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51. 发明授权

US5252540A Sulfonamides 失效
标题翻译：磺胺类
公开(公告)号：US5252540A
公开(公告)日：1993-10-12
申请号：US760156
申请日：1991-09-16
申请人： Elisabeth Heistracher , Klaus Fischer , Horst Mayer , Thomas Saupe , Gerhard Hamprecht , Klaus Ditrich , Thomas Kuekenhoehner , Matthias Gerber , Helmut Walter , Karl-Otto Westphalen
发明人： Elisabeth Heistracher , Klaus Fischer , Horst Mayer , Thomas Saupe , Gerhard Hamprecht , Klaus Ditrich , Thomas Kuekenhoehner , Matthias Gerber , Helmut Walter , Karl-Otto Westphalen
IPC分类号： A01N43/08 , A01N43/10 , A01N43/36 , A01N43/50 , A01N43/56 , A01N43/78 , A01N43/80 , C07D207/34 , C07D207/416 , C07D231/14 , C07D231/16 , C07D231/54 , C07D231/56 , C07D233/90 , C07D261/18 , C07D263/34 , C07D271/04 , C07D271/06 , C07D271/08 , C07D271/10 , C07D277/20 , C07D277/32 , C07D277/34 , C07D277/56 , C07D285/06 , C07D307/68 , C07D307/71 , C07D333/38 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12
CPC分类号： C07D231/16 , C07D207/34 , C07D231/14 , C07D231/54 , C07D231/56 , C07D233/90 , C07D261/18 , C07D263/34 , C07D277/32 , C07D277/34 , C07D285/06 , C07D307/68 , C07D307/71 , C07D333/38 , C07D401/12 , C07D409/12
摘要： Sulfonamides of the formula I ##STR1## where A is an unsubstituted or substituted aromatic or heteroaromatic radical; W is oxygen or sulfur; B is an unsubstituted or substituted furyl, thienyl, pyrrolyl, oxazolyl, isothiazolyl, imidazolyl, pyrazolyl, thiadiazolyl, oxadiazolyl or triazolyl radical, and the environmentally compatible salts thereof are prepared as described and are used as herbicides.
摘要翻译：式I的磺酰胺（I）其中A是未取代或取代的芳族或杂芳族基团; W是氧或硫; B是未取代或取代的呋喃基，噻吩基，吡咯基，恶唑基，异噻唑基，咪唑基，吡唑基，噻二唑基，恶二唑基或三唑基，并且其环境相容的盐如所述制备并用作除草剂。

