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1. 发明授权

US08158575B2 Agent for the prevention and treatment of sexually transmitted diseases-I 有权
标题翻译：预防和治疗性传播疾病的代理 - 我
公开(公告)号：US08158575B2
公开(公告)日：2012-04-17
申请号：US12498077
申请日：2009-07-06
申请人： Barry Ross Matthews , George Holan , Peter Karellas , Scott Andrew Henderson , David Francis O'Keefe
发明人： Barry Ross Matthews , George Holan , Peter Karellas , Scott Andrew Henderson , David Francis O'Keefe
IPC分类号： A01N61/00
CPC分类号： B82Y5/00 , A61K47/59 , A61K47/595 , A61K47/645 , A61K47/6949 , C08G69/10 , C08G83/003 , Y10S977/754
摘要： Use of a polylysine, polyamidoamine or polypropylenimine dendrimer having naphthyl disulphonate terminal groups as a topically applied agent in prophylaxis or treatment of sexually transmitted diseases.
摘要翻译：具有萘基二磺酸酯末端基团的聚赖氨酸，聚酰胺胺或聚丙烯亚胺树枝状大分子作为局部施用剂在预防或治疗性传播疾病中的应用。

2. 发明申请

US20090269298A1 AGENT FOR THE PREVENTION AND TREATMENT OF SEXUALLY TRANSMITTED DISEASES-I 有权
标题翻译：预防和治疗性传播疾病的代理 - 一
公开(公告)号：US20090269298A1
公开(公告)日：2009-10-29
申请号：US12498077
申请日：2009-07-06
申请人： Barry Ross MATTHEWS , George HOLAN , Peter KARELLAS , Scott Andrew HENDERSON , David Francis O'KEEFE
发明人： Barry Ross MATTHEWS , George HOLAN , Peter KARELLAS , Scott Andrew HENDERSON , David Francis O'KEEFE
IPC分类号： A61K31/785 , A61P31/22
CPC分类号： B82Y5/00 , A61K47/59 , A61K47/595 , A61K47/645 , A61K47/6949 , C08G69/10 , C08G83/003 , Y10S977/754
摘要： Use of a polylysine, polyamidoamine or polypropylenimine dendrimer having naphthyl disulphonate terminal groups as a topically applied agent in prophylaxis or treatment of sexually transmitted diseases.
摘要翻译：具有萘基二磺酸酯末端基团的聚赖氨酸，聚酰胺胺或聚丙烯亚胺树枝状大分子作为局部施用的药物用于预防或治疗性传播疾病。

3. 发明授权

US4753960A Oxime insecticides 失效
标题翻译：肟类杀虫剂
公开(公告)号：US4753960A
公开(公告)日：1988-06-28
申请号：US847903
申请日：1986-03-10
申请人： George Holan , Kurt Rihs , Wynona M. P. Johnson
发明人： George Holan , Kurt Rihs , Wynona M. P. Johnson
IPC分类号： A01N35/10 , A01N43/30 , C07D317/58 , A61K31/30
CPC分类号： A01N43/30 , A01N35/10 , C07D317/58
摘要： Compounds with anthropodicidal activities having the general formula (1) ##STR1## and their isomeric forms wherein R represents F, Cl, Br, ethoxy, methoxy or propxy and n is an integer between 1 and 5; or R represents 3,4-methylenedioxyl; and R.sup.40 represents di- or trichloromethyl, fluorodichloromethyl or trifluoromethyl.
摘要翻译： PCT No.PCT / AU85 / 00164 Sec。 371日期：1986年3月10日 102（e）1986年3月10日PCT PCT日期：1985年7月22日PCT公布。出版物WO86 / 00894 日期：1986年2月13日。具有通式（1）及其异构体形式的具有杀虫活性的化合物，其中R表示F，Cl，Br，乙氧基，甲氧基或丙氧基，n为1至5的整数; 或R代表3,4-亚甲二氧基; R40表示二氯或三氯甲基，氟代二氯甲基或三氟甲基。

