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81. 发明申请

US20050277672A1 Benzimidazolone carboxylic acid derivatives 失效
标题翻译：苯并咪唑酮羧酸衍生物
公开(公告)号：US20050277672A1
公开(公告)日：2005-12-15
申请号：US11153766
申请日：2005-06-14
申请人： Koji Ando , Satoru Iguchi , Noriaki Murase , Yoshinori Murata , Toyoharu Numata , Hiroki Sone , Chikara Uchida , Tatsuo Ueki
发明人： Koji Ando , Satoru Iguchi , Noriaki Murase , Yoshinori Murata , Toyoharu Numata , Hiroki Sone , Chikara Uchida , Tatsuo Ueki
IPC分类号： A61K31/4184 , A61K31/454 , C07D401/12 , C07D401/14 , C07D405/14 , C07D43/02
CPC分类号： C07D401/12 , C07D401/14 , C07D405/14
摘要： This invention relates to compounds of the formula (I): wherein R1, R2, R3, A and m are each as described herein or a pharmaceutically acceptable salt or solvate thereof, and compositions containing such compounds and the use of such compounds in the treatment of a condition mediated by 5-HT4 receptor activity such as, but not limited to, gastroesophageal reflux disease, gastrointestinal disease, gastric motility disorder, non-ulcer dyspepsia, functional dyspepsia, irritable bowel syndrome (IBS), constipation, dyspepsia, esophagitis, gastroesophageral disease, nausea, central nervous system disease, Alzheimer's disease, cognitive disorder, emesis, migraine, neurological disease, pain, cardiovascular disorders such as cardiac failure and heart arrhythmia, diabetes and apnea syndrome.
摘要翻译：本发明涉及式（I）化合物：其中R 1，R 2，R 3，A和m各自如上所述本文或其药学上可接受的盐或溶剂合物，以及含有这些化合物的组合物以及这些化合物在治疗由5-HT 4受体活性介导的病症中的用途，所述活性例如但不限于，胃食管反流病，胃肠道疾病，胃动力障碍，非溃疡性消化不良，功能性消化不良，肠易激综合征（IBS），便秘，消化不良，食管炎，胃肠疾病，恶心，中枢神经系统疾病，阿尔茨海默病，认知障碍，呕吐，偏头痛，神经系统疾病，疼痛，心血管疾病如心力衰竭和心律失常，糖尿病和呼吸暂停综合征。

82. 发明申请

US20050277671A1 Benzimidazolone carboxylic acid derivatives 失效
公开(公告)号：US20050277671A1
公开(公告)日：2005-12-15
申请号：US11153757
申请日：2005-06-14
申请人： Koji Ando , Satoru Iguchi , Noriaki Murase , Yoshinori Murata , Toyoharu Numata , Hiroki Sone , Chikara Uchida , Tatsuo Ueki
发明人： Koji Ando , Satoru Iguchi , Noriaki Murase , Yoshinori Murata , Toyoharu Numata , Hiroki Sone , Chikara Uchida , Tatsuo Ueki
IPC分类号： A61K31/41 , A61K31/4184 , A61K31/4245 , A61K31/433 , A61K31/453 , A61K31/454 , A61P1/00 , A61P1/04 , A61P1/06 , A61P3/10 , A61P9/00 , A61P25/00 , A61P25/06 , A61P25/28 , C07D401/12 , C07D401/14 , C07D403/00 , C07D403/14 , C07D405/14 , C07D413/14 , C07D417/14 , C07D43/02
CPC分类号： C07D401/12 , C07D211/26 , C07D401/06 , C07D401/14 , C07D405/06 , C07D405/14
摘要： This invention relates to compounds of the formula (I): wherein R1, R2, R3, A and m are each as described herein or a pharmaceutically acceptable salt or solvate thereof, and compositions containing such compounds and the use of such compounds in the treatment of a condition mediated by 5-HT4 receptor activity such as, but not limited to, gastroesophageal reflux disease, gastrointestinal disease, gastric motility disorder, non-ulcer dyspepsia, functional dyspepsia, irritable bowel syndrome (IBS), constipation, dyspepsia, esophagitis, gastroesophageral disease, nausea, central nervous system disease, Alzheimer's disease, cognitive disorder, emesis, migraine, neurological disease, pain, cardiovascular disorders such as cardiac failure and heart arrhythmia, diabetes and apnea syndrome.

