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1. 发明申请

US20060217440A1 Porcess for production of 2-cyano-3-hydroxy-n-(4-trifluoromethylphenyl)hept-2-en-6-ynamide and process for production of polymorphs thereof 审中-公开
标题翻译： 2-氰基-3-羟基 - 正（4-三氟甲基苯基）庚-2-烯-6-基酰胺的生产工艺及其多晶型物的制备方法
公开(公告)号：US20060217440A1
公开(公告)日：2006-09-28
申请号：US10550099
申请日：2004-03-23
申请人： Hiroki Omori , Satoshi Hirabayashi , Ariyoshi Kubota , Takeshi Kawakami , Yosuke Fujii , Ikuo Matsumoto , Masato Kitayama , Shunsuke Goto
发明人： Hiroki Omori , Satoshi Hirabayashi , Ariyoshi Kubota , Takeshi Kawakami , Yosuke Fujii , Ikuo Matsumoto , Masato Kitayama , Shunsuke Goto
IPC分类号： A61K31/277 , C07C253/30
CPC分类号： C07C253/30 , C07C255/23
摘要： A compound (II) is reacted with a compound (III) or a reactive derivative at the carboxyl group thereof to obtain a compound (IV), which is reacted with a mixed acid anhydride of a compound (V) to prepare a compound (I). In recrystallization of the compound (I), temperature for the recrystallization and/or time for the crystal precipitation is controlled to selectively produce A-form crystals, B-form crystals and C-form crystals of the compound (I).
摘要翻译：使化合物（II）与化合物（III）或其羧基上的活性衍生物反应，得到化合物（IV），其与化合物（V）的混合酸酐反应，制备化合物（I ）。在化合物（I）的重结晶中，控制用于重结晶的温度和/或晶体沉淀的时间，以选择性地生成化合物（I）的A-型晶体，B型晶体和C型晶体。

2. 发明授权

US07229992B2 Process for the preparation of a piperazine derivative 失效
标题翻译：哌嗪衍生物的制备方法
公开(公告)号：US07229992B2
公开(公告)日：2007-06-12
申请号：US10297592
申请日：2001-06-08
申请人： Keiichi Koga , Ryoki Orii , Yosuke Fujii , Shunsuke Goto , Satoshi Hirabayashi
发明人： Keiichi Koga , Ryoki Orii , Yosuke Fujii , Shunsuke Goto , Satoshi Hirabayashi
IPC分类号： A61K31/5377 , C07D265/30
CPC分类号： C07D413/06 , C07D241/04
摘要： (2R)-1-[3,5-bis(trifluoromethyl)benzoyl]-4-[2-[(2S)-2-(methoxymethyl)morpholino]ethyl]-2-(3-hydroxy-4-methylbenzyl)piperazine dihydrochloride is obtained by debenzylating (2R)-4-benzyl-1-[3,5-bis(trifluoromethyl)-benzoyl]-2-(3-hydroxy-4-methylbenzyl)piperazine, then N-alkylating and converting to hydrochloride.
摘要翻译：（2R）-1- [3,5-双（三氟甲基）苯甲酰基] -4- [2 - [（2S）-2-（甲氧基甲基）吗啉代]乙基] -2-（3-羟基-4-甲基苄基）通过使（2R）-4-苄基-1- [3,5-双（三氟甲基） - 苯甲酰基] -2-（3-羟基-4-甲基苄基）哌嗪脱苄化，然后N-烷基化并转化成盐酸盐得到二盐酸盐。

