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1. 发明申请

US20110029125A1 APPARATUS FOR CONTROLLING A MACHINE TOOL 审中-公开
标题翻译：用于控制机床的装置
公开(公告)号：US20110029125A1
公开(公告)日：2011-02-03
申请号：US12845647
申请日：2010-07-28
申请人： Achim Feinauer , Uwe Bräuning , Matthias Schwarz
发明人： Achim Feinauer , Uwe Bräuning , Matthias Schwarz
IPC分类号： G05B19/402 , G09G5/00
CPC分类号： G05B19/409 , G05B2219/23018 , G05B2219/23029 , G05B2219/32128 , G05B2219/35508
摘要： An apparatus on a machine tool for machining workpieces, preferably for machining workpieces by removing material, is provided to control functions of the machine tool and to program and/or test the machining of workpieces and/or to test the machine tool itself. The apparatus is provided with at least one display unit and at least one input unit, whereby masks for displaying and/or for inputting, via the input unit, machine and/or control parameters are displayable on the display unit. A start matrix having a grid of fields, which are stored in a geometrically addressable manner and are preferably arranged in rows and columns, can be displayed on the display unit, the input unit which is separate from the display unit being able to be used to select each field via its geometrical position in the grid at which it is displayed on the display unit, and the assigned function being able to be immediately triggered or a mask being able to be immediately displayed on the display unit by activating a field.
摘要翻译：用于加工工件的机床上的装置，优选用于通过移除材料来加工工件，用于控制机床的功能，以及编程和/或测试工件的加工和/或测试机床本身。该装置设置有至少一个显示单元和至少一个输入单元，由此可以在显示单元上显示用于显示和/或经由输入单元输入机器和/或控制参数的掩模。可以在显示单元上显示具有以几何可寻址方式存储并优选地以行和列布置的具有场格的起始矩阵，与显示单元分离的输入单元能够被用于通过其在显示单元上显示的网格中的几何位置来选择每个场，并且可以立即触发所分配的功能，或者通过激活场立即在显示单元上显示掩模。

2. 发明授权

US08202856B2 Triazole oxadiazoles derivatives 有权
标题翻译：三唑恶二唑衍生物
公开(公告)号：US08202856B2
公开(公告)日：2012-06-19
申请号：US12809816
申请日：2008-12-17
申请人： Anna Quattropani , Christophe Cleva , Eric Sebille , Matthias Schwarz , Delphine Marin , Agnes Bombrun , Wesley Blackaby , Charles Baker-Glenn , Chris Knight , Craig Rouse
发明人： Anna Quattropani , Christophe Cleva , Eric Sebille , Matthias Schwarz , Delphine Marin , Agnes Bombrun , Wesley Blackaby , Charles Baker-Glenn , Chris Knight , Craig Rouse
IPC分类号： A61K31/397 , A61K31/4545 , A61K31/444 , A61K31/5377 , A61K31/4245 , A61K31/4439 , A61K31/4725 , A61K31/497 , C07D413/04 , C07D413/14 , C07D401/14 , A61P19/02 , A61P3/10 , A61P9/10 , A61P29/00 , A61P1/04 , A61P17/06 , A61P11/06
CPC分类号： C07D413/04 , C07D413/14
摘要： The invention relates to compounds of formula I: wherein R1, R2,Ra, Rb, X have the meanings given in claim 16. The compounds are useful e.g. in the treatment of autoimmune disorders, such as multiple sclerosis.
摘要翻译：本发明涉及式I化合物：其中R1，R2，Ra，Rb，X具有权利要求1中给出的含义。治疗自身免疫性疾病，如多发性硬化症。

