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1. 发明授权

US5606070A Process for the preparation of alkoxytriazolinones 失效
标题翻译：制备烷氧基三唑啉酮的方法
公开(公告)号：US5606070A
公开(公告)日：1997-02-25
申请号：US528585
申请日：1995-09-15
申请人： Heinz-J urgen Wroblowsky , Klaus K onig , Joachim Kluth , Klaus-Helmut M uller
发明人： Heinz-J urgen Wroblowsky , Klaus K onig , Joachim Kluth , Klaus-Helmut M uller
IPC分类号： C07D249/12
CPC分类号： C07D249/12
摘要： Alkoxytriazolinones of the general formula (I), ##STR1## in which R.sup.1 and R.sup.2 independently of one another represent in each case optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl,(which can be used as intermediates for the preparation of herbicidal active compounds) are obtained in very good yields and in high purity by reacting iminothiocarbonic diester (II) with carbazinic esters (III) ##STR2## in which R.sup.3 and R.sup.4 in each case represent, for example, alkyl or aryl, at -20.degree. C. to +50.degree. C. (1st step) and subjecting the semicarbazide derivatives (IV) formed in this process with elimination of R.sup.3 -SH ##STR3## to a cyclizing condensation reaction and if appropriate in the presence of a base at 20.degree. C. to 100.degree. C. with elimination of R.sup.4 --OH, if appropriate after intermediate isolation (2nd step).
摘要翻译：通式（I）的烷氧基三唑啉酮，其中R 1和R 2彼此独立地表示在各种情况下为任选取代的烷基，烯基，炔基，环烷基，环烷基烷基，芳基或芳烷基（其可以用作用于制备除草活性化合物的中间体）以非常好的产率和高纯度通过亚氨基碳二酸酯（II）与咔嗪酸酯（III）反应获得，其中R 3和R 4在每种情况下代表例如烷基或芳基，在-20℃至+ 50℃（第一步），并将在该过程中形成的氨基脲衍生物（IV）与R3-SH的消除进行环化缩合反应，并且如果在适当的情况下存在的碱在20℃至100℃，如果适当，在中间分离（第二步）后消除R4-OH。

2. 发明授权

US5552369A Sulphonylaminocarbonyltriazolinones 失效
标题翻译：磺酰氨基羰基三唑啉酮
公开(公告)号：US5552369A
公开(公告)日：1996-09-03
申请号：US411718
申请日：1995-04-07
申请人： Kurt Findeisen , Karl-Heinz Linker , Joachim Kluth , Klaus-Helmut M uller , Hans-Jochem Riebel , Klaus K onig , Hans-Joachim Santel , Robert R. Schmidt
发明人： Kurt Findeisen , Karl-Heinz Linker , Joachim Kluth , Klaus-Helmut M uller , Hans-Jochem Riebel , Klaus K onig , Hans-Joachim Santel , Robert R. Schmidt
IPC分类号： A01N47/38 , A01N57/32 , A01P13/00 , C07D249/12 , C07D249/14 , C07F9/6518 , C07D413/04
CPC分类号： A01N47/38 , C07D249/12 , C07D249/14
摘要： The invention relates to new sulphonylaminocarbonyltriazolinones of the formula (I) ##STR1## in which Q represents oxygen, sulphur or one of the following groups ##STR2## (in which the radicals R.sup.1, R.sup.2, R.sup.3 and R.sup.4 have the meanings given in the description),as well as to salts of compounds of the formula (I), to processes and novel intermediates for the preparation of the novel compounds, and to their use as herbicides.
摘要翻译： PCT No.PCT / EP93 / 02706 Sec。 371日期：1995年4月7日 102（e）日期1995年4月7日PCT提交1993年10月4日PCT公布。公开号WO94 / 08979 日期：1994年04月28日本发明涉及式（I）的新的磺酰基氨基羰基三唑啉酮，其中Q表示氧，硫或以下基团之一：其中基团R 1，R 2，R 3和 R4具有说明书中给出的含义）以及式（I）化合物的盐，用于制备新化合物的方法和新型中间体，以及它们作为除草剂的用途。