3. 发明授权

US06344559B1 Process for producing quinazoline derivatives 失效
标题翻译：喹唑啉衍生物的制备方法
公开(公告)号：US06344559B1
公开(公告)日：2002-02-05
申请号：US09380609
申请日：1999-10-13
申请人： Hiroki Omori , Shunsuke Goto , Hiroyuki Tsuboi , Masayasu Fukagawa , Kooji Kagara
发明人： Hiroki Omori , Shunsuke Goto , Hiroyuki Tsuboi , Masayasu Fukagawa , Kooji Kagara
IPC分类号： C07D23996
CPC分类号： C07D239/96
摘要： This invention provides an industrially useful process for producing a quinazoline derivative (I) of the general formula: [wherein R1 is hydrogen or halogen; R2 is carboxy or protected carboxy; A is lower alkylene] or its salt on a commercial scale which comprises reacting a compound of the general formula: [wherein R1 is hydrogen or halogen] or its salt with a silylating agent and then with a compound of the general formula: Cl—A—R2 (III) [wherein R2 is carboxy or protected carboxy; A is lower alkylene] or its salt, optionally followed by desilylation.
摘要翻译：本发明提供了一种工业上有用的制备具有以下通式的喹唑啉衍生物（I）的方法：其中R 1是氢或卤素; R2是羧基或被保护的羧基; A是低级亚烷基]或其盐，其包括使通式为[其中R 1为氢或卤素]的化合物或其盐与甲硅烷基化试剂反应，然后与下列通式的化合物反应：其中R 2 是羧基或被保护的羧基; A是低级亚烷基]或其盐，任选地随后脱甲硅烷基化。

4. 发明授权

US06538007B1 N-[(R)-1-[3-(4-piperidyl)propionyl]-3-piperidylcarbonyl]-2(S)-acetylamino-&bgr;-alanine trihydrate, compositions thereof, and methods for its use 失效
标题翻译： N - [（R）-1- [3-（4-哌啶基）丙酰] -3-哌啶基羰基] -2（S） - 乙酰氨基-β-丙氨酸三水合物，其组合物及其使用方法
公开(公告)号：US06538007B1
公开(公告)日：2003-03-25
申请号：US09806483
申请日：2001-04-12
申请人： Mitsuru Ohkubo , Satoru Kuroda , Hideko Nakamura , Hisashi Takasugi , Yosuke Fujii , Keiichi Koga , Eiki Oikawa , Ryoki Orii , Shunsuke Goto
发明人： Mitsuru Ohkubo , Satoru Kuroda , Hideko Nakamura , Hisashi Takasugi , Yosuke Fujii , Keiichi Koga , Eiki Oikawa , Ryoki Orii , Shunsuke Goto
IPC分类号： A61K31445
CPC分类号： C07D211/60 , Y02P20/55
摘要： The trihydrates of &bgr;-alanine of the formula Are disclosed. Also method of antogonizing glycoprotein IIb/IIIa activity using these compounds is also disclosed.
摘要翻译：公开了β-丙氨酸的三水合物。还公开了使用这些化合物使糖蛋白IIb / IIIa活性钝化的方法。

5. 发明授权

US5675011A Process for producing pyrrolidine derivative and salt thereof 失效
标题翻译：制备吡咯烷衍生物及其盐的方法
公开(公告)号：US5675011A
公开(公告)日：1997-10-07
申请号：US487521
申请日：1995-06-07
申请人： Kohji Kagara , Shunsuke Goto , Satoshi Yonishi , Muneharu Ikushima , Yukihisa Baba , Haruo Horiai
发明人： Kohji Kagara , Shunsuke Goto , Satoshi Yonishi , Muneharu Ikushima , Yukihisa Baba , Haruo Horiai
IPC分类号： C07D207/14 , C07D401/06
CPC分类号： C07D401/06 , C07D207/14
摘要： A process for producing a compound of the general formula: ##STR1## wherein R.sup.1 is heterocyclic(lower)alkyl, R.sup.2 is acyl, and R.sup.3 is carboxy(lower)alkyl or protected carboxy(lower)alkyl, which is useful as a medicament or a salt thereof.
摘要翻译：制备通式如下的化合物的方法：其中R 1为杂环（低级）烷基，R 2为酰基，且R 3为羧基（低级）烷基或被保护的羧基（低级）烷基，其可用作药物或其盐。

