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51. 发明授权

US07608564B2 3-heterocyclyl-substituted benzoyl derivatives 有权
标题翻译： 3-杂环基取代的苯甲酰基衍生物
公开(公告)号：US07608564B2
公开(公告)日：2009-10-27
申请号：US11739928
申请日：2007-04-25
申请人： Wolfgang von Deyn , Regina Luise Hill , Uwe Kardorff , Ernst Baumann , Stefan Engel , Guido Mayer , Matthias Witschel , Michael Rack , Norbert Götz , Joachim Gebhardt , Ulf Miβlitz , Helmut Walter , Karl-Otto Westphalen , Martina Otten , Joachim Rheinheimer
发明人： Wolfgang von Deyn , Regina Luise Hill , Uwe Kardorff , Ernst Baumann , Stefan Engel , Guido Mayer , Matthias Witschel , Michael Rack , Norbert Götz , Joachim Gebhardt , Ulf Miβlitz , Helmut Walter , Karl-Otto Westphalen , Martina Otten , Joachim Rheinheimer
IPC分类号： A01N43/76 , C07D263/02
CPC分类号： C07D413/10 , A01N43/76 , A01N43/80 , C07D231/20 , C07D261/04 , C07D261/20 , C07D403/12 , C07D417/10
摘要： Benzoyl derivatives of the formula I where the variables have the following meanings: R1, R2 are hydrogen, nitro, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl or C1-C6-haloalkylsulfonyl; R3 is hydrogen, halogen or alkyl; R4, R5 are hydrogen, halogen, cyano, nitro, alkyl, alkoxy, alkylthio, dialkylamino, phenyl or carbonyl, it being possible for the 6 last-mentioned radicals to be substituted; X is O, S, NR9, CO or CR10R11; Y is O, S, NR12, CO or CR13R14; R15 is pyrazole which is unsubstituted or substituted, linked in the 4-position and has attached to it in the 5-position a hydroxyl or sulfonyloxy radical; and the agriculturally useful salts thereof; processes and intermediates for the preparation of the 3-heterocyclyl-substituted benzoyl derivatives; compositions comprising them; and the use of these derivatives or compositions comprising them for controlling undesirable plants.
摘要翻译：式I的苯甲酰基衍生物，其中变量具有以下含义：R 1，R 2是氢，硝基，卤素，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基或C 1 -C 6卤代烷基磺酰基; R3是氢，卤素或烷基; R4，R5是氢，卤素，氰基，硝基，烷基，烷氧基，烷硫基，二烷基氨基，苯基或羰基，最后提到的6个基团可以被取代; X是O，S，NR 9，CO或CR 10 R 11; Y为O，S，NR 12，CO或CR 13 R 14; R15是未取代或取代的吡唑，其在4-位连接并在5-位上连接羟基或磺酰氧基; 及其农业上有用的盐; 用于制备3-杂环基取代的苯甲酰基衍生物的方法和中间体; 包含它们的组合物; 以及包含它们的这些衍生物或组合物用于控制不期望的植物的用途。