52. 发明授权

US06204222B1 Substituted cyclohexene-1,2-dicarboxylic acid derivatives and intermediates for their preparation 失效
标题翻译：取代的环己烯-1,2-二羧酸衍生物及其制备中间体
公开(公告)号：US06204222B1
公开(公告)日：2001-03-20
申请号：US09085769
申请日：1998-05-29
申请人： Ralf Klintz , Elisabeth Heistracher , Peter Schaefer , Gerhard Hamprecht , Peter Plath , Uwe Kardorff , Matthias Gerber , Karl-Otto Westphalen , Helmut Walter
发明人： Ralf Klintz , Elisabeth Heistracher , Peter Schaefer , Gerhard Hamprecht , Peter Plath , Uwe Kardorff , Matthias Gerber , Karl-Otto Westphalen , Helmut Walter
IPC分类号： A01N4336
CPC分类号： C07D209/48 , A01N37/30 , A01N37/32 , A01N37/34 , A01N37/46 , A01N43/12 , A01N43/16 , A01N43/40 , A01N43/74 , C07C233/61 , C07C233/63 , C07C255/13 , C07C255/46 , C07D295/185 , C07D307/12 , C07D307/90 , C07D309/06 , C07D339/08 , C07D401/10 , C07D413/10 , C07D417/10
摘要： Substituted cyclohexene-1,2-dicarboxylic acid derivatives I (R1 and R2 are each H, unsubstituted or substituted C1-C6-alkyl, C3-C6-alkenyl or C3-C6-alkynyl, C3-C8-cycloalkyl, unsubstituted or substituted phenyl or heterocyclyl and, if R1 is H or C1-C6-alkyl, R2 is additionally OH, C1-C6-alkoxy, C3-C6-alkenyloxy, C3-C6-alkynyloxy, C3-C6-cycloalkoxy, C5-C7-cycloalkenyloxy, C1-C6-haloalkoxy, C3-C6-haloalkenyloxy, C3-C7-cycloalkyl-C1-C6-alkoxy, C1-C6-alkyl-carbonyloxy, C1-C6-cyanoalkoxy, hydroxy-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C1-C6-alkoxycarbonyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C1-C6-alkylamino-C1-C6-alkoxy, C1-C6-dialkylamino-C1-C6-alkoxy, unsubstituted or substituted phenyl-C1-C6-alkoxy, phenyl-C3-C6-alkenyloxy or phenyl-C3-C7-alkynyloxy or unsubstituted or substituted amino, or R1 and R2, together with the nitrogen atom to which they are bonded, form an unsubstituted or substituted 3-membered to 8-membered heterocyclic structure, R3 is H or C1-C6-alkyl, R4 is H or halogen, R5 is H, halogen, NO2, CN or CF3, R6 is an unsubstituted or substituted 3-membered to 8-membered heterocyclic group, —A—CN, —A—CO—B, OR9, —C(R10)═O, —C(R10)═S, —C(R10)═N—R16, —CHR10)—CHR11—CO—B, —C(X1R14)(X2R15)R10 or —P(R12)(R13)═O, where the stated radicals have the meanings listed in the description, or R5 and R6 together form a 3-membered to 5-membered substituted carbon chain, and the agriculturally useful salts of Ia and Ib and intermediates for their preparation. The compounds Ia and Ib and their intermediates are suitable as herbicides and for the desiccation/defoliation of plants.
摘要翻译：取代的环己烯-1,2-二羧酸衍生物I（R 1和R 2各自为H，未取代或取代的C 1 -C 6 - 烷基，C 3 -C 6 - 烯基或C 3 -C 6炔基，C 3 -C 8 - 环烷基，未取代或取代的苯基或者杂环基，如果R 1是H或C 1 -C 6烷基，则R 2又是OH，C 1 -C 6 - 烷氧基，C 3 -C 6 - 烯氧基，C 3 -C 6 - 炔氧基，C 3 -C 6 - 环烷氧基，C 5 -C 7 - 环烯基氧基， C 1 -C 6 - 卤代烷氧基，C 3 -C 6 - 卤代链烯氧基，C 3 -C 7 - 环烷基-C 1 -C 6 - 烷氧基，C 1 -C 6烷基 - 羰氧基，C 1 -C 6 - 氰基烷氧基，羟基-C 1 -C 6烷氧基，烷氧基-C 1 -C 6烷氧基，C 1 -C 6烷氧基-C 1 -C 6烷氧基，C 1 -C 6烷氧基-C 1 -C 6烷氧基，C 1 -C 6烷基氨基-C 1 -C 6烷氧基，C 1 -C 6二烷基氨基 - C 1 -C 6 - 烷氧基，未取代或取代的苯基-C 1 -C 6 - 烷氧基，苯基-C 3 -C 6 - 烯氧基或苯基-C 3 -C 7 - 炔氧基或未取代或取代的氨基，或R 1和R 2与它们是键合的，形成未取代或取代的3元至8元杂环结构，R 3是H或C 1 -C 6 - 烷基，R 4是H或卤代 n为5，卤素，NO 2，CN或CF 3，R 6为未取代或取代的3元至8元杂环基，-A-CN，-A-CO-B，OR 9，-C（R 10） O，-C（R 10）= S，-C（R 10）= N-R 16，-CHR 10）-CHR 11 -CO-B，-C（X 1 R 14）（X 2 R 15）R 10或-P（R 12）其中所述基团具有本说明书所列的含义，或者R5和R6一起形成3元至5元取代的碳链，以及Ia和Ib的农业上有用的盐及其制备的中间体。化合物Ia和 Ib及其中间体适合作为除草剂和植物的干燥/脱叶作用。

