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61. 发明授权

US5744426A Substituted 3-phenylpyrazoles 失效
标题翻译：取代的3-苯基吡唑
公开(公告)号：US5744426A
公开(公告)日：1998-04-28
申请号：US750231
申请日：1996-11-26
申请人： Christoph-Sweder von dem Bussche-Hunnefeld , Ralf Klintz , Gerhard Hamprecht , Elisabeth Heistracher , Peter Schafer , Klaus Ditrich , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
发明人： Christoph-Sweder von dem Bussche-Hunnefeld , Ralf Klintz , Gerhard Hamprecht , Elisabeth Heistracher , Peter Schafer , Klaus Ditrich , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
IPC分类号： C07D231/18 , A01N43/56 , A01N47/12 , A01N47/34 , A01N47/40 , C07D231/20 , C07D231/22 , C07D401/06 , C07D401/10 , C07D403/06 , C07D403/10 , C07D405/06 , C07D405/10 , C07D409/06
CPC分类号： C07D401/10 , A01N43/56 , C07D231/22 , C07D403/10 , C07D405/10
摘要： Substituted 3-phenylpyrazoles I ##STR1## are used as herbicides.
摘要翻译： PCT No.PCT / EP95 / 02062 Sec。 371日期1996年11月26日 102（e）日期1996年11月26日PCT提交1995年5月31日PCT公布。出版物WO95 / 33728 PCT 日期1995年12月14日取代的3-苯基吡唑I被用作除草剂。

62. 发明授权

US5677283A .alpha.-heteroaryloxymethyl ketones as interleukin - 1 .beta. converting enzyme inhibitors 失效
标题翻译： α-杂环氧基甲基酮作为白细胞介素-1β转换酶抑制剂
公开(公告)号：US5677283A
公开(公告)日：1997-10-14
申请号：US732173
申请日：1996-10-16
申请人： Roland E. Dolle , Jasbir Singh , David A. Whipple , Catherine Prouty , Prasad V. Chaturvedula , Stanley J. Schmidt , Mohamed M. A. Awad , Denton W. Hoyer , Tina Morgan Ross
发明人： Roland E. Dolle , Jasbir Singh , David A. Whipple , Catherine Prouty , Prasad V. Chaturvedula , Stanley J. Schmidt , Mohamed M. A. Awad , Denton W. Hoyer , Tina Morgan Ross
IPC分类号： C12N9/99 , A61K31/397 , A61K31/415 , A61K31/42 , A61K31/421 , A61K31/47 , A61K31/472 , A61K31/535 , A61K31/5375 , A61K31/5377 , A61K31/55 , A61K38/00 , A61P29/00 , A61P37/00 , A61P43/00 , C07D205/04 , C07D207/38 , C07D209/12 , C07D215/14 , C07D217/16 , C07D223/08 , C07D231/20 , C07D231/22 , C07D261/12 , C07D263/06 , C07D265/06 , C07D265/30 , C07D311/46 , C07D311/50 , C07D311/56 , C07D401/12 , C07D409/12 , C07D413/04 , C07D417/12 , C07D453/02 , C07D471/04 , C07K5/02 , C07K5/06 , C07K5/062 , C07K5/078 , C07K5/08 , C07K5/083 , C07K5/09 , C07K5/097 , C07D231/04 , C07K5/00
CPC分类号： C07D401/12 , C07D207/38 , C07D231/20 , C07D231/22 , C07D261/12 , C07D311/46 , C07D311/56 , C07D409/12 , C07D413/04 , C07D417/12 , C07D453/02 , C07K5/0202 , A61K38/00
摘要： Compounds which Inhibit interleukin-1.beta. protease activity, pharmaceutical compositions containing the compounds and methods using the compounds are provided. The compounds have the formula ##STR1## wherein n is 0-2; each AA is Independently L-valine or L-alanine; R.sub.1 is selected from the group consisting of N-�4(N,N-dimethylaminomethyl)!benzoyl, N-benzoyloxycarbonyl, N-methyl-N-�4-(pyridyl)methyl!, N-�4-(pyddyl)methyl!carbonyl, N-3-(piperidinopropionyl), N-�4-(morpholinoethoxy)benzoyl, N-2-(quinuclidinyl)carbonyl, N-(3-pyridyl)methoxy carbonyl, N-(2-pyddyl)methoxy carbonyl, N-methyl-N-benzyl carbonyl, N-methyl-N-�2-(4-pyridyl)ethyl!carbonyl, and N-(N-phenylpiperazino) carbonyl; and R.sub.8, R.sub.9 and R.sub.10 are as defined below.
摘要翻译：提供了抑制白细胞介素-1β蛋白酶活性的化合物，含有这些化合物的药物组合物和使用该化合物的方法。化合物具有式（1）其中n为0-2; 每个AA是独立的L-缬氨酸或L-丙氨酸; R1选自N- [4（N，N-二甲基氨基甲基）]苯甲酰基，N-苯甲酰氧基羰基，N-甲基-N- [4-（吡啶基）甲基]，N- [4-（吡啶基）甲基 ]羰基，N-3-（哌啶基丙酰基），N- [4-（吗啉代乙氧基）苯甲酰基，N-2-（奎宁环基）羰基，N-（3-吡啶基）甲氧基羰基，N-（2- N-甲基-N-苄基羰基，N-甲基-N- [2-（4-吡啶基）乙基]羰基和N-（N-苯基哌嗪基）羰基; 并且R 8，R 9和R 10如下所定义。

