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1. 发明申请

US20080249113A1 Fungicidal Mixtures 审中-公开
标题翻译：杀菌混合物
公开(公告)号：US20080249113A1
公开(公告)日：2008-10-09
申请号：US11659192
申请日：2005-07-28
申请人： Carsten Blettner , Jochen Dietz , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Jochen Dietz , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： A01N43/90 , C07D487/04 , A01N25/26 , A01P3/00
CPC分类号： A01N43/90 , A01N43/653 , A01N47/14 , A01N43/50 , A01N57/12 , A01N47/04 , A01N37/34 , A01N43/40 , A01N37/50 , A01N37/46 , A01N43/84 , A01N37/38 , A01N43/28 , A01N47/38 , A01N43/54 , A01N43/32 , A01N59/20 , A01N2300/00
摘要： Fungicidal mixtures, comprising as active components 1) a 5-chloro-6-phenyl-7-heterocyclylaminotriazolopyrimidine of the formula I, in which D together with the nitrogen atom forms a pyrrolidine, piperidine or azepine ring, which rings are unsubstituted or substituted by one or two methyl groups or by an ethyl, propyl or butyl group; and L is methyl, fluorine or chlorine; and 2) at least one active compound II selected from the following groups: A) azoles; B) strobilurins; C) acylalanines; D) amine derivatives; E) anilinopyrimidines; F) dicarboximides; G) cinnamides and analogs; H) antibiotics; K) dithiocarbamates; L) heterocyclic compounds according to the description; M) sulfur and copper fungicides; N) nitrophenyl derivatives; O) phenylpyrroles; P) sulfenic acid derivatives; Q) other fungicides according to the description; or R) growth retardants; in a synergistically effective amount, novel triazolopyrimidines, methods for controlling harmful fungi using compounds or mixtures of a compound I with an active compound of groups A) to R) and the use of the compounds I with the active compounds of groups A) to R) for preparing such mixtures, and also compositions comprising these compounds or mixtures.
摘要翻译：包含作为活性组分的杀真菌混合物1）式I的5-氯-6-苯基-7-杂环基氨基三唑并嘧啶，其中D与氮原子一起形成吡咯烷，哌啶或氮杂环，该环是未取代的或被一个或两个甲基或乙基，丙基或丁基; L为甲基，氟或氯; 和2）至少一种选自以下组的活性化合物II：A）唑类; B）嗜球果伞素 C）酰基丙氨酸; D）胺衍生物; E）苯胺嘧啶嘧啶; F）二羧酰亚胺; G）肉桂酸酯类似物; H）抗生素; K）二硫代氨基甲酸盐; L）杂环化合物; M）硫和铜杀菌剂; N）硝基苯基衍生物; O）苯基吡咯; P）亚磺酸衍生物; Q）其他杀菌剂根据说明; 或R）生长阻滞剂; 协同有效量的新型三唑并嘧啶，使用化合物或化合物I与A）至R）的活性化合物的混合物来控制有害真菌的方法以及将化合物I与基团A）至R的活性化合物），以及包含这些化合物或混合物的组合物。

2. 发明申请

US20080032889A1 6-(2-Fluorophenyl)-Triazolopyrimidines, Method For The Production Thereof, Use Thereof For Controlling Harmful Fungi, And Agents Containing The Same 审中-公开
标题翻译： 6-（2-氟苯基） - 三唑并嘧啶，其生产方法，用于控制有害真菌及其含有药剂
公开(公告)号：US20080032889A1
公开(公告)日：2008-02-07
申请号：US11630558
申请日：2005-06-14
申请人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： A01N43/90 , A01C1/06 , C07D487/04
CPC分类号： A01N43/90 , C07D487/04
摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, halocycloalkyl, alkenyl, cycloalkyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen, alkyl or one of the groups mentioned under R1; R1 and/or R2 may carry one to four identical or different groups Ra: Ra is chlorine, bromine, iodine, cyano, nitro, hydroxyl, alkyl, alkylcarbonyl, cycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, alkylthio, alkylamino, dialkyl-amino, alkenyl, cycloalkenyl, alkenyloxy, haloalkenyloxy, alkynyl, halo-alkynyl, alkynyloxy, haloalkynyloxy, cycloalkoxy, cycloalkenyloxy, oxyalkylenoxy, naphthyl, a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, where these aliphatic, alicyclic or aromatic groups for their part may be substituted according to the description; and X is halogen; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要翻译：取代基如下定义的式I的取代三唑并嘧啶：R 1是烷基，卤代环烷基，烯基，环烷基，环烯基，卤代环烯基，炔基，卤代炔基或萘基，或五或六元环，包含一至四个由O，N和S组成的组的杂原子的2-元饱和的，部分不饱和的或芳族的杂环，R 2是氢，烷基或R 1上提到的基团之一， / SUP>; R 1和/或R 2可以携带一至四个相同或不同的基团R a是：R a是氯，溴，碘，氰基，硝基，羟基，烷基，烷基羰基，环烷基，烷氧基，卤代烷氧基，烷氧基羰基，烷硫基，烷基氨基，二烷基氨基，烯基，环烯基，烯氧基，卤代烯氧基，炔基，卤代炔基，炔氧基，卤代炔氧基，环烷氧基，环烯氧基，氧亚烷基氧基，萘基，五至十元饱和的部分不饱和或芳族杂环，其包含一至四个由O，N和S组成的组的杂原子，其中这些脂族，脂环族或芳族基团可以根据描述进行替代; X为卤素; 制备这些化合物的方法，包含它们的组合物及其用于控制植物病原性有害真菌的用途。