53. 发明授权

US6013606A Substituted cinnamic oxime and hydroxamide derivatives 失效
标题翻译：取代的肉桂肟和羟基酰胺衍生物
公开(公告)号：US6013606A
公开(公告)日：2000-01-11
申请号：US765180
申请日：1997-06-30
申请人： Ralf Klintz , Gerhard Hamprecht , Elisabeth Heistracher , Peter Schafer , Christoph-Sweder von dem Bussche-Hunnefeld , Peter Munster , Reinhard Kirstgen , Albrecht Harreus , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
发明人： Ralf Klintz , Gerhard Hamprecht , Elisabeth Heistracher , Peter Schafer , Christoph-Sweder von dem Bussche-Hunnefeld , Peter Munster , Reinhard Kirstgen , Albrecht Harreus , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
IPC分类号： C07D239/52 , A01N37/32 , A01N37/50 , A01N43/38 , A01N43/54 , C07C251/40 , C07C259/06 , C07C265/14 , C07C271/28 , C07C271/58 , C07C331/28 , C07D209/48 , C07D239/54 , C07D239/56 , C07D239/58 , C07D413/10 , A01N43/50 , C07D223/10 , C07D235/26
CPC分类号： C07D209/48 , A01N37/32 , A01N37/50 , A01N43/54 , C07C251/40 , C07C259/06 , C07C265/14 , C07C271/28 , C07C271/58 , C07C331/28 , C07D239/54
摘要： Substituted cinnamic oxime derivatives I and cinnamic hydroxamide derivatives II ##STR1## (R.sup.1= halogen, NO.sub.2, CN, CF.sub.3 ; R.sup.2 =H, halogen; R.sup.3= H, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, hydroxy-C.sub.1 -C.sub.6 -alkyl;R.sup.4= H, halogen, CN, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl orR.sup.3 +R.sup.4 =chemical bond;Y=--O--, --S--, --O--CO--, --O--SO.sub.2 -- or chemical bond;Y'=--O-- or --S--;R.sup.5= unsubst. or subst. C.sub.1 -C.sub.6 -alkyl or C.sub.1 -C.sub.6 -haloalkyl; C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, unsubst. or subst. phenyl or phenyl-C.sub.1 -C.sub.6 -alkyl, or, if Y is --O--, --S-- or a chemical bond, is (C.sub.1 -C.sub.6 -alkyl)carbonyl or (C.sub.1 -C.sub.6 -alkoxy)carbonyl; or, if Y is a chemical bond, is hydrogen or halogen;R.sup.5 '=R.sup.5, H or (C.sub.1 -C.sub.6 -haloalkyl)carbonyl;R.sup.6= H, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, hydroxy-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkylthio-C.sub.1 -C.sub.6 -alkyl, cyano-C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkoxy) carbonyl-C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkyl) carbonyl-C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkyl)carbonyloxy-C.sub.1 -C.sub.6 -alkyl or unsubst. or subst. phenyl-C.sub.1 -C.sub.6 -alkyl;or, if Y is oxygen or sulfur, R.sup.5 +R.sup.6 together=unsubst. or subst. C.sub.1 -C.sub.3 -alkylene;Cyc=N-(3,4,5,6-tetrahydrophthalimido) or ##STR2## X.sup.1, X.sup.2 =oxygen or sulfur; R.sup.7 =H, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, NH.sub.2 ;R.sup.8, R.sup.9 =H, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl or unsubst. or subst. phenyl);and salts of I and II.Use: herbicides; desiccation/defoliation of plants.
摘要翻译： PCT No.PCT / EP95 / 02584第 371日期：1997年6月30日 102（e）日期1997年6月30日PCT提交1995年7月4日PCT公布。第WO96 / 02518号公报日期1996年2月1日取代肉桂肟衍生物I和肉桂酸羟基酰胺衍生物II（R1 =卤素，NO2，CN，CF3; R2 = H，卤素; R3 = H，卤素，C1-C6-烷基，C1-C6-卤代烷基， C3-C6-环烷基，C3-C6-烯基，C3-C6-炔基，羟基-C1-C6-烷基; R4 = H，卤素，CN，C1-C6-烷基，C1-C6-卤代烷基或R3 + R4 = 化学键; Y = -O-，-S-，-O-CO-，-O-SO2-或化学键; Y'= -O-或-S-; R5 =未取代或未取代的C1-C6- 烷基或C 1 -C 6 - 卤代烷基; C 3 -C 6 - 环烷基，C 3 -C 6 - 烯基，C 3 -C 6炔基，未取代或取代的苯基或苯基-C 1 -C 6烷基，或者如果Y是-O- （C 1 -C 6烷基）羰基或（C 1 -C 6 - 烷氧基）羰基;或者如果Y是化学键，则是氢或卤素; R 5'= R 5，H或（C 1 -C 6 - -C 6 - 卤代烷基）羰基; R 6 = H，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 3 -C 6环烷基，C 3 -C 6 - 烯基，C 3 -C 6炔基，羟基-C 1 -C 6烷基， C 1 -C 6烷氧基-C 1 -C 6烷基，C 1 -C 6烷硫基-C 1 -C 6烷基，氰基-C 1 -C 6烷基，（C 1 -C 6 - 烷氧基）羰基-C 1 -C 6烷基，（C 1 -C 6 - 烷基）羰基-C 1 -C 6 - 烷基，（C 1 -C 6 - 烷基）羰基氧基 -C 1 -C 6 - 烷基或未取代基。或subst。苯基-C 1 -C 6 - 烷基; 或者如果Y是氧或硫，则R5 + R6一起=不成立。或subst。 C1-C3-亚烷基; Cyc = N-（3,4,5,6-四氢邻苯二甲酰亚氨基）或X1，X2 =氧或硫; R7 = H，C1-C6-烷基，C1-C6-卤代烷基，NH2; R8，R9 = H，卤素，C1-C6-烷基，C1-C6-卤代烷基或未取代基。或subst。苯基）; 和I和II的盐。用途：除草剂; 植物的干燥/脱叶。