3. 发明授权

US5597939A Herbicidal sulphonylaminocarbonyltriazolinones having substituents bonded via oxygen of the formula 失效
标题翻译：具有通过下式的氧连接的取代基的除草磺酰基氨基羰基三唑啉酮
公开(公告)号：US5597939A
公开(公告)日：1997-01-28
申请号：US630569
申请日：1996-04-10
申请人： Klaus-Helmut M uller , Klaus K onig , Joachim Kluth , Klaus L urssen , Hans-Joachim Santel , Robert R. Schmidt
发明人： Klaus-Helmut M uller , Klaus K onig , Joachim Kluth , Klaus L urssen , Hans-Joachim Santel , Robert R. Schmidt
IPC分类号： A01N47/38 , C07D249/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07C275/70
CPC分类号： C07D403/12 , A01N47/38 , C07D249/12 , C07D405/12 , C07D409/12
摘要： R.sup.2 represents an optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, aralkyl or aryl radical, andR.sup.3 represents an optionally substituted alkyl, aralkyl, aryl or heteroaryl radical,and salts thereof, with the exception of the compounds:2-(2-methoxycarbonyl-phenylsulphonylaminocarbonyl)-4-methyl-5-methoxy-2,4-dihydro-3H-1,2,4-triazol-3-one,2-(2-trifluoromethoxy-phenylsulphonylaminocarbonyl)-4-cyclopropnl-5-methoxy-2,4-dihydro-3H-1,2,4-triazol-3-one,2-(2-difluoromethoxy-phenylsulphonylaminocarbonyl)-cyclobutyl-5-ethoxy-2,4-dihydro-3H-1,2,4-triazol-3-one, and2-(2-methoxycarbonyl-phenylsulphonylaminocarbonyl)-4-ethyl-5-ethoxy-2,4-dihydro-3H-1,2,4-triazol-3-one.
摘要翻译：链烯基，环烷基，芳烷基，芳基，烷基氨基，环烷基氨基或二烷基氨基，R 2表示任选取代的烷基，烯基，炔基，环烷基，环烯基，芳烷基或芳基，R 3表示任选取代的烷基，芳烷基，芳基或杂芳基及其盐，除了化合物：2-（2-甲氧基羰基 - 苯基磺酰基氨基羰基）-4-甲基-5-甲氧基 -2,4-二氢-3H-1,2,4-三唑-3-酮，2-（2-三氟甲氧基 - 苯基磺酰基氨基羰基）-4-环丙基-5-甲氧基-2,4-二氢-3H-1， 2,4-二氟甲氧基 - 苯基磺酰基氨基羰基） - 环丁基-5-乙氧基-2,4-二氢-3H-1,2,4-三唑-3-酮和2-（ 2-甲氧基羰基 - 苯基磺酰基氨基羰基）-4-乙基-5-乙氧基-2,4-二氢-3H-1,2,4-三唑-3-酮。

4. 发明授权

US5541337A Substituted 5-alkoxy-1,2,4-triazol-3-(thi)ones 失效
标题翻译：取代的5-烷氧基-1,2,4-三唑-3-（硫）
公开(公告)号：US5541337A
公开(公告)日：1996-07-30
申请号：US269875
申请日：1994-06-30
申请人： Klaus-Helmut M uller , Klaus K onig , Joachim Kluth , Klaus L urssen , Hans-Joachim Santel , Robert R. Schmidt
发明人： Klaus-Helmut M uller , Klaus K onig , Joachim Kluth , Klaus L urssen , Hans-Joachim Santel , Robert R. Schmidt
IPC分类号： A01N47/38 , A01N51/00 , C07D249/12 , C07D249/14 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04
CPC分类号： C07D401/12 , A01N47/38 , A01N51/00 , C07D249/12 , C07D249/14 , C07D403/12 , C07D405/12 , C07D409/12 , C07D471/04 , C07D487/04
摘要： Herbicidal 5-alkoxy-1,2,4-triazol-3-(thi)ones of the gerneral formula ##STR1## (in which the radicals R.sup.1, R.sup.2, R.sup.3, X and Y have the meanings given in the description), processes for their preparation, and their use as herbicides, and also new intermediates of the formula (II) ##STR2##
摘要翻译：（I）（其中基团R 1，R 2，R 3，X和Y具有在说明书中给出的含义）的除草剂5-烷氧基-1,2,4-三唑-3-（thi）），它们的制备方法和它们作为除草剂的用途，以及式（II）的新的中间体<图像（II）

