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1. 发明申请

US20050234110A1 Novel 2-pyridylethylbenzamide derivative 有权
标题翻译：新型2-吡啶基乙基苯甲酰胺衍生物
公开(公告)号：US20050234110A1
公开(公告)日：2005-10-20
申请号：US10524345
申请日：2003-08-08
申请人： Darren Mansfield , Tracey Cooke , Peter Thomas , Pierre-Yves Coqueron , Jean-Pierre Vors , Geoffrey Briggs , Helene Lachaise , Heiko Rieck , Philippe Desbordes
发明人： Darren Mansfield , Tracey Cooke , Peter Thomas , Pierre-Yves Coqueron , Jean-Pierre Vors , Geoffrey Briggs , Helene Lachaise , Heiko Rieck , Philippe Desbordes
IPC分类号： A01N25/30 , A01N43/40 , C07D213/40 , C07D213/61 , C07D213/89 , A61K31/44 , C07D213/56
CPC分类号： C07D213/89 , A01N43/40 , C07D213/40 , C07D213/61
摘要： Compound of general formula (I) in which p is an integer equal to 1, 2, 3 or 4; q is an integer equal to 1, 2, 3, 4 or 5; each substituent X is chosen, independently of the others, as being halogen, alkyl or haloalkyl, at least one of the substituents being a haloalkyl; each substituent Y is chosen, independently of the others, as being halogen, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, amino, phenoxy, alkylthio, dialkylamino, acyl, cyano, ester, hydroxy, aminoalkyl, benzyl, haloalkoxy, halosulphonyl, halothioalkyl, alkoxyalkenyl, alkylsulphonamide, nitro, alkylsulphonyl, phenylsulphonyl or benzylsulphonyl; as to the N-oxides of 2-pyridine thereof; with the exception of N-{2-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-ethyl}-2,6-dichlorobenzamide. Method for preparing the compound of general formula (I). Fungicidal composition comprising the compound of general formula (I). Method for treating phytopathogenic diseases.
摘要翻译：通式（I）的化合物，其中p是等于1,2,3或4的整数; q是等于1,2,3,4或5的整数; 每个取代基X独立地选自卤素，烷基或卤代烷基，至少一个取代基是卤代烷基; 氰基，酯，羟基，氨基烷基，苄基，卤代烷氧基，卤代磺酰基，卤代烷基，卤代烷基，卤代烷基，烷氧基烯基，烷基磺酰胺，硝基，烷基磺酰基，苯基磺酰基或苄基磺酰基; 关于其2-吡啶的N-氧化物; 除了N- {2- [3-氯-5-（三氟甲基）-2-吡啶基] - 乙基} -2,6-二氯苯甲酰胺外。制备通式（I）化合物的方法。包含通式（I）的化合物的杀真菌组合物。治疗植物病原性疾病的方法

2. 发明授权

US06630495B1 Fungicides 有权
标题翻译：杀菌剂
公开(公告)号：US06630495B1
公开(公告)日：2003-10-07
申请号：US10049981
申请日：2002-07-22
申请人： Tracey Cooke , Tennyson Ekwuru , David Hardy , Peter Millward , Brian Moloney , Andrew Pettinger , Peter Stanley Thomas , Richard Michael Turner
发明人： Tracey Cooke , Tennyson Ekwuru , David Hardy , Peter Millward , Brian Moloney , Andrew Pettinger , Peter Stanley Thomas , Richard Michael Turner
IPC分类号： C07D21302
CPC分类号： A01N43/90 , A01N43/40 , A01N43/42 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/78 , A01N43/80 , A01N43/82 , A01N47/24 , A01N47/38 , A01N47/40 , A01N53/00
摘要： Compounds of formula (I) or (II): or salts therefor are used as phytopathogenic fungicides wherein the various radicals and substitutents are as defined in the description. Pesticidal compositions contain these compounds together with an agriculturally acceptable diluent or carrier. The compounds and compositions are applied in methods for combating pests.
摘要翻译：式（I）或（II）的化合物或其盐用作植物病原性杀真菌剂，其中各种基团和取代基如说明书中所定义。杀虫组合物含有这些化合物以及农业上可接受的稀释剂或载体。化合物和组合物应用于防治害虫的方法中。