52. 发明申请

US20080039327A1 3-HETEROCYCLYL-SUBSTITUTED BENZOYL DERIVATIVES 有权
标题翻译： 3-杂环取代的苯甲酰基衍生物
公开(公告)号：US20080039327A1
公开(公告)日：2008-02-14
申请号：US11739928
申请日：2007-04-25
申请人： Wolfgang Deyn , Regina Hill , Uwe Kardorff , Ernst Baumann , Stefan Engel , Guido Mayer , Matthias Witschel , Michael Rack , Norbert Gotz , Joachim Gebhardt , Ulf MiBlitz , Helmut Walter , Karl-Otto Westphalen , Martina Otten , Joachim Rheinheimer
发明人： Wolfgang Deyn , Regina Hill , Uwe Kardorff , Ernst Baumann , Stefan Engel , Guido Mayer , Matthias Witschel , Michael Rack , Norbert Gotz , Joachim Gebhardt , Ulf MiBlitz , Helmut Walter , Karl-Otto Westphalen , Martina Otten , Joachim Rheinheimer
IPC分类号： A01N43/80 , A01P13/00 , C07D261/04
CPC分类号： C07D413/10 , A01N43/76 , A01N43/80 , C07D231/20 , C07D261/04 , C07D261/20 , C07D403/12 , C07D417/10
摘要： Benzoyl derivatives of the formula I where the variables have the following meanings: R1, R2 are hydrogen, nitro, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl or C1-C6-haloalkylsulfonyl; R3 is hydrogen, halogen or alkyl; R4, R5 are hydrogen, halogen, cyano, nitro, alkyl, alkoxy, alkylthio, dialkylamino, phenyl or carbonyl, it being possible for the 6 last-mentioned radicals to be substituted; X is O, S, NR9, CO or CR10R11; Y is O, S, NR12, CO or CR13R14; R15 is pyrazole which is unsubstituted or substituted, linked in the 4-position and has attached to it in the 5-position a hydroxyl or sulfonyloxy radical; and the agriculturally useful salts thereof; processes and intermediates for the preparation of the 3-heterocyclyl-substituted benzoyl derivatives; compositions comprising them; and the use of these derivatives or compositions comprising them for controlling undesirable plants.
摘要翻译：式I的苯甲酰基衍生物，其中变量具有以下含义：R 1，R 2是氢，硝基，卤素，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基或C 1 -C 6 - 卤代烷基磺酰基; R 3是氢，卤素或烷基; R 4，R 5是氢，卤素，氰基，硝基，烷基，烷氧基，烷硫基，二烷基氨基，苯基或羰基，对于最后提到的6个基团是可能的被替代 X是O，S，NR 9，CO或CR 10 R 11， Y是O，S，NR 12，CO或CR 13 R 14; R 15是未取代或取代的吡唑，其在4-位连接并在5-位上连接羟基或磺酰氧基; 及其农业上有用的盐; 用于制备3-杂环基取代的苯甲酰基衍生物的方法和中间体; 包含它们的组合物; 以及包含它们的这些衍生物或组合物用于控制不期望的植物的用途。

53. 发明授权

US06716989B2 Preparation of 2-alkyl-3-(4,5-dihydroisoxazol-3-yl) halobenzenes 有权
标题翻译： 2-烷基-3-（4,5-二氢异恶唑-3-基）卤代苯的制备
公开(公告)号：US06716989B2
公开(公告)日：2004-04-06
申请号：US10462903
申请日：2003-06-18
申请人： Michael Rack , Norbert Götz , Helmut Hagen , Wolfgang von Deyn , Ernst Baumann , Rene Lochtman , Joachim Gebhardt
发明人： Michael Rack , Norbert Götz , Helmut Hagen , Wolfgang von Deyn , Ernst Baumann , Rene Lochtman , Joachim Gebhardt
IPC分类号： C07D26118
CPC分类号： C07D261/04
摘要： A novel process for preparing the compounds of the formula I where: n is 0, 1 or 2; R1, R2 are C1-C6-alkyl; R3, R4, R5 are hydrogen or C1-C6-alkyl, or R4 and R5 together form a bond; R6 is Cl, Br, which comprises a synthesis sequence starting from 1,2-dialkylbenzenes of the formula II with subsequent halogenation to give 3,6-dihalo-1,2-dialkylbenzenes, haloalkylation to give benzyl bromides, oxidation to give benzaldehydes, oximation, reaction with alkenes to give isoxazoles, conversion into thioethers and, if appropriate, oxidation to give sulfenyl or sulfonyl derivatives of the formula I.
摘要翻译：一种制备式I化合物的新方法，其中n为0,1或2; R 1，R 2为C 1 -C 6 - 烷基; R 3，R 4，R 5，或者R 4和R 5一起形成键; R 6是Cl，Br，其包含从式II的1,2-二烷基苯开始的合成序列，随后卤化得到3,6-二卤代-1,2-二烷基苯，卤代烷基化得到苄基溴，氧化得到苯甲醛，肟化，与烯烃反应得到异恶唑，转化成硫醚，如果合适，氧化得到亚硫酰基或磺酰基衍生物的式I。