3. 发明申请

US20120028959A1 DIHYDROOROTATE DEHYDROGENASE INHIBITORS 有权
标题翻译： DIHYDROOROTATE DEHYDROGENASE抑制剂
公开(公告)号：US20120028959A1
公开(公告)日：2012-02-02
申请号：US13262640
申请日：2010-03-26
申请人： Siva Sanjeeva Rao Thunuguntla , Hosahalli Subramanya , Satish Reddy Kunnam , Sekhar Reddy Sanivaru Vijay , Chakrapani Bingi , Raviraj Kusanur , Matthias Schwarz , Michael Arlt
发明人： Siva Sanjeeva Rao Thunuguntla , Hosahalli Subramanya , Satish Reddy Kunnam , Sekhar Reddy Sanivaru Vijay , Chakrapani Bingi , Raviraj Kusanur , Matthias Schwarz , Michael Arlt
IPC分类号： A61K31/55 , A61K31/4184 , C07D263/57 , A61K31/423 , C07D409/10 , C07D403/10 , C07D417/10 , A61K31/428 , C07D401/04 , A61K31/4439 , C07D413/10 , A61K31/5377 , A61P25/00 , A61P29/00 , A61P35/00 , A61P1/00 , C07D235/18
CPC分类号： C07D209/08 , C07D235/18 , C07D401/04 , C07D401/10 , C07D403/04 , C07D409/10 , C07D413/10 , C07D417/10 , C07D471/04
摘要： The invention relates to compounds of formula (I) wherein R1, R2, X1, X2, Y, Ra, Rb, Q have the meanings given in claim 1. The compounds are useful e.g. in the treatment of autoimmune disorders, such as multiple sclerosis and also in the treatment of cancer disorders.
摘要翻译：本发明涉及式（I）化合物，其中R 1，R 2，X 1，X 2，Y，R a，R b，Q具有权利要求1中给出的含义。在治疗自身免疫性疾病如多发性硬化以及治疗癌症中。

4. 发明申请

US20100305137A1 PIPERAZINE DERIVATIVES AND METHODS OF USE 审中-公开
标题翻译：哌嗪衍生物及其使用方法
公开(公告)号：US20100305137A1
公开(公告)日：2010-12-02
申请号：US12792665
申请日：2010-06-02
申请人： Sharad Magar , Andreas Goutopulos , Yihua Liao , Matthias Schwarz , Russel J. Thomas
发明人： Sharad Magar , Andreas Goutopulos , Yihua Liao , Matthias Schwarz , Russel J. Thomas
IPC分类号： A61K31/496 , A61P15/00 , A61P15/08
CPC分类号： C07D409/14 , A61K31/496 , C07D401/14 , C07D403/12 , C07D403/14 , C07D471/04 , C07D487/04
摘要： The invention provides 2-carboxamide piperazine compounds, and methods of treatment and pharmaceutical compositions that utilize or comprise one or more such compounds. Compounds of the invention are useful for the treatment of mammalian infertility.
摘要翻译：本发明提供2-甲酰胺哌嗪化合物，以及使用或包含一种或多种这些化合物的治疗方法和药物组合物。本发明的化合物可用于治疗哺乳动物不育症。

5. 发明申请

US20090215749A9 THIAZOLIDINE CARBOXAMIDE DERIVATIVES AS MODULATORS OF THE PROSTAGLANDIN F RECEPTOR 有权
标题翻译：作为PROSTAGLANDIN F受体的调节剂的噻唑烷羧酰胺衍生物
公开(公告)号：US20090215749A9
公开(公告)日：2009-08-27
申请号：US12140682
申请日：2008-06-17
申请人： Patrick Naxos PAGE , Catherine Jorand-Lebrun , Anna Quattropani , Vincent Pomel , Matthias Schwarz , Estelle Hamelin , Russell J. Thomas
发明人： Patrick Naxos PAGE , Catherine Jorand-Lebrun , Anna Quattropani , Vincent Pomel , Matthias Schwarz , Estelle Hamelin , Russell J. Thomas
IPC分类号： A61K31/55 , C07D277/06 , A61K31/426 , A61P15/06 , A61P15/04 , C07D417/12
CPC分类号： C07D417/12 , A61K31/426 , A61K31/427 , C07D277/06 , C07D417/14 , Y02P20/582
摘要： The present invention is related to thiazolidine carboxamide derivatives of formula (II) for the treatment and/or prophylaxis of preterm labor, premature birth, dysmenorrhea and for stopping labor prior to cesarean delivery.
摘要翻译：本发明涉及式（II）的噻唑烷羧酰胺衍生物，其用于治疗和/或预防早产，早产，痛经和用于在剖宫产分娩前停止劳动。