3. 发明授权

US6080871A Sulfonamides and sulfamides as H.sub.3 receptor antagonists 失效
标题翻译：磺酰胺和磺酰胺作为H3受体拮抗剂
公开(公告)号：US6080871A
公开(公告)日：2000-06-27
申请号：US117808
申请日：1998-10-06
申请人： Sarkis Barret Kalindjian , Nigel Paul Shankley , Matthew John Tozer , Iain Mair McDonald , Michael John Pether , Elaine Anne Harper , Gillian Fairfull Watt , Tracey Cooke , Caroline Minli Rachel Low
发明人： Sarkis Barret Kalindjian , Nigel Paul Shankley , Matthew John Tozer , Iain Mair McDonald , Michael John Pether , Elaine Anne Harper , Gillian Fairfull Watt , Tracey Cooke , Caroline Minli Rachel Low
IPC分类号： A61K31/00 , A61K31/415 , A61K31/4164 , A61K31/417 , A61P43/00 , C07D233/54 , C07D233/64 , C07D401/12
CPC分类号： C07D233/64 , C07D401/12
摘要： Compounds of formula (I) or (II) wherein R.sup.1 is C.sub.4 to C.sub.20 hydrocarbyl (in which one or more hydrogen atoms may be replaced by halogen, and up to three carbon atoms may be replaced by oxygen, nitrogen or sulphur atoms, provided that R.sup.1 does not contain an --O--O-- group), R.sup.2 is H or C.sub.1 to C.sub.3 alkyl, m is from 1 to 15, n is from 2 to 6, each X group is independently (a), or one X group is --N(R.sup.4)--, --O-- or --S-- and the remaining X groups are independently (a), wherein R.sup.3 is H, C.sub.1 to C.sub.6 alkyl, --CO.sub.2 R.sup.5, --CONR.sup.5.sub.2, --CR.sup.5.sub.2 OR.sup.6 or --OR.sup.5 (in which R.sup.5 and R.sup.6 are H or C.sub.1 to C.sub.3 alkyl), and R.sup.4 is H or C.sub.1 to C.sub.6 alkyl, each Y group is independently --C(R.sup.3)R.sup.4 --, or up to two Y groups are --N(R.sup.4)--, --O-- or --S-- and the remaining Y groups are independently --C(R.sup.3)R.sup.4 --, wherein R.sup.3 is as defined above, one R.sup.4 group in the structure is imidazoyl or imidazoylalkyl and the remaining R.sup.4 groups are H or C.sub.1 to C.sub.6 alkyl, and Z is >C(R.sup.7)NR.sup.2 -- or >N--, wherein R.sup.7 is any of the groups recited above for R.sup.3, and pharmaceutically acceptable salts thereof are ligands at histamine H.sub.3 receptors. ##STR1##
摘要翻译： PCT No.PCT / GB97 / 00358 Sec。 371 1998年10月6日第 102（e）日期1998年10月6日PCT 1997年2月10日提交PCT公布。第WO97 / 29092号公报日期1997年8月14日其中R 1为C 4至C 20烃基（其中一个或多个氢原子可以被卤素取代，并且最多三个碳原子）可以被氧，氮或氮取代的式（I）或（II）硫原子，条件是R1不含有-OO-基），R2为H或C1至C3烷基，m为1至15，n为2-6，X基团独立地为（a）或一个 X基团是-N（R 4） - ， - O-或-S-，其余的X基团独立地是（a），其中R 3是H，C 1 -C 6烷基，-CO 2 R 5，-CONR 52，-CR 52 OR 6或-OR 5（其中R5和R6是H或C1-C3烷基），R4是H或C1-C6烷基，每个Y基团独立地是-C（R3）R4-，或者最多两个Y基团是-N（R4） - ，-O-或-S-，其余的Y基团独立地为-C（R 3）R 4 - ，其中R 3如上定义，结构中的一个R 4基团为咪唑基或咪唑基烷基，其余的R 4基团为H或C 1至 C6烷基，并且Z是> C（R7）NR2-或> N-，其中R7是上述对R3所述的任何基团，并且药物其可用的盐是组胺H3受体的配体。

4. 发明授权

US06821992B1 Fungicides 有权
标题翻译：杀菌剂
公开(公告)号：US06821992B1
公开(公告)日：2004-11-23
申请号：US10049976
申请日：2002-07-09
申请人： Tracey Cooke , David Hardy , Brian Moloney , Peter Stanley Thomas , Chris Richard Steele , Geoffrey Gower Briggs
发明人： Tracey Cooke , David Hardy , Brian Moloney , Peter Stanley Thomas , Chris Richard Steele , Geoffrey Gower Briggs
IPC分类号： A01N4340
CPC分类号： C07D231/12 , A01N43/40 , A01N47/30 , C07D213/61 , C07D233/56 , C07D249/08 , C07D401/06 , C07D401/12 , C07D409/12 , C07D417/12
摘要： The invention relates to compounds of general formula I, where A1, R1, R2 and Y are as defined in the description; and to their use as phytopathogenic fungicides.
摘要翻译：本发明涉及通式I的化合物，其中A 1，R 1，R 2和Y如说明书中所定义; 并将其用作植物病原性杀真菌剂。

