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1. 发明授权

US4020164A Benzomorphan derivatives 失效
标题翻译：苯并吗啉衍生物
公开(公告)号：US4020164A
公开(公告)日：1977-04-26
申请号：US550611
申请日：1975-02-18
申请人： Dieter Rahtz , Eberhard Schroder , Reinhard Horowski , Gert Paschelke , Dieter Palenschat , Helmut Wachtel , Wolfgang Kehr
发明人： Dieter Rahtz , Eberhard Schroder , Reinhard Horowski , Gert Paschelke , Dieter Palenschat , Helmut Wachtel , Wolfgang Kehr
IPC分类号： C07D221/26 , A61K31/445
CPC分类号： C07D221/26
摘要： Benzomorphans of the formula ##STR1## wherein R.sub.1 is H, CH.sub.3 or C.sub.2 H.sub.5 ; R.sub.2 is CH.sub.3 or C.sub.2 H.sub.5 and R.sub.3 and R.sub.4, which can be alike or different, each are lower alkyl, and the acid addition salts thereof with physiologically acceptable acids have CNS activity, including analgesic, morphine antagonistic, anti-convulsive, muscle relaxant, sedative and neuroleptic activity.
摘要翻译：其中R 1是H，CH 3或C 2 H 5的式[IMAGE]的苯并吗啡; R2是CH3或C2H5，R3和R4可以相同或不同，各自为低级烷基，其与生理上可接受的酸的酸加成盐具有CNS活性，包括止痛，吗啡拮抗，抗惊厥，肌肉松弛剂，镇静剂和精神安定药活动。

2. 发明授权

US3952007A Processes for preparing 5-nitro-1-methyl-2-(2-dialkylaminovinyl)-imidazole and 5-nitro-1-methyl-2-imidazolyl carboxaldehyde 失效
标题翻译：制备5-硝基-1-甲基-2-（2-二烷基氨基乙烯基） - 咪唑和5-硝基-1-甲基-2-咪唑基甲醛的方法
公开(公告)号：US3952007A
公开(公告)日：1976-04-20
申请号：US316928
申请日：1972-12-20
申请人： Clemens Rufer , Eberhard Schroder
发明人： Clemens Rufer , Eberhard Schroder
IPC分类号： B01J23/00 , C07D233/92 , C07D233/94 , C07D233/95 , C07D401/06 , C07D405/06 , C07D413/12 , C07D295/22
CPC分类号： C07D233/95 , C07D233/92 , C07D233/94
摘要： 1-SUBSTITUTED 5-NITRO-2-(2-DIALKYLAMINOVINYL)-IMIDAZOLES HAVING TRICHOMONACIDAL ACTIVITY OF THE FORMULA: ##SPC1##Wherein R is H, CH.sub.3 or C.sub.2 H.sub.5 and X is hydrocarbon or hydrocarbon substituted with a halogen or a hydroxy, ether, ester or amino group, are produced by reacting the 1-substituted-5-nitro-2-alkyl-imidazoles with an aminal ester or amidoacetal of orthoformic acid or like functionally reactive derivative thereof.
摘要翻译： 1-取代的5-硝基-2-（2-二烷基氨基乙基） - 具有公式的三氯杀菌活性的咪达唑仑：