6. 发明授权

US07557136B2 Pyrrolidine derivatives as oxytocin antagonists 失效
标题翻译：吡咯烷衍生物作为催产素拮抗剂
公开(公告)号：US07557136B2
公开(公告)日：2009-07-07
申请号：US10547032
申请日：2004-02-16
申请人： Matthias Schwarz , Catherine Jorand-Lebrun , Delphine Valognes
发明人： Matthias Schwarz , Catherine Jorand-Lebrun , Delphine Valognes
IPC分类号： A61K31/40 , A61K31/4245 , A61K31/4184 , C07D207/14 , C07D271/06 , C07D403/06
CPC分类号： C07D413/06 , C07D207/22
摘要： The present invention relates to novel pyrrolidine derivatives of Formula (I), its geometrical isomers, its optically active forms as enantiomers, diastercomers, mixtures of these and its racemate forms, as well as salts thereof, wherein: R1is selected from the group comprising or consisting of H and C1-C6-alkyl; R2 is selected from the group comprising or consisting of hydrogen, C1-C6-alkyl, C1-C6 alkyl aryl, heteroaryl, C1-C6 alkyl heteroaryl, C2-C6-alkenyl, C2-C6-alkenyl aryl, C2-C6 alkenyl heteroaryl, C2-C6-alkynyl, C2-C6-alkynyl aryl, C2C6-alkynyl heteroaryl, C3-C8 cycloalkyl, heterocycloalkyl, CI-C6-alkyl cycloallcyl, CI-C6-alkyl heterocycloalkyl, CIC6 alkyl carboxy, acyl, C1-C6-alkyl acyl, C1-C6-alkyl acyloxy, C1-C6-alkyl alkoxy, alkoxycarbonyl, C1-C6-alkyl alkoxycarbonyl, aminocarbonyl, C1-C6-alkyl aminocarbonyl, C1-C6-alkyl acylarnino, C1-C6-alkyl ureido, amino, C1-C6-alkyl amino, sulfonyloxy, C1-C6 alkyl sulfonyloxy, sulfonyl, C1-C6-alkyl sulfonyl, sulfinyl, C1-C6-alkyl sulfinyl, C1-C6alkyl sulfanyl, C1-C6-alkyl sulfonylamino.
摘要翻译：本发明涉及式（I）的新型吡咯烷衍生物，其几何异构体，其作为对映异构体的光学活性形式，diastercomers，它们的混合物及其外消旋体形式及其盐，其中：R 1选自包括或由H和C 1 -C 6 - 烷基组成; R 2选自氢，C 1 -C 6 - 烷基，C 1 -C 6烷基芳基，杂芳基，C 1 -C 6烷基杂芳基，C 2 -C 6 - 烯基，C 2 -C 6烯基芳基，C 2 -C 6烯基杂芳基，C 2 -C 6 - 炔基芳基，C 2 -C 6炔基杂芳基，C 3 -C 8环烷基，杂环烷基，C 1 -C 6烷基环烷基，C 1 -C 6烷基杂环烷基，CIC 6烷基羧基，酰基，C 1 -C 6 - 烷基酰基，C 1 -C 6烷基酰氧基，C 1 -C 6烷基烷氧基，烷氧基羰基，C 1 -C 6烷基烷氧基羰基，氨基羰基，C 1 -C 6烷基氨基羰基，C 1 -C 6烷基酰基氨基，C 1 -C 6烷基脲基，氨基，C 1 -C 6烷基氨基，磺酰氧基，C 1 -C 6烷基磺酰氧基，磺酰基，C 1 -C 6烷基磺酰基，亚磺酰基，C 1 -C 6烷基亚磺酰基，C 1 -C 6烷基硫烷基，C 1 -C 6烷基磺酰基氨基。