5. 发明授权

US5550244A Process for preparing sulphonylaminocarbonyltriazolinones 失效
标题翻译：制备磺酰氨基羰基三唑啉酮的方法
公开(公告)号：US5550244A
公开(公告)日：1996-08-27
申请号：US355724
申请日：1994-12-14
申请人： Joachim Kluth , Klaus-Helmut M uller
发明人： Joachim Kluth , Klaus-Helmut M uller
IPC分类号： A01N47/38 , C07D249/12 , C07D409/12 , C07D401/12 , C07D403/12
CPC分类号： A01N47/38 , C07D249/12
摘要： Substituted (herbicidally active) sulphonylaminocarbonyltriazolinones of the formula (I) ##STR1## in which R.sup.1 represents hydrogen, hydroxyl or amino, or represents an optionally substituted radical from the group comprising alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy, cycloalkylamino, cycloalkylalkyl, aryl or arylalkyl,R.sup.2 represents hydrogen, hydroxyl, mercapto, amino or halogen, or represents an optionally substituted radical from the group comprising alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy, alkylthio, alkenylthio, alkinylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino, cycloalkyl, cycloalkenyl, cycloalkyloxy, cycloalkenyloxy, cycloalkylthio, cycloalkenylthio, cycloalkylamino, cycloalkenylamino, cycloalkylalkyl, cycloalkenylalkyl, aryl, aryloxy, arylthio, arylamino, arylalkyl, arylalkyloxy, arylalkylthio or arylalkylamino, andR.sup.3 represents an optionally substituted radical from the group comprising alkyl, cycloalkyl, cycloalkylalkyl, aryl, arylalkyl, heterocyclyl or heterocyclylalkyl,are obtained in Good yields and at high purity by reacting, in a three-component reaction, triazolinones of the general formula (II) ##STR2## with sulphonylhalides of the general formula (III)R.sup.3 --SO.sub.2 --X (III)X=Halogen,and metal cyanates of the General formula (IV)MOCN (IV)in which M represents an alkali metal or one alkaline earth metal equivalent, optionally in the presence of a reaction auxiliary and optionally in the presence of a diluent at temperatures of between 20.degree. C. and 150.degree. C.
摘要翻译：式（I）的取代（除草活性）磺酰基氨基羰基三唑啉酮其中R 1表示氢，羟基或氨基，或代表任选取代的基团，其包括烷基，烯基，炔基，烷氧基，烯氧基，烷基氨基，二烷基氨基，环烷基，环烷基氧基，环烷基氨基，环烷基烷基，芳基或芳基烷基，R2代表氢，羟基，巯基，氨基或卤素，或代表任选取代的基团，包括烷基，烯基，炔基，烷氧基，烯氧基，烷氧基，烷硫基，链烯硫基，炔基硫基，烷基亚磺酰基，烷基磺酰基，烷基氨基，二烷基氨基，环烷基，环烯基，环烷基氧基，环烯基氧基，环烷硫基，环烯基硫基，环烷基氨基，环烯基氨基，环烷基烷基，环烯基烷基，芳基，芳氧基，芳硫基，芳基氨基，芳基烷基，芳基烷氧基，芳基烷硫基或芳烷基氨基，表示来自该组的任选取代的基团通过在三组分反应中使通式（II）的三唑啉酮与磺酰卤反应，以良好的产率和高纯度获得烷基，环烷基，环烷基烷基，芳基，芳烷基，杂环基或杂环基烷基。通式（III）中R 3 -SO 2 -X（III）X =卤素和通式（IV）MOCN（IV）的金属氰酸酯，其中M表示碱金属或一种碱土金属当量，任选地在存在反应助剂，任选在稀释剂存在下，温度在20℃至150℃之间。

6. 发明授权

US09006266B2 Heteroarylpiperidine and -piperazine derivatives as fungicides 有权
标题翻译：杂芳基哌啶和哌嗪衍生物作为杀真菌剂
公开(公告)号：US09006266B2
公开(公告)日：2015-04-14
申请号：US13993262
申请日：2011-08-24
申请人： Tomoki Tsuchiya , Pierre Wasnaire , Sebastian Hoffmann , Pierre Cristau , Thomas Seitz , Joachim Kluth , Stefan Hillebrand , Juergen Benting , Daniela Portz , Ulrike Wachendorff-Neumann
发明人： Tomoki Tsuchiya , Pierre Wasnaire , Sebastian Hoffmann , Pierre Cristau , Thomas Seitz , Joachim Kluth , Stefan Hillebrand , Juergen Benting , Daniela Portz , Ulrike Wachendorff-Neumann
IPC分类号： A61K31/445 , C07D405/00 , A01N43/78 , A01N43/80 , A01N47/38 , A01N55/00 , C07D417/14
CPC分类号： A01N43/80 , A01N43/78 , A01N47/22 , A01N47/38 , A01N55/00 , C07D417/14 , C07F7/0812
摘要： Heteroarylpiperidine and -piperazine derivatives of the formula (I) in which the symbols A, X, Y, L1, L2, G, Q, p, R1, R2 and R10 are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).
摘要翻译：符号A，X，Y，L1，L2，G，Q，p，R1，R2和R10各自如说明书中所定义的式（I）的杂芳基哌啶和哌嗪衍生物，以及盐，金属络合物和式（I）化合物的N-氧化物及其用于控制植物病原性有害真菌的用途及其制备式（I）化合物的方法。

