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1. 发明申请

US20110319617A1 Rosuvastatin and Atorvastatin Derivatives 失效
标题翻译：罗苏伐他汀和阿托伐他汀衍生物
公开(公告)号：US20110319617A1
公开(公告)日：2011-12-29
申请号：US13255700
申请日：2010-03-10
申请人： Derek Lindsay , Peter Jackson , Stephen Hindley , Inder Bhamra
发明人： Derek Lindsay , Peter Jackson , Stephen Hindley , Inder Bhamra
IPC分类号： C07D239/42
CPC分类号： C07D405/06 , A61K31/40 , A61K31/506 , C07D405/14
摘要： This invention relates to the discovery of novel rosuvastatin and atorvastatin analogues.
摘要翻译：本发明涉及新型罗苏伐他汀和阿托伐他汀类似物的发现。

2. 发明授权

US08877945B2 Redox drug derivatives 有权
标题翻译：氧化还原药物衍生物
公开(公告)号：US08877945B2
公开(公告)日：2014-11-04
申请号：US13319377
申请日：2010-05-17
申请人： Derek Lindsay , Peter Jackson
发明人： Derek Lindsay , Peter Jackson
IPC分类号： C07D401/10 , C07D209/48 , C07D317/30 , C07D405/06
CPC分类号： C07D215/233 , C07C233/52 , C07D209/46 , C07D317/28 , C07D405/06 , C07D498/06
摘要： The present invention provides redox drug derivatives. In particular, 9-fluoro-2,3-dihydro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-7H-pyrido[1,2,3-de]-1,4-benzoxazine-6-carboxylic acid, 1-ethyl-6-fluoro-1,4-dihydro-7-(4-methyl-1-piperazinyl)-4-oxo-3-quinolinecarboxylic acid, (3R,4R,5S)-4-(acetylamino)-5-amino-3-(1-ethylpropoxy)-1-cyclohexene-1-carboxylic acid ethyl ester, (3S)-3-(aminomethyl)-5-methylhexanoic acid, (3S)-1-[2-(2,3-dihydro-5-benzofuranyl)ethyl]-α-α-diphenyl-3-pyrrolidineacetamide, (1S,2S,3S,4R)-3-[(1S)-1-acetamido-2-ethyl-butyl]-4-(diaminomethylideneamino)-2-hydroxy-cyclopentane-1-carboxylic acid and (2R,3R,4S)-4-[(diaminomethylidene)amino]-3-acetamido-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acid redox derivatives.
摘要翻译：本发明提供了氧化还原药物衍生物。特别地，9-氟-2,3-二氢-3-甲基-10-（4-甲基-1-哌嗪基）-7-氧代-7H-吡啶并[1,2,3-de] 苯并恶嗪-6-羧酸，1-乙基-6-氟-1,4-二氢-7-（4-甲基-1-哌嗪基）-4-氧代-3-喹啉羧酸（3R，4R，5S） - 4-（乙酰氨基）-5-氨基-3-（1-乙基丙氧基）-1-环己烯-1-羧酸乙酯，（3S）-3-（氨基甲基）-5-甲基己酸，（3S）-1- 乙基]-α-α-二苯基-3-吡咯烷乙酰胺，（1S，2S，3S，4R）-3 - [（1S）-1-乙酰氨基-2- 乙基 - 丁基] -4-（二氨基亚甲基氨基）-2-羟基 - 环戊烷-1-羧酸和（2R，3R，4S）-4 - [（二氨基亚甲基）氨基] -3-乙酰氨基-2 - [（1R，2R ）-1,2,3-三羟丙基] -3,4-二氢-2H-吡喃-6-羧酸氧化还原衍生物。

3. 发明申请

US20120004408A1 Use of Rosuvastatin Lactols as Medicaments 审中-公开
标题翻译：使用罗苏伐他汀乳糖作为药物
公开(公告)号：US20120004408A1
公开(公告)日：2012-01-05
申请号：US13255705
申请日：2010-03-10
申请人： Derek Lindsay , Peter Jackson
发明人： Derek Lindsay , Peter Jackson
IPC分类号： C07D405/14 , C07D405/06
CPC分类号： C07D405/06 , A61K31/505 , C07D405/14
摘要： This invention relates to the discovery of novel rosuvastatin analogues. More specifically, the invention relates to novel rosuvastatin analogues which have utility in treating conditions treatable by the inhibition of HMG-CoA reductase.
摘要翻译：本发明涉及新型瑞舒伐他汀类似物的发现。更具体地，本发明涉及可用于治疗可通过抑制HMG-CoA还原酶治疗的病症的新型瑞舒伐他汀类似物。