3. 发明申请

US20070208038A1 6-(2-Fluorophenyl)-Triazolopyrimidines, Method for Producing Them, Their use for Controlling Parasitic Fungi and Agents Containing the Same 审中-公开
公开(公告)号：US20070208038A1
公开(公告)日：2007-09-06
申请号：US10594738
申请日：2005-03-26
申请人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Michael Rack , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Michael Rack , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： A61K31/519 , C07D487/04 , A01N43/90
CPC分类号： A01N43/90 , C07D487/04
摘要： 6-(2-Fluorophenyl)-triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is C4-C8-alkyl, C4-C8-haloalkyl, substituted C3-C8-cycloalkyl, C3-C8-halocycloalkyl, C5-C8-alkenyl, C2-C8-haloalkenyl, C3-C6-cycloalkenyl, C3-C6-halocycloalkenyl, C2-C8-alkynyl, C2-C8-haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen, C1-C3-alkyl or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and contain one to three further heteroatoms from the group consisting of O, N and S as ring member, except for piperidin-1-yl optionally substituted by methyl groups; R1 and/or R2 may be substituted according to the description; L1 is chlorine or fluorine; L2 is hydrogen, is, if L1 is fluorine, also fluorine; X is alkyl; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

4. 发明申请

US20070142404A1 6-(2,6-Dichlorophenyl)-triazolopyrimidines, methods for the production thereof, use thereof for controlling pathogenic fungi, and agents containing the same 审中-公开
标题翻译： 6-（2,6-二氯苯基） - 三唑并嘧啶，其制备方法，用于控制致病真菌的用途及含有它们的试剂
公开(公告)号：US20070142404A1
公开(公告)日：2007-06-21
申请号：US10590924
申请日：2005-03-29
申请人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Michael Rack , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Michael Rack , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： A61K31/519 , C07D487/04
CPC分类号： A01N43/90 , C07D487/04
摘要： 6-(2,6-Dichlorophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring member and which is substituted according to the description; X is alkyl, cyano, alkoxy, haloalkoxy, alkenyloxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要翻译：其中取代基如下定义的式I的6-（2,6-二氯苯基）三唑并嘧啶：R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五元或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子 R 1和R 2连同它们所连接的氮原子一起也可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员，并且根据描述被取代; X是烷基，氰基，烷氧基，卤代烷氧基，烯氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制植物病原性有害真菌的用途。