54. 发明授权

US06407245B2 Substituted thiopyridines 失效
标题翻译：取代的硫代吡啶
公开(公告)号：US06407245B2
公开(公告)日：2002-06-18
申请号：US09791688
申请日：2001-02-26
申请人： Gerhard Hamprecht , Joachim Gebhardt , Heinz Isak , Michael Rack , Joachim Rheinheimer , Peter Schäfer
发明人： Gerhard Hamprecht , Joachim Gebhardt , Heinz Isak , Michael Rack , Joachim Rheinheimer , Peter Schäfer
IPC分类号： C07D21371
CPC分类号： C07D213/71
摘要： Substituted thiopyridines of the general formula I where n is 1 or 2; R1 is chlorine, C1-C3-fluoroalkyl, nitro or methylsulfonyl; R2 is a C1-C10-alkyl, C2-C10-alkenyl or C2-C10-alkynyl radical, in each case unsubstituted or substituted by halogen, C1-C4-alkoxy, C1-C4-alkoxycarbonyl, di-(C1-C4-alkylamino)carbonyl, cyano or nitro, a C3-C8-cycloalkyl radical, or a C1-C4-alkyl-enephenyl, phenyl or naphthyl radical which is unsubstituted or substituted in the phenyl moiety by halogen, C1-C3-alkyl, C1-C3-alkoxy, trifluoromethyl, cyano or nitro.
摘要翻译：通式Iwheren的取代的硫代吡啶为1或2; R 1为氯，C 1 -C 3 - 氟代烷基，硝基或甲基磺酰基; R 2为C 1 -C 10 - 烷基，C 2 -C 10 - 烯基或C 2 -C 10 - 炔基 C 1 -C 4 - 烷氧基羰基，C 1 -C 4 - 烷基氨基羰基，氰基或硝基，C 3 -C 8环烷基或C 1 -C 4 - 烷基 - 苯基，苯基或萘基，其未被取代或在苯基部分被卤素，C 1 -C 3 - 烷基，C 1 -C 3 - 烷氧基，三氟甲基，氰基或硝基取代。

55. 发明授权

US06169184A Process for the production of substituted phenylpyridines 失效
标题翻译：制备取代苯基吡啶的方法
公开(公告)号：US06169184A
公开(公告)日：2001-01-02
申请号：US09254456
申请日：1999-03-10
申请人： Gerhard Hamprecht , Joachim Gebhardt , Heinz Isak , Michael Rack , Joachim Rheinheimer , Peter Sch{umlaut over (a)}fer
发明人： Gerhard Hamprecht , Joachim Gebhardt , Heinz Isak , Michael Rack , Joachim Rheinheimer , Peter Sch{umlaut over (a)}fer
IPC分类号： C02D2472
CPC分类号： C07D213/62
摘要： A process for preparing substituted phenylpyridines of the formula I comprises reacting substituted pyridines of the formula II with an aryl compound of the formula III.
摘要翻译：制备式I取代的苯基吡啶的方法包括使式II的取代的吡啶与式III的芳基化合物反应。