83. 发明授权

US4213517A Elevator control system 失效
标题翻译：电梯控制系统
公开(公告)号：US4213517A
公开(公告)日：1980-07-22
申请号：US922430
申请日：1978-07-06
申请人： Koji Ando
发明人： Koji Ando
IPC分类号： B66B1/28 , H02P27/02 , B66B1/30
CPC分类号： H02P27/026 , B66B1/308
摘要： An elevator control system includes a power source which supplies AC power to an induction motor for driving an elevator car through a first thyristor gate circuit. Another induction motor provided for braking the elevator car is connected to the power source through a second thyristor gate circuit. A tachometer generator connected to the induction motors produces an speed signal indicative of the speed of the elevator car. The speed signal is compared with a reference signal and the difference therebetween is used to control the first and second thyristor gate circuits for controlling the elevator car speed.
摘要翻译：电梯控制系统包括：电源，其通过第一晶闸管门电路向用于驱动电梯轿厢的感应电动机提供AC电力。设置用于制动电梯轿厢的另一感应电动机通过第二晶闸管门电路连接到电源。连接到感应电动机的转速计发生器产生指示电梯轿厢的速度的速度信号。将速度信号与参考信号进行比较，并且其差值用于控制用于控制电梯轿厢速度的第一和第二晶闸管门电路。

84. 发明授权

US08383819B2 Method for producing 4-oxoquinoline compound 有权
标题翻译： 4-氧代喹啉化合物的制备方法
公开(公告)号：US08383819B2
公开(公告)日：2013-02-26
申请号：US12281889
申请日：2007-03-06
申请人： Koji Matsuda , Koji Ando , Shigeji Ohki , Jun-ichi Hoshi , Takahiro Yamasaki
发明人： Koji Matsuda , Koji Ando , Shigeji Ohki , Jun-ichi Hoshi , Takahiro Yamasaki
IPC分类号： C07D215/00
CPC分类号： C07C229/30 , C07C43/215 , C07C57/72 , C07C57/76 , C07C61/40 , C07C67/333 , C07C67/343 , C07C69/708 , C07C69/716 , C07C69/738 , C07C69/92 , C07C69/94 , C07C229/34 , C07D215/56
摘要： The present invention provides a compound useful as a synthetic intermediate for an anti-HIV agent having an integrase inhibitory activity, and a production method thereof, and a production method of an anti-HIV agent using the synthetic intermediate. Specifically, for example, a compound represented by the formula (2′): wherein R is a fluorine atom or a methoxy group, and R400 is a hydrogen atom or a C1-C4 alkyl group, or a salt thereof, and a production method thereof, and a production method of an anti-HIV agent using the synthetic intermediate.
摘要翻译：本发明提供了可用作具有整合酶抑制活性的抗HIV剂的合成中间体的化合物及其制备方法，以及使用该合成中间体的抗HIV剂的制备方法。具体而言，例如，式（2'）表示的化合物或其盐，其中R为氟原子或甲氧基，R400为氢原子或C1-C4烷基，以及使用该合成中间体的抗HIV剂的制造方法。

85. 发明授权

US07964732B2 Substituted bicyclocarboxyamide compounds 失效
标题翻译：取代的双环羧基酰胺化合物
公开(公告)号：US07964732B2
公开(公告)日：2011-06-21
申请号：US12063159
申请日：2007-11-09
申请人： Koji Ando , Andrew Anthony Calabrese , Matthew Alexander James Duncton , Kentaro Futatsugi , Misato Hirano , Satochi Nagayama
发明人： Koji Ando , Andrew Anthony Calabrese , Matthew Alexander James Duncton , Kentaro Futatsugi , Misato Hirano , Satochi Nagayama
IPC分类号： A61P25/00 , A61P29/00 , A61P11/00 , A61P1/00
CPC分类号： C07D401/12 , C07D231/12
摘要： This invention provides a compound of the formula These compounds are useful for the treatment of disease conditions caused by overactivation of the VR1 receptor such as pain, or the like in mammal. This invention also provides a pharmaceutical composition comprising the above compound.
摘要翻译：本发明提供下式的化合物这些化合物可用于治疗哺乳动物VR1受体过度活化（如疼痛等）引起的疾病状况。本发明还提供了包含上述化合物的药物组合物。