63. 发明授权

US5663365A Process for the preparation of pyrazolones 失效
标题翻译：制备吡唑啉酮的方法
公开(公告)号：US5663365A
公开(公告)日：1997-09-02
申请号：US739695
申请日：1996-10-29
申请人： Yasuo Yamamoto , Naoki Shirakawa , Shinichi Takano , Yoshio Kawai
发明人： Yasuo Yamamoto , Naoki Shirakawa , Shinichi Takano , Yoshio Kawai
IPC分类号： C07D231/20 , C07D231/22
CPC分类号： C07D231/22 , C07D231/20
摘要： A process for the preparation of pyrazolone derivatives represented by the general formula ##STR1## wherein R is a hydrogen atom, an alkyl group, an allyl group, an aryl group or an aralkyl group, and R.sub.1 and R.sub.2 are, respectively, a hydrogen atom, an alkyl group or a phenyl group which may have a substituent, comprising reacting a 2,3-dihalocarboxylic acid derivative or a 2-haloacrylic acid derivative with a hydrazine derivative. A pyrazolone or 1-substituted-3-pyrazolones useful as intermediate starting materials for the synthesis of agricultural chemicals, medicine and chemical compounds can be easily and cheaply prepared from widely used industrial starting materials.
摘要翻译：制备由通式“IMAGE”表示的吡唑啉酮衍生物的方法，其中R是氢原子，烷基，烯丙基，芳基或芳烷基，R 1和R 2分别是氢原子，可以具有取代基的烷基或苯基，包括使2,3-二卤代羧酸衍生物或2-卤代丙烯酸衍生物与肼衍生物反应。用作合成农药，药物和化合物的中间原料的吡唑啉酮或1-取代-3-吡唑啉酮可以从广泛使用的工业起始原料中容易地和廉价地制备。