6. 发明授权

US4973693A Novel pentacyclic compound and stereoselective synthesis thereof 失效
标题翻译：新型五环化合物及其立体选择性合成
公开(公告)号：US4973693A
公开(公告)日：1990-11-27
申请号：US401746
申请日：1989-09-01
申请人： Shunsuke Goto , Tohru Fukuyama
发明人： Shunsuke Goto , Tohru Fukuyama
IPC分类号： A61K31/535 , A61P31/04 , A61P35/00 , C07D498/22
CPC分类号： C07D498/22
摘要： Novel pentacyclic compounds having antimicrobial and antitumor activity and a process for preparing the same. The pentacyclic compounds are also usefual as intermediates in the production of known tetracyclic antitumor compounds.
摘要翻译：具有抗微生物和抗肿瘤活性的新型五环化合物及其制备方法。五环化合物在生产已知的四环抗肿瘤化合物中也是有用的中间体。

7. 发明授权

US07973379B2 Photovoltaic ultraviolet sensor 有权
标题翻译：光伏紫外线传感器
公开(公告)号：US07973379B2
公开(公告)日：2011-07-05
申请号：US11388052
申请日：2006-03-23
申请人： Mayo Sugibuchi , Kohsuke Takahashi , Shunsuke Goto , Yasube Kashiwaba , Haruyuki Endo , Tatsuo Hasegawa , Fukunori Izumida , Eriko Ohshima
发明人： Mayo Sugibuchi , Kohsuke Takahashi , Shunsuke Goto , Yasube Kashiwaba , Haruyuki Endo , Tatsuo Hasegawa , Fukunori Izumida , Eriko Ohshima
IPC分类号： H01L31/07
CPC分类号： G01J1/429 , H01L31/0296 , H01L31/108
摘要： A photovoltaic ultraviolet sensor comprises a zinc oxide single crystal substrate. On the +c face of the zinc oxide single crystal substrate, an ultraviolet receiver is formed. The exemplary ultraviolet receiver includes a Schottky electrode which, when receiving ultraviolet rays, produces a voltage in cooperation with the zinc oxide single crystal substrate. The ultraviolet sensor does not have any sensitivity to the visible rays. The ultraviolet sensor has a relatively fast response of several microseconds.
摘要翻译：光伏紫外线传感器包括氧化锌单晶基板。在氧化锌单晶基板的+ c面上形成紫外线接收体。示例性紫外线接收器包括肖特基电极，当接收紫外线时，与氧化锌单晶衬底配合产生电压。紫外线传感器对可见光线没有任何敏感性。紫外线传感器具有几微秒的相对较快的响应。

8. 发明授权

US09429322B2 Glow plug 有权
标题翻译：辉光插头
公开(公告)号：US09429322B2
公开(公告)日：2016-08-30
申请号：US13983162
申请日：2012-04-12
申请人： Yuki Doi , Shunsuke Goto
发明人： Yuki Doi , Shunsuke Goto
IPC分类号： F23Q7/00 , H01T13/08
CPC分类号： F23Q7/001 , H01T13/08
摘要： A glow plug (1) including a metallic shell (2) having a forward end portion (20) having an outer peripheral surface whose diameter increases toward the rear end side with respect to the axial direction, the forward end portion (20) coming into contact with a seat surface (55) formed on an internal combustion engine (50). The outer peripheral surface of the forward end portion (20) includes a first, second and third contact surfaces (21), (22) and (23), respectively, which differ in imaginary line angle from one another, the imaginary line angle of each contact surface being an angle which is formed, as viewed on a cross section including an axis C1, between two straight imaginary lines connecting inflection points of the contact surface at opposite ends of the contact surface. At least one of the contact surfaces is a curved surface which bulges outward.
摘要翻译：一种电热塞（1），包括具有前端部（20）的金属壳（2），所述前端部具有相对于所述轴向朝向后端侧的直径增大的外周面，所述前端部（20）进入与形成在内燃机（50）上的座面（55）接触。前端部（20）的外周面分别具有第一，第二和第三接触面（21），（22）和（23），它们的虚拟线角度彼此不同，假想线角度每个接触表面是在连接接触表面的相对端处的接触表面的拐点之间的两条直线假想线之间形成的角度，在包括轴线C1的横截面上观察。至少一个接触表面是向外凸出的曲面。

