专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

标题翻译：咪唑化合物和杀生物组合物，其组成物包含用于控制有害生物体的化合物

公开(公告)号：US4995898A

公开(公告)日：1991-02-26

申请号：US168070

申请日：1988-03-14

申请人： Rikuo Nasu , Terumasa Komyoji , Toshio Nakajima , Kazumi Suzuki , Keiichiro Ito , Takeshi Oshima , Hideshi Yoshimura

发明人： Rikuo Nasu , Terumasa Komyoji , Toshio Nakajima , Kazumi Suzuki , Keiichiro Ito , Takeshi Oshima , Hideshi Yoshimura

IPC分类号： A01N43/50 , A01N31/14 , A01N33/00 , A01N37/34 , A01N43/08 , A01N43/84 , A01N55/00 , A01P3/00 , C07D233/84 , C07D233/90 , C07D233/92 , C07D401/04 , C07D401/12 , C07D405/04 , C07D405/14 , C07D409/04 , C07D409/12 , C07F7/08

CPC分类号： C07D401/04 , A01N43/50 , A01N55/00 , C07D233/90 , C07D401/12 , C07D405/04 , C07D405/14 , C07D409/04 , C07F7/0814

摘要： Novel imidazole compounds are disclosed, which are represented by the following general formula: ##STR1## wherein: R.sub.1 represents a cyano group or a --CSNHR.sub.5 group, wherein R.sub.5 represents a hydrogen atom, a C.sub.1-4 alkyl group, or a --COR.sub.6 group, wherein R.sub.6 represents a C.sub.1-4 alkyl group, a halogenated C.sub.1-4 alkyl group, or a phenyl group;R.sub.2 and R.sub.3 each represents a hydrogen atom; a halogen atom; a nitro group; a cyano group; a trimethylsilyl group; a C.sub.3-6 cycloalkyl group; a naphthyl group; a C.sub.1-12 alkyl group which is optionally substituted with one or more halogen atoms, hydroxyl groups, acetoxy groups, C.sub.1-4 alkoxy groups, halogenated C.sub.1-4 alkoxy groups, phenyl groups, halogenated phenyl groups, or C.sub.1-4 alkylated phenyl groups; a C.sub.2-10 alkenyl group which is optionally substituted with one or more halogen atoms; a C.sub.1-6 alkoxy group which is optionally substituted with one or more halogen atoms; a phenyl group which is optionally substituted with one or more halogen atoms, C.sub.1-4 alkyl groups, halogenated C.sub.1-4 alkyl groups, C.sub.1-4 alkoxy groups, halogenated C.sub.1-4 alkoxy groups, C.sub.1-4 alkylthio groups, halogenated C.sub.1-4 alkylthio groups, nitro groups, cyano groups, or 3,4-methylenedioxy groups; a furyl group which is optionally substituted with one or more halogen atoms or C.sub.1-4 alkyl groups; a thienyl group which is optionally substituted with one or more halogen atoms or C.sub.1-4 alkyl groups; a pyridyl group which is optionally substituted with one or more halogen atoms or C.sub.1-4 alkyl groups; an --SO.sub.n R.sub.7 group, wherein R.sub.7 represents a C.sub.1-6 alkyl group, a C.sub.2-6 alkenyl group, a phenyl group which is optionally substituted with one or more halogen atoms, a benzyl group, a pyridyl group which is optionally substituted with one or more halogen atoms, C.sub.1-4 alkyl groups, or halogenated C.sub.1-4 alkyl groups; or an --NR.sub.8 R.sub.9 group, wherein R.sub.8 and R.sub.9 each represents a C.sub.1-4 alkyl group, and n is 0, 1, or 2; or a --CO(NH).sub.m R.sub.10 group, wherein R.sub.10 represents a C.sub.1-4 alkyl group which is optionally substituted with one or more halogen atoms, a C.sub.1-4 alkoxy group which is optionally substituted with one or more halogen atoms, or a phenyl group which is optionally substituted with one or more halogen atoms; and m is 0 or 1; andR.sub.4 represents a C.sub.1-6 alkyl group which is optionally substituted with one or more halogen atoms; a C.sub.3-6 cycloalkyl group; a phenyl group; a thienyl group; or an --NR.sub.11 R.sub.12 group, wherein R.sub.11 and R.sub.12 each represents a hydrogen atom, a C.sub.1-4 alkyl group which is optionally substituted with one or more halogen atoms, a C.sub.2-4 alkenyl group, or R.sub.11 and R.sub.12 are combined with each other together with a nitrogen atoms adjacent thereto to form a pyrrolidinyl group, a piperidinyl group, a morpholino group, or a thiomorpholino group, provided that R.sub.11 and R.sub.12 are not simultaneously a hydrogen atom;provided that R.sub.2 and R.sub.3 are not simultaneously a halogen atom. The compounds are effective as biocides.

摘要翻译：由通式I表示的咪唑化合物：其中：R1表示氰基或-CSNHR5基团，其中R5表示氢原子，C1-4烷基或-COR6基团，其中R6表示C1- 4烷基，卤代C 1-4烷基或苯基; R2和R3各自表示氢原子; 卤素原子; 硝基; 氰基; 三甲基甲硅烷基 C 3-6环烷基; 萘基; 任选取代的C 1-12烷基，C 2-10烯基，C 1-6烷氧基，苯基，呋喃基，亚硫酰基或吡啶基; a-SO n R 7基，其中R 7表示C 1-6烷基，C 2-6烯基，苄基，任选取代的苯基或吡啶基; NR8R9基团，其中R8和R9各自表示C1-4烷基，n为0,1或2; 或-CO（NH）m R 10 gorup，其中R 10表示任选取代的C 1-4烷基，C 1-4烷氧基或苯基，m为0或1; 并且R 4表示任选被一个或多个卤素原子取代的C 1-6烷基; C 3-6环烷基; 苯基; 噻吩基; 或-NR 11 R 12基团，其中R 11和R 12各自表示氢原子，任选被一个或多个卤素原子取代的C 1-4烷基，C 2-4链烯基或R 11和R 12一起彼此结合与其相邻的氮原子形成吡咯烷基，哌啶基，吗啉代基或硫代吗啉基，条件是R 11和R 12不同时为氢原子; 条件是R2和R3不同时为卤素原子。这些化合物作为杀生物剂是有效的。

IPRDB

热门服务

关于我们

友情链接

联系方式