7. 发明授权

US08822693B2 Heteroarylpiperidine and-piperazine derivatives as fungicides 有权
标题翻译：杂芳基哌啶和哌嗪衍生物作为杀真菌剂
公开(公告)号：US08822693B2
公开(公告)日：2014-09-02
申请号：US13364168
申请日：2012-02-01
申请人： Sebastian Hoffmann , Pierre Wasnaire , Tomoki Tsuchiya , Pierre Cristau , Thomas Seitz , Joachim Kluth , Jürgen Benting , Ulrike Wachendorff-Neumann
发明人： Sebastian Hoffmann , Pierre Wasnaire , Tomoki Tsuchiya , Pierre Cristau , Thomas Seitz , Joachim Kluth , Jürgen Benting , Ulrike Wachendorff-Neumann
IPC分类号： C07D417/14 , A01N43/40 , C07D417/04 , A01N43/80
CPC分类号： C07D417/14 , A01N43/80 , C07D417/04
摘要： Heteroarylpiperidine and -piperazine derivatives of the formula (I) in which the symbols are each as defined in the description, and agrochemically active salts thereof, and use thereof for controlling phytopathogenic harmful fungi, and also processes for preparing compounds of the formula (I).
摘要翻译：符号分别如说明书中所定义的式（I）的杂芳基哌啶和哌嗪衍生物及其农业化学活性盐及其用于控制植物病原性有害真菌的用途，以及制备式（I）化合物的方法，。

8. 发明申请

US20110098287A1 Novel Heteroaromatic Amides And Thioamides As Pesticides 有权
标题翻译：新型杂芳族酰胺和硫代酰胺作为农药
公开(公告)号：US20110098287A1
公开(公告)日：2011-04-28
申请号：US12997803
申请日：2009-06-04
申请人： Thomas Bretschneider , Eva-Maria Franken , Ulrich Görgens , Martin Fusslein , Achim Hense , Joachim Kluth
发明人： Thomas Bretschneider , Eva-Maria Franken , Ulrich Görgens , Martin Fusslein , Achim Hense , Joachim Kluth
IPC分类号： A01N43/88 , C07D417/04 , C07D417/14 , C07D401/04 , C07D401/12 , C07D413/14 , A01N43/40 , A01N43/78 , A01N43/836 , A01N43/54 , A01P7/04 , A01P7/00
CPC分类号： A01N43/78 , A01N43/54 , A01N43/56 , A01N43/80 , A01N43/82 , A01N43/84 , A01N43/88 , A01N47/12 , A01N47/24 , C07D401/04 , C07D401/14 , C07D413/14 , C07D417/04 , C07D417/14
摘要： The present application relates to novel amides and thioamides, to processes for preparation thereof and to use thereof for controlling animal pests, in particular arthropods and especially insects.
摘要翻译：本申请涉及新型酰胺和硫代酰胺，其制备方法及其用于控制动物害虫，特别是节肢动物，特别是昆虫的用途。

9. 发明申请

US20050130843A1 Substituted thien-3-yl-sulphonylamino(thio)carbonyl-triazolin(ethi)ones 有权
标题翻译：取代的噻吩-3-基 - 磺酰基氨基（硫代）羰基 - 三唑啉（ethi）
公开(公告)号：US20050130843A1
公开(公告)日：2005-06-16
申请号：US11044969
申请日：2005-01-27
申请人： Ernst Gesing , Joachim Kluth , Klaus-Helmut Muller , Mark Drewes , Peter Dahmen , Dieter Feucht , Rolf Pontzen
发明人： Ernst Gesing , Joachim Kluth , Klaus-Helmut Muller , Mark Drewes , Peter Dahmen , Dieter Feucht , Rolf Pontzen
IPC分类号： A01N43/653 , A01N47/38 , A01P13/00 , C07D249/08 , C07D333/38 , C07D409/12 , C07D49/02
CPC分类号： C07D409/12 , A01N47/38 , C07D333/38
摘要： The invention relates to novel substituted thien-3-yl-sulphonylamino(thio)carbonyl-triazolin(ethi)ones of the general formula (I) in which Q1, Q2, R1, R2, R3 and R4 are each as defined in the description, and to salts of the compounds according to formula (I), to processes and to novel intermediates for their preparation and to their use as herbicides.
摘要翻译：本发明涉及通式（I）中的新的取代的噻吩-3-基 - 磺酰基氨基（硫代）羰基 - 三唑啉（ethi），其中Q 1，Q 2， R 1，R 2，R 3，R 4和R 4各自如说明书中所定义，和涉及式（I）化合物的盐，其制备方法和新型中间体及其作为除草剂的用途。

