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71. 发明授权

US4876270B1 失效
公开(公告)号：US4876270B1
公开(公告)日：1992-06-02
申请号：US15466188
申请日：1988-02-10
申请人： HANS RUDOLF WAESPE
发明人： HANS-RUDOLF WAESPE
IPC分类号： A01N43/28 , A01N43/30 , A01N43/32 , C07D317/50 , C07D317/52 , C07D317/54 , C07D317/64 , C07D327/04 , C07D405/10
CPC分类号： C07D405/10 , A01N43/28 , A01N43/30 , A01N43/32 , C07D317/50 , C07D317/52 , C07D317/54 , C07D317/64 , C07D327/04

72. 发明授权

US5004594A Benzylidenecamphor sulphonamides derived from amino acids and their application in cosmetics, particularly as sunscreens 失效
标题翻译：衍生自氨基酸的亚苄基樟脑磺酰胺及其在化妆品中的应用，特别是作为防晒剂
公开(公告)号：US5004594A
公开(公告)日：1991-04-02
申请号：US287054
申请日：1988-12-21
申请人： Herve Richard , Madeleine Leduc , Serge Forestier , Gerard Lang
发明人： Herve Richard , Madeleine Leduc , Serge Forestier , Gerard Lang
IPC分类号： A61K8/00 , A61K8/33 , A61K8/34 , A61K8/35 , A61K8/37 , A61K8/41 , A61K8/44 , A61K8/46 , A61K8/92 , A61K8/97 , A61K31/18 , A61Q1/00 , A61Q5/00 , A61Q17/04 , C07C309/25 , C07C311/00 , C07C311/02 , C07C311/13 , C07C311/15 , C07C311/19 , C07C323/58 , C07C323/62 , C07D317/50 , C07D317/54 , C09K3/00
CPC分类号： A61Q17/04 , A61K8/466 , C07C311/13 , C07C311/19 , C07D317/54 , C07C2102/42 , Y10S424/05 , Y10S514/844 , Y10S514/845 , Y10S514/846 , Y10S514/847 , Y10S514/937 , Y10S514/938 , Y10S514/944
摘要： Cosmetic screening composition containing a benzylidene camphor sulphonamide and its use for the protection of human skin against ultraviolet radiation.
摘要翻译：含有亚苄基樟脑磺酰胺的化妆品筛选组合物及其用于保护人体皮肤免受紫外线辐射的用途。