54. 发明授权

US5939558A N-phenyltetrahydroindazoles, their preparation, and their use as crop protection agents 失效
公开(公告)号：US5939558A
公开(公告)日：1999-08-17
申请号：US793124
申请日：1997-02-18
申请人： Elisabeth Heistracher , Lothar Rub , Christoph-Sweder von dem Bussche-Hunnefeld , Gerhard Hamprecht , Ralf Klintz , Peter Schafer , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
发明人： Elisabeth Heistracher , Lothar Rub , Christoph-Sweder von dem Bussche-Hunnefeld , Gerhard Hamprecht , Ralf Klintz , Peter Schafer , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
IPC分类号： C07D231/56 , A01N43/56
CPC分类号： A01N43/56
摘要： N-Phenyltetrahydroindazoles of formula (I), where R.sub.1 is H or C.sub.1-4 -alkyl; R.sup.2 is halogen, C.sub.1-4 -alkyl or C.sub.1-4 -haloalkyl; R.sup.3 is H or halogen; R.sup.4 is NO.sub.2, halogen, C.sub.1-4 -alkyl or C.sub.1-4 -haloalkyl; R.sup.5 is --XR.sup.6 ; X is --O--, --S--, --SO-- or --SO.sub.2 --; R.sup.6 is --Alk--R.sup.7 ; Alk is a substituted or unsubstituted methylene, ethylene, propylene, butylene or pentamethylene chain, where one chain member can carry a spiro-linked 2- to 5-membered C chain or where 2 ring members can be bridged via a C.sub.1-5 -alkylene chain; R.sup.7 is CN, SCN, halogen or --YR.sup.11, where Y is --O--, --S--, --SO-- or --SO.sub.2 --; R.sup.10 is H, OH, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.3 -C.sub.5 -cycloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.3 -C.sub.5 -cycloalkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkylthio, --NH--R.sup.12, --N(C.sub.1 -C.sub.4 -alkyl)--R.sup.12, --N(C.sub.3 -C.sub.4 -alkenyl)-R.sup.12, --N(C.sub.3 -C.sub.4 -alkynyl)-R.sup.12, pyrrolidin-1-yl, piperid-1-yl, morpholin-4-yl, azepan-1-yl, (i) unsubstituted or substituted phenyl, benzyl, phenoxy or benzyloxy; R.sup.11 is C.sub.1-6 -alkyl, C.sub.1-6 -haloalkyl or C.sub.1-6 -cycloalkyl; R.sup.12 is H, OH, C.sub.1-4 -alkyl, C.sub.3-4 -alkenyl, C.sub.3-4 -alkynyl, C.sub.3-6 -cycloalkyl, C.sub.1-4 -alkoxy, C.sub.3-4 -alkenyloxy, C.sub.3-4 -alkenyloxy, C.sub.3-4 -alkynyloxy, or substituted or unsubstituted phenyl or benzyl; and the agriculturally utilizable salts of formula (I), with the provisoes that the simultaneous meaning of R.sup.6 as dihalomethyl, R.sup.2 and R.sup.4 as chlorine and R.sup.3 as halogen is excluded; the simultaneous meaning of X as oxygen and R.sup.7 as --OR.sup.11 or C.sub.1 -C.sub.6 -alkylthio is excluded; Alk must not carry a spiro-linked three-membered ring if R.sup.7 is halogen and R.sup.11 is not C.sub.1-6 -alkyl if R.sup.1 is H, R.sup.2 is C.sub.1-4 -haloalkyl, R.sup.3 is F, R.sup.4 is halogen and R.sup.7 is --R.sup.11. Use: as herbicides; for desiccating/defoliating plants.