4. 发明授权

US4474815A Insecticidal oximes 失效
标题翻译：杀虫肟
公开(公告)号：US4474815A
公开(公告)日：1984-10-02
申请号：US370971
申请日：1982-04-02
申请人： George Holan , Wynona M. P. Johnson
发明人： George Holan , Wynona M. P. Johnson
IPC分类号： A01N35/10 , C07C67/00 , C07C239/00 , C07C251/50 , A61K31/15 , C07C131/00
CPC分类号： A01N35/10
摘要： Compounds of the general formula (I) ##STR1## wherein R represents F, Cl, Br, I, ethoxy, methoxy or propoxy and n is an integer between 1 and 5; orR represents 3,4-methylenedioxy; andR.sup.1 represents di- or tri-chloromethyl.The compounds have arthropodicidal (especially insecticidal and acaricidal) activity.
摘要翻译：通式（I）的化合物其中R表示F，Cl，Br，I，乙氧基，甲氧基或丙氧基，n为1至5之间的整数; 或R表示3,4-亚甲二氧基; 并且R 1表示二 - 或三 - 氯甲基。这些化合物具有节肢动物（特别是杀虫和杀螨）活性。

5. 发明授权

US4390715A Pentafluorobenzyl esters 失效
标题翻译：五氟苄基酯
公开(公告)号：US4390715A
公开(公告)日：1983-06-28
申请号：US282190
申请日：1981-07-10
申请人： George Holan , David F. O'Keefe
发明人： George Holan , David F. O'Keefe
IPC分类号： C07C69/753 , A01N37/08 , A01N37/38 , A01N43/30 , A01N53/00 , A01N53/06 , C07C69/757 , C07D317/60 , C07C69/76
CPC分类号： A01N37/38 , A01N37/08 , A01N53/00
摘要： The (+), (-) and (.+-.) forms of the compounds of the general formula (I) ##STR1## characterized in that R.sup.1 is a halo group; or a lower alkyl, lower alkoxy or lower alkylthio group, each of which may be substituted with one or more halo groups;R.sup.2 is hydrogen or a methyl group; or R.sup.1 and R.sup.2 together form a methylenedioxy, or a difluoromethylenedioxy group or, with the carbon atoms to which they are attached, an aromatic or heteroaromatic ring; andA is one of the groups X or Y ##STR2## wherein X.sup.1 and X.sup.2 are the same or different and each is hydrogen or a fluoro, chloro, bromo or methyl group, with the proviso that if X.sup.1 is a fluoro group, then X.sup.2 should not be a bromo group; and X.sup.3 and X.sup.4 are the same or different and each is hydrogen or a fluoro group; andY.sup.1, Y.sup.2, Y.sup.3, Y.sup.4, Y.sup.5 and Y.sup.6 are the same or different groups and each is hydrogen or a fluoro, bromo, chloro, or methyl group.The compounds (I) are insecticidally active.
摘要翻译：通式（I）化合物（I）的（+），（ - ）和（+/-）形式，其特征在于R1为卤素基团; 或低级烷基，低级烷氧基或低级烷硫基，每一个可被一个或多个卤素基团取代; R2是氢或甲基; 或R 1和R 2一起形成亚甲二氧基或二氟亚甲二氧基，或与其连接的碳原子一起形成芳族或杂芳族环; 并且A是X或Y之一，其中X 1和X 2相同或不同，并且各自是氢或氟，氯，溴或甲基，条件是如果X 1是氟基，则X 2 不应该是溴族; X3和X4相同或不同，各自为氢或氟基; Y 1，Y 2，Y 3，Y 4，Y 5和Y 6为相同或不同的基团，各自为氢或氟，溴，氯或甲基。