5. 发明授权

US07572818B2 2-pyridylethylbenzamide derivative 有权
标题翻译： 2-吡啶基乙基苯甲酰胺衍生物
公开(公告)号：US07572818B2
公开(公告)日：2009-08-11
申请号：US10524345
申请日：2003-08-08
申请人： Darren James Mansfield , Tracey Cooke , Peter Stanley Thomas , Pierre-Yves Coqueron , Jean-Pierre Vors , Geoffrey Gower Briggs , Hélène Lachaise , Heiko Rieck , Philippe Desbordes , Marie-Claire Grosjean-Cournoyer
发明人： Darren James Mansfield , Tracey Cooke , Peter Stanley Thomas , Pierre-Yves Coqueron , Jean-Pierre Vors , Geoffrey Gower Briggs , Hélène Lachaise , Heiko Rieck , Philippe Desbordes , Marie-Claire Grosjean-Cournoyer
IPC分类号： A61K31/44
CPC分类号： C07D213/89 , A01N43/40 , C07D213/40 , C07D213/61
摘要： Compound of general formula (I) in which p is an integer equal to 1, 2, 3 or 4; q is an integer equal to 1, 2, 3, 4 or 5; each substituent X is chosen, independently of the others, as being halogen, alkyl or haloalkyl, at least one of the substituents being a haloalkyl; each substituent Y is chosen, independently of the others, as being halogen, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, amino, phenoxy, alkylthio, dialkylamino, acyl, cyano, ester, hydroxy, aminoalkyl, benzyl, haloalkoxy, halosulphonyl, halothioalkyl, alkoxyalkenyl, alkylsulphonamide, nitro, alkylsulphonyl, phenylsulphonyl or benzylsulphonyl; as to the N-oxides of 2-pyridine thereof; with the exception of N-{2-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-ethyl}-2,6-dichlorobenzamide. Method for preparing the compound of general formula (I). Fungicidal composition comprising the compound of general formula (I). Method for treating phytopathogenic diseases.
摘要翻译：通式（I）的化合物，其中p是等于1,2,3或4的整数; q是等于1,2,3,4或5的整数; 每个取代基X独立地选自卤素，烷基或卤代烷基，至少一个取代基是卤代烷基; 每个取代基Y独立地选自卤素，烷基，烯基，炔基，卤代烷基，烷氧基，氨基，苯氧基，烷硫基，二烷基氨基，酰基，氰基，酯，羟基，氨基烷基，苄基，卤代烷氧基，卤代磺酰基，卤代烷基烷氧基烯基，烷基磺酰胺，硝基，烷基磺酰基，苯基磺酰基或苄基磺酰基; 关于其2-吡啶的N-氧化物; 除了N- {2- [3-氯-5-（三氟甲基）-2-吡啶基] - 乙基} -2,6-二氯苯甲酰胺外。制备通式（I）化合物的方法。包含通式（I）的化合物的杀真菌组合物。治疗植物病原性疾病的方法

6. 发明授权

US06939882B1 Fungicides 有权
标题翻译：杀菌剂
公开(公告)号：US06939882B1
公开(公告)日：2005-09-06
申请号：US10049980
申请日：2000-08-11
申请人： Tracey Cooke , David Hardy , Brian Anthony Moloney , Mary Josephine O'Mahony , Michael George Pettett , Gita Patel , Stefan Schnatterer
发明人： Tracey Cooke , David Hardy , Brian Anthony Moloney , Mary Josephine O'Mahony , Michael George Pettett , Gita Patel , Stefan Schnatterer
IPC分类号： A01N37/28 , A01N43/40 , A01N43/42 , A01N43/54 , A01N43/60 , A01N43/78 , A01N43/80 , A01N43/90 , A01N47/12 , A01N47/30 , A01N47/36 , A01N53/00 , A01N57/16 , C07C243/38 , C07D213/61 , C07D213/64 , C07D213/76 , C07D213/81 , C07D239/52 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D498/04 , C07F9/58 , C07D213/00
CPC分类号： C07D401/12 , A01N43/40 , A01N43/54 , A01N43/60 , A01N43/78 , A01N43/80 , A01N43/90 , A01N53/00 , A01N57/16 , C07C243/38 , C07D213/61 , C07D239/52 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07F9/58
摘要： Use of compounds of general formula (I) or salts thereof as phytopathogenic fungicides wherein the various radicals and substituents are as defined in the description, pesticidal compositions containing them and method for combatting pests which comprises applying these.
摘要翻译：使用通式（I）的化合物或其盐作为植物病原性杀真菌剂，其中各种基团和取代基如描述中所定义，含有它们的杀虫组合物和用于防治害虫的方法包括应用它们。