9. 发明申请

US20130306017A1 GLOW PLUG 有权
标题翻译： GLOW插头
公开(公告)号：US20130306017A1
公开(公告)日：2013-11-21
申请号：US13983162
申请日：2012-04-12
申请人： Yuki Doi , Shunsuke Goto
发明人： Yuki Doi , Shunsuke Goto
IPC分类号： F23Q7/00
CPC分类号： F23Q7/001 , H01T13/08
摘要： A glow plug (1) including a metallic shell (2) having a forward end portion (20) having an outer peripheral surface whose diameter increases toward the rear end side with respect to the axial direction, the forward end portion (20) coming into contact with a seat surface (55) formed on an internal combustion engine (50). The outer peripheral surface of the forward end portion (20) includes a first, second and third contact surfaces (21), (22) and (23), respectively, which differ in imaginary line angle from one another, the imaginary line angle of each contact surface being an angle which is formed, as viewed on a cross section including an axis C1, between two straight imaginary lines connecting inflection points of the contact surface at opposite ends of the contact surface. At least one of the contact surfaces is a curved surface which bulges outward.
摘要翻译：一种电热塞（1），包括具有前端部（20）的金属壳（2），所述前端部具有相对于所述轴向朝向后端侧的直径增大的外周面，所述前端部（20）进入与形成在内燃机（50）上的座面（55）接触。前端部（20）的外周面分别具有第一，第二和第三接触面（21），（22）和（23），它们的虚拟线角度彼此不同，假想线角度每个接触表面是在连接接触表面的相对端处的接触表面的拐点之间的两条直线假想线之间形成的角度，在包括轴线C1的横截面上观察。至少一个接触表面是向外凸出的曲面。

10. 发明申请

US20070145499A1 Photovoltaic ultraviolet sensor 有权
标题翻译：光伏紫外线传感器
公开(公告)号：US20070145499A1
公开(公告)日：2007-06-28
申请号：US11388052
申请日：2006-03-23
申请人： Mayo Sugibuchi , Kohsuke Takahashi , Shunsuke Goto , Yasube Kashiwaba , Haruyuki Endo , Tatsuo Hasegawa , Fukunori Izumida , Eriko Ohshima
发明人： Mayo Sugibuchi , Kohsuke Takahashi , Shunsuke Goto , Yasube Kashiwaba , Haruyuki Endo , Tatsuo Hasegawa , Fukunori Izumida , Eriko Ohshima
IPC分类号： H01L29/82
CPC分类号： G01J1/429 , H01L31/0296 , H01L31/108
摘要： A photovoltaic ultraviolet sensor comprises a zinc oxide single crystal substrate. On the +c face of the zinc oxide single crystal substrate, an ultraviolet receiver is formed. The exemplary ultraviolet receiver includes a Schottky electrode which, when receiving ultraviolet rays, produces a voltage in cooperation with the zinc oxide single crystal substrate. The ultraviolet sensor does not have any sensitivity to the visible rays. The ultraviolet sensor has a relatively fast response of several microseconds.
摘要翻译：光伏紫外线传感器包括氧化锌单晶基板。在氧化锌单晶基板的+ c面上形成紫外线接收体。示例性紫外线接收器包括肖特基电极，当接收紫外线时，与氧化锌单晶衬底配合产生电压。紫外线传感器对可见光线没有任何敏感性。紫外线传感器具有几微秒的相对较快的响应。

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