64. 发明授权

US5502069A 1-thiocarbamoyl-5-hydroxy-pyrazoles as microbicides 失效
标题翻译： 1-硫代氨基甲酰基-5-羟基 - 吡唑作为杀微生物剂
公开(公告)号：US5502069A
公开(公告)日：1996-03-26
申请号：US302076
申请日：1994-09-07
申请人： Klaus Sasse , Peter Wachtler , Georg-Wilhelm Ludwig , Wilfried Paulus
发明人： Klaus Sasse , Peter Wachtler , Georg-Wilhelm Ludwig , Wilfried Paulus
IPC分类号： A01N47/38 , C07D231/14 , C07D231/20 , C07D231/22 , C07D231/28 , C07D231/54 , C07D231/56 , A01N43/56
CPC分类号： C07D231/56 , C07D231/22 , C07D231/28
摘要： 1-Thiocarbamoyl-5-hydroxy-pyrazoles have a microbicidal action and are therefore suitable for use for the preservation of materials. Since, in contrast to other microbicides, they are ecologically acceptable and do not discolour plastics, paints and paint films, they are particularly recommended for use in these substances.
摘要翻译： 1-硫代氨基甲酰基-5-羟基 - 吡唑具有杀微生物作用，因此适用于保存材料。由于与其他杀微生物剂相反，它们在生态上是可以接受的，并且不会使塑料，油漆和油漆膜变色，因此特别推荐用于这些物质。

65. 发明授权

US5374644A Fungicides 失效
标题翻译：杀菌剂
公开(公告)号：US5374644A
公开(公告)日：1994-12-20
申请号：US815588
申请日：1991-12-31
申请人： John M. Clough , Christopher R. A. Godfrey , Ian T. Streeting
发明人： John M. Clough , Christopher R. A. Godfrey , Ian T. Streeting
IPC分类号： A01N43/824 , A01N43/76 , A01N43/90 , C07D207/34 , C07D207/36 , C07D209/30 , C07D209/34 , C07D209/36 , C07D231/18 , C07D231/20 , C07D231/22 , C07D231/56 , C07D233/70 , C07D233/84 , C07D249/04 , C07D249/12 , C07D257/04 , C07D261/10 , C07D261/12 , C07D261/20 , C07D263/38 , C07D263/40 , C07D263/42 , C07D263/46 , C07D263/58 , C07D275/00 , C07D275/02 , C07D275/03 , C07D275/04 , C07D277/20 , C07D277/32 , C07D277/34 , C07D277/36 , C07D277/58 , C07D277/68 , C07D285/08 , C07D285/12 , C07D285/13 , C07D307/58 , C07D307/64 , C07D307/82 , C07D307/83 , C07D333/32 , C07D333/34 , C07D333/42 , C07D333/44 , C07D333/62 , C07D333/64 , C07D513/04 , C03D263/58
CPC分类号： C07D231/56 , A01N43/90 , C07D207/36 , C07D209/30 , C07D209/34 , C07D209/36 , C07D231/18 , C07D231/22 , C07D261/10 , C07D261/12 , C07D261/20 , C07D263/40 , C07D263/42 , C07D263/58 , C07D275/03 , C07D275/04 , C07D277/58 , C07D285/13 , C07D307/58 , C07D307/64 , C07D307/82 , C07D307/83 , C07D333/32 , C07D333/34 , C07D333/44 , C07D333/62 , C07D333/64 , C07D513/04
摘要： Compounds of formula: ##STR1## and stereoisomers thereof, wherein X, Y and Z, which are the same or different, are hydrogen, halogen, hydroxy, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted aryl, optionally substituted alkynyl, optionally substituted alkoxy, optionally substituted aryloxy, optionally substituted aralkyl, optionally substituted arylalkoxy, optionally substituted aryloxyalkyl, optionally substituted acyloxy, optionally substituted amino, acylamino, nitro, cyano, --CO.sub.2 R.sup.1, --CONR.sup.2 R.sup.3, or --COR.sup.4 ; or X and Y, when they are in adjacent positions of the phenyl ring, join to form a fused ring, either aromatic or aliphatic, optionally containing one or more heteroatoms; W is a C-linked optionally substituted five membered heterocylic ring, containing one to four hetero-atoms, which are the same or different, and which are nitrogen, sulphur or oxygen and wherein adjacent substituents may together form a fused aromatic or hetero-aromatic ring; A is an oxygen or sulphur atom; and R.sup.1, R.sup.2, R.sup.3 and R.sup.4, which are the same or different, are hydrogen, alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, optionally substituted aryl or optionally substituted aralkyl; and metal complexes thereof. The compounds are useful as fungicides and also insecticides.
摘要翻译：式（I）化合物及其立体异构体，其中X，Y和Z相同或不同，为氢，卤素，羟基，任选取代的烷基，任选取代的烯基，任选取代的芳基，任选取代的炔基任选取代的芳氧基，任选取代的芳基烷氧基，任选取代的芳氧基烷基，任选取代的酰氧基，任选取代的氨基，酰氨基，硝基，氰基，-CO 2 R 1，-CONR 2 R 3或-COR 4; 或X和Y，当它们在苯环的相邻位置时，连接形成任选含有一个或多个杂原子的芳环或脂族稠环; W是C连接的任选取代的五元杂环，其含有一至四个杂原子，它们相同或不同，并且是氮，硫或氧，并且其中相邻的取代基可以一起形成稠合芳族或杂芳族环; A是氧或硫原子; R 1，R 2，R 3和R 4相同或不同，为氢，烷基，环烷基，环烷基烷基，烯基，炔基，任选取代的芳基或任选取代的芳烷基; 及其金属络合物。这些化合物可用作杀真菌剂和杀虫剂。

