会员体验
专利管家(专利管理)
工作空间(专利管理)
风险监控(情报监控)
数据分析(专利分析)
侵权分析(诉讼无效)
联系我们
交流群
官方交流:
QQ群: 891211   
微信请扫码    >>>
现在联系顾问~
热词
    • 3. 发明授权
    • Oxime esters of substituted quinoline-8-carboxylic acids and use thereof
as herbicides
    • 取代喹啉-8-羧酸的肟酯及其作为除草剂的用途
    • US4808212A
    • 1989-02-28
    • US944519
    • 1986-12-22
    • Peter PlathKarl EickenBernd ZeehUlrich EichenauerHelmut HagenRolf-Dieter KohlerNorbert MeyerBruno Wuerzer
    • Peter PlathKarl EickenBernd ZeehUlrich EichenauerHelmut HagenRolf-Dieter KohlerNorbert MeyerBruno Wuerzer
    • C07D333/00A01N43/42A01N43/48A01N43/653C07D215/32C07D215/48C07D335/00C07D401/12C07D405/12C07D409/12C07D521/00
    • C07D231/12A01N43/42A01N43/653C07D215/32C07D233/56C07D249/08C07D405/12C07D409/12
    • Oxime esters of substituted quinoline-8-carboxylic acids of the formula ##STR1## where X is hydrogen, C.sub.1 -C.sub.4 -alkyl or halogen, Z is hydrogen or methyl, R.sup.1 is C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkoxymethyl, C.sub.1 -C.sub.4 -alkoxyethyl, C.sub.1 -C.sub.4 -alkylthiomethyl, C.sub.1 -C.sub.4 -alkylthioethyl, C.sub.1 -C.sub.4 -alkoxycarbonyl, C.sub.3 -C.sub.6 -alkenyl or C.sub.5 -C.sub.8 -cycloalkyl, each of which is unsubstituted or bears up to 3 methyl substituents, hydrogen, cyano, acetyl, benzoyl, unsubstituted benzyl or phenyl, or benzyl or phenyl bearing up to 3 substitutents selected from the group consisting of halogen, cyano, trifluoromethyl, C.sub.1 -C.sub.4 -haloalkyloxy, C.sub.1 -C.sub.6 -alkylthio, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkyl, hydroxy, dimethylamino or acetamino, R.sup.2 is hydrogen if R.sup.1 is not hydrogen, R.sup.2 further denotes C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkoxymethyl, chloromethyl, azolylmethyl, 1,1-dimethoxymethyl, cyano, C.sub.1 -C.sub.4 -alkoxycarbony, C.sub.1 -C.sub.4 -alkoxy, phenyl if R.sup.1 is H, CH.sub.3 or acetyl, or R.sup.2 denotes, when R.sup.1 is H or methyl, furyl, tetrahydrofuryl, thienyl, tetrahydropyranyl, tetrahydrothiopyranyl, dihydro-.DELTA..sup.3 -pyranyl or dihydro-.DELTA..sup.3 -thiopyranyl; further, R.sup.1 and R.sup.2, together with the carbon atom to which they are linked, denote C.sub.1 -C.sub.12 -cycloalkylidene, C.sub.5 -C.sub.6 -cycloalkenylidene or 4-oxacyclohexadienylidene, each of which is unsubstituted or bears up to 3 methyl substituents, it being possible, where the ring is 5-membered or 6-membered, or doubly unsaturated 6-membered, for it to contain an oxygen or sulfur atom, their preparation, and their use as herbicides.