5. 发明申请

US20080248952A1 Substituted 6-Phenyl-7-Aminotriazolopyrimidines, Method for the Production Thereof, Their Use for Controlling Pathogenic Fungi, and Agents Containing These Compounds 审中-公开
标题翻译：取代的6-苯基-7-氨基三唑并嘧啶，其制备方法，其用于控制致病真菌和含有这些化合物的试剂
公开(公告)号：US20080248952A1
公开(公告)日：2008-10-09
申请号：US11631004
申请日：2005-07-06
申请人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： C07D487/04 , A01N43/90 , A01N25/00
CPC分类号： A01N43/90 , C07D487/04
摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or a group R1, R1 and R2 together with the nitrogen atom, to which they are attached, may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and which may comprise one to three further heteroatoms from the groups consisting of O, N and S as ring member and/or may be substituted according to the description; L is fluorine, chlorine or methyl; X is cyano, C1-C4-alkyl, C1-C4-alkoxy or C1-C2-haloalkoxy, where X is not methyl if R1 and R2 together are n-pentylene or 3-methyl-n-pentylene and L is fluorine, or R1 and R2 together are 3-methyl-n-pentylene and L is chlorine; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要翻译：取代基如下定义：式I的取代三唑并嘧啶：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，包含一至四个由O，N和S组成的组的杂原子的五或六元饱和的部分不饱和或芳族杂环，R 2是氢或基团R 1， R 1，R 2和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基或杂芳基，它们是通过N连接并且其可以包含一个至三个由O，N和S组成的基团的另外的杂原子作为环成员和/或可以根据描述被取代; L是氟，氯或甲基; X是氰基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基或C 1 -C 4 - 如果R 1和R 2一起都是正 - 亚戊基，其中X不是甲基，其中X不是甲基或3-甲基 - 正戊烯，L是氟，R 1和R 2一起是3-甲基 - 正戊烯，L是氯; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制植物病原性有害真菌的用途。

6. 发明申请

US20080039319A1 Fungicidal Mixtures and Novel Triazolopyrimidines 审中-公开
标题翻译：杀菌混合物和新型三唑并嘧啶
公开(公告)号：US20080039319A1
公开(公告)日：2008-02-14
申请号：US11596464
申请日：2005-05-11
申请人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Barbara Nave , Maria Scherer , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： A01N43/90 , A01N25/34 , A01N59/20
CPC分类号： A01N43/90 , A01N59/06 , A01N59/02 , A01N57/12 , A01N47/38 , A01N47/34 , A01N47/24 , A01N47/04 , A01N43/50 , A01N43/76 , A01N43/653 , A01N43/36 , A01N43/40 , A01N43/32 , A01N37/48 , A01N37/46 , A01N37/38 , A01N37/34 , A01N2300/00
摘要： The invention relates to fungicidal mixtures containing in the form of active components 1) 5-methyl-7-amino-triazolopyrimidine of formula (I), wherein R1 is alkyl, halogenalkyl, alkenyl or cyclopentyl, R2 is hydrogen or alkyl, R1 and R2 together with the nitrogen atom to which they are bound may form a piperidinyl cycle substitutable by a methyl group, L1 is fluorine or chlorine, L2, L3 are independently from each other hydrogen, fluorine or chlorine and 2) at least one type of active substance selected from groups A) azoles, B) strobilurins, C) acyl alanines, D) amine derivatives, E) anilinopyrimidines; F) dicarboximides; G) cinnamic acid amides and analogues thereof, H) antibiotics, K) dithiocarbamates, L) heterocyclic compounds, M) sulphur and copper fungicides, N) nitrophenyl derivatives, O) phenylpyrroles, P) sulfenic acid derivatives, Q) other fungicides and R) growth retardants according to the descriptions, wherein said mixtures contain the compounds in a synergically efficient amount. Novel triazolopyrimidines, methods for controlling pathogenic fungi using the mixtures of the compound (1) with active substances of the groups A) and R), the use the compounds (I) with the active substances of the groups A) and R) for producing said mixtures and agents containing said mixtures are also disclosed.
摘要翻译：本发明涉及含有活性组分形式的杀真菌混合物1）式（I）的5-甲基-7-氨基 - 三唑并嘧啶，其中R 1是烷基，卤代烷基，烯基或环戊基，R R 2是氢或烷基，R 1和R 2与它们所连接的氮原子一起可以形成可被甲基，L 1是氟或氯，L 2，L 3，3彼此独立地为氢，氟或氯，以及2）在至少一种活性物质选自A）唑类，B）嗜球果伞素，C）酰基丙氨酸，D）胺衍生物，E）苯胺基嘧啶; F）二羧酰亚胺; G）肉桂酸酰胺及其类似物，H）抗生素，K）二硫代氨基甲酸盐，L）杂环化合物，M）硫和铜杀真菌剂，N）硝基苯基衍生物，O）苯基吡咯，P）亚磺酸衍生物，Q）其他杀真菌剂和R ）生长阻滞剂，其中所述混合物包含协同有效量的化合物。新型三唑并嘧啶，使用化合物（1）与A）和R）基团的活性物质的混合物来控制致病真菌的方法，将化合物（I）与A）和R）基团的活性物质一起用于生产还公开了含有所述混合物的所述混合物和试剂。