3. 发明授权

US5859373A Apparatus and process for determining the instantaneous and continuous loads on a lifting mechanism 失效
标题翻译：用于确定提升机构上的瞬时和连续负载的装置和过程
公开(公告)号：US5859373A
公开(公告)日：1999-01-12
申请号：US840859
申请日：1997-04-17
申请人： Anton Munzebrock , Eberhard Schroder , Michael Hulsmann
发明人： Anton Munzebrock , Eberhard Schroder , Michael Hulsmann
IPC分类号： G01L5/00 , B66C13/16 , B66D1/46 , B66D1/54 , G07C3/00 , H02P29/40 , G01L1/04
CPC分类号： G07C3/00 , B66C13/16 , B66D1/54 , H02P29/40
摘要： A process and apparatus for determining a load on a lifting mechanism including a load measuring device and a three-phase induction motor operable for lifting and lowering the load. The effective power consumption of the induction motor is determined by the load measuring device based on a measured current and measured voltage of the induction motor. The measured effective power consumption is then compared with a reference power, which is calculated as the power output of the induction motor driving a nominal load of the lifting mechanism, to calculated an instantaneous load on the lifting mechanism. The inventive apparatus and process advantageously requires no modifications or additions to load carrying parts of a lifting mechanism or carrying gear and provides accurate real time measurement of the load.
摘要翻译：一种用于确定提升机构上的负载的方法和装置，包括负载测量装置和用于提升和降低负载的三相感应电动机。感应电动机的有效功率消耗由负载测量装置基于测量的电流和感应电动机的测量电压来确定。然后将测量的有效功率消耗与参考功率进行比较，该参考功率是以驱动提升机构的额定负载的感应电动机的功率输出计算的，以计算提升机构上的瞬时负载。本发明的装置和方法有利地不需要对提升机构或承载装置的承载部件进行修改或添加，并提供负载的精确的实时测量。

4. 发明授权

US3956295A Carbazole derivatives 失效
标题翻译：咔唑衍生物
公开(公告)号：US3956295A
公开(公告)日：1976-05-11
申请号：US489162
申请日：1974-07-17
申请人： Helmut Biere , Hanns Ahrens , Clemens Rufer , Eberhard Schroder , Henning Koch
发明人： Helmut Biere , Hanns Ahrens , Clemens Rufer , Eberhard Schroder , Henning Koch
IPC分类号： A61K31/405 , C07D209/88 , C07D209/82
CPC分类号： C07D209/88 , A61K31/405 , Y10S514/887
摘要： Carbazoles of the formula ##SPC1##Wherein R.sub.1 is hydroxymethyl, alkanoyloxymethyl, tetrazolyl, cyano, oximinocarbonyl, aminocarbonyl, carboxyl and salts thereof with physiologically acceptable bases and the esters thereof with physiologically acceptable alcohols and amides thereof with physiologically acceptable amines,R.sub.2 through R.sub.6 each are a hydrogen atom, halogen atom, lower alkyl, trifluoromethyl, or lower alkoxy, orR.sub.5 and R.sub.6 collectively are a five- or six-membered isocyclic ring, andR.sub.7 is a hydrocarbon of 3-8 carbon atoms or, when at least one of the R.sub.2 through R.sub.6 is other than a hydrogen atom, a hydrogen atom, methyl or ethyl,And the corresponding compounds wherein R.sub.7 is a hydrogen atom, methyl or ethyl,And the 5,6,7,8-tetrahydrocarbazoles, possess topical anti-inflammatory activity.
摘要翻译：式VIII的咔唑，其中R1是羟甲基，烷酰氧基甲基，四唑基，氰基，肟基羰基，氨基羰基，羧基及其盐与生理上可接受的碱，其酯与其生理上可接受的醇和酰胺与生理上可接受的胺，R2至R6各自为氢原子，卤素原子，低级烷基，三氟甲基或低级烷氧基，或者R5和R6共同是五元或六元的环状环，并且R 7是3-8个碳原子的烃，或者当R2中的至少一个通过R6不同于氢原子，氢原子，甲基或乙基，以及其中R7是氢原子，甲基或乙基的相应化合物，以及5,6,7,8-四氢四硼化物，POSSESS局部抗炎活性。