55. 发明授权

US5783522A Substituted 2-phenylpyridines 失效
标题翻译：取代的2-苯基吡啶
公开(公告)号：US5783522A
公开(公告)日：1998-07-21
申请号：US592355
申请日：1996-01-11
申请人： Peter Schaefer , Gerhard Hamprecht , Elisabeth Heistracher , Hartmann Koenig , Ralf Klintz , Peter Muenster , Harald Rang , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
发明人： Peter Schaefer , Gerhard Hamprecht , Elisabeth Heistracher , Hartmann Koenig , Ralf Klintz , Peter Muenster , Harald Rang , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
IPC分类号： A01N43/40 , A01N43/42 , A01N43/60 , A01N43/647 , A01N43/76 , A01N43/78 , A01N43/84 , A01N47/22 , C07D213/30 , C07D213/61 , C07D213/65 , C07D213/70 , C07D213/89 , C07D265/36 , C07D401/04 , C07D405/04 , C07D405/14 , C07D409/04 , C07D409/12 , C07D413/04 , C07D417/04
CPC分类号： C07D213/30 , C07D213/61 , C07D265/36 , C07D409/12
摘要： Substituted 2-phenylpyridines I ##STR1## R.sup.1,R.sup.3 =H, halogen, alkyl, haloalkyl, alkoxyalkyl, alkoxy, alkoxyalkoxy, OH, haloalkoxy, alkylcarbonyloxy, haloalkylcarbonyloxy, SH, alkylthio, alkylsulfinyl, alkylsulfonyl, haloalkylthio, haloalkylsulfinyl, haloalkylsulfonyl, CHO, CN, CO.sub.2 H, alkoxycarbonyl, alkoxyalkoxycarbonyl, haloalkoxycarbonyl, alkylcarbonyl, haloalkylcarbonyl, alkoxyalkylcarbonyl, CONH.sub.2, alkyl-aminocarbonyl, dialkylaminocarbonyl, pyrrolidinyl-carbonyl piperidylcarbonyl, morpholinylcarbonyl, NO.sub.2, NH.sub.2, alkylamino, dialkylamino, pyrrolidinyl, piperidinyl, morpholinyl, alkylcarbonylamino, haloalkylcarbonylamino, alkylsulfonylamino; R.sup.2 =halogen, CN, NO.sub.2, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio; or R.sup.1 +R.sup.2 or R.sup.2 +R.sup.3 =trimethylene or tetramethylene chain;R.sup.4 =halogen, alkyl, haloalkyl, alkoxyalkyl, alkoxy, alkoxyalkoxy, OH, haloalkoxy, alkylcarbonyloxy, haloalkylcarbonyloxy, SH, alkylthio, alkylsulfinyl, alkylsulfonyl, haloalkylthio, haloalkylsulfinyl, haloalkylsulfonyl, CHO, CN, CO.sub.2 