73. 发明授权

US4971981A Substituted dioxolan and dioxan derivatives useful as pesticides 失效
公开(公告)号：US4971981A
公开(公告)日：1990-11-20
申请号：US145432
申请日：1988-01-19
申请人： Friedrich Karrer
发明人： Friedrich Karrer
IPC分类号： C07D317/18 , A01N43/28 , A01N43/30 , A01N43/32 , A01N43/40 , A01N47/12 , C07D317/22 , C07D317/50 , C07D317/54 , C07D317/64 , C07D317/72 , C07D319/12 , C07D319/14 , C07D319/16 , C07D405/04 , C07D407/04 , C07D409/04
CPC分类号： C07D405/04 , A01N43/28 , A01N43/30 , A01N43/32 , A01N43/40 , A01N47/12 , C07D317/22 , C07D317/64 , C07D317/72 , C07D319/12 , C07D407/04 , C07D409/04
摘要： Novel substituted 1,3-dioxolan and 1,4-dioxan derivatives of formula I ##STR1## in which R.sub.1, R.sub.2, R.sub.3, R.sub.4, R.sub.5 and R.sub.6 each independently of the others represents hydrogen or C.sub.1 -C.sub.4 -alkyl or, if n=1,R.sub.2 and R.sub.4 together represent one of the radicals ##STR2## R.sub.7 represents hydrogen, halogen, methyl, ethyl, C.sub.1 -C.sub.2 -alkyl substituted by 1 to 5 halogen atoms, methoxy, ethoxy or C.sub.1 -C.sub.2 -alkoxy substituted by 1 to 5 halogen atoms;R.sub.8 represents a halogen, C.sub.1 -C.sub.3 -alkyl, C.sub.1 -C.sub.3 -alkyl substituted by 1 to 7 halogen atoms, C.sub.1 -C.sub.3 -alkoxy, C.sub.1 -C.sub.3 -alkoxy substituted by 1 to 7 halogen atoms, or cyano;U represents a grouping --CH.dbd. or --N.dbd.;X represents --O--, --S-- or --N(R.sub.9)--;Y represents --O--, --S--, --S(O)--, --S(O.sub.2)--, --CH.sub.2 --, --CO-- or --N(R.sub.9)--, whereinR.sub.9 represents hydrogen, C.sub.1 -C.sub.4 -alkyl or alkylcarbonyl having a total of from 2 to 4 carbon atoms;n is a number 0 or 1;m is a number 0, 1 or 2;p is a number 1, 2 or 3; andZ represents one of the radicals ##STR3## wherein R.sub.10 represents hydrogen, methyl or ethyl;R.sub.11 represents hydrogen, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.2 -C.sub.4 -alkenyl, C.sub.2 -C.sub.4 -alkynyl, alkoxyalkyl having a total of 2 to 6 carbon atoms, C.sub.1 -C.sub.6 -alkyl substituted by 1 to 7 halogen atoms, benzyl or benzyl substituted in the nucleus by a halogen atom, by a C.sub.1 -C.sub.3 -alkyl radical or by a C.sub.1 -C.sub.3 -alkoxy radical, cyanomethyl, (C.sub.1 -C.sub.2 -alkoxy)-carbonyl or the radical --CH.sub.2 --NH--COO--(C.sub.1 -C.sub.2 -alkyl);R.sub.12 represents hydrogen, C.sub.1 -C.sub.6 -alkyl, phenyl, phenyl substituted by 1 to 3 substituents from the group consisting of halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.3 -alkyl substituted by 1 to 7 halogen atoms, C.sub.2 -C.sub.4 -alkenyl, C.sub.2 -C.sub.4 -alkynyl, C.sub.1l -C.sub.3 -alkoxy, C.sub.1 -C.sub.3 -alkoxy substituted by from 1 to 7 halogen atoms, alkoxyalkyl having a total of from 2 to 5 carbon atoms, C.sub.3 -C.sub.4 -alkenyloxy, C.sub.3 -C.sub.4 -alkynyloxy and C.sub.1 -C.sub.3 -alkylthio, or represents pyridyl, furan-2-yl, thien-2-yl or the radical ##STR4## R.sub.12 and R.sub.11 together represent one of the groups ##STR5## and R.sub.13 and R.sub.14 each independently of the other represents hydrogen, halogen or C.sub.1 -C.sub.3 -alkyl; orR.sub.13 and R.sub.14 together represent the group ##STR6## Processes for the preparation of these compounds and their use in pest control, especially for controlling insects and representatives of the order Acarina, are described.

74. 发明授权

US4806604A Photosensitive calcium chelators 失效
标题翻译：感光钙螯合剂
公开(公告)号：US4806604A
公开(公告)日：1989-02-21
申请号：US49658
申请日：1987-05-13
申请人： Roger Yonchien Tsien , Stephen R. Adams
发明人： Roger Yonchien Tsien , Stephen R. Adams
IPC分类号： G01N31/00 , C07C67/00 , C07C227/00 , C07C229/18 , C07C309/04 , C07D317/50 , C07D317/52 , C07D317/54 , C07D317/58 , C07D317/62 , C07D319/18 , C07F9/09 , C09K3/00 , G01N33/84 , C07D407/02 , C07D207/12 , C07D211/40 , C07D307/20 , C07D309/10 , C07D317/48 , C07D333/32 , C07D335/02
CPC分类号： C07D317/62
摘要： The present invention discloses a new class of calcium chelating compounds which have a decreased affinity for calcium following illumination. These new compounds contain a photolabile nitrobenzyl derivative coupled to a tetracarboxylate Ca.sup.2+ chelating parent compound having the octacoordinate chelating groups characteristic of EGTA or BAPTA. However unlike EGTA or BAPTA-like compounds, in which the two halves of the chelator are linked by a simple 1,2-ethanediyl moiety, the compounds of the present invention modify the stereochemical conformation of this linkage by adding bulky substituents or incorporating the linkage into a carbocyclic or heterocyclic ring. In a first form, the new compounds are comprised of a BAPTA-like chelator coupled to a single 2-nitrobenzyl derivative, which in turn is a photochemical precursor of a 2-nitrosobenzophenone. In a second form, the new compounds are comprised of a BAPTA-like chelator coupled to two 2-nitrobenzyl derivatives, themselves photochemical precursors of the related 2-nitrosobenzophenones.