7. 发明授权

US06355665B1 1H-4(5)-substituted imidazole derivatives, their preparation and their use as histamine H3 receptor ligands 失效
标题翻译： 1H-4（5） - 取代咪唑衍生物，其制备及其作为组胺H3受体配体的用途
公开(公告)号：US06355665B1
公开(公告)日：2002-03-12
申请号：US09463012
申请日：2000-03-14
申请人： Matthew John Tozer , Sarkis Barret Kalindjian , Ian Duncan Linney , Katherine Isabel Mary Steel , Michael John Pether , Tracey Cooke
发明人： Matthew John Tozer , Sarkis Barret Kalindjian , Ian Duncan Linney , Katherine Isabel Mary Steel , Michael John Pether , Tracey Cooke
IPC分类号： C07D23354
CPC分类号： C07D233/64 , C07D417/04
摘要： A compound of the formula wherein R2 is an optionally substituted Cz to Cg alkylene or alkylene chain; R3 is C2 to C15 optionally substituted hydrocarbyl; X is a bond or —NR4—, wherein R4 is hydrogen or non-aromatic C1 to C5 optionally substituted hydrocarbyl, or aryl(C1 to C3)alkyl, or a pharmaceutically acceptable salt thereof. A method of modifing histamine activity in a patient comprising administering to said patient a pharmaceutical composition containing an effective amount of a compound of formula wherein R1 is selected from C1 to C6 alkyl, C1 to C6 alkoxy, C1 to C6 alkylthio, carboxy, carboxy(C1 to C6)alkyl, formyl, C1 to C6 alkylcarbonyl, C1 to C6 alkylcarbonylalkoxy, nitro, trihalomethyl, hydroxy, amino, C1 to C6 alkylcarbonylalkoxy, nitro, trihalomethyl, hydroxy, amino, C1 to C6 alkylamino, di(C1 to C6 alkyl)amino, aryl, C1 to C6 alkylaryl, halo, sulfamoyl and cyano; R2 is optionally substituted C2 to C20 hydrocarbylene, in which one or more hydrogen atoms may be replaced by halogen atoms and up to 6 carbon atoms may be replaced by oxygen or nitrogen atoms, R2 being in the form of an optionally substituted C2 to C8 alkylene or alkenylene chain; R3 is hydrogen or C1 to C15 optionally substituted hydrocarbyl; X is a bond or —NR4—; and a is from 0 to 2, or a pharmaceutically acceptable salt thereof.
摘要翻译：化学式R 2的化合物是任选取代的C 1至C 8亚烷基或亚烷基链; R3是C2至C15任选取代的烃基; X是键或-NR 4 - ，其中R 4是氢或非芳族C 1至C 5任选取代的烃基或芳基（C 1至C 3）烷基或其药学上可接受的盐。1，一种修饰患者组胺活性的方法，向所述患者施用含有有效量的蛔虫素R1化合物的药物组合物选自C1至C6烷基，C1至C6烷氧基，C1至C6烷硫基，羧基，羧基（C1至C6）烷基，甲酰基，C1至C6 烷基羰基，C 1至C 6烷基羰基烷氧基，硝基，三卤代甲基，羟基，氨基，C 1至C 6烷基羰基烷氧基，硝基，三卤甲基，羟基，氨基，C 1至C 6烷基氨基，二（C 1至C 6烷基）氨基，芳基，C 1至C 6烷基芳基，，氨磺酰基和氰基; R2是任选取代的C 2至C 20亚烃基，其中一个或多个氢原子可以被卤素原子取代，并且最多6个碳原子可被氧或氮原子取代，R 2为任选取代的C 2至C 8亚烷基或亚烯基链; R 3是氢或C 1至C 15任选取代的烃基; X是键或-NR4-; 和a为0至2，或其药学上可接受的盐。

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