    • 其中X是氢,C 1 -C 4烷基或卤素,Z是氢或甲基的取代喹啉-8-羧酸的肟酯,R 1是C 1 -C 6烷基,C 1 -C 4烷氧基甲基, C 1 -C 4 - 烷氧基乙基,C 1 -C 4 - 烷硫基甲基,C 1 -C 4 - 烷硫基乙基,C 1 -C 4 - 烷氧基羰基,C 3 -C 6 - 烯基或C 5 -C 8 - 环烷基,其各自为未取代的或至多含有3个甲基取代基 ,氰基,乙酰基,苯甲酰基,未取代的苄基或苯基,或带有至多3个选自卤素,氰基,三氟甲基,C 1 -C 4卤代烷氧基,C 1 -C 6 - 烷硫基,C 1 -C 4 - 烷氧基的取代基的苄基或苯基 C1-C4烷基,羟基,二甲基氨基或乙酰氨基,如果R1不是氢,R2是氢,R2还表示C1-C6-烷基,C1-C4-烷氧基甲基,氯甲基,唑基甲基,1,1-二甲氧基甲基,氰基,C1 -C 1-4烷氧基羰基,C 1 -C 4 - 烷氧基,如果R 1为H,CH 3或乙酰基,则为苯基,或R 2表示当R 1为H或甲基时,呋喃基,四氢呋喃基,噻吩基,四氢吡喃基,四氢噻喃基,二 水合-3β-吡喃基或二氢-D-3,3-噻喃基; 此外,R 1和R 2与它们所连接的碳原子一起表示C 1 -C 12 - 亚环烷基,C 5 -C 6 - 环亚烯基或4-氧杂环己二亚苯基,其各自是未取代的或最多含有3个甲基取代基,可能是 ,其中环为5元或6元,或双不饱和6元,含有氧或硫原子,其制备及其作为除草剂的用途。
    • 7. 发明授权
    • 2,3-substituted 1,8-naphthyridines, their preparation and their use as
antidotes
    • 2,3-取代的1,8-萘啶,其制备及其作为抗体使用
    • US5059240A
    • 1991-10-22
    • US486867
    • 1990-03-01
    • Helmut HagenJuergen PfisterHans ZieglerBruno WuerzerKarl-Otto Westphalen
    • Helmut HagenJuergen PfisterHans ZieglerBruno WuerzerKarl-Otto Westphalen
    • A01N25/32A01N43/90C07D471/04C07D471/14
    • C07D471/04A01N25/32C07D471/14
    • 2,3-substituted 1,8-naphthyridines of the general formula I ##STR1## where: R is hydrogen or C.sub.1 -C.sub.4 -alkyl (n=1 or 2)R.sup.1 is amino or substituted amino,XR.sup.5, where X is oxygen or sulfur and R.sup.5 is hydrogen, C.sub.1 -C.sub.12 -alkyl, C.sub.1 -C.sub.4 -alkoxycarbonyl-((C.sub.1 -C.sub.4)-alkyl, C.sub.5 -C.sub.8 -cycloakyl, substituted or unsubstituted phenyl, substituted or unsubstituted phenyl-(C.sub.1 -C.sub.3)-alkyl,halogen,isothiorhonium halide,C.sub.1 -C.sub.12 -alkyl,C.sub.1 -C.sub.4 -alkoxycarbonyl-C.sub.1 -C.sub.4 -alkyl,substituted or unsubstituted phenyl or phenyl-(C.sub.1 -C.sub.3)-alkyl,R.sup.2 is C.sub.1 -C.sub.4 -alkyl, cyano, carboxyl or a group ##STR2## where X is oxygen or sulfur,B is C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxy or alkylthio, amino, mono- or dialkylamino, where each alkyl radical is of 1 to 4 carbon atoms, morpholino, piperidyl, chlorine, bromine or substituted or unsubstituted phenyl,D is C.sub.1 -C.sub.4 alkyl or NH.sub.2 andR.sup.6 is hydrogen, C.sub.1 -C.sub.8 -alkyl or alkylcarbonyl,or R.sup.1 and R.sup.2 together are --NH--N.dbd.C(CH.sub.2)--,and their environmentally tolerated saltswith the proviso that R.sup.2 is not cyano, carboxyl or a carboxamido or carboxylic ester group when R.sup.1 is methyl, hydroxyl or amino (NH.sub.2), processes for their manufacture, and herbicidal agents containing a naphthyridine I as safener and at least one herbicidal active ingredient selected from the group consisting ofa) 2-(4-heteroaryloxy)- or 2-(4-aryloxy)-phenoxyacetic acid derivatives andb) cyclohexenone derivatives.