10. 发明授权

US06525211B1 Herbicidal sulphonylamino(thio)carbonyl compounds 失效
标题翻译：除草磺酰氨基（硫代）羰基化合物
公开(公告)号：US06525211B1
公开(公告)日：2003-02-25
申请号：US09838812
申请日：2001-04-20
申请人： Klaus-Helmut Müller , Rolf Kirsten , Ernst Rudolf F. Gesing , Joachim Kluth , Mark Wilhelm Drewes , Kurt Findeisen , Johannes Rudolf Jansen , Klaus König , Hans-Jochem Riebel , Otto Schallner , Markus Dollinger , Hans-Joachim Santel
发明人： Klaus-Helmut Müller , Rolf Kirsten , Ernst Rudolf F. Gesing , Joachim Kluth , Mark Wilhelm Drewes , Kurt Findeisen , Johannes Rudolf Jansen , Klaus König , Hans-Jochem Riebel , Otto Schallner , Markus Dollinger , Hans-Joachim Santel
IPC分类号： C07C30941
CPC分类号： C07D263/34 , A01N43/74 , A01N43/76 , A01N43/82 , A01N47/38 , C07C249/12 , C07C309/87 , C07C311/29 , C07C311/65 , C07C331/32 , C07D249/12 , C07D249/14 , C07D263/42 , C07D271/06 , C07D271/10 , C07D487/04
摘要： The invention relates to novel sulphonylamino(thio)carbonyl compounds of the formula (I), in which A represents a single bond, oxygen, sulphur or the group N—R, in which R represents hydrogen, alkyl, alkenyl, alkinyl or cycloalkyl, Q represents oxygen or sulphur, R1 represents hydrogen or formyl or represents in each case optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, cycloalkyl, cycloalkylcarbonyl or cycloalkylsulphonyl, R2 represents cyano or halogen or represents in each case optionally substituted alky, alkenyl, alkinyl, alkoxy, alkenyloxy or alkinyloxy, and R3 represents in each case optionally substituted heterocyclyl having 5 ring members of which at least one is oxygen, sulphur or nitrogen and from one to three further ring members can be nitrogen, and salts of compounds of the formula (I), the previously known compounds 4,5-dimethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one, 4,5-diethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one and N-(2,5-dimethoxy-phenylsulphonyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide being excluded by disclaimer; and also to processes and novel intermediates for the preparation of the novel substances and to their use as herbicides.
摘要翻译：本发明涉及式（I）的新型磺酰基氨基（硫代）羰基化合物，其中A表示单键，氧，硫或基团NR，其中R表示氢，烷基，烯基，炔基或环烷基，Q表示氧或硫，R1表示氢或甲酰基，或表示在各种情况下任选取代的烷基，烯基，炔基，烷基羰基，烷氧基羰基，烷基磺酰基，环烷基，环烷基羰基或环烷基磺酰基，R2表示氰基或卤素，或表示在各情况下任选取代的烷基，烯基，炔基，烷氧基，烯氧基或烷氧基，R 3在各自的情况下表示具有5个环成员的任选取代的杂环基，其中至少一个是氧，硫或氮，并且一至三个其它的环成员可以是氮， I），先前已知的化合物4,5-二甲氧基-2-（2,5-二甲氧基 - 苯基磺酰基氨基羰基）-2,4-二氢-3H-1,2,4-三唑-3-酮，4,5-二乙氧基 -2-（2,5-二甲氧基 - 苯基磺酰基氨基羰基）-2,4-二氢-3H-1,2,4-三唑-3-酮和N-（2,5-二甲氧基 - 苯基磺酰基）-1,5-二甲基-1H-吡唑-3-甲酰胺被排除在免责声明之外;还涉及用于制备新物质和用作除草剂的方法和新型中间体。

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