6. 发明授权

US4355042A Insecticidal esters 失效
公开(公告)号：US4355042A
公开(公告)日：1982-10-19
申请号：US195600
申请日：1980-10-09
申请人： George Holan , David F. O'Keefe
发明人： George Holan , David F. O'Keefe
IPC分类号： C07C69/74 , A01N33/20 , A01N37/08 , A01N37/10 , A01N37/34 , A01N37/38 , A01N37/48 , A01N43/08 , A01N43/30 , C07C51/00 , C07C61/15 , C07C61/39 , C07C61/40 , C07C62/12 , C07C62/34 , C07C67/00 , C07C69/753 , C07C69/757 , C07C201/00 , C07C205/55 , C07C253/00 , C07C255/38 , C07C313/00 , C07C323/62 , C07D307/42 , C07D317/60 , C07D317/68 , C07D307/40
CPC分类号： A01N37/48 , A01N37/08 , A01N37/10 , A01N37/34 , A01N37/38 , A01N43/08 , A01N43/30 , C07C61/15 , C07C61/40 , C07C62/12 , C07C62/34 , C07C69/753 , C07C69/757 , C07D317/60
摘要： Compounds of the general formula I ##STR1## wherein R.sup.1 is hydrogen or a methoxy, ethoxy, propoxy, butoxy, tetrafluoroethoxy, methylthio, ethylthio, propylthio, fluoro, chloro, bromo, methyl, ethyl, or nitro group, and R.sup.2 is hydrogen or a methyl group, orR.sup.1 and R.sup.2 together form a methylenedioxy group;R.sup.3 is hydrogen, or a lower alkyl group, or one of the following groups (a) to (f):(a) 3-phenoxybenzyl(b) 2-benzyl-4-furylmethyl(c) .alpha.-cyano-3-phenoxybenzyl(d) 3,4-methylenedioxybenzyl(e) .alpha.-ethynyl-3-phenoxybenzyl(f) .alpha.-cyano-3-(4'-chlorophenoxy)-benzyland Y.sup.1, Y.sup.2, Y.sup.3, Y.sup.4, Y.sup.5 and Y.sup.6 are the same or different groups and each is hydrogen or a fluoro, bromo or chloro group, with the proviso that when R.sup.1 is hydrogen, fluoro, chloro, bromo or methyl and R.sup.2 is hydrogen, then one of Y.sup.1 to Y.sup.6 is other than hydrogen.The compounds in which R.sup.3 is one of groups (a) to (f) are insecticides.

7. 发明授权

US4262014A Insecticidal esters 失效
标题翻译：杀虫剂
公开(公告)号：US4262014A
公开(公告)日：1981-04-14
申请号：US932549
申请日：1978-08-10
申请人： George Holan , Reimund A. Walser
发明人： George Holan , Reimund A. Walser
IPC分类号： C07C69/007 , A01N53/00 , A01N53/02 , A01N53/04 , A01N53/08 , A01N53/10 , A01N57/00 , C07C51/00 , C07C51/353 , C07C61/28 , C07C61/39 , C07C61/40 , C07C62/34 , C07C67/00 , C07C69/612 , C07C69/618 , C07C69/73 , C07C69/734 , C07C69/74 , C07C69/747 , C07C69/753 , C07C69/757 , C07C201/00 , C07C205/55 , C07C205/56 , C07C227/00 , C07C227/16 , C07C227/18 , C07C229/46 , C07C253/00 , C07C255/38 , C07C255/39 , C07C255/42 , C07C313/00 , C07C323/62 , C07D307/36 , C07D307/42 , C07D307/45 , C07D307/54 , C07D317/06 , C07D317/46 , C07D317/54 , C07D317/60 , A01N43/16
CPC分类号： C07D307/42 , A01N53/00 , C07C255/00 , C07D307/54 , C07D317/60 , Y10S514/919
摘要： The (+), (-) and (.+-.) forms of the compounds of formula I ##STR1## wherein R.sup.1 is hydrogen or a methoxy, ethoxy, propoxy, methylthio, ethylthio, propylthio, fluoro, chloro, bromo, methyl, ethyl, nitro or amino group,andR.sup.2 is a hydrogen or methyl group or R.sup.1 and R.sup.2 together form a methylenedioxy group;R.sup.3 is hydrogen, or a lower alkyl group, or one of the following groups (a) to (d):(a) m-phenoxybenzyl(b) 2-benzyl-4-furylmethyl(c) .alpha.-cyano-m-phenoxybenzyl(d) 3-4-methylenedioxy-benzyl,andR.sup.4 and R.sup.5 are the same or different groups and each is a fluoro, bromo, chloro or methyl group.The compounds of formula I in which R.sup.3 is one of groups (a) to (d) are extremely active as insecticides (except when R.sup.1 is an amino group). The compounds also possess the property of contact repellency to insects.
摘要翻译：其中R 1是氢或甲氧基，乙氧基，丙氧基，甲硫基，乙硫基，丙硫基，氟，氯，溴，甲基，或它们的（+），（ - ）和（+/-）乙基，硝基或氨基，R 2为氢或甲基，或者R 1和R 2一起形成亚甲二氧基; R3是氢或低级烷基，或以下基团之一（a）至（d）：（a）间苯氧基苄基（b）2-苄基-4-呋喃基甲基（c）α-氰基间苯氧基苄基（d）3-4-亚甲二氧基 - 苄基，R 4和R 5是相同或不同的基团，并且各自是氟，溴，氯或甲基。其中R3是基团（a）至（d）之一的式I化合物作为杀虫剂是非常有活性的（除了当R1是氨基时）。该化合物还具有与昆虫接触排斥性的性质。

