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1. 发明授权

US08034931B2 Process for producing substituted aminoquinazolinone derivative, intermediate therefor, and pest control agent 有权
标题翻译：制备取代氨基喹唑啉酮衍生物，其中间体和害虫防治剂的方法
公开(公告)号：US08034931B2
公开(公告)日：2011-10-11
申请号：US10556218
申请日：2004-05-11
申请人： Osamu Sanpei , Masahiro Uehara , Nobuyuki Niino , Hiroki Kodama , Kazuyuki Sakata
发明人： Osamu Sanpei , Masahiro Uehara , Nobuyuki Niino , Hiroki Kodama , Kazuyuki Sakata
IPC分类号： C07D239/80
CPC分类号： A01N43/54 , A01N47/16 , C07D401/12
摘要： A process for producing a substituted aminoquinazolinone derivative of formula (I), characterized by reducing a substituted iminoquinazolinone derivative of formula (II) with hydrogen in the presence of a catalyst and either of a halogen compound and a sulfur compound; a substituted iminoquinazolinone derivative of formula (II′); and a pest control agent containing the derivative of formula (II′) or a salt thereof as an active ingredient and a method of using the same (in the formulae, R represents hydrogen, formyl, (C1-C6) alkyl, (C1-C6)alkoxy(C1-C3)alkyl, (C1-C6) alkylsulfonyl, optionally substituted phenylcarbonyl, etc.; R1 represents an optionally substituted, 5- or 6-membered heterocycle having one to three heteroatoms selected among oxygen, sulfur, and nitrogen; R2 represents hydrogen or (C1-C3) alkyl; X and X′ may be the same or different and each represents (C1-C6) haloalkyl, (C1-C6) haloalkoxy, etc.; n is an integer of 0; and n′ is an integer of 1-4).
摘要翻译：一种制备式（I）的取代氨基喹唑啉酮衍生物的方法，其特征在于在催化剂和卤素化合物和硫化合物中的任一种存在下，用氢还原式（II）的取代亚氨基喹唑啉酮衍生物; 式（II'）的取代亚氨基喹唑啉酮衍生物; 和含有式（II'）的衍生物或其盐作为有效成分的害虫控制剂及其使用方法（式中，R表示氢，甲酰基，（C1-C6）烷基，（C1- C6烷氧基（C1-C3）烷基，（C1-C6）烷基磺酰基，任选取代的苯基羰基等; R 1表示具有一至三个选自氧，硫和氮的杂原子的任选取代的五元或六元杂环 ; R 2表示氢或（C 1 -C 3）烷基; X和X'可以相同或不同，表示（C1-C6）卤代烷基，（C1-C6）卤代烷氧基等; n为0的整数; n'是1-4的整数）。