66. 发明授权

US5342837A Fungicides dizinyl oxime ethers 失效
标题翻译：杀真菌剂二嗪基肟醚
公开(公告)号：US5342837A
公开(公告)日：1994-08-30
申请号：US87706
申请日：1993-01-22
申请人： John M. Clough , Christopher R. A. Godfrey , Paul J. de Fraine , Ian R. Matthews
发明人： John M. Clough , Christopher R. A. Godfrey , Paul J. de Fraine , Ian R. Matthews
IPC分类号： A01N37/18 , A01N37/50 , A01N43/06 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/74 , C07C251/60 , C07C255/62 , C07C317/28 , C07C323/47 , C07D207/06 , C07D207/32 , C07D207/335 , C07D213/26 , C07D213/53 , C07D213/61 , C07D213/63 , C07D213/64 , C07D213/84 , C07D215/18 , C07D215/50 , C07D231/20 , C07D231/22 , C07D233/54 , C07D237/14 , C07D239/26 , C07D239/34 , C07D239/38 , C07D239/42 , C07D239/52 , C07D241/12 , C07D241/18 , C07D241/24 , C07D249/08 , C07D251/02 , C07D263/14 , C07D277/28 , C07D277/54 , C07D277/64 , C07D307/52 , C07D307/81 , C07D307/82 , C07D333/20 , C07D333/22 , C07D333/28 , C07D333/38 , C07D333/58 , C07D521/00 , C07F9/40 , A61K31/50 , A61K31/505 , C07D237/06 , C07D239/24
CPC分类号： C07D207/335 , A01N37/50 , A01N43/06 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/74 , C07C251/60 , C07D213/26 , C07D213/53 , C07D213/61 , C07D213/63 , C07D213/64 , C07D213/84 , C07D231/22 , C07D239/26 , C07D239/34 , C07D239/38 , C07D239/42 , C07D239/52 , C07D241/12 , C07D241/18 , C07D241/24 , C07D277/54 , C07D307/52 , C07D307/82 , C07D333/22 , C07D333/28 , C07D333/58 , C07C2101/14
摘要： Fungicidal compounds having the formula (I): ##STR1## and stereoisomers thereof, wherein A is hydrogen, halo, hydroxy, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-4 haloalkyl, C.sub.1-4 haloalkoxy, C.sub.1-4 alkylcarbonyl, C.sub.1-4 alkoxycarbonyl, phenoxy, nitro or cyano; R.sup.1 and R.sup.2, which may be the same or different, are hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted heterocyclylalkyl, optionally substituted cycloalkylalkyl, optionally substituted aralkyl, optionally substituted aryloxyalkyl, optionally substituted heterocyclyloxyalkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted alkoxy, optionally substituted aryl, optionally substituted heterocyclyl, optionally substituted aryloxy, optionally substituted heterocyclyloxy, nitro halo cyano, --NR.sup.3 R.sup.4, --CO.sub.2 R.sup.3, --CONR.sup.3 R.sup.4, --COR.sup.3, --S(O).sub.n R.sup.3 wherein is 0, 1 or 2, (CH.sub.2).sub.m PO(OR.sup.3).sub.2 wherein m is 0 or 1, or R.sup.1 and R.sup.2 join to form a carbocyclic or heterocyclic ring system; R.sup.3 and R.sup.4, which are the same or different, are hydrogen, optionally substituted alkyl, optionally substituted aralkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted aryl or optionally substituted heteroaryl, or R.sup.3 and R.sup.4 join to form an optionally substituted heterocyclic ring; and R.sup.5 and R.sup.6 are independently hydrogen or C.sub.1-4 alkyl.
摘要翻译：具有式（I）的杀真菌化合物及其立体异构体，其中A为氢，卤素，羟基，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基，C 1-4卤代烷氧基， 4-烷基羰基，C 1-4烷氧基羰基，苯氧基，硝基或氰基; R 1和R 2可以相同或不同，为氢，任选取代的烷基，任选取代的环烷基，任选取代的杂环基烷基，任选取代的环烷基烷基，任选取代的芳烷基，任选取代的芳氧基烷基，任选取代的杂环基烷基，任选取代的烯基，任选取代的炔基，任选取代的烷氧基，任选取代的芳基，任选取代的杂环基，任选取代的芳氧基，任选取代的杂环氧基，硝基卤代氰基，-NR 3 R 4，-CO 2 R 3，-CONR 3 R 4，-COR 3，-S（O）n R 3，其中0,1或2 ，（CH 2）m PO（OR 3）2，其中m为0或1，或R 1和R 2连接形成碳环或杂环系; R 3和R 4相同或不同，为氢，任选取代的烷基，任选取代的芳烷基，任选取代的烯基，任选取代的炔基，任选取代的芳基或任选取代的杂芳基，或R 3和R 4连接形成任选取代的杂环 ; 并且R 5和R 6独立地是氢或C 1-4烷基。