75. 发明授权

US4803290A Nonanol/nonene antimicrobial compositions 失效
标题翻译：壬醇/壬烯抗菌组合物
公开(公告)号：US4803290A
公开(公告)日：1989-02-07
申请号：US55645
申请日：1987-05-29
申请人： Basil A. Burke , Muraleedharan Nair
发明人： Basil A. Burke , Muraleedharan Nair
IPC分类号： A01N43/30 , C07D317/50 , C07D317/54
CPC分类号： A01N43/30 , C07D317/50
摘要： Substituted 5'-nonanol/5'-nonene compounds which exhibit important antimicrobial and antifungal activity, compositions and methods of delivery against pathovars and pathogens, and methods of synthesis from commonly available reactants. The antimicrobial composition active ingredient is one or more substituted 1,2-alkylidenedioxybenzene compounds of the formula: ##STR1## where R.sub.3 is selected from 5'-nonanol and 5'-nonene, and R.sub.1 and R.sub.2 are selected from H and C.sub.1 -C.sub.5 alkyl, alkenyl and alkynyl groups. The preferred compounds are 5-(5'-hydroxy- 5'- nonanyl)-1,1-methylenedioxybenzene and 4-(5'-non-4'-enyl)-1,2-methylenedioxybenzene. Compositions including these compounds exhibit antimicrobial activity against a variety of pathogens and pathovars, e.g., Xanthomonas campestris spp. bacteria, antifungal activity against a variety of fungi and bacteria, and are highly specific, e.g., having antifungal activity against wheat powdery mildew and cucumber downy mildew, but do not affect seed germination or have appreciable herbicidal or insecticidal activity. Methods and compositions for delivery of these agents against such pathogens, and methods of chemical synthesis of the compounds are disclosed.
摘要翻译：表现出重要的抗微生物和抗真菌活性的替代的5'-壬醇/ 5'-壬烯化合物，对病原体和病原体递送的组合物和方法，以及通常可得到的反应物的合成方法。抗微生物组合物活性成分是一种或多种下式的取代的1,2-亚烷基二氧基苯化合物：其中R 3选自5'-壬醇和5'-壬烯，并且R 1和R 2选自H和C 1 -C 5 烷基，烯基和炔基。优选的化合物是5-（5'-羟基-5'-壬酰基）-1,1-亚甲二氧基苯和4-（5'-非-4'-烯基）-1,2-亚甲二氧基苯。包括这些化合物的组合物对各种病原体和病原体表现出抗菌活性，例如野油菜黄单胞菌（Xanthomonas campestris spp。）细菌，针对各种真菌和细菌的抗真菌活性，并且高度特异性，例如对小麦白粉病和黄瓜霜霉病具有抗真菌活性，但不影响种子萌发或具有明显的除草或杀虫活性。公开了用于递送这些试剂以抵抗这种病原体的方法和组合物，以及化合物的化学合成方法。

76. 发明授权

US4714786A Vinylphenol derivatives, their preparation and their use 失效
标题翻译：乙烯基苯酚衍生物，其制备及其用途
公开(公告)号：US4714786A
公开(公告)日：1987-12-22
申请号：US7586
申请日：1987-01-28
申请人： Hans-Heiner Wuesi , Bernd Janssen , Fritz-Frieder Frickel , Axel Nuerrenbach
发明人： Hans-Heiner Wuesi , Bernd Janssen , Fritz-Frieder Frickel , Axel Nuerrenbach
IPC分类号： A61K31/05 , A61K31/047 , A61K31/085 , A61K31/135 , A61K31/19 , A61K31/195 , A61K31/215 , A61K31/22 , A61K31/357 , A61K31/36 , A61P17/00 , A61P29/00 , A61P35/00 , C07C27/00 , C07C39/23 , C07C39/42 , C07C41/00 , C07C43/20 , C07C43/215 , C07C51/00 , C07C59/125 , C07C59/68 , C07C59/72 , C07C62/38 , C07C67/00 , C07C69/07 , C07C69/157 , C07C69/24 , C07C69/78 , C07C213/00 , C07C217/18 , C07D317/50 , C07D325/00
CPC分类号： C07C43/215 , C07C39/23 , C07C59/72 , C07D317/50 , C07C2102/10 , Y10S514/859 , Y10S514/863
摘要： Vinylphenol derivatives of the formula I ##STR1## where A and R.sup.1 to R.sup.7 have the meanings stated in claim 1 and in the description, and their physiologically tolerated salts, drugs prepared from these, and their use for the treatment of various disorders of the skin, the mucous membranes and the internal organs, and of rheumatic disorders.
摘要翻译：式I的乙烯基苯酚衍生物，其中A和R 1至R 7具有权利要求1和描述中所述的含义及其生理上耐受的盐，由它们制备的药物及其用于治疗皮肤各种疾病的用途，粘膜和内脏，以及风湿病。