7. 发明申请

US20070249633A1 1,2,4-Triazolo[1,5a] Pyrimidines and Use Thereof for Controlling Plant-Pathogenic Fungi 审中-公开
公开(公告)号：US20070249633A1
公开(公告)日：2007-10-25
申请号：US11597379
申请日：2005-06-08
申请人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Michael Rack , Barbara Nave , Maria Scherer , Siegfried Strahmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Michael Rack , Barbara Nave , Maria Scherer , Siegfried Strahmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： A01N43/90 , C07D487/04
CPC分类号： A01N43/90 , C07D487/04
摘要： The invention relates to triazolopyrimidines of the formula I in which the index n and the substituents R, R1, R2 and X are as defined below: X is nitro, a group —C(S)NR3R4, a group —C(═N—OR5)(NR6R7) or a group —C(═N—NR8R9)(NR10R11), R is halogen, cyano, hydroxyl, cyanato, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one, two, three or four heteroatoms from the group consisting of O, N or S; R1 is alkyl in which one carbon atom may be replaced by a silicon atom, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via a carbon atom and which contains one, two, three or four heteroatoms, independently of one another selected from the group consisting of O, N and S, as ring members; where R1 may be substituted as defined in the description; R2 is alkyl, alkenyl or alkynyl which may be substituted as defined in the description; R3, R4, R5, R6, R7, R8, R9, R10 and R11 are, independently of one another, selected from the group consisting of hydrogen, alkyl, cycloalkyl, alkenyl or alkynyl, where the 4 lastmentioned radicals may be substituted as defined in the description; or R3 and R4, R6 and R7, R8 and R9 and/or R10 and R11 together with the nitrogen atom to which they are attached form a four-, five- or six-membered saturated or partially unsaturated ring which may be substituted as defined in the description; and n is 0 or an integer 1, 2, 3 or 4; and the agriculturally acceptable salts thereof, to crop protection compositions comprising at least one compound of the formula I and/or an agriculturally acceptable salt thereof and at least one liquid or solid carrier and to a method for controlling phytopathogenic harmful fungi.

8. 发明申请

US20070238744A1 Use of 6-(2-Tolyl)-Triazolopyrimidines as Fungicides, Novel 6-(2-Tolyl)-Triazolopyrimidines, Method for the Production Thereof, Used There of for Controlling Harmful Fungi, and Agents Containing the Same 审中-公开
标题翻译： 6-（2-甲苯基） - 三唑并嘧啶类作为杀真菌剂，新型6-（2-甲苯基） - 三唑并嘧啶类，其生产方法，用于控制有害真菌及含有其的药剂
公开(公告)号：US20070238744A1
公开(公告)日：2007-10-11
申请号：US11629126
申请日：2005-06-14
申请人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Barbara Nave , Maria Scherer , Sigfried Strathmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bernd Muller , Matthias Niedenbruck , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Barbara Nave , Maria Scherer , Sigfried Strathmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： A61K31/519 , C07D487/02
CPC分类号： A01N43/90 , C07D487/04
摘要： The use of substituted triazolopyrimidines of the formula I in which R1 is alkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or a group R1, where R1 and/or R2 may be substituted according to the description, and X is halogen; as fungicides, novel 6-(2-tolyl)triazolopyrimidines, processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要翻译：使用式I的取代三唑并嘧啶，其中R 1是烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或萘基，或五或六元饱和，包含一至四个由O，N和S组成的组的杂原子的部分不饱和或芳族杂环，R 2是氢或基团R 1，其中R 0 > 1和/或R 2可以根据描述被取代，X是卤素; 作为杀真菌剂，新颖的6-（2-甲苯基）三唑并嘧啶，制备这些化合物的方法，包含它们的组合物及其用于控制植物病原性有害真菌的用途。