67. 发明授权

US5202442A Process for preparing pyrazolecarboxylic acid compounds 失效
标题翻译：吡唑羧酸化合物的制备方法
公开(公告)号：US5202442A
公开(公告)日：1993-04-13
申请号：US722533
申请日：1991-06-27
申请人： Shinichiro Takigawa , Shuzo Shinke
发明人： Shinichiro Takigawa , Shuzo Shinke
IPC分类号： C07D231/14 , C07D231/16 , C07D231/18 , C07D231/22 , C07D231/38 , C07D401/04
CPC分类号： C07D231/38 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/22 , C07D401/04
摘要： A process for preparing a pyrazolecarboxylic acid compound of the formula (II): ##STR1## wherein Y and Z each represent a hydrogen, a halogen, a nitro, a cyano, COOR.sub.1, NR.sub.1 R.sub.2, CONR.sub.1 R.sub.2, SR.sub.1, SO.sub.2 NR.sub.1 R.sub.2, SO.sub.2 R.sub.3, R.sub.3 CO, OR.sub.4, CHX.sub.2 or CX.sub.3 ; A represents a hydrogen, an alkyl having 2 to 4 carbons, a phenyl, a pyridyl or OR.sub.5 ; where R.sub.1 and R.sub.2 each represent a hydrogen or an alkyl having 1 to 10 carbons; R.sub.3 represents an alkyl having 1 to 10 carbons; R.sub.4 represents a hydrogen, an alkyl having 1 to 10 carbons, a phenyl, CHF.sub.2, CF.sub.3 or CF.sub.3 CH.sub.2 ; R.sub.5 represents an alkyl having 1 to 10 carbons; and X represents a halogen, which comprises oxidizing a pyrazole compound of the formula (I): ##STR2## wherein Y, Z and A have the same meanings as above, by contacting the compound of formula (I) with an oxygen-containing gas in the presence of a metal catalyst at 20.degree. to 200.degree. C., the partial pressure of the oxygen-containing gas being from atmospheric pressure to 80 kg/cm.sup.2 and the metal catalyst is in an amount of 0.1 to 20 gram-atom based on 100 moles of the compound of formula (I) and is at least one compound selected from the group consisting of iron compounds, cobalt compounds, nickel compounds, manganese compounds, cerium compounds and zirconium compounds.
摘要翻译：制备式（II）的吡唑甲酸化合物的方法：其中Y和Z各自表示氢，卤素，硝基，氰基，COOR1，NR1R2，CONR1R2，SR1，SO2NR1R2，SO2R3 ，R3CO，OR4，CHX2或CX3; A表示氢，具有2至4个碳的烷基，苯基，吡啶基或OR 5; 其中R 1和R 2各自表示氢或具有1至10个碳的烷基; R3表示碳原子数1〜10的烷基， R4表示氢，碳原子数1〜10的烷基，苯基，CHF 2，CF 3或CF 3 CH 2; R5表示碳原子数1〜10的烷基，并且X表示卤素，其包括使式（I）的吡唑化合物氧化：其中Y，Z和A具有与上述相同的含义，通过使式（I）化合物与氧在金属催化剂存在下，在20〜200℃下，含氧气体的分压为大气压至80kg / cm2，金属催化剂的量为0.1〜20g - 原子，基于100摩尔式（I）化合物，并且是至少一种选自铁化合物，钴化合物，镍化合物，锰化合物，铈化合物和锆化合物的化合物。

68. 发明授权

US5174808A Herbicidal pyrazolin-5-one derivatives, compositions and use 失效