8. 发明授权

US4097599A Triazoles 失效
标题翻译：三唑
公开(公告)号：US4097599A
公开(公告)日：1978-06-27
申请号：US776187
申请日：1977-03-10
申请人： John James Alexander Evans , George Holan
发明人： John James Alexander Evans , George Holan
IPC分类号： A01N43/78 , C07D249/08 , A01N9/22 , C07D401/04
CPC分类号： A01N43/78
摘要： 3-Trihalomethyl-1,2,4-triazoles either unsubstituted or having substituents in the 4 and/or 5, 1 and/or 5, and 2 and/or 5 positions; and methods for their preparation. The compounds show biological activity; at least some have acaricidal activity.
摘要翻译：在4和/或5,1和/或5和2和/或5位未被取代或具有取代基的3-三卤代甲基-1,2,4-三唑; 及其制备方法。

9. 发明授权

US3576818A 2-cyanobenzimidazoles and a process for their preparation 失效
标题翻译： 2-氰基苯并咪唑及其制备方法
公开(公告)号：US3576818A
公开(公告)日：1971-04-27
申请号：US3576818D
申请日：1967-09-18
申请人： EVA LEA SAMUEL , GEORGE HOLAN
发明人： SAMUEL EVA LEA , HOLAN GEORGE
IPC分类号： C07D235/10 , C07D235/24 , C07D49/38
CPC分类号： C07D235/24 , C07D235/10
摘要： 2-CYANOBENZIMIDAZOLES OF THE FORMULA:

2-(CN-),R1,R2-BENZIMIDAZOLE

WHEREIN R1 AND R2 ARE INDEPENDENTLY SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, CHLORINE, BROMINE, NITRO, ALKYL OF NOT MORE THAN FOUR CARBON ATOMS, AND ALKOXY OF NOT MORE THAN FOUR CARBON ATOMS, EXHIBIT ANTISEPTIC AND BACTERICIDAL ACTIVITY. THE 2-CYANOBENZIMIDAZOLES ARE PREPARED BY THE REACTION OF A BENZIMIDAZOLE OF THE FORMULA

2-A,R1,R2-BENZIMIDAZOLE

WHEREIN R1 AND R2 ARE AS DEFINED ABOVE AND A IS SELECTED FROM TRICHLOROMETHYL, MONOCHLORODIFLUOROMETHYL NAD MONOFLUORODICHLOROMETHYL, WITH AMMONIA.

10. 发明申请

US20050008611A1 Agent for the prevention and treatment of sexually transmitted diseases-I 有权
标题翻译：预防和治疗性传播疾病的代理 - 我
公开(公告)号：US20050008611A1
公开(公告)日：2005-01-13
申请号：US10472439
申请日：2002-03-28
申请人： Barry Matthews , George Holan , Peter Karellas , Scott Henderson , David O'Keefe
发明人： Barry Matthews , George Holan , Peter Karellas , Scott Henderson , David O'Keefe
IPC分类号： A61K38/00 , A61K31/785 , A61K47/48 , A61P15/00 , A61P31/04 , A61P31/12 , A61P31/18 , A61P31/22 , C07K14/00 , C08G69/10 , C08G83/00 , A61K31/74 , C08G69/08 , C08G73/10
CPC分类号： B82Y5/00 , A61K47/59 , A61K47/595 , A61K47/645 , A61K47/6949 , C08G69/10 , C08G83/003 , Y10S977/754
摘要： Use of a polylysine, polyamidoamine or polypropylenimine dendrimer having naphthyl disulphonate terminal groups as a topically applied agent in prophylaxis or treatment of sexually transmitted diseases.
摘要翻译：具有萘基二磺酸酯末端基团的聚赖氨酸，聚酰胺胺或聚丙烯亚胺树枝状大分子作为局部施用的药物用于预防或治疗性传播疾病。

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