    • 具有通式I的2,3-取代的1,8-萘啶,其中:R是氢或C 1 -C 4 - 烷基(n = 1或2)R 1是氨基或取代的氨基,XR 5,其中X是氧 或(C 1 -C 4) - 烷基,C 5 -C 8 - 环烷基,取代或未取代的苯基,取代或未取代的苯基 - (C 1 -C 3) - 烷基,卤素,异卤卤化物,C 1 -C 12 - 烷基,C 1 -C 4 - 烷氧基羰基-C 1 -C 4烷基,取代或未取代的苯基或苯基 - (C 1 -C 3) - 烷基,R 2为C 1 -C 4烷基,氰基, 羧基或基团,其中X为氧或硫,B为C 1 -C 6 - 烷基,C 1 -C 6 - 烷氧基或烷硫基,氨基,单或二烷基氨基,其中每个烷基为1至4个碳原子,吗啉代 ,哌啶基,氯,溴或取代或未取代的苯基,D是C 1 -C 4烷基或NH 2,R 6是氢,C 1 -C 8 - 烷基或烷基羰基,或者R 1和R 2一起是-NH-N = C(CH 2) 其环境耐受性盐,条件是R2不是氰基,羧基或a 当R1是甲基,羟基或氨基(NH2)时,羧酰胺基或羧酸酯基,其制备方法和含有萘啶I作为安全剂的除草剂和至少一种除草活性成分,其选自a)2-(4 - 杂芳氧基) - 或2-(4-芳氧基) - 苯氧基乙酸衍生物和b)环己烯酮衍生物。
    • 9. 发明授权
    • Novel 4'(benzisothiazo-5-yloxy)-phenylurea derivatives, their
preparation and their use as herbicides
    • 新型4'(苯并异噻唑-5-基氧基) - 苯基脲衍生物,其制备及其作为除草剂的用途
    • US4589910A
    • 1986-05-20
    • US727628
    • 1985-04-30
    • Helmut HagenHans ZieglerBruno Wuerzer
    • Helmut HagenHans ZieglerBruno Wuerzer
    • A01N47/30C07D275/04A01N47/38
    • C07D275/04A01N47/30
    • A 4'-(Benzisothiazol-5-yloxy)-phenylureas of the formula ##STR1## where R.sup.1 and R.sup.2 are each a saturated straight-chain or branched aliphatic radical of 1 to 10 carbon atoms, an unsaturated straight-chain or branched aliphatic radical of 3 to 10 carbon atoms, or an araliphatic or aromatic radical which may be substituted by 1, 2 or 3 C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, cyano, halogen, nitro, monofluoromethyl or trifluoromethyl groups, or are each alkoxy of 1 to 6 carbon atoms, R.sup.2 may furthermore be hydrogen, or R.sup.1 and R.sup.2, together with the nitrogen atom, may be members of a 5-membered or 6-membered ring which may contain further nitrogen and/or oxygen atoms as heteroatoms, and X is hydrogen, trifluoromethyl or chlorine, processes for their preparation, and herbicides containing ureas of the formula I as active ingredients.
    • 式Ⅰ的4' - (苯并异噻唑-5-基氧基) - 苯基,其中R 1和R 2各自是1-10个碳原子的饱和直链或支链脂族基团,不饱和直链或支链脂族基 或可被1,2或3个C 1 -C 4 - 烷基,C 1 -C 4 - 烷氧基,氰基,卤素,硝基,单氟甲基或三氟甲基取代的芳脂族或芳族基团,或各自为 具有1至6个碳原子的烷氧基,R 2还可以是氢,或者R 1和R 2与氮原子一起可以是可以含有另外的氮原子和/或氧原子作为杂原子的5元或6元环的成员 ,X为氢,三氟甲基或氯,其制备方法,以及含有式I的脲的除草剂作为活性成分。