4. 发明申请

US20120077974A1 REDOX DRUG DERIVATIVES 有权
标题翻译： REDOX药物衍生物
公开(公告)号：US20120077974A1
公开(公告)日：2012-03-29
申请号：US13319377
申请日：2010-05-17
申请人： Derek Lindsay , Peter Jackson
发明人： Derek Lindsay , Peter Jackson
IPC分类号： C07D401/10 , C07D209/48 , C07D317/30 , C07D405/06 , C07C271/24 , C07D498/06 , C07D209/46
CPC分类号： C07D215/233 , C07C233/52 , C07D209/46 , C07D317/28 , C07D405/06 , C07D498/06
摘要： The present invention provides redox drug derivatives. In particular, 9-fluoro-2,3-dihydro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-7H-pyrido[1,2,3-de]-1,4-benzoxazine-6-carboxylic acid, 1-ethyl-6-fluoro-1,4-dihydro-7-(4-methyl-1-piperazinyl)-4-oxo-3-quinolinecarboxylic acid, (3R,4R,5S)-4-(acetylamino)-5-amino-3-(1-ethylpropoxy)-1-cyclohexene-1-carboxylic acid ethyl ester, (3S)-3-(aminomethyl)-5-methylhexanoic acid, (3S)-1-[2-(2,3-dihydro-5-benzofuranyl)ethyl]-α-α-diphenyl-3-pyrrolidineacetamide, (1S,2S,3S,4R)-3-[(1S)-1-acetamido-2-ethyl-butyl]-4-(diaminomethylideneamino)-2-hydroxy-cyclopentane-1-carboxylic acid and (2R,3R,4S)-4-[(diaminomethylidene)amino]-3-acetamido-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acid redox derivatives.
摘要翻译：本发明提供了氧化还原药物衍生物。特别地，9-氟-2,3-二氢-3-甲基-10-（4-甲基-1-哌嗪基）-7-氧代-7H-吡啶并[1,2,3-de] 苯并恶嗪-6-羧酸，1-乙基-6-氟-1,4-二氢-7-（4-甲基-1-哌嗪基）-4-氧代-3-喹啉羧酸（3R，4R，5S） - 4-（乙酰氨基）-5-氨基-3-（1-乙基丙氧基）-1-环己烯-1-羧酸乙酯，（3S）-3-（氨基甲基）-5-甲基己酸，（3S）-1- 乙基]-α-α-二苯基-3-吡咯烷乙酰胺，（1S，2S，3S，4R）-3 - [（1S）-1-乙酰氨基-2- 乙基 - 丁基] -4-（二氨基亚甲基氨基）-2-羟基 - 环戊烷-1-羧酸和（2R，3R，4S）-4 - [（二氨基亚甲基）氨基] -3-乙酰氨基-2 - [（1R，2R ）-1,2,3-三羟丙基] -3,4-二氢-2H-吡喃-6-羧酸氧化还原衍生物。

5. 发明授权

US08513412B2 Rosuvastatin and atorvastatin derivatives 失效
公开(公告)号：US08513412B2
公开(公告)日：2013-08-20
申请号：US13255700
申请日：2010-03-10
申请人： Derek Lindsay , Peter Jackson , Stephen Hindley , Inder Bhamra
发明人： Derek Lindsay , Peter Jackson , Stephen Hindley , Inder Bhamra
IPC分类号： C07D239/02
CPC分类号： C07D405/06 , A61K31/40 , A61K31/506 , C07D405/14
摘要： This invention relates to the discovery of novel rosuvastatin and atorvastatin analogues.

6. 发明申请

US20110319626A1 Use of Atorvastatin Lactols as Medicaments 审中-公开
标题翻译：使用阿托伐他汀乳糖作为药物
公开(公告)号：US20110319626A1
公开(公告)日：2011-12-29
申请号：US13255707
申请日：2010-03-10
申请人： Derek Lindsay , Peter Jackson
发明人： Derek Lindsay , Peter Jackson
IPC分类号： C07D401/14 , C07D405/06
CPC分类号： A61K31/40
摘要： This invention relates to the discovery of novel atorvastatin analogues. More specifically, the invention relates to novel atorvastatin analogues which have utility in treating conditions treatable by the inhibition of HMG-CoA reductase.
摘要翻译：本发明涉及新型阿托伐他汀类似物的发现。更具体地，本发明涉及可用于治疗可通过抑制HMG-CoA还原酶治疗的病症的新型阿托伐他汀类似物。