56. 发明申请

US20100222586A1 Methods for Producing Sulfonic Acid Diamides 有权
标题翻译：生产磺酸二酰胺的方法
公开(公告)号：US20100222586A1
公开(公告)日：2010-09-02
申请号：US12681843
申请日：2008-10-10
申请人： Axel Pleschke , Thomas Schmidt , Joachim Gebhardt , Sandra Loehr , Michael Keil , Jan Hendrik Wevers
发明人： Axel Pleschke , Thomas Schmidt , Joachim Gebhardt , Sandra Loehr , Michael Keil , Jan Hendrik Wevers
IPC分类号： C07D239/10 , C07C309/63
CPC分类号： C07C303/34 , A01N43/54 , C07C307/06 , C07C381/00 , C07D239/54
摘要： The present invention relates to a process for preparing sulfuric diamides of the general formula I R1R2N—S(O)2—NH2 (I) in which R1 and R2 are each independently a primary alkyl radical having from 1 to 8 carbon atoms, a secondary alkyl radical having from 3 to 8 carbon atoms or a cycloalkyl radical having from 5 to 8 carbon atoms, or, together with the nitrogen atom, form a 5- to 8-membered, saturated nitrogen heterocycle which, as well as the nitrogen atom, may have a further heteroatom selected from O and S as a ring member, where the nitrogen heterocycle is unsubstituted or may have 1, 2, 3 or 4 alkyl groups having in each case from 1 to 4 carbon atoms as substituents. The process comprises the following steps: i) the reaction of a secondary amine of the formula II R1R2NH (II) in which R1 and R2 are each as defined above with sulfuryl chloride in an inert solvent, especially an aromatic solvent, in the presence of a tertiary amine to give a sulfamoyl chloride of the formula III R1R2N—S(O)2—Cl (III) in which R1 and R2 are each as defined above, and ii) reaction of the sulfamoyl chloride of the formula III obtained in step i) with ammonia, the sulfamoyl chloride of the formula III being used in step ii) in the form of the solution obtained in step i) in the inert solvent, especially the aromatic solvent.
摘要翻译：本发明涉及制备通式为R 1 R 2 N-S（O）2 -NH 2（I）的硫酸二酰胺的方法，其中R 1和R 2各自独立地为具有1至8个碳原子的伯烷基，二级具有3至8个碳原子的烷基或具有5至8个碳原子的环烷基，或与氮原子一起形成5-8元饱和氮杂环，其氮原子，可以具有选自O和S的另外的杂原子作为环成员，其中氮杂环是未取代的或可以具有1,2,3或4个烷基，每个情况下具有1至4个碳原子作为取代基。该方法包括以下步骤：i）在惰性溶剂，特别是芳族溶剂中，在惰性溶剂，特别是芳族溶剂的存在下，使式II的R 1 R 2 NH（II）的仲胺与R 1和R 2各自如上所述与磺酰氯反应，得到式III的R 1 R 2 N-S（O）2 -C（III）的氨磺酰氯，其中R 1和R 2各自如上所定义，和ii）在步骤（a）中获得的式III的氨磺酰氯的反应， i）与氨，式III的氨磺酰氯以步骤ⅱ）中的步骤i）中获得的溶液的形式在惰性溶剂中，特别是芳族溶剂中使用。

57. 发明申请

US20110152522A1 METHOD FOR THE PRODUCTION OF 3-PHENYL(THIO) URACILS AND DITHIOURACILS 有权
标题翻译：生产3-苯基（硫脲）尿素和二氧化硅的方法
公开(公告)号：US20110152522A1
公开(公告)日：2011-06-23
申请号：US13040292
申请日：2011-03-04
申请人： Sandra Löhr , Joachim Gebhardt , Guido Mayer , Michael Keil , Thomas Schmidt , Bernd Wolf
发明人： Sandra Löhr , Joachim Gebhardt , Guido Mayer , Michael Keil , Thomas Schmidt , Bernd Wolf
IPC分类号： C07D239/54 , C07C303/40
CPC分类号： C07D239/54
摘要： The present invention relates to a process for preparing 3-phenyl(thio)uracils and -dithiouracils of the formula I where the variables are each as defined in the description, and also intermediates for their preparation.
摘要翻译：本发明涉及一种制备式I的3-苯基（硫代）尿嘧啶和二硫尿嘧啶的方法，其中各变量各自如说明书中所定义，以及它们制备的中间体。