5. 发明授权

US3966732A Nitroimidazolyl pyrimidines 失效
标题翻译：硝基咪唑基嘧啶
公开(公告)号：US3966732A
公开(公告)日：1976-06-29
申请号：US568117
申请日：1975-04-14
申请人： Clemens Rufer , Eberhard Schroder , Hans-Joachim Kessler
发明人： Clemens Rufer , Eberhard Schroder , Hans-Joachim Kessler
IPC分类号： C07D403/04 , C07D409/14 , C07D277/06
CPC分类号： C07D409/14 , C07D403/04
摘要： Nitroimidazolyl pyrimidines of the formula ##SPC1##And physiologically acceptable acid addition salts thereon wherein X is alkyl of 1-4 carbon atoms, R.sub.1 and R.sub.2 each are a hydrogen atom, alkyl of 1-4 carbon atoms, phenyl triflouromethyl or a monocyclic heterocyclic ring and R.sub.3 is a hydrogen atoms, alkyl of 1-4 carbon atoms, hydroxyalkoxy of 2-4 carbon atoms or an ester thereof of an alkanocarboxylic acid of 1-4 carbon atoms, oxoalkyl of 8-6 carbon atoms, or, when R.sub.1 or R.sub.2 is phenyl, alkylene having 1-2 carbon atoms in the chain joined to the 2-position of the phenyl ring possess trichomonicidal activity.
摘要翻译：式的硝基咪唑基嘧啶及其生理学上可接受的酸的添加剂其中X是1-4个碳原子的烷基，R1和R2各自是氢原子，1-4个碳原子的烷基，苯基三氟乙基或单环杂环，R3是 1-4个碳原子的烷基，2-4个碳原子的羟基烷氧基或其1-4个碳原子的链烷酸的酯，8-6个碳原子的氧代烷基，或当R1或R2是苯基时在与苯环的2-位连接的链中具有1-2个碳原子的亚烷基具有杀虫活性。

6. 发明授权

US3962453A Novel pyrazolyloxyacetic acid derivatives and process for the preparation thereof 失效
标题翻译：新型吡唑氧基乙酸衍生物及其制备方法
公开(公告)号：US3962453A
公开(公告)日：1976-06-08
申请号：US505208
申请日：1974-09-12
申请人： Hans Ahrens , Helmut Biere , Clemens Rufer , Eberhard Schroder , Henning Koch
发明人： Hans Ahrens , Helmut Biere , Clemens Rufer , Eberhard Schroder , Henning Koch
IPC分类号： C07D231/20 , A61K31/415 , A61P29/00 , C07D231/22 , C07D231/18
CPC分类号： C07D231/22
摘要： Compounds of the formula ##SPC1##Wherein X and Y each are a bond or methylene, R is H or lower-alkyl and Z is a carboxyl, amide, nitrile or alkoxycarbonyl of 1-6 carbon atoms in the alkoxy group and the corresponding compounds bearing 1-2 halogen, lower-alkyl or lower-alkoxy groups on one or both benzene rings and, when Z is carboxyl, salts thereof with physiologically acceptable bases, possess anti-inflammatory and antipyretic activities.
摘要翻译：式WHEREIN X和Y各自为键或亚甲基的化合物，R为H或低级烷基，Z为烷氧基中1-6个碳原子的羧基，酰胺，腈或烷氧基羰基，一个或两个苯环上的2个卤素，低级烷基或低级烷氧基，当Z为羧基时，其盐与生理上可接受的碱基具有抗炎和解热活性。