7. 发明授权

US09035259B2 Level measurement system 有权
标题翻译：液位测量系统
公开(公告)号：US09035259B2
公开(公告)日：2015-05-19
申请号：US13119607
申请日：2009-09-18
申请人： Paul David Featonby , Peter Jackson , Benjamin Metcalfe , Thomas John Partington
发明人： Paul David Featonby , Peter Jackson , Benjamin Metcalfe , Thomas John Partington
IPC分类号： G01F23/00 , G01F23/288
CPC分类号： G01F23/288 , G01F23/2885
摘要： An instrument adapted for the determination of fluid levels within a vessel by the comparison of the density of the fluid along the length of the instrument, said instrument comprising: (i) at least one generally linear source array comprising a plurality of sources of penetrating radiation, shielding and collimation means and a source supporting structure for supporting the sources and shielding and collimation means in a linear array (ii) at least one generally linear detector array comprising a plurality of radiation detectors, supported on a detector support structure, capable of detecting radiation emitted by the sources, and (iii) means to position the source and a respective detector array such that (a) radiation emitted from each of the sources is capable of following a linear path from the source, through the vessel and material to at least a respective one of the detectors forming a part of the respective detector array, and (b) the linear axis of the source array and the linear axis of its respective detector array are substantially parallel to each other (iv) means for analyzing the detector output signals to determine the density of the medium traversed by the beams of radiation in passing from a source to a detector characterized in that the detector support structure and/or its associated electrical circuits and connectors is formed from a plurality of modular portions, each modular portion being adapted to be joined to an adjacent portion to provide a detector array of the required length.
摘要翻译：一种适于通过比较沿着仪器长度的流体密度来确定容器内液体水平的仪器，所述仪器包括：（i）至少一个大致线性的源阵列，其包括多个穿透辐射源，屏蔽和准直装置以及用于支撑源的源支撑结构，以及线性阵列中的屏蔽和准直装置（ii）至少一个大致线性的检测器阵列，其包括支撑在检测器支撑结构上的多个辐射检测器，能够检测由源发射的辐射，以及（iii）用于定位源和相应检测器阵列的装置，使得（a）从每个源发射的辐射能够跟随来自源的线性路径，通过容器和材料到达形成检测器阵列的一部分的检测器中的相应的一个检测器阵列，以及（b）源极阵列和线的轴线相应检测器阵列的耳轴基本上彼此平行（iv）用于分析检测器输出信号以确定由源到检测器的辐射束穿过的介质的密度的装置，其特征在于检测器支撑结构和/或其相关联的电路和连接器由多个模块化部分形成，每个模块化部分适于连接到相邻部分以提供所需长度的检测器阵列。

8. 发明申请

US20120128906A1 CROSSLINKED CHLORINATED POLYOLEFIN COMPOSITIONS 审中-公开
标题翻译：交联氯化聚烯烃组合物
公开(公告)号：US20120128906A1
公开(公告)日：2012-05-24
申请号：US13112859
申请日：2011-05-20
申请人： Peter Jackson , Joseph R. Prema
发明人： Peter Jackson , Joseph R. Prema
IPC分类号： C08L23/28 , B65B53/02 , C08K3/22 , C08L51/00 , C08K3/10
CPC分类号： C08F8/42 , Y10T428/1331
摘要： A chlorinated polyolefin composition suitable for use in the manufacture of crosslinked, thermoset, flame-retardant articles such as jackets for electrical or fiber optic cables, insulating coatings or layers for electrical conductors, and heat-shrinkable tubing, sheets or other shapes for protection of cable connectors and splices. The composition is thermosetting and moisture curable and comprises a chlorinated polyolefin such as chlorinated polyethylene or chlorosulfonated polyethylene and a non-chlorinated polyolefin which contains moisture crosslinkable silane groups. The non-chlorinated polyolefin preferably comprises polyethylene or a copolymer thereof. Exposure of the composition to moisture causes the formation of intermolecular crosslinks between molecules of the non-chlorinated polyolefin. The compositions can be formed by blending the non-chlorinated polyolefin with a silanated non-chlorinated polyolefin or by silane-grafting a blend of the chlorinated polyolefin and the non-chlorinated polyolefin.
摘要翻译：适合用于制造交联，热固性阻燃制品的氯化聚烯烃组合物，例如用于电缆或光纤电缆的夹套，用于电导体的绝缘涂层或层，以及用于保护的热收缩管，片或其它形状电缆连接器和接头。组合物是热固性和湿固化性的，并且包含氯化聚烯烃如氯化聚乙烯或氯磺化聚乙烯和含有水分可交联硅烷基团的非氯化聚烯烃。非氯化聚烯烃优选包含聚乙烯或其共聚物。将组合物暴露于水分导致在非氯化聚烯烃的分子之间形成分子间交联。组合物可以通过将非氯化聚烯烃与硅烷化非氯化聚烯烃共混或通过硅烷接枝氯化聚烯烃和非氯化聚烯烃的共混物来形成。