77. 发明授权

US4661501A Certain aryl-alkane-2-pyridyloxy-phenyl derivatives having insecticidal and acaricidal activity 失效
标题翻译：某些具有杀虫和杀螨活性的芳烷基-2-吡啶氧基 - 苯基衍生物
公开(公告)号：US4661501A
公开(公告)日：1987-04-28
申请号：US833675
申请日：1986-02-26
申请人： Kiyoshi Nakatani , Satoshi Numata , Kenji Kodaka , Kengo Oda , Shiro Shiraishi , Takatoshi Udagawa
发明人： Kiyoshi Nakatani , Satoshi Numata , Kenji Kodaka , Kengo Oda , Shiro Shiraishi , Takatoshi Udagawa
IPC分类号： C07D209/48 , A01N25/02 , A01N25/14 , A01N25/30 , A01N31/08 , A01N31/14 , A01N31/16 , A01N35/00 , A01N35/04 , A01N37/32 , A01N37/34 , A01N37/38 , A01N43/00 , A01N43/06 , A01N43/08 , A01N43/30 , A01N43/38 , A01N43/40 , A01P7/04 , C07C15/12 , C07C41/00 , C07C41/18 , C07C43/02 , C07C43/205 , C07C43/215 , C07C43/257 , C07C43/263 , C07C43/275 , C07C43/29 , C07C45/00 , C07C45/62 , C07C45/72 , C07C45/74 , C07C49/213 , C07C49/223 , C07C49/255 , C07C49/76 , C07C49/84 , C07C67/00 , C07C69/94 , C07C253/00 , C07C255/00 , C07C255/37 , C07C255/53 , C07C313/00 , C07C319/20 , C07C323/09 , C07C323/18 , C07D213/64 , C07D307/34 , C07D307/38 , C07D307/56 , C07D317/50 , C07D317/54
CPC分类号： C07D317/54 , A01N31/14 , A01N31/16 , A01N35/04 , A01N37/38 , A01N43/08 , A01N43/30 , A01N43/40 , C07C323/00 , C07C43/205 , C07C43/215 , C07C43/257 , C07C45/004 , C07C45/62 , C07C45/72 , C07C45/74 , C07C49/213 , C07C49/223 , C07C49/255 , C07C49/84
摘要： The present invention relates to novel aromatic alkane derivatives represented by the following general formula (I): ##STR1## wherein Ar stands for a substituted or unsubstituted phenyl or naphthyl group, R.sup.1 stands for a methyl, ethyl or isopropyl group and R.sup.2 stands for a hydrogen atom or a methyl group, or R.sup.1 and R.sup.2 together with the carbon to which they are attached jointly represent a substituted or unsubstituted cycloalkyl group and R.sup.3, stands for a fundamental group of an alcohol which is usually used in a form of R.sup.3 OH as to natural or synthetic pyrethroids, and also to the uses of these compounds.These compounds of the present invention have excellent insecticidal and acaricidal activities while the toxicities of these compounds are very low.
摘要翻译：本发明涉及由以下通式（I）表示的新型芳族烷烃衍生物：其中Ar表示取代或未取代的苯基或萘基，R 1表示甲基，乙基或异丙基，R 2表示代表氢原子或甲基，或R 1和R 2与它们所连接的碳一起表示取代或未取代的环烷基，R3代表醇的基本基团，其通常以 R3OH关于天然或合成拟除虫菊酯，以及这些化合物的用途。本发明的这些化合物具有优异的杀虫和杀螨活性，而这些化合物的毒性非常低。

78. 发明授权

US4302615A Synthesis of 2-alkoxyphenols 失效
标题翻译： 2-烷氧基苯酚的合成
公开(公告)号：US4302615A
公开(公告)日：1981-11-24
申请号：US175475
申请日：1980-08-05
申请人： John D. Hagarty
发明人： John D. Hagarty
IPC分类号： C07C43/23 , C07D317/50 , C07C41/01 , C07C41/28
CPC分类号： C07C43/23 , C07D317/50
摘要： A reductive hydrogenolysis of a 2-substituted 1,3-benzodioxole is carried out employing a hydride-donating reducing agent system to produce a 2-alkoxyphenol.
摘要翻译：使用氢化物供给还原剂体系进行2-取代的1,3-苯并间二氧杂环戊烯的还原氢解以制备2-烷氧基苯酚。

