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1. 发明授权

US09708313B2 Substituted pyrido[3,4-b]pyrazines as GPR6 modulators 有权
公开(公告)号：US09708313B2
公开(公告)日：2017-07-18
申请号：US14883174
申请日：2015-10-14
申请人： Jason W. Brown , Stephen Hitchcock , Maria Hopkins , Shota Kikuchi , Holger Monenschein , Holly Reichard , Kristin Schleicher , Huikai Sun , Todd Macklin
发明人： Jason W. Brown , Stephen Hitchcock , Maria Hopkins , Shota Kikuchi , Holger Monenschein , Holly Reichard , Kristin Schleicher , Huikai Sun , Todd Macklin
IPC分类号： C07D241/38 , C07D471/04
CPC分类号： C07D471/04
摘要： This present invention provides compounds of formula II: which are useful as modulators of GPR6, pharmaceutical compositions thereof, methods for treatment of conditions associated with GPR6, processes for making the compounds and intermediates thereof.

2. 发明申请

US20160031881A1 TETRAHYDROPYRIDOPYRAZINES AS MODULATORS OF GPR6 有权
标题翻译：作为GPR6的调节剂的四氢吡咯并吡喃
公开(公告)号：US20160031881A1
公开(公告)日：2016-02-04
申请号：US14883174
申请日：2015-10-14
申请人： Jason W. Brown , Stephen Hitchcock , Maria Hopkins , Shota Kikuchi , Holger Monenschein , Holly Reichard , Kristin Schleicher , Huikai Sun , Todd Macklin
发明人： Jason W. Brown , Stephen Hitchcock , Maria Hopkins , Shota Kikuchi , Holger Monenschein , Holly Reichard , Kristin Schleicher , Huikai Sun , Todd Macklin
IPC分类号： C07D471/04
CPC分类号： C07D471/04
摘要： The present invention provides compounds of formula I: which are useful as modulators of GPR6, pharmaceutical compositions thereof, methods for treatment of conditions associated with GPR6, processes for making the compounds and intermediates thereof.
摘要翻译：本发明提供式I化合物：其可用作GPR6的调节剂，其药物组合物，用于治疗与GPR6相关的病症的方法，用于制备化合物的方法及其中间体。

3. 发明申请

US20170174677A1 TETRAHYDROPYRIDOPYRAZINES MODULATORS OF GPR6 审中-公开
公开(公告)号：US20170174677A1
公开(公告)日：2017-06-22
申请号：US15118447
申请日：2015-02-13
申请人： Stephen Hitchcock , Maria Hopkins , Shota Kikuchi , Holger Monenschein , Holly Reichard , Huikai Sun , Todd Macklin
发明人： Stephen Hitchcock , Maria Hopkins , Shota Kikuchi , Holger Monenschein , Holly Reichard , Huikai Sun , Todd Macklin
IPC分类号： C07D471/04
CPC分类号： C07D471/04
摘要： The present invention provides compounds of formula I: which are useful as modulators of GPR6, pharmaceutical compositions thereof, methods for treatment of conditions associated with GPR6, processes for making the compounds and intermediates thereof.

4. 发明授权

US09346829B2 5-HT3 receptor antagonists 有权
标题翻译： 5-HT3受体拮抗剂
公开(公告)号：US09346829B2
公开(公告)日：2016-05-24
申请号：US14645639
申请日：2015-03-12
申请人： Stephen Hitchcock , Holger Monenschein , Holly Reichard , Huikai Sun , Shota Kikuchi , Todd Macklin , Maria Hopkins
发明人： Stephen Hitchcock , Holger Monenschein , Holly Reichard , Huikai Sun , Shota Kikuchi , Todd Macklin , Maria Hopkins
IPC分类号： A61K31/19 , A61K31/5386 , C07D519/00 , C07D498/08 , C07D451/12 , C07D471/04 , C07D221/22
CPC分类号： C07D498/08 , A61K31/19 , A61K31/5386 , C07C53/18 , C07C53/40 , C07D221/22 , C07D451/12 , C07D453/02 , C07D471/04 , C07D471/08 , C07D519/00
摘要： The present invention provides a method of treating nicotine addiction comprising administering a 5-HT3 receptor antagonists of Formula (I):
摘要翻译：本发明提供了一种治疗尼古丁成瘾的方法，包括给予式（I）的5-HT 3受体拮抗剂：

5. 发明申请

US20150182533A1 5-HT3 RECEPTOR ANTAGONISTS 审中-公开
标题翻译： 5-HT3受体拮抗剂
公开(公告)号：US20150182533A1
公开(公告)日：2015-07-02
申请号：US14645639
申请日：2015-03-12
申请人： Stephen Hitchcock , Holger Monenschein , Holly Reichard , Huikai Sun , Shota Kikuchi , Todd Macklin , Maria Hopkins
发明人： Stephen Hitchcock , Holger Monenschein , Holly Reichard , Huikai Sun , Shota Kikuchi , Todd Macklin , Maria Hopkins
IPC分类号： A61K31/5386 , A61K31/19
CPC分类号： C07D498/08 , A61K31/19 , A61K31/5386 , C07C53/18 , C07C53/40 , C07D221/22 , C07D451/12 , C07D453/02 , C07D471/04 , C07D471/08 , C07D519/00
摘要： The present invention provides a method of treating nicotine addiction comprising administering a 5-HT3 receptor antagonists of Formula (I):
摘要翻译：本发明提供了一种治疗尼古丁成瘾的方法，包括给予式（I）的5-HT 3受体拮抗剂：