标题翻译：除草剂吡唑啉-5-酮衍生物，组合物和用途
公开(公告)号：US5174808A
公开(公告)日：1992-12-29
申请号：US610597
申请日：1990-11-08
申请人： Heinz-Jurgen Wroblowsky , Peter Babczinski , Klaus Lurssen , Hans-Joachim Santel , Robert R. Schmidt
发明人： Heinz-Jurgen Wroblowsky , Peter Babczinski , Klaus Lurssen , Hans-Joachim Santel , Robert R. Schmidt
IPC分类号： A01N43/56 , C07D231/22 , C07D401/04 , C07D405/04 , C07D405/06 , C07D409/04 , C07D409/06
CPC分类号： C07D401/04 , C07D231/22 , C07D405/04 , C07D409/04 , C07D409/06
摘要： Herbicidal pyrazolin-5-one derivatives of the formula ##STR1## in which R.sup.1 represents alkyl, cycloalkyl, halogenoalkyl, alkenyl, alkynyl, alkenyl or alkynyl substituted by optionally substituted phenyl, halogenoalkenyl, alkoxy, alkoxyalkyl, alkylthioalkyl, alkylsulphonylalkyl, alkylsulphinylalkyl, alkoxycarbonylalkyl, in each case optionally substituted aryl, aralkyl, aryloxyalkyl or arylthioalkyl, an optionally substituted heterocycle, heterocyclylalkyl or the --NH--CO--R.sup.3 or --CO--O--R.sup.4 groups, in which R.sup.3 and R.sup.4 in each case independently of one another represent alkyl or aryl,R.sup.2 represents hydrogen, alkyl, cycloalkyl, halogenoalkyl, alkenyl, alkinyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, alkylsulphonylalkyl, alkylsuslphinylalkyl or alkoxycarbonylalkyl andAr represents optionally substituted aryl or a heterocycle which is optionally substituted and optionally fused,excluding the compounds 1-(3-chlorophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazoline-5-one, 1-(4-chlorophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazolin-5-one, 1-(4-trifluoronethylphenyl-3-methylthiomethyl-4-(N-hydroxyaminomethylidene))-pyrazolin-5-one and 1-(4-n-nitrophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazolin-5-one.
摘要翻译：式（Ⅰ）的除草吡唑啉-5-酮衍生物，其中R 1表示被任选取代的苯基，卤代烯基，烷氧基，烷氧基烷基，烷基硫代烷基，烷基磺酰基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷氧基羰基烷基，在各种情况下均为任选取代的芳基，芳烷基，芳氧基烷基或芳硫基烷基，任选取代的杂环，杂环基烷基或-NH-CO-R 3或-CO-O-R 4基团，其中R 3和R 4各自独立地为另一个代表烷基或芳基，R 2表示氢，烷基，环烷基，卤代烷基，烯基，炔基，卤代烯基，烷氧基烷基，烷基硫代烷基，烷基磺酰基烷基，烷基磺酰基烷基或烷氧基羰基烷基，Ar表示任选取代的芳基或任选被取代和任选稠合的杂环，化合物1-（3-氯苯基）-3-甲硫基甲基-4-（N-羟基氨基亚甲基） - 吡唑并-5-酮， 1-（4-氯苯基）-3-甲基硫代甲基-4-（N-羟基氨基亚甲基） - 吡唑啉-5-酮，1-（4-三氟甲基苯基-3-甲硫基甲基-4-（N-羟基氨基甲基二烯） 5-（1-硝基苯基）-3-甲基硫代甲基-4-（N-羟基氨基亚甲基） - 对]吡唑-5-酮。