86. 发明申请

US20090318702A1 PROCESS FOR PRODUCTION OF 4-OXOQUINOLINE COMPOUND 有权
标题翻译： 4-氧杂环戊烯化合物的生产方法
公开(公告)号：US20090318702A1
公开(公告)日：2009-12-24
申请号：US12281921
申请日：2007-03-06
申请人： Koji Matsuda , Koji Ando , Shigeji Ohki , Takahiro Yamasaki , Jun-ichi Hoshi
发明人： Koji Matsuda , Koji Ando , Shigeji Ohki , Takahiro Yamasaki , Jun-ichi Hoshi
IPC分类号： C07D215/233 , C07C229/34 , C07C69/612 , C07C49/303
CPC分类号： C07C229/30 , C07C65/21 , C07C69/716 , C07C229/34 , C07D215/233 , C07D215/56 , C07F7/1804 , Y02P20/55
摘要： The present invention provides a compound useful as a synthetic intermediate for an anti-HIV agent having an integrase inhibitory activity, a production method thereof, and a production method of an anti-HIV agent using the synthetic intermediate. Specifically, the present invention provides, for example, compounds represented by the formulas (6), (7-1), (7-2) and (8): wherein R is a fluorine atom or a methoxy group, R1 is a C1-C4 alkyl group, R2 is a hydroxyl-protecting group, and X2 is a halogen atom, a production method thereof, and a production method of an anti-HIV agent using the synthetic intermediate.
摘要翻译：本发明提供了可用作具有整合酶抑制活性的抗HIV剂的合成中间体的化合物，其制备方法和使用该合成中间体的抗HIV药物的制备方法。具体地说，本发明提供例如由式（6），（7-1），（7-2）和（8）表示的化合物：其中R是氟原子或甲氧基，R1是C1 -C4烷基，R2为羟基保护基，X2为卤素原子，其制造方法以及使用该合成中间体的抗HIV剂的制造方法。

87. 发明申请

US20090036684A1 METHOD FOR PRODUCING 4-OXOQUINOLINE COMPOUND 有权
标题翻译：生产4-氧杂环戊烯化合物的方法
公开(公告)号：US20090036684A1
公开(公告)日：2009-02-05
申请号：US12281889
申请日：2007-03-06
申请人： Koji Matsuda , Koji Ando , Shigeki Ohki , Jun-ichi Hoshi , Takahiro Yamasaki
发明人： Koji Matsuda , Koji Ando , Shigeki Ohki , Jun-ichi Hoshi , Takahiro Yamasaki
IPC分类号： C07D215/00 , C07C69/76 , C07C65/00 , C07C49/105
CPC分类号： C07C229/30 , C07C43/215 , C07C57/72 , C07C57/76 , C07C61/40 , C07C67/333 , C07C67/343 , C07C69/708 , C07C69/716 , C07C69/738 , C07C69/92 , C07C69/94 , C07C229/34 , C07D215/56
摘要： The present invention provides a compound useful as a synthetic intermediate for an anti-HIV agent having an integrase inhibitory activity, and a production method thereof, and a production method of an anti-HIV agent using the synthetic intermediate. Specifically, for example, a compound represented by the formula (2′): wherein R is a fluorine atom or a methoxy group, and R400 is a hydrogen atom or a C1-C4 alkyl group, or a salt thereof, and a production method thereof, and a production method of an anti-HIV agent using the synthetic intermediate.
摘要翻译：本发明提供了可用作具有整合酶抑制活性的抗HIV剂的合成中间体的化合物及其制备方法，以及使用该合成中间体的抗HIV剂的制备方法。具体而言，例如，式（2'）表示的化合物或其盐，其中R为氟原子或甲氧基，R400为氢原子或C1-C4烷基，以及使用该合成中间体的抗HIV剂的制造方法。