7. 发明授权

US3960949A 1,2-Biguanides 失效
标题翻译： 1,2双胍
公开(公告)号：US3960949A
公开(公告)日：1976-06-01
申请号：US486758
申请日：1974-07-09
申请人： Hanns Ahrens , Clemens Rufer , Helmut Biere , Eberhard Schroder , Wolfgang Losert , Olaf Loge , Ekkehard Schillinger
发明人： Hanns Ahrens , Clemens Rufer , Helmut Biere , Eberhard Schroder , Wolfgang Losert , Olaf Loge , Ekkehard Schillinger
IPC分类号： C07C279/26 , C07C129/16
CPC分类号： C07C279/26
摘要： 1,2-Substituted biguanides of the formula ##EQU1## wherein R.sub.1 is saturated or unsaturated, straight-chain or branched hydrocarbon of 1-12 carbon atoms which is unsubstituted or substituted by one or more fluorine atoms; a cycloalkyl group of 3-6 carbon atoms; or an aryl or aralkyl group of the formula ##SPC1##With n being the integer 0, 1 or 2 and X being hydrogen or halogen; and R'.sub.1 is a hydrogen atom or a saturated or unsaturated, straight-chain or branched hydrocarbon group of 1-12 carbon atoms; or R.sub.1 and R'.sub.1 collectively with the nitrogen atom to which they are attached are a heterocyclic ring containing one or more hetero atoms; and R.sub.2 is saturated or unsaturated, straight-chain or branched hydrocarbon of 1-12 carbon atoms which is unsubstituted or substituted by one or more fluorine atoms; or cycloalkyl of 3-6 carbon atoms, alkoxyalkyl containing a total of 2-12 carbon atoms, or alkoxy of 1-6 atoms; mixtures thereof, and pharmaceutically acceptable acid addition salts thereof, are useful in the treatment of diabetes mellitus.
摘要翻译： 1,2-取代的式R'1 | R1-NC-NH-C-NH2的平行二亚胺平行平行NNH | R2其中R1是1-12个碳原子的饱和或不饱和的直链或支链烃，未取代或未取代的被一个或多个氟原子取代; 3-6个碳原子的环烷基; 或下式的芳基或芳烷基：其中N为整数0,1或2且X为氢或卤素; 并且R'1是1-12个碳原子的氢原子或饱和或不饱和的直链或支链烃基; 或者R1和R'1与它们所连接的氮原子一起是含有一个或多个杂原子的杂环; R2是未被取代或被一个或多个氟原子取代的1-12个碳原子的饱和或不饱和的直链或支链烃基; 或3-6个碳原子的环烷基，总共2-12个碳原子的烷氧基烷基或1-6个原子的烷氧基; 其混合物及其药学上可接受的酸加成盐可用于治疗糖尿病。

8. 发明申请

US20050110451A1 Method for stabilizing the movement of an articulated chain of a chain block, especially to prevent the formation of a resonance oscillation of the chain, and a chain block apparatus 失效
标题翻译：用于稳定链块的铰接链的运动的方法，特别是用于防止链的共振振荡的形成，链节装置
公开(公告)号：US20050110451A1
公开(公告)日：2005-05-26
申请号：US10814902
申请日：2004-03-31
申请人： Eberhard Schroder , Giuliano Persico
发明人： Eberhard Schroder , Giuliano Persico
IPC分类号： B66D3/20 , B66D1/48 , B66D3/26 , H02P29/00 , G05B5/01
CPC分类号： B66D1/485
摘要： The invention concerns a method for stabilizing the motion of an articulated chain of a chain block, especially to prevent the formation of resonance oscillation of the chain, in which an articulated chain is led across a polygonal chain wheel with non-uniform pitch, which is driven by an electric motor. In order to create a method to prevent the formation of a resonance oscillation of the articulated chain, it is proposed that a periodic and/or stochastic and dampening actuating variable is superimposed on the velocity of the chain wheel (4) and the dampening actuating variable produces a change in the chain velocity so as to prevent a formation of a resonance oscillation. The chain drive with reduced polygon effect is characterized in that an electronic damper (8) is hooked up in front of the electric motor (2), which produces a control of the electric motor (2) such that a formation of a resonance oscillation of the articulated chain (5) is prevented.
摘要翻译：本发明涉及一种用于稳定链块的铰接链的运动的方法，特别是用于防止链条的共振振荡的形成，其中铰接链被引导穿过具有非均匀间距的多边形链轮，由电动机驱动。为了创建一种防止关节链形成共振振荡的方法，提出周期性和/或随机衰减和阻尼致动变量叠加在链轮（4）的速度和阻尼致动变量产生链速度的变化，以防止形成共振振荡。具有减少的多边形效应的链条驱动器的特征在于，电子阻尼器（8）被钩在电动机（2）的前面，其产生电动机（2）的控制，使得形成共振振荡铰链链（5）被防止。