69. 发明授权

US5112384A 3-(substituted phenyl) pyrazole derivatives herbicidal composition containing the same and method of controlling weeds using said composition 失效
标题翻译： 3-（取代的苯基）吡唑衍生物含有它们的除草组合物和使用合成组合物控制的方法
公开(公告)号：US5112384A
公开(公告)日：1992-05-12
申请号：US659729
申请日：1991-02-25
申请人： Yuzo Miura , Masanobu Ohnishi , Tsutomu Mabuchi , Isao Yanai
发明人： Yuzo Miura , Masanobu Ohnishi , Tsutomu Mabuchi , Isao Yanai
IPC分类号： A01N43/56 , C07D231/22
CPC分类号： C07D231/22 , A01N43/56
摘要： A 3-(substituted phenyl)pyrazole derivative or a salt thereof, the derivative being represented by the general formula ##STR1## wherein, X denotes halogen, R.sup.1 denotes lower alkyl, R.sup.2 denotes halogen and R.sup.3 denotes lower alkyl, lower alkenyl or benzyl group, a process for producing said pyrazole derivative, a herbicidal composition containing said pyrazole derivative as an active ingredient, and a method of controlling weeds by applying said composition.

70. 发明授权

US5032165A 3-(substituted phenyl)pyrazole derivatives, salts thereof, and herbicides therefrom 失效
标题翻译： 3-（取代苯基）吡唑衍生物，其盐，和除草剂
公开(公告)号：US5032165A
公开(公告)日：1991-07-16
申请号：US400791
申请日：1989-08-30
申请人： Yuzo Miura , Tsutomu Mabuchi , Mitsuru Kajioka , Isao Yanai
发明人： Yuzo Miura , Tsutomu Mabuchi , Mitsuru Kajioka , Isao Yanai
IPC分类号： C07D231/16 , A01N20060101 , A01N43/56 , C07D20060101 , C07D231/12 , C07D231/18 , C07D231/20 , C07D231/22 , C07D231/38 , C07D405/12 , C07F7/08 , C07F9/6503
CPC分类号： C07F7/0812 , A01N43/56 , C07D231/18 , C07D231/22 , C07F9/65033
摘要： There are disclosed a (3-substituted phenyl)pyrazole derivative represented by the general formula ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4 and X are various substituents and a salt thereof, and its production process. Said pyrazole derivative or its salt is useful as a herbicide for controlling various injurious weeds.

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