9. 发明授权

US08158703B2 Paintable primer system 有权
标题翻译：可涂漆底漆系统
公开(公告)号：US08158703B2
公开(公告)日：2012-04-17
申请号：US10591313
申请日：2005-03-02
申请人： Gerard Short , Boris Bobyreff , Peter Jackson
发明人： Gerard Short , Boris Bobyreff , Peter Jackson
IPC分类号： C08L67/00
CPC分类号： C09D5/002
摘要： A paintable primer composition comprising a dispersion, or chip is disclosed. the chip is produced from a dispersion comprising a thermoplastic polymer, a phthalate ester of a C1-C6 alkylated aromatic alcohol, a surfactant and other components selected from a metal carbonate, a white metal oxide pigment, an alkaline earth metal salt of a C9-C20 aliphatic fatty acid, a lower alkyl methacrylate polymer, a solvent and a rust inhibitor. The paintable primer composition is particularly suitable for painting surfaces, such as metals, composite materials and thermoplastic polyolefins including polyethylene, polypropylene, polystyrene, thermoplastic elastomer or ethylene-propylene rubbers. Painting of polyethylene surfaces may be assisted by precoating with an adhesion promoter comprising an aromatic hydrocarbon, a co-polymer of a C2-C6 alkene and a vinyl ester and a chlorinated polyolefin.
摘要翻译：公开了包含分散体或芯片的可涂漆底漆组合物。该芯片由包含热塑性聚合物，C1-C6烷基化芳族醇的邻苯二甲酸酯，表面活性剂和其它选自金属碳酸盐，白色金属氧化物颜料，C 9 -C 12烷基化芳族醇的碱土金属盐， C20脂肪族脂肪酸，甲基丙烯酸低级烷基酯聚合物，溶剂和防锈剂。可涂漆底漆组合物特别适用于涂漆表面，如金属，复合材料和热塑性聚烯烃，包括聚乙烯，聚丙烯，聚苯乙烯，热塑性弹性体或乙烯 - 丙烯橡胶。聚乙烯表面的涂布可以通过用包含芳族烃，C 2 -C 6烯烃和乙烯基酯的共聚物和氯化聚烯烃的粘合促进剂预涂覆来辅助。

10. 发明授权

US07923121B2 Photo-crosslinkable polyolefin compositions 有权
标题翻译：光交联聚烯烃组合物
公开(公告)号：US07923121B2
公开(公告)日：2011-04-12
申请号：US12780399
申请日：2010-05-14
申请人： Peter Jackson , Eileen Wan
发明人： Peter Jackson , Eileen Wan
IPC分类号： B32B27/00 , C08L23/00 , C08F10/00 , C08F220/10 , C08K3/22
CPC分类号： C08J3/243 , C08J2323/00 , C08K7/14 , C08L21/00 , C08L23/04 , C08L23/06 , C08L23/0884 , C08L23/10 , C08L23/16 , C08L51/06 , C08L2205/02 , C08L2312/06 , C08L2314/06 , C09D151/06 , Y10T428/31909 , Y10T428/31938 , C08L2666/06 , C08L2666/08 , C08L2666/24 , C08L2666/04 , C08L2666/02
摘要： A photo-crosslinkable polyolefin composition comprises a polyolefin, a source of functionality receptive to crosslinking by UV radiation, a cationic photoinitiator and optionally includes a free-radical photoinitiator, a crosslinking accelerator or sensitizer, and other additives such as compatibilizers, inorganic fillers, nanofillers, glass, polymeric and ceramic microspheres, glass fibers, flame retardants, antioxidants, stabilizers, processing aids, foaming agents and pigments. A method for manufacturing a UV-crosslinked polyolefin article comprises forming an article by extruding, molding or otherwise forming the UV-crosslinkable polyolefin composition and subjecting the article to UV radiation on-line with the extrusion, molding or other forming operation.
摘要翻译：光交联聚烯烃组合物包含聚烯烃，可接受紫外线辐射交联的功能源，阳离子光引发剂，任选地包括自由基光引发剂，交联促进剂或敏化剂，以及其它添加剂，例如增容剂，无机填料，纳米填料玻璃，聚合物和陶瓷微球，玻璃纤维，阻燃剂，抗氧化剂，稳定剂，加工助剂，发泡剂和颜料。 UV交联聚烯烃制品的制造方法包括通过挤出，成型或以其它方式形成UV可交联聚烯烃组合物并通过挤出，模塑或其它成型操作在线进行UV辐射来制造制品。

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