6. 发明申请

US20170174659A1 PYRAZINES MODULATORS OF GPR6 有权
公开(公告)号：US20170174659A1
公开(公告)日：2017-06-22
申请号：US15118461
申请日：2015-02-13
申请人： Mark E. Adams , Jason W. Brown , Stephen Hitchcock , Maria Hopkins , Shota Kikuchi , Betty Lam , Holger Monenschein , Holly Reichard , Huikai Sun
发明人： Mark E. Adams , Jason W. Brown , Stephen Hitchcock , Maria Hopkins , Shota Kikuchi , Betty Lam , Holger Monenschein , Holly Reichard , Huikai Sun
IPC分类号： C07D401/14 , C07D401/04 , C07D241/28
CPC分类号： C07D401/14 , C07D241/26 , C07D241/28 , C07D401/04
摘要： The present invention provides compounds of formula I: which are useful as modulators of GPR6, pharmaceutical compositions thereof, methods for treatment of conditions associated with GPR6, processes for making the compounds and intermediates thereof.

7. 发明授权

US08823473B2 Latching relay 有权
标题翻译：闭锁继电器
公开(公告)号：US08823473B2
公开(公告)日：2014-09-02
申请号：US13885310
申请日：2011-11-24
申请人： Ken Fujita , Shota Kikuchi , Noriyoshi Machida
发明人： Ken Fujita , Shota Kikuchi , Noriyoshi Machida
IPC分类号： H01H3/00 , H01H9/00 , H01H51/27 , H01H50/18 , H01H50/24 , H01H51/22 , H01H50/64
CPC分类号： H01H50/18 , H01H50/24 , H01H50/641 , H01H51/2263 , H01H51/27
摘要： A latching relay has a fixed iron core including an exciting coil wound around an intermediate portion and a magnetic pole piece at two ends; movable iron pieces sandwiching a permanent magnet between two bar-shaped iron pieces disposed in parallel with each other, and are fixed with a holder; and a switchable electrical contact portion. The fixed iron core and the movable iron pieces are disposed facing each other to insert each of the magnetic pole pieces on two sides of the fixed iron core to be spaced apart in a space between the two bar-shaped iron pieces of two end portions of the movable iron pieces. The movable iron pieces are supported pivotally in a direction in which the two bar-shaped iron pieces are aligned. The movable iron pieces are linked to the electrical contact portion, and the movable iron pieces perform a switching of the electrical contact portion.
摘要翻译：闭锁继电器具有固定铁芯，包括缠绕在中间部分上的励磁线圈和两端的磁极片; 在彼此平行设置的两个棒状铁片之间夹持永久磁铁的可动铁片，并用固定器固定; 和可切换的电接触部分。固定铁芯和可动铁片彼此面对地设置，以将每个磁极片插入固定铁芯的两侧，以分开在两个两端部的两个棒状铁片之间的空间内可动铁件。可动铁片沿着两个条形铁片对准的方向枢转地支撑。可动铁片与电接触部分连接，并且可动铁片执行电接触部分的切换。

8. 发明申请

US20130229246A1 LATCHING RELAY 有权
标题翻译：锁定继电器
公开(公告)号：US20130229246A1
公开(公告)日：2013-09-05
申请号：US13885310
申请日：2011-11-24
申请人： Ken Fujita , Shota Kikuchi , Noriyoshi Machida
发明人： Ken Fujita , Shota Kikuchi , Noriyoshi Machida
IPC分类号： H01H50/18
CPC分类号： H01H50/18 , H01H50/24 , H01H50/641 , H01H51/2263 , H01H51/27
摘要： A latching relay has a fixed iron core including an exciting coil wound around an intermediate portion and a magnetic pole piece at two ends; movable iron pieces sandwiching a permanent magnet between two bar-shaped iron pieces disposed in parallel with each other, and are fixed with a holder; and a switchable electrical contact portion. The fixed iron core and the movable iron pieces are disposed facing each other to insert each of the magnetic pole pieces on two sides of the fixed iron core to be spaced apart in a space between the two bar-shaped iron pieces of two end portions of the movable iron pieces. The movable iron pieces are supported pivotally in a direction in which the two bar-shaped iron pieces are aligned. The movable iron pieces are linked to the electrical contact portion, and the movable iron pieces perform a switching of the electrical contact portion.
摘要翻译：闭锁继电器具有固定铁芯，包括缠绕在中间部分上的励磁线圈和两端的磁极片; 在彼此平行设置的两个棒状铁片之间夹持永久磁铁的可动铁片，并用固定器固定; 和可切换的电接触部分。固定铁芯和可动铁片彼此面对地设置，以将每个磁极片插入固定铁芯的两侧，以分开在两个两端部的两个棒状铁片之间的空间内可动铁件。可动铁片沿着两个条形铁片对准的方向枢转地支撑。可动铁片与电接触部分连接，并且可动铁片执行电接触部分的切换。

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