7. 发明授权

US07468385B2 Triazoles as oxytocin antagonists 失效
标题翻译：三唑作为催产素拮抗剂
公开(公告)号：US07468385B2
公开(公告)日：2008-12-23
申请号：US10498356
申请日：2002-12-19
申请人： Anna Quattropani , Matthias Schwarz , Russell J. Thomas , Thomas Coulter
发明人： Anna Quattropani , Matthias Schwarz , Russell J. Thomas , Thomas Coulter
IPC分类号： A61K31/41 , C07D249/08
CPC分类号： C07D403/12 , C07D249/10 , C07D249/12 , C07D249/14 , C07D405/06 , C07D405/12
摘要： The present invention relates to triazole derivatives of formula (I) notably for use as pharmaceutically active compounds, as well as pharmaceutical formulations containing such triazole derivatives. Said triazoles are useful in the treatment and/or prevention of preterm labor, premature birth, dysmenorrhea, inappropriate secretion of vasopressin, congestive heart failure, arterial hypertension, liver cirrhosis, nephrotic syndrome and ocular hypertension. In particular, the present invention is related to triazole derivatives displaying a substantial modulatory, in particular antagonistic activity, of the oxytocin and/or vasopressin receptor. More preferably, said compounds are useful in the treatment and/or prevention of disease states mediated by oxytocin and/or vasopressin. The present invention is furthermore related to novel triazole derivatives as well as to methods of their preparation.
摘要翻译：本发明涉及特别用作药物活性化合物的式（I）的三唑衍生物以及含有这种三唑衍生物的药物制剂。所述三唑可用于治疗和/或预防早产，早产，痛经，不适当的血管加压素分泌，充血性心力衰竭，动脉高血压，肝硬化，肾病综合征和高眼压症。特别地，本发明涉及显示催产素和/或加压素受体的显着调节，特别是拮抗活性的三唑衍生物。更优选地，所述化合物可用于治疗和/或预防催产素和/或加压素介导的疾病状态。本发明还涉及新的三唑衍生物及其制备方法。

8. 发明申请

US20080287474A1 Antiproliferative Pyrimidyl, Fused Pyrimidyl and Pyrimidyl Hydrazones 失效
标题翻译：抗增生嘧啶，熔融的嘧啶基和嘧啶基腙
公开(公告)号：US20080287474A1
公开(公告)日：2008-11-20
申请号：US12096110
申请日：2006-12-08
申请人： Brian Healey , Zhong Zhao , Amanda Sutton , Matthias Schwarz
发明人： Brian Healey , Zhong Zhao , Amanda Sutton , Matthias Schwarz
IPC分类号： A61K31/517 , C07D239/94 , A61K31/506 , C07D401/04 , C12N5/06 , A61P35/00
CPC分类号： C07D239/94 , C07D239/42 , C07D239/47 , C07D239/48 , C07D401/04 , C07D413/04
摘要： The present invention is related to a novel series of pyrimidyl or fused pyrimidyl hydrazones. Compounds of Formula (I) wherein A is selected from the group consisting of Formulas (A1), (A2), (A3), (A4), (A5) are useful for the treatment and/or prevention of a proliferative disease.
摘要翻译：本发明涉及新的一系列嘧啶基或稠合的嘧啶基腙。其中A选自式（A1），（A2），（A3），（A4），（A5）的式（I）化合物可用于治疗和/或预防增殖性疾病。