88. 发明申请

US20080108660A1 Benzimidazolone Carboxylic Acid Derivatives 审中-公开
标题翻译：苯并咪唑酮羧酸衍生物
公开(公告)号：US20080108660A1
公开(公告)日：2008-05-08
申请号：US11971265
申请日：2008-01-09
申请人： Koji Ando , Satoru Iguchi , Noriaki Murase , Yoshinori Murata , Toyoharu Numata , Hiroki Sone , Chikara Uchida , Tatsuo Ueki
发明人： Koji Ando , Satoru Iguchi , Noriaki Murase , Yoshinori Murata , Toyoharu Numata , Hiroki Sone , Chikara Uchida , Tatsuo Ueki
IPC分类号： A61K31/445 , C07D403/02 , A61P1/00 , C07D211/06 , A61K31/4164
CPC分类号： C07D401/12 , C07D211/26 , C07D401/06 , C07D401/14 , C07D405/06 , C07D405/14
摘要： This invention relates to compounds of the formula (I): wherein R1, R2, R3, A and m are each as described herein or a pharmaceutically acceptable salt or solvate thereof, and compositions containing such compounds and the use of such compounds in the treatment of a condition mediated by 5-HT4 receptor activity such as, but not limited to, gastroesophageal reflux disease, gastrointestinal disease, gastric motility disorder, non-ulcer dyspepsia, functional dyspepsia, irritable bowel syndrome (IBS), constipation, dyspepsia, esophagitis, gastroesophageal disease, nausea, central nervous system disease, Alzheimer's disease, cognitive disorder, emesis, migraine, neurological disease, pain, cardiovascular disorders such as cardiac failure and heart arrhythmia, diabetes and apnea syndrome.
摘要翻译：本发明涉及式（I）化合物：其中R 1，R 2，R 3，A和m各自如上所述本文或其药学上可接受的盐或溶剂合物，以及含有这些化合物的组合物以及这些化合物在治疗由5-HT 4受体活性介导的病症中的用途，所述活性例如但不限于，胃食管反流病，胃肠道疾病，胃动力障碍，非溃疡性消化不良，功能性消化不良，肠易激综合征（IBS），便秘，消化不良，食管炎，胃食管疾病，恶心，中枢神经系统疾病，阿尔茨海默病，认知障碍，呕吐，偏头痛，神经系统疾病，疼痛，心血管疾病如心力衰竭和心律失常，糖尿病和呼吸暂停综合征。

89. 发明申请

US20070273531A1 Communication antenna and pole with built-in antenna 审中-公开
标题翻译：内置天线通信天线和极
公开(公告)号：US20070273531A1
公开(公告)日：2007-11-29
申请号：US11798461
申请日：2007-05-14
申请人： Koji Ando , Takehiro Kawai
发明人： Koji Ando , Takehiro Kawai
IPC分类号： G08B13/14 , H04Q5/22
CPC分类号： H01Q3/26 , H01Q1/2216 , H01Q21/20
摘要： An antenna array part constituting a communication antenna is composed of a plurality of antenna elements. The antenna elements are arranged on an arc. This allows radio waves to be irradiated also in the exact transverse direction of the antenna array part, thereby making available the communications with an RFID tag positioned in the exact transverse direction. By shifting the phase of a radio frequency signal supplied to each antenna element or adjusting the amplitude of the radio frequency signal, it is possible to change the direction of radio beams irradiated from the antenna array part or expand the width of the radio beams thus making available with RFID tags present in a wider area.
摘要翻译：构成通信天线的天线阵列部分由多个天线元件构成。天线元件布置在弧形上。这样也能够在天线阵列部分的精确的横向上照射无线电波，从而使得与位于精确横向方向的RFID标签的通信成为可能。通过移动提供给每个天线元件的射频信号的相位或调节射频信号的幅度，可以改变从天线阵列部分照射的无线电波束的方向或扩大无线电波束的宽度，从而使得可用于存在于更广泛区域的RFID标签。

90. 发明授权

US07207325B2 Engine ignition system having noise protection circuit 有权
标题翻译：发动机点火系统具有噪声保护电路
公开(公告)号：US07207325B2
公开(公告)日：2007-04-24
申请号：US11194477
申请日：2005-08-02
申请人： Koji Ando
发明人： Koji Ando
IPC分类号： F02P3/05 , F02P3/055
CPC分类号： F02P3/0554
摘要： An ignition system for an internal combustion engine includes a switch circuit connected to an ignition coil to switch on or off current supplied to the ignition coil, a control circuit for providing a control signal for controlling the switch circuit based on the ignition signal and a protection circuit including an input terminal that receives the ignition signal, an NPN transistor having a collector connected to the input terminal, an emitter connected to a ground, a base and the collector and a parasitic diode between the collector and the emitter of the NPN transistor, in which a prescribed capacitance is formed between the base and the collector of the NPN transistor. If an electric surge that has an ascending slope comes into the input terminal, the NPN transistor to turn on to discharge the electric surge to a ground. If an electric surge that has an descending slope comes into the input terminal, it passes through the parasitic diode toward the input terminal.
摘要翻译：一种用于内燃机的点火系统包括连接到点火线圈的开关电路，以接通或断开供应到点火线圈的电流;控制电路，用于根据点火信号和保护来提供用于控制开关电路的控制信号包括接收点火信号的输入端子，具有连接到输入端子的集电极的NPN晶体管，连接到地的发射极，基极和集电极以及NPN晶体管的集电极和发射极之间的寄生二极管，其中在NPN晶体管的基极和集电极之间形成规定的电容。如果具有上升斜坡的电涌进入输入端，则NPN晶体管导通以将电涌放电到地。如果具有下降斜坡的电涌进入输入端，则其通过寄生二极管朝向输入端。

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