9. 发明申请

US20070249634A1 Triazolopyrimidine Compounds and Use Thereof for Controlling Harmful Fungi 审中-公开
公开(公告)号：US20070249634A1
公开(公告)日：2007-10-25
申请号：US11597409
申请日：2005-06-08
申请人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bern Muller , Matthias Niedenbruck , Joachim Rheinheimer , Petere Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Liliana Rapado , Michael Rack , Barbara Nave , Maria Schere , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
发明人： Carsten Blettner , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Udo Hunger , Bern Muller , Matthias Niedenbruck , Joachim Rheinheimer , Petere Schafer , Frank Schieweck , Anja Schwogler , Oliver Wagner , Liliana Rapado , Michael Rack , Barbara Nave , Maria Schere , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
IPC分类号： A01N43/90 , A01P3/00
CPC分类号： A01N43/90
摘要： The invention relates to the use of triazolopyrimidines of the formula I In which: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl, C3-C6-cycloalkynyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one, two, three or four heteroatoms from the group consisting of O, N and S, where R1, R2 may be substituted as defined in the description or R1 and R2 together with the nitrogen atom to which they are attached may form five- to eight-membered heterocyclyl or heteroaryl which is attached via nitrogen and may contain one, two or three further heteroatoms from the group consisting of O, N and S as ring members and/or may be substituted as defined in the description; L independently of one another are halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyloxy, cyano, C(═O)A1, S(═O)mA2, NRcRd or NRc—(C═O)—Rd, where A1, A2, Rc, Rd and m are as defined in the description; L1 is halogen, alkyl or haloalkyl; L2 is nitro, a group —C(S)NR3R4, a group —C(═N—OR5)(NR6R7) or a group —C(═N—NR8R9)(NR10OR11); X is halogen, cyano, alkyl, alkoxy, haloalkyl or haloalkoxy; R3, R4, R5, R6, R7, R8, R9, R10 and R11 are independently of one another selected from the group consisting of hydrogen, alkyl, cycloalkyl, alkenyl and alkynyl, where the 4 last-mentioned radicals may be substituted as defined in the description; or R3 and R4, or R6 and R7, or R8 and R9 or R10 and R11 together with the nitrogen atom to which they are attached form a four, five, or six-membered saturated or partially unsaturated ring which may be substituted as defined in the description; n is 0, 1, 2 or 3; and the agriculturally acceptable salts thereof, novel triazolopyrimidines, crop protection compositions comprising at least one compound of the formula I and at least one solid or liquid carrier, and a method for controlling phytopathogenic harmful fungi.

10. 发明申请

US20080146593A1 Substituted 5-Phenyl Pyrimidines I In Therapy 审中-公开
公开(公告)号：US20080146593A1
公开(公告)日：2008-06-19
申请号：US11815042
申请日：2006-01-30
申请人： Joachim Rheinheimer , Thomas Grote , Bernd Muller , Barbara Nave , Frank Schieweck , Anja Schwogler , Thorsten Jabs , Carsten Blettner
发明人： Joachim Rheinheimer , Thomas Grote , Bernd Muller , Barbara Nave , Frank Schieweck , Anja Schwogler , Thorsten Jabs , Carsten Blettner
IPC分类号： A61K31/505 , A61K31/513 , A61P35/00
CPC分类号： C07D239/48 , C07D239/42 , C07D401/04 , C07D403/04 , C07D417/04
摘要： The present invention relates to substituted 5-phenyl pyrimidines I, which carry a radical X in the 4-position of the pyrimidine ring, a radical Y in the 6-position of the pyrimidine ring, the radical X denoting a group of the formula NR1R2, OR1a or SR1a, in which R1, R2, independently of each other, denote hydrogen, C1-C10-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C1-C10-haloalkyl, C3-C8-cycloalkyl, C3-C8-halocycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which radicals may be unsubstituted or may carry 1, 2, 3 or 4 radicals Ra1; or the radical NR1R2 may also form a 5- or 6-membered optionally substituted heterocyclic ring, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which are non-adjacent to the nitrogen of NR1R2, in which two adjacent C atoms or one N atom and one adjacent C atom can be linked by a C1-C4-alkylene chain and wherein the heterocyclic ring may be unsubstituted or may carry 1, 2, 3 or 4 radicals Ra1 as defined in claim 1, R1a has one of the meanings given for R1 except for hydrogen; the radical Y being selected from the group consisting of halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C3-C6-cycloalkyl, C1-C4-alkoxy, C3-C4-alkenyloxy, C3-C4-alkynyloxy, C1-C6-alkylthio, di-(C1-C6-alkyl)amino or C1-C6-alkylamino, where the alkyl, alkenyl and alkynyl radicals of Y may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl; and wherein the pyrimidine radical may also carry a radical different from hydrogen in the 2-position and wherein the phenyl ring in the 5-position of the pyrimidine ring may be unsubstituted or carry 1, 2, 3, 4 or 5 radicals L which are different from hydrogen, and the pharmaceutically acceptable salts substituted 5-phenyl pyrimidines for use in therapy, in particular in therapy or treatment of cancerous diseases.

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