2. 发明申请

US20070185142A1 Process for producing substituted aminoquinazolinone derivative, intermediate therefor, and pest control agent 有权
标题翻译：制备取代氨基喹唑啉酮衍生物，其中间体和害虫防治剂的方法
公开(公告)号：US20070185142A1
公开(公告)日：2007-08-09
申请号：US10556218
申请日：2004-05-11
申请人： Osamu Sanpei , Masahiro Uehara , Nobuyuki Niino , Hiroki Kodama , Kazuyuki Sakata
发明人： Osamu Sanpei , Masahiro Uehara , Nobuyuki Niino , Hiroki Kodama , Kazuyuki Sakata
IPC分类号： A61K31/517 , C07D239/92
CPC分类号： A01N43/54 , A01N47/16 , C07D401/12
摘要： A process for producing a substituted aminoquinazolinone derivative represented by the formula (I), characterized by reducing a substituted iminoquinazolinone derivative represented by the formula (II) with hydrogen in the presence of a catalyst and either of a halogen compound and a sulfur compound; a substituted iminoquinazolinone derivative represented by the formula (II′), which is an intermediate in the production process; and a pest control agent containing the derivative of the formula (II′) or a salt thereof as an active ingredient and a method of using the same (in the formulae, R represents hydrogen, formyl, (C1-C6) alkyl, (C1-C6)alkoxy(C1-C3)alkyl, (C1-C6) alkylsulfonyl, optionally substituted phenylcarbonyl, etc.; R1 represents an optionally substituted, 5- or 6-membered heterocycle having one to three heteroatoms selected among oxygen, sulfur, and nitrogen; R2 represents hydrogen or (C1-C3) alkyl; X and X′ may be the same or different and each represents (C1-C6) haloalkyl, (C1-C6) haloalkoxy, etc.; n is an integer of 0 to 4; and n′ is an integer of 1 to 4).
摘要翻译：一种制备由式（I）表示的取代氨基喹唑啉酮衍生物的方法，其特征在于在催化剂和卤素化合物和硫化合物之一中，用氢还原式（II）表示的取代亚氨基喹唑啉酮衍生物; 由式（II'）表示的取代亚氨基喹唑啉酮衍生物，其为生产过程中的中间体; 和含有式（II'）的衍生物或其盐作为有效成分的害虫防除剂及其使用方法（式中，R表示氢，甲酰基，（C 1〜 C 1 -C 6烷基，（C 1 -C 6 -C 6）烷氧基（C 1 -C 6亚烷基）烷基，（C 1 -C 6 -C 6）烷基磺酰基，任选取代的苯基羰基等; R 1表示任选取代的具有一至三个选自氧，硫和氮的杂原子的5-或6-元杂环; R 2表示氢或（C 1 -C 3 -C （C 1 -C 6）烷基; X和X'可以相同或不同，并且各自表示（C 1 -C 6 -C 6）卤代烷基，（C 1 -C 6烷基） C 1 -C 6卤代烷氧基等; n为0〜4的整数，n'为1〜4的整数。

3. 发明授权

US06639109B1 Process for production of thioalkylamine derivatives 有权
标题翻译：硫代烷基胺衍生物的制备方法
公开(公告)号：US06639109B1
公开(公告)日：2003-10-28
申请号：US10089114
申请日：2002-05-29
申请人： Osamu Sanpei , Kenji Tsubata
发明人： Osamu Sanpei , Kenji Tsubata
IPC分类号： C07C32324
CPC分类号： C07D213/70 , C07C323/25 , C07C2601/08 , C07D213/89 , C07D249/12 , C07D295/088 , C07D333/34
摘要： The present invention relates to a thioalkylamine derivative represented by general formula (I); and a process for production thereof: wherein each of R1 and R2 is H, (C1-C4)alkyl, (C3-C8)cycloalkyl, (C3-C8)cycloalkyl(C1-C4)alkyl, (substituted) phenyl, (substituted) phenyl(C1-C4)alkyl, or the like; each of R3 and R4 is H or a (C1-C4)alkyl group; each of R5 and R6 is H, (C1-C4)alkyl, a (substituted) phenyl group or a (substituted) phenyl(C1-C4)alkyl group; alternatively each of R1 and R2, R1 and R3 or R5, R3 and R4, R3 and R5 or R5 and R6 may together form lower alkylene; and R is (C1-C12)alkyl, (C3-C8)cycloalkyl, (C3-C8)cycloalkyl(C1-C4)alkyl, (substituted) phenyl, (substituted) phenyl(C1-C4)alkyl, a naphthyl group, a (substituted) aromatic heterocyclic, or the like.
摘要翻译：本发明涉及由通式（I）表示的硫代烷基胺衍生物。及其制备方法：其中R 1和R 2各自为H，（C 1 -C 4）烷基，（C 3 -C 8）环烷基，（C 3 -C 8）环烷基（C 1 -C 4）烷基，（取代的））苯基（C 1 -C 4）烷基等; R 3和R 4各自为H或（C 1 -C 4）烷基; R5和R6各自为H，（C1-C4）烷基，（取代）苯基或（取代）苯基（C1-C4）烷基; 或者R1和R2中的每一个，R 1和R 3或R 5，R 3和R 4，R 3和R 5或R 5和R 6可以一起形成低级亚烷基; 和（C 1 -C 4）烷基，（C 3 -C 8）环烷基，（C 3 -C 8）环烷基（C 1 -C 4）烷基，（取代的）苯基，（取代的）（取代的）芳族杂环基等。