58. 发明授权

US08362026B2 Crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2H)-pyrimidinyl]-4-fluoro-N-[[methyl(1-methyl-ethyl)amino]sulfonyl]benzamide 有权
标题翻译：结晶形式的2-氯-5- [3,6-二氢-3-甲基-2,6-二氧代-4-（三氟甲基）-1-（2H） - 嘧啶基] -4-氟-N - [[甲基（1-甲基 - 乙基）氨基]磺酰基]苯甲酰胺
公开(公告)号：US08362026B2
公开(公告)日：2013-01-29
申请号：US12444653
申请日：2007-10-12
申请人： Thomas Schmidt , Joachim Gebhardt , Sandra Löhr , Michael Keil , Jan Hendrik Wevers , Peter Erk , Heidi Emilia Saxell , Gerhard Hamprecht , Werner Seitz , Guido Mayer , Bernd Wolf , Gerhard Cox , Alfred Michel , Cyrill Zagar , Robert Reinhard , Bernd Sievernich
发明人： Thomas Schmidt , Joachim Gebhardt , Sandra Löhr , Michael Keil , Jan Hendrik Wevers , Peter Erk , Heidi Emilia Saxell , Gerhard Hamprecht , Werner Seitz , Guido Mayer , Bernd Wolf , Gerhard Cox , Alfred Michel , Cyrill Zagar , Robert Reinhard , Bernd Sievernich
IPC分类号： A01N43/54 , A61K31/505
CPC分类号： C07D239/54
摘要： The present invention relates to a crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2H)pyrimidinyl]-4-fluoro-N-[[methyl(1-methylethyl)-amino]sulfonyl]benzamide. The invention also relates to a process for the preparation of this crystalline form and to plant protection formulations which comprise this crystalline form of the phenyluracil.
摘要翻译：本发明涉及2-氯-5- [3,6-二氢-3-甲基-2,6-二氧代-4-（三氟甲基）-1-（2H）嘧啶基] -4-氟 - N - [[甲基（1-甲基乙基） - 氨基]磺酰基]苯甲酰胺。本发明还涉及制备该结晶形式的方法以及包含该苯基尿嘧啶的该结晶形式的植物保护制剂。

59. 发明申请

US20120289706A1 Method for Producing Triazolinthione Derivatives and Intermediates Thereof 审中-公开
标题翻译：生产三唑啉衍生物及其中间体的方法
公开(公告)号：US20120289706A1
公开(公告)日：2012-11-15
申请号：US13515064
申请日：2010-12-13
申请人： Jens Renner , Jochen Dietz , Thomas Grote , Joachim Gebhardt , Markus Nett , Michael Keil
发明人： Jens Renner , Jochen Dietz , Thomas Grote , Joachim Gebhardt , Markus Nett , Michael Keil
IPC分类号： C07D405/06 , C07D303/36
CPC分类号： C07D249/12
摘要： The present invention relates to a new process for the preparation of substituted thiotriazolo groups of the general formula (I) wherein the variables have the meanings as given in the claims and the description.
摘要翻译：本发明涉及制备通式（I）的取代的三优唑基的新方法，其中变量具有权利要求书和说明书中给出的含义。

60. 发明授权

US08252925B2 Method for the production of 3-phenyl(thio)uracils and dithiouracils 有权
标题翻译：制备3-苯基（硫代）尿嘧啶和二硫尿嘧啶的方法
公开(公告)号：US08252925B2
公开(公告)日：2012-08-28
申请号：US11631972
申请日：2005-07-13
申请人： Sandra Löhr , Joachim Gebhardt , Guido Mayer , Michael Keil , Thomas Schmidt , Bernd Wolf
发明人： Sandra Löhr , Joachim Gebhardt , Guido Mayer , Michael Keil , Thomas Schmidt , Bernd Wolf
IPC分类号： C07D239/00 , C07D239/02
CPC分类号： C07D239/54
摘要： The present invention relates to a process for preparing 3-phenyl(thio)uracils and -dithiouracils of the formula I where the variables are each as defined in the description, and also intermediates for their preparation.
摘要翻译：本发明涉及一种制备式I的3-苯基（硫代）尿嘧啶和二硫尿嘧啶的方法，其中各变量各自如说明书中所定义，以及它们制备的中间体。

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