9. 发明申请

US20080167318A1 Pharmaceutically active pyrrolidine derivatives 审中-公开
标题翻译：药用活性吡咯烷衍生物
公开(公告)号：US20080167318A1
公开(公告)日：2008-07-10
申请号：US11783341
申请日：2007-04-09
申请人： Serge Halazy , Anna Quattropani , Alexander Scheer , Matthias Schwarz , Russell J. Thomas , Anthony Baxter
发明人： Serge Halazy , Anna Quattropani , Alexander Scheer , Matthias Schwarz , Russell J. Thomas , Anthony Baxter
IPC分类号： A61K31/497 , A61K31/40 , A61K31/403 , A61P15/06 , C07D209/56 , C07D455/02 , C07D403/02 , C07D207/02 , A61P15/02 , A61K31/47
CPC分类号： C07D401/12 , C07D207/22 , C07D403/04 , C07D403/06 , C07D403/14 , C07D405/06 , C07D405/12 , C07D405/14 , C07D409/12 , C07D417/12
摘要： The present invention is related to pyrrolidine derivatives of formula I. Said compounds are preferably for use as pharmaceutically active compounds. Specifically, pyrrolidine derivatives of formula I are useful in the treatment and/or prevention of premature labor, premature birth and dysmenorrhea. In particular, the present invention is related to pyrrolidine derivatives displaying a substantial modulatory, notably an antagonist activity of the oxytocin receptor. More preferably, said compounds are useful in the treatment and/or prevention of disease states mediated by oxytocin, including premature labor, premature birth and dysmenorrhea. The present invention is furthermore related to novel pyrrolidine derivatives as well as to methods of their preparation. wherein X is selected from the group consisting of CR6R7, NOR6, NNR6R7; A is selected from the group consisting of —(C═O)—, —(C═O)—O—, —C(═NH)—, —(C═O)—NH—, —(C═S)—NH, —SO2—, —SO2NH—, —CH2—, B is either a group —C═O)—NR8R9 or represents a heterocyclic residue having the formula wherein Q is NR10, O or S; n is an integer selected of 0, 1 or 2; Y, Z and E form together with the 2 carbons to which they are attached a 5-6 membered aryl or heteroaryl ring.
摘要翻译：本发明涉及式I的吡咯烷衍生物。所述化合物优选用作药物活性化合物。具体地，式I的吡咯烷衍生物可用于治疗和/或预防早产，早产和痛经。特别地，本发明涉及显示出显着调节，特别是催产素受体拮抗剂活性的吡咯烷衍生物。更优选地，所述化合物可用于治疗和/或预防催产素介导的疾病状态，包括早产，早产和痛经。本发明还涉及新型吡咯烷衍生物及其制备方法。其中X选自CR 6，S 6，S 6，N 6，R 6，O 6， > 7 ; A选自 - （CO） - ， - （CO）-O-，-C（-NH） - ， - （CO）-NH-， - （CS）-NH， 2 - ， - SO 2 NH - ， - CH 2 - ， - B是基团-CO）-NR 8 - 或者表示具有下式的杂环残基：其中Q是NR 10，O或S; n是选自0,1或2的整数; Y，Z和E与它们所连接的2个碳原子一起形成5-6元芳基或杂芳基环。

10. 发明申请

US20070283829A1 METHOD AND APPARATUS FOR COLLECTING OPERATING DATA FROM MACHINES USED IN THE PRINTING INDUSTRY 审中-公开
标题翻译：用于从印刷行业使用的机器中收集操作数据的方法和装置
公开(公告)号：US20070283829A1
公开(公告)日：2007-12-13
申请号：US11760620
申请日：2007-06-08
申请人： Matthias Schwarz , Guenter Reimers , Joachim Ruf , Gregor Enke , Claus Stenger
发明人： Matthias Schwarz , Guenter Reimers , Joachim Ruf , Gregor Enke , Claus Stenger
IPC分类号： B41F33/00
CPC分类号： B41F33/0009 , B41F33/16
摘要： A method and apparatus for collecting operating data from machines used in the printing industry, in particular from printing presses, is disclosed. At least one machine linked to a control device, or an operating data collection device, automatically transmits data during operation of the machine to the control device, or the operating data collection device, and a time frame for operating data collection is generated automatically from the machine data such that machine activity time intervals about the operating time of the machine on the one hand and machine downtime intervals on the other hand are derived from the machine data. Reasons for downtime are automatically assigned to the established machine downtime intervals and/or can be assigned semi-automatically.
摘要翻译：公开了一种用于从印刷工业中使用的机器收集操作数据的方法和装置，特别是用于印刷机。链接到控制装置或操作数据收集装置的至少一个机器在机器的操作期间自动地将数据传送到控制装置或操作数据收集装置，并且用于操作数据收集的时间框架从机器数据，一方面机器的运行时间间隔一方面与另一方面机器停机时间间隔是从机床数据得出的。停机时间的原因将自动分配给已建立的机器停机时间间隔，和/或可以半自动分配。

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