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1. 发明授权

US3971814A Benzo(b)thiophene derivatives 失效
标题翻译：苯并（b）噻吩衍生物
公开(公告)号：US3971814A
公开(公告)日：1976-07-27
申请号：US566469
申请日：1975-04-09
申请人： Peter Johannes Stoss , Manfred Franz Reinhold Herrmann , Gerhard Satzinger
发明人： Peter Johannes Stoss , Manfred Franz Reinhold Herrmann , Gerhard Satzinger
IPC分类号： C07D413/04 , C07D333/64
CPC分类号： C07D413/04
摘要： The present invention relates to novel benzo(b)thiophene derivatives of the general formula: ##SPC1##Wherein Y represents a hydrogen or halogen atom; A represents a hydrogen atom or a phenyl group which may be substituted with a halogen atom or a lower alkoxy group; B represents a radical of the formula OR' or NR.sup.2 R.sup.3, wherein R' is an alkyl radical of 1 to 5 carbons which may be substituted with hydroxy, lower alkoxy, phenyl or phenoxy groups or a cycloalkyl or phenyl group which may be substituted by lower alkoxy or halogen atoms; R.sup.2 and R.sup.3, which may be identical or different, represent, if identical, hydrogen, alkyl radicals of 1 to 5 carbon atoms which may be substituted by hydroxy, lower alkoxy, phenoxy, di-lower alkylamino, or phenyl groups; or, if R.sup.2 is hydrogen, R.sup.3 represents either a hydroxyl or an amino group which may be substituted by lower alkyl, dialkyl, alkylidene, phenyl of acyl groups or a lower alkyl group which may be substituted by hydroxy, lower alkoxy, phenoxy, dialkylamino, pyrrolidino, piperidino or morpholino groups; R.sup.3 further is a cycloalkyl or phenyl group, which may be substituted by a halogen or a lower alkoxy radical; or R.sup.2 and R.sup.3 together with the nitrogen atom to which they are attached, may form an aziridine, pyrrolidine, piperidine, morpholine or piperazine ring which may be substituted by lower alkyl, hydroxyalkyl, phenylalkyl, phenyl or acetyl groups; or A and B together with the C=N group may form a 5, 6, or 7-membered heterocyclic ring.
摘要翻译：本发明涉及以下通式的新型苯并（b）噻吩衍生物：

2. 发明授权

US4056526A Benzo(b)thiophene derivatives 失效
标题翻译： BENZO（B）噻吩衍生物
公开(公告)号：US4056526A
公开(公告)日：1977-11-01
申请号：US691109
申请日：1976-05-28
申请人： Peter Johannes Stoss , Manfred Franz Reinhold Herrmann , Gerhard Satzinger
发明人： Peter Johannes Stoss , Manfred Franz Reinhold Herrmann , Gerhard Satzinger
IPC分类号： C07D413/04 , C07D413/02
CPC分类号： C07D413/04
摘要： The present invention relates to novel benzo(b)thiophene derivatives of the general formula: ##STR1## wherein Y represents a hydrogen or halogen atom; A represents a hydrogen atom or a phenyl group which may be substituted with a halogen atom or a lower alkoxy group; B represents a radical of the formula OR' or NR.sup.2 R.sup.3, wherein R' is an alkyl radical of 1 to 5 carbons which may be substituted with hydroxy, lower alkoxy, phenyl or phenoxy groups or a cycloalkyl or phenyl group which may be substituted by lower alkoxy or halogen atoms; R.sup.2 and R.sup.3, which may be identical or different, represent, if identical, hydrogen, alkyl radicals of 1 to 5 carbon atoms which may be substituted by hydroxy, lower alkoxy, phenoxy, di-lower alkylamino, or phenyl groups; or, if R.sup.2 is hydrogen, R.sup.3 represents either a hydroxyl or an amino group which may be substituted by lower alkyl, dialkyl, alkylidene, phenyl or acyl groups or a lower alkyl group which may be substituted by hydroxy, lower alkoxy, phenoxy, dialkylamino, pyrrolidino, piperidino or morpholino groups; R.sup.3 further is a cycloalkyl or phenyl group, which may be substituted by a halogen or a lower alkoxy radical; or R.sup.2 and R.sup.3 together with the nitrogen atom to which they are attached, may form an aziridine, pyrrolidine, piperidine, morpholine or piperazine ring which may be substituted by lower alkyl, hydroxyalkyl, phenylalkyl, phenyl or acetyl groups; or A and B together with the C.dbd.N group may form a 5, 6, or 7-membered heterocyclic ring.

