12，R 5是未被取代或取代的C 3 -C 5炔基或C 1 -C 4烷基或未被取代或被卤素或C 1 -C 4 - 烷氧基取代的C 3 -C 5烯基，R 6和R 9各自独立地为C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 4烷氧基， C5链烯基，C3-C5炔基，苯基或苄基，R7和R8各自独立地为氢，C1-C4烷基，C1-C4卤代烷基，C2-C4烷氧基烷基，C3-C5烯基，C3-C5炔基，苯基或苄基，R10为C1-C4烷基，C1- C4烷氧基，C1-C4卤代烷氧基或-NR13R14，R11和R12各自为吲哚基 R 1和R 4各自独立地为氢，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基，C 3 -C 5炔基，苯基或苄基，X为氧或硫或其盐具有良好的芽前和出苗后选择性除草和生长调节性质。

6. 发明授权

US08003626B2 Pyrazole-4-carboxamide derivatives as microbiocides 失效
标题翻译：吡唑-4-甲酰胺衍生物作为杀微生物剂
公开(公告)号：US08003626B2
公开(公告)日：2011-08-23
申请号：US11996094
申请日：2006-07-17
申请人： Clemens Lamberth , Camilla Corsi , Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Clemens Lamberth , Camilla Corsi , Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A01N57/00 , C07D231/06
CPC分类号： C07D409/12 , C07D231/06 , C07D401/12
摘要： Compounds of the formula I in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
摘要翻译：其中取代基如权利要求1中所定义的式I化合物适合用作杀微生物剂。

7. 发明授权

US07994341B2 Process for the production of amides 有权
标题翻译：酰胺生产工艺
公开(公告)号：US07994341B2
公开(公告)日：2011-08-09
申请号：US12066683
申请日：2006-09-14
申请人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi , Fanny Giordano , Martin Zeller , Gottfried Seifert , Shailesh Shah , Neil George , Ian Kevin Jones , Paul Edward Bonnett
发明人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi , Fanny Giordano , Martin Zeller , Gottfried Seifert , Shailesh Shah , Neil George , Ian Kevin Jones , Paul Edward Bonnett
IPC分类号： C07D231/14
CPC分类号： C07C211/61 , A01N43/56 , C07C205/06 , C07C209/325 , C07C209/70 , C07C2603/66 , C07D231/14
摘要： The present invention relates to a process for the preparation of compounds of formula (I) wherein R1 and R2 are each independently of the other hydrogen or C1-C5alkyl and R3 is CF3 or CF2H, by a) reaction of a compound of formula (II) wherein R1 and R2 are as defined for formula (I), with at least one reducing agent to form a compound of formula (III) wherein R1 and R2 are as defined for formula (I), and b) reaction of that compound with at least one reducing agent to form a compound of formula (IV) wherein R1 and R2 are as defined for formula (I), and (c) reaction of that compound with a compound of formula (V) wherein Q is chlorine, fluorine, bromine, iodine, hydroxy or C1-C6alkoxy and R3 is as defined for formula (I), to form the compound of formula (I); and to novel intermediates for use in that process.
摘要翻译：本发明涉及制备式（I）化合物的方法，其中R 1和R 2各自独立地为氢或C 1 -C 5烷基，R 3为CF 3或CF 2 H，通过a）式（Ⅱ）化合物）其中R1和R2如式（I）所定义，与至少一种还原剂形成式（III）化合物，其中R 1和R 2如式（I）所定义，和b）该化合物与至少一种还原剂形成式（Ⅳ）化合物，其中R1和R2如式（Ⅰ）所定义，和（c）该化合物与式（Ⅴ）化合物的反应其中Q是氯，氟，溴，碘，羟基或C 1 -C 6烷氧基，R 3如式（I）所定义，形成式（I）化合物; 以及用于该过程的新型中间体。

8. 发明授权

US07956194B2 Microbiocidal (E.G. fungicidal) 1,2,3-triazole derivatives 有权
标题翻译：杀微生物剂（E.G.杀真菌剂）1,2,3-三唑衍生物
公开(公告)号：US07956194B2
公开(公告)日：2011-06-07
申请号：US12463449
申请日：2009-05-11
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： C07D403/00 , C07C211/60
CPC分类号： C07D401/12 , A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08
摘要： A compound of formula (I): where A is an ortho-substituted ring selected from a number of specified rings; R1 is halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy or optionally substituted C2-4 alkenyl, optionally substituted C2-4 alkynyl or optionally substituted SO2(C1-4)alkyl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R2 is C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl or C1-4 alkylthio(C1-4)alkyl or [optionally substituted aryl](C1-4)alkyl- or [optionally substituted aryl]oxy(C1-4)alkyl-(where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R3 is hydrogen, CH2C≡CR4, CH2CR4═C(H)R4, CH═C═CH2 or COR5 or optionally substituted C1-4 alkyl, optionally substituted C1-4 alkoxy or optionally substituted (C1-4) alkylC(═O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy, C1-4 alkyl, C1-2 haloalkoxy, hydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl); each R4 is, independently, hydrogen, halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkoxy(C1-4)alkyl; and R5 is hydrogen or optionally substituted C1-6 alkyl, optionally substituted C1-4 alkoxy, optionally substituted C1-4 alkoxy(C1-4)alkyl, optionally substituted C1-4 alkylthio(C1-4)alkyl or optionally substituted aryl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen, C1-6 alkoxy, C1-6 haloalkoxy, cyano, hydroxy, methoxycarbonyl and ethoxycarbonyl).
摘要翻译：式（I）的化合物：其中A是选自多个指定环的邻位取代的环; R 1是卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基或任选取代的C 2-4烯基，任选取代的C 2-4炔基或任选取代的SO 2（C 1-4）烷基（其中任选取代的部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 2是C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基或C 1-4烷硫基（C 1-4）烷基或[任意取代的芳基]（C 1-4）烷基 - 或[ 芳基]氧基（C 1-4）烷基 - （其中任选取代的芳基部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 3是氢，CH 2C≡CR4，CH 2 CR 4 = C（H）R 4，CH = C = CH 2或COR 5或任选取代的C 1-4烷基，任选取代的C 1-4烷氧基或任选取代的（C 1-4）烷基C（= O（其中任选取代的部分可以各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基，C 1-4烷基，C 1-2卤代烷氧基，羟基，氰基，羧基，甲氧基羰基，乙氧基羰基，甲基磺酰基和乙基磺酰基） ; 每个R 4独立地是氢，卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4烷氧基（C 1-4）烷基; 并且R 5为氢或任选取代的C 1-6烷基，任选取代的C 1-4烷氧基，任选取代的C 1-4烷氧基（C 1-4）烷基，任选取代的C 1-4烷硫基（C 1-4）烷基或任选取代的芳基（其中任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素，C 1-6烷氧基，C 1-6卤代烷氧基，氰基，羟基，甲氧基羰基和乙氧基羰基）。