9. 发明授权

US4289777A Quinolonecarboxylic acid derivatives and pharmaceutical preparations thereof for treatment of an allergic disease of the respiratory tract 失效
标题翻译：喹诺酮羧酸衍生物及其药物制剂，用于治疗呼吸道过敏性疾病
公开(公告)号：US4289777A
公开(公告)日：1981-09-15
申请号：US107676
申请日：1979-12-27
申请人： Rudolf Albrecht , Eberhard Schroder , Irmgard Bottcher
发明人： Rudolf Albrecht , Eberhard Schroder , Irmgard Bottcher
IPC分类号： A61K31/47 , A61P29/00 , A61P31/04 , A61P37/08 , C07D215/56 , C07D401/12
CPC分类号： C07D215/56
摘要： Quinolonecarboxylic acid derivatives of the formula ##STR1## wherein the grouping ##STR2## is independently in the 6-, 7- or 8-position of each of the quinolone residues;m and n independently are each 1-4;R.sub.1 is hydrogen or alkyl of 1-6 carbon atoms;R.sub.2 is hyrogen, alkanoyl of 1-8 carbon atoms or benzoyl; andX is hydrogen, alkyl of 1-6 carbon atoms or the cation of a base which produces a physiologically acceptable salt with the quinolonecarboxylic acid,have valuable pharmacological properties.
摘要翻译：喹诺酮羧酸衍生物，其分子式“IMAGE”独立地在每个喹诺酮残基的6-，7-或8-位; m和n各自独立地为1-4; R1是氢或1-6个碳原子的烷基; R2为氢，1-8个碳原子的烷酰基或苯甲酰基; X为氢，1-6个碳原子的烷基或与喹诺酮羧酸产生生理上可接受的盐的碱的阳离子，具有有价值的药理学性质。

10. 发明授权

US4057640A 5,6,7,8:Tetrahydrocarbazole-1-carboxylic acid derivatives 失效
标题翻译： 5,6,7,8：四氢咔唑-1-羧酸衍生物
公开(公告)号：US4057640A
公开(公告)日：1977-11-08
申请号：US683752
申请日：1976-05-06
申请人： Helmut Biere , Hanns Ahrens , Clemens Rufer , Eberhard Schroder , Henning Koch
发明人： Helmut Biere , Hanns Ahrens , Clemens Rufer , Eberhard Schroder , Henning Koch
IPC分类号： A61K31/405 , C07D209/88 , A61K31/40
CPC分类号： C07D209/88 , A61K31/405
摘要： Carbazoles of the formula ##STR1## wherein R.sub.1 is hydroxymethyl, alkanoyloxymethyl, tetrazolyl, cyano, oximinocarbonyl, aminocarbonyl, carboxyl and salts thereof with physiologically acceptable bases and the esters thereof with physiologically acceptable alcohols and amides thereof with physiologically acceptable amines,R.sub.2 through R.sub.6 each are a hydrogen atom, halogen atom, lower alkyl, trifluoromethyl, or lower alkoxy, orR.sub.5 and R.sub.6 collectively are a five- or six-membered isocyclic ring, andR.sub.7 is a hydrocarbon of 3-8 carbon atoms or, when at least one of the R.sub.2 through R.sub.6 is other than a hydrogen atom, a hydrogen atom, methyl or ethyl,And the corresponding compounds wherein R.sub.7 is a hydrogen atom, methyl or ethyl,And the 5,6,7,8-tetrahydrocarbazoles, possess topical anti-inflammatory activity.
摘要翻译：其中R 1为羟甲基，烷酰氧基甲基，四唑基，氰基，肟基羰基，氨基羰基，羧基及其盐与生理上可接受的碱，其酯与其生理上可接受的醇和酰胺与生理上可接受的胺，R 2至R 6各自相同是氢原子，卤素原子，低级烷基，三氟甲基或低级烷氧基，或者R5和R6共同是五元或六元的环状环，而R7是3-8个碳原子的烃，或者当至少一个 R 2至R 6不是氢原子，氢原子，甲基或乙基，并且R 7是氢原子，甲基或乙基的相应化合物，以及5,6,7,8-四氢四硼化物，POSSESS主题抗体 -INFLAMMATORY活动。

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