3. 发明授权

US4082770A Benzo(b)thiophene derivatives 失效
标题翻译： BENZO（B）噻吩衍生物
公开(公告)号：US4082770A
公开(公告)日：1978-04-04
申请号：US785809
申请日：1977-04-08
申请人： Peter Johannes Stoss , Manfred Franz Reinhold Herrmann , Gerhard Satzinger
发明人： Peter Johannes Stoss , Manfred Franz Reinhold Herrmann , Gerhard Satzinger
IPC分类号： C07D333/70 , C07D333/64
CPC分类号： C07D333/70
摘要： The present invention relates to novel benzo(b)thiophene derivatives of the general formula: ##STR1## wherein Y represents a hydrogen or halogen atom; A represents a hydrogen atom or a phenyl group which may be substituted with a halogen atom or a lower alkoxy group; B represents a radical of the formula OR' or NR.sup.2 R.sup.3, wherein R' is an alkyl radical of 1 to 5 carbon atoms which may be substituted with hydroxy, lower alkoxy, phenyl or phenoxy groups or a cycloalkyl or phenyl group which may be substituted by lower alkoxy or halogen atoms; R.sup.2 and R.sup.3, which may be identical or different, represent, if identical, hydrogen, alkyl radicals of 1 to 5 carbon atoms which may be substituted by hydroxy, lower alkoxy, phenoxy, di-lower alkylamino, or phenyl groups; or, if R.sup.2 is hydrogen, R.sup.3 represents either a hydroxyl or an amino group which may be substituted by lower alkyl, dialkyl, alkylidene, phenyl or acyl groups or a lower alkyl group which may be substituted by hydroxy, lower alkoxy, phenoxy, dialkylamino, pyrrolidino, piperidino or morpholino groups; R.sup.3 further is a cycloalkyl or phenyl group, which may be substituted by a halogen or a lower alkoxy radical; R.sup.2 and R.sup.3 together with the nitrogen atom to which they are attached, may form an aziridine, pyrrolidine, piperidine, morpholine or piperazine ring which may be substituted by lower alkyl, hydroxyalkyl, phenylalkyl, phenyl or acetyl groups; or A and B together with the C--N group may form a 5, 6, or 7-membered heterocyclic ring.The present invention further relates to the processes for the preparation of these derivatives and to the salts of these compounds with physiologically acceptable inorganic and organic acids such as hydrochloric acid, sulfuric acid, phosphoric acid, fumaric acid, oxalic acid, citric acid, etc., and the quaternary ammonium compounds.

4. 发明授权

US4018793A Benzo (b) thiophene derivatives 失效
标题翻译：苯并（b）噻吩衍生物
公开(公告)号：US4018793A
公开(公告)日：1977-04-19
申请号：US685600
申请日：1976-05-12
申请人： Peter Johannes Stoss , Manfred Franz Reinhold Herrmann , Gerhard Satzinger
发明人： Peter Johannes Stoss , Manfred Franz Reinhold Herrmann , Gerhard Satzinger
IPC分类号： C07D333/70 , C07D413/04 , C07D333/66
CPC分类号： C07D413/04 , C07D333/70
摘要： The present invention relates to novel benzo(b)thiophene derivatives of the general formula: ##STR1## wherein Y represents a hydrogen or halogen atom; A represents a hydrogen atom or a phenyl group which may be substituted with a halogen atom or a lower alkoxy group; B represents a radical of the formula OR' or NR.sup.2 N.sup.3, wherein R' is an alkyl radical of 1 to 5 carbons which may be substituted with hydroxy, lower alkoxy, phenyl or phenoxy groups or a cycloalkyl or phenyl group which may be substituted by lower alkoxy or halogen atoms; R.sup.2 and R.sup.3, which may be identical or different, represent, if identical, hydrogen, alkyl radicals of 1 to 5 carbon atoms which may be substituted by hydroxy, lower alkoxy, phenoxy, di-lower alkylamino, or phenyl groups; or, if R.sup.2 is hydrogen, R.sup.3 represents either a hydroxyl or an amino group which may be substituted by lower alkyl, dialkyl, akylidene, phenyl or acyl groups or a lower alkyl group which may be substituted by hydroxy, lower alkoxy, phenoxy, dialkylamino, pyrrolidino, piperidino or morpholino groups; R.sup. 3 further is a cycloalkyl or phenyl group, which may be substituted by a halogen or a lower alkoxy radical; or R.sup.2 and R.sup.3 together with the nitrogen atom to which they are attached, may form an aziridine, pyrrolidine, piperidine, morpholine or piperazine ring which may be substituted by lower alkyl, hydroxyalkyl, phenylalkyl, phenyl or acetyl groups; or A and B together with the C=N group may form a 5, 6, or 7-membered heterocyclic ring.The present invention further relates to the processes for the preparation of these derivatives and to the salts of these compounds with physiologically acceptable inorganic and organic acids such as hydrochloric acid, sulfuric acid, phosphoric acid, fumaric acid, oxalic acid, citric acid, etc., and the quaternary ammonium compounds.
摘要翻译：本发明涉及以下通式的新的苯并（b）噻吩衍生物：其中Y代表氢或卤素原子; A表示氢原子或可被卤素原子或低级烷氧基取代的苯基; B表示式OR'或NR 2 N 3的基团，其中R'为可被羟基，低级烷氧基，苯基或苯氧基取代的1至5个碳的烷基或可以被低级烷基取代的环烷基或苯基烷氧基或卤素原子; R 2和R 3可以相同或不同，表示氢，氢原子可以被羟基，低级烷氧基，苯氧基，二低级烷基氨基或苯基取代的具有1-5个碳原子的烷基; 或者如果R 2为氢，则R 3表示可被低级烷基，二烷基，亚烷基，苯基或酰基取代的羟基或氨基，或可被羟基，低级烷氧基，苯氧基，二烷基氨基取代的低级烷基，吡咯烷子基，哌啶子基或吗啉代基团; R 3还可以是可被卤素或低级烷氧基取代的环烷基或苯基; 或R 2和R 3与它们所连接的氮原子一起形成可被低级烷基，羟基烷基，苯基烷基，苯基或乙酰基取代的氮丙啶，吡咯烷，哌啶，吗啉或哌嗪环; 或A和B与C = N基团一起可以形成5,6或7元杂环。

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