9. 发明授权

US07737301B2 Process for the production of anilines 有权
标题翻译：生产苯胺的方法
公开(公告)号：US07737301B2
公开(公告)日：2010-06-15
申请号：US12065304
申请日：2006-08-28
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Hans Tobler
IPC分类号： C07C209/62 , C07C209/10 , C07C211/45 , C07C211/48
CPC分类号： C07C209/10 , C07C209/62 , C07C2601/02 , C07C211/45 , C07C211/48
摘要： The present invention relates to a process for the preparation of compounds of formula wherein R1, R2 and R3 are each independently of the others hydrogen or C1-C4alkyl, by a) reacting compounds of formula (II) wherein R1, R2 and R3 are as defined for formula (I) and X is bromine or chlorine, with a compound of formula (III) wherein R4 is hydrogen or C1-C4alkyl, in the presence of a base and catalytic amounts of at least one palladium complex compound, to form compounds of formula (IV) wherein R1, R2, R3 and R4 are as defined for formula (I), and b) converting those compounds, using a reducing agent, into compounds of formula (I).
摘要翻译：本发明涉及制备下式化合物的方法，其中R 1，R 2和R 3各自独立地为氢或C 1 -C 4烷基，通过a）使式（Ⅱ）化合物（其中R 1，R 2和R 3为与式（Ⅲ）化合物（其中R 4是氢或C 1 -C 4烷基）在碱和催化量的至少一种钯络合物的存在下形成化合物（I），X是溴或氯，其中R 1，R 2，R 3和R 4如式（I）所定义，并且b）使用还原剂将这些化合物转化为式（I）化合物。

10. 发明授权

US07732469B2 Heterocyclic amide derivatives useful as microbiocides 有权
标题翻译：用作杀微生物剂的杂环酰胺衍生物
公开(公告)号：US07732469B2
公开(公告)日：2010-06-08
申请号：US12091189
申请日：2006-10-23
申请人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi
发明人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi
IPC分类号： A01N43/78 , C07D277/56 , C07C205/11 , A01P1/00
CPC分类号： C07C205/06 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/647 , A01N43/76 , A01N43/78 , C07C205/11 , C07C205/12 , C07C205/37 , C07C205/45 , C07C211/61 , C07C2603/66 , C07D207/34 , C07D207/46 , C07D213/89 , C07D231/14 , C07D249/04 , C07D263/34 , C07D277/56 , C07D327/06
摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R6, R7 and R8; R1 is hydrogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy, C1-4 haloalkoxy, CH2 C≡CR9, CH2 CR10═CHR11, CH═C═CH2 or COR12; R2 and R3 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl or C1-4 haloalkoxy; R4 and R5 are each independently selected from halo, cyano and nitro; or one of R4 and R5 is hydrogen and the other is selected from halo, cyano and nitro; R6, R7 and R8 are each, independently, hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4 haloalkoxy(C1-4)alkyl or C1-4 haloalkoxy, provided that at least one of R6, R7 and R8 is not hydrogen; R9, R10 and R11 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 haloalkyl or C1-4 alkoxy(C1-4)alkyl; and R12 is hydrogen, C1-6 alkyl, C1-6 haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4 alkylthio(C1-4)-alkyl, C1-4 alkoxy or aryl; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被R6基团取代，R7和R8; R 1是氢，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基，CH 2C≡CR9，CH 2 CR 10 = CHR 11，CH = C = CH 2或COR 12; R 2和R 3各自独立地为氢，卤素，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基或C 1-4卤代烷氧基; R4和R5各自独立地选自卤素，氰基和硝基; 或者R4和R5之一是氢，另一个选自卤素，氰基和硝基; R 6，R 7和R 8各自独立地为氢，卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4卤代烷氧基（C 1-4）烷基或 C 1-4卤代烷氧基，条件是R 6，R 7和R 8中的至少一个不是氢; R 9，R 10和R 11各自独立地为氢，卤素，C 1-4烷基，C 1-4卤代烷基或C 1-4烷氧基（C 1-4）烷基; 和R 12是氢，C 1-6烷基，C 1-6卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4烷硫基（C 1-4） - 烷基，C 1-4烷氧基或芳基; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

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