4. 发明授权

US06239077B1 Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof 有权
标题翻译：氨基乙腈衍生物农业和园艺杀虫剂含有相同的用途
公开(公告)号：US06239077B1
公开(公告)日：2001-05-29
申请号：US09295319
申请日：1999-04-21
申请人： Nobuharu Andoh , Osamu Sanpei , Kazuyuki Sakata
发明人： Nobuharu Andoh , Osamu Sanpei , Kazuyuki Sakata
IPC分类号： A01N3734
CPC分类号： C07D213/30 , A01N37/26 , A01N37/34 , C07C255/26 , C07C255/57 , C07C309/65 , C07C311/09 , C07C317/22 , C07C317/44 , C07C317/50 , C07C323/19 , C07C323/20 , C07C323/60 , C07C323/62 , C07C2601/02 , C07C2601/14 , C07D213/64 , C07D213/65 , C07D213/69 , C07D213/81 , C07D213/82 , C07D213/85
摘要： An aminoacetonitrile derivative of the formula (I): (wherein Ar1 and Ar2 represents phenyl group; substituted phenyl group having at least one subsituent selected from halogen atom, nitro group, cyano group, (halo) C1-C6 alkyl group, (halo) C1-C6 alkoxyl group, (substituted) pheny group, (substituted) phenyloxy group and (substituted) phenylacetylene group; (substituted) pyridyl group; and (substituted) naphthyl group, Q represents —C(R1)(R2)— (wherein R1 and R2 represent hydrogen atom, halogen atom, (halo) C1-C6 alkyl group, (halo) C1-C6 alkoxy group, (substituted) C3-C6 cycloalkyl group), or R1 and R2 may be bound to represent C2-C6 alkylene group), —CH═CH— or —C≡C—, d is 0 or an integer of 1, R3 represents hydrogen atom, (halo) C1-C6 alkyl group, R4, R5, R6, R7 and R8 represent hydrogen atom, halogen atom, (halo) C1-C6 alkyl group, W is —O—, —S—, —SO2— or —N(R9)— (wherein R9 is a hydrogen atom or C1-C6 alkyl group), and a and b are 0 or an integer of 1 to 4)), an agricultural and hortecultural insecticide containing as an active ingredient said derivative, and a method for using the insecticide.
摘要翻译：式（I）的氨基乙腈衍生物:(其中Ar1和Ar2表示苯基;具有至少一个选自卤素原子，硝基，氰基，（卤代）C 1 -C 6烷基，（卤素） C1-C6烷氧基，（取代）苯基，（取代）苯氧基和（取代）苯乙炔基;（取代）吡啶基;（取代）萘基，Q表示-C（R1）（R2） - （其中 R 1和R 2表示氢原子，卤素原子，（卤素）C 1 -C 6烷基，（卤素）C 1 -C 6烷氧基，（取代的）C 3 -C 6环烷基），或者R 1和R 2可以结合表示C 2 -C 6 亚烷基），-CH = CH-或-C = C-，d为0或整数1，R 3表示氢原子，（卤素）C 1 -C 6烷基，R 4，R 5，R 6，R 7和R 8表示氢原子，卤素原子，（卤素）C 1 -C 6烷基，W是-O - ， - S - ， - SO 2 - 或-N（R 9） - （其中R 9是氢原子或C 1 -C 6烷基） a和b为0或1〜4的整数）），农业和水平含有作为活性成分的所述衍生物的文化杀虫剂以及使用杀虫剂的方法。

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