79. 发明授权

US4212885A Insecticidal compositions containing certain tetraorganotin compounds and method for using same 失效
标题翻译：含有某些四有机锡化合物的杀虫剂组合物及其使用方法
公开(公告)号：US4212885A
公开(公告)日：1980-07-15
申请号：US966947
申请日：1978-12-06
申请人： Melvin H. Gitlitz , John E. Engelhart , Carlos M. Mery
发明人： Melvin H. Gitlitz , John E. Engelhart , Carlos M. Mery
IPC分类号： A01N55/04 , A01N57/22 , C07D213/24 , C07D213/60 , C07D317/50 , C07D319/18 , C07F7/22 , A01N9/00 , A01N9/36
CPC分类号： A01N55/04 , A01N57/22 , C07D213/24 , C07D213/60 , C07D317/50 , C07D319/18 , C07F7/2212
摘要： Many varieties of harmful insects which attack useful plant crops can be controlled by treating the plants with compositions containing at least one tetraorganotin compound wherein three of the four hydrocarbon groups bonded to the tin atom are methyl and the remaining group is substituted aromatic or heterocyclic that is either bonded directly to the tin atom or separated from the tin atom by one methylene group. These compounds exhibit unexpectedly superior insecticidal activity relative to organotin compounds containing three methyl groups and a phenyl or an alkyl-substituted phenyl group.
摘要翻译：可以通过用含有至少一种四有机锡化合物的组合物处理植物来控制许多有害昆虫品种，其中与锡原子键合的四个烃基中的三个是甲基，剩余的基团是取代的芳族或杂环，或直接与锡原子键合或与锡原子分离一个亚甲基。相对于含有三个甲基和苯基或烷基取代的苯基的有机锡化合物，这些化合物出乎意料地优异的杀虫活性。

80. 发明授权

US4158099A Production of aromatic compounds containing ethylene double bonds 失效
标题翻译：生产含乙烯双键的芳香族化合物
公开(公告)号：US4158099A
公开(公告)日：1979-06-12
申请号：US673317
申请日：1976-04-05
申请人： Adolf E. Siegrist , Peter Liechti , Hans R. Meyer , Kurt Weber
发明人： Adolf E. Siegrist , Peter Liechti , Hans R. Meyer , Kurt Weber
IPC分类号： C07C2/86 , C07C17/26 , C07C41/30 , C07C43/215 , C07D213/06 , C07D213/16 , C07D213/30 , C07D317/50 , C07D317/54 , C07D333/08 , C07D333/16 , C07C41/06
CPC分类号： C07D213/16 , C07C17/263 , C07C2/86 , C07C41/30 , C07D213/06 , C07D213/30 , C07D317/50 , C07D317/54 , C07D333/08 , C07D333/16 , C07C2103/24 , C07C2103/26 , C07C2103/50
摘要： The invention provides a new process for the manufacture of aromatic compounds which at least once contain a benzene ring of an aromatic carbocyclic ring system bonded by an ethylene double bond in conjugation with a further aromatic ring system, i.e. contain the stilbene skeleton or stilbene analogon as central structural element, as well as certain classes of new compounds of this type. The process is characterized by the reaction of a Schiff base of an aromatic aldehyde with an aromatic carbocyclic six-membered ring compound which contains one to four methyl groups bonded to ring carbon atoms of a benzene ring, which furthermore contains aromatic rings which are exclusively six-membered carbocyclic rings, and wherein those benzene rings whose methyl groups are to be caused to react are free of other substituents which contain atoms wich are replaceable by alkali metal. The reaction is carried out in the presence of (a) a strongly basic alkali compound and (b) an N-dialkyl-acylamide as solvent. The compounds obtainable according to this process show a marked fluorescence emission and therefore are suitable for all purposes where fluorescence properties are used, as for instance optical brighteners, scintillators fluorescence dyes, etc.
摘要翻译：本发明提供了一种制备芳族化合物的新方法，所述芳族化合物至少一次含有通过乙烯双键与另外的芳族环系统共轭的芳族碳环系统的苯环，即含有二苯乙烯骨架或1,2-二苯乙烯类似物作为中心结构元素，以及某些类型的这类新化合物。该方法的特征在于芳族醛的席夫碱与芳族碳环六元环化合物的反应，所述芳族碳环六元环化合物含有与苯环的环碳原子键合的一至四个甲基，其还包含仅六个芳环的芳环并且其中将要使甲基反应的那些苯环不含可被碱金属替代的原子的其它取代基。反应在（a）强碱性碱性化合物和（b）N-二烷基 - 酰基酰胺作为溶剂的存在下进行。根据该方法可获得的化合物显示出显着的荧光发射，因此适用于所有使用荧光性质的目的，例如荧光增白剂，闪烁体荧光染料等。

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