H, alkoxycarbonyl, alkoxyalkoxycarbonyl, haloalkoxycarbonyl, alkylcarbonyl, haloalkylcarbonyl, alkoxyalkylcarbonyl, NO.sub.2, NH.sub.2, alkylamino, dialkylamino, pyrrolidinyl, piperidinyl, morpholinyl, alkylcarbonylamino, haloalkylcarbonylamino, alkylsulfonylamino; R.sup.5 =hydrogen or halogen; R.sup.6 =halogen, CN, NO.sub.2, OH, CF.sub.3, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkoxy; R.sup.7 =various radicals; and the N-oxides of I and the agriculturally utilizable salts of I where these exist, excepting those compounds I where R.sup.2 is C.sub.1 -C.sub.4 -alkoxy and R.sup.1 and/or R.sup.3 is carboxyl or the salt, ester or amide thereof.
摘要翻译： PCT No.PCT / EP94 / 02263 371日期1996年1月11日 102（e）日期1996年1月11日PCT提交1994年7月11日PCT公布。公开号WO95 / 02580 日期1995年1月26日取代的2-苯基吡啶I R1，R3 = H，卤素，烷基，卤代烷基，烷氧基烷基，烷氧基，烷氧基烷氧基，OH，卤代烷氧基，烷基羰基氧基，卤代烷基羰氧基，SH，烷硫基，烷基亚磺酰基，烷基磺酰基，卤代烷硫基，卤代烷基亚磺酰基，卤代烷基磺酰基，CHO，CN，CO 2 H，烷氧基羰基，烷氧基烷氧基羰基，卤代烷氧基羰基，烷基羰基，卤代烷基羰基，烷氧基烷基羰基，CONH 2，烷基氨基羰基，二烷基氨基羰基，吡咯烷基 - 羰基哌啶基羰基，吗啉基羰基，NO 2，NH 2，烷基氨基，二烷基氨基，吡咯烷基，哌啶基，吗啉基，烷基羰基氨基，卤代烷基羰基氨基，烷基磺酰基氨基; R 2 =卤素，CN，NO 2，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基; 或R1 + R2或R2 + R3 =三亚甲基或四亚甲基链; R 4 =卤素，烷基，卤代烷基，烷氧基烷基，烷氧基，烷氧基烷氧基，OH，卤代烷氧基，烷基羰基氧基，卤代烷基羰氧基，烷硫基，烷基亚磺酰基，烷基磺酰基，卤代烷硫基，卤代烷基亚磺酰基，卤代烷基磺酰基，CHO，CN，CO 2 H，烷氧基羰基，烷氧基烷氧基羰基，卤代烷氧基羰基，烷基羰基，卤代烷基羰基，烷氧基烷基羰基，NO 2，NH 2，烷基氨基，二烷基氨基，吡咯烷基，哌啶基，吗啉基，烷基羰基氨基，卤代烷基羰基氨基，烷基磺酰基氨基。 R5 =氢或卤素; R6 =卤素，CN，NO2，OH，CF3，C1-C6-烷基，C1-C4-烷氧基; R7 =各种基团; 和I的N-氧化物和其中存在的I的农业上可利用的盐，除了其中R 2是C 1 -C 4 - 烷氧基且R 1和/或R 3是羧基的化合物I或其盐，酯或酰胺。

56. 发明授权

US06169184A Process for the production of substituted phenylpyridines 失效
标题翻译：制备取代苯基吡啶的方法
公开(公告)号：US06169184A
公开(公告)日：2001-01-02
申请号：US09254456
申请日：1999-03-10
申请人： Gerhard Hamprecht , Joachim Gebhardt , Heinz Isak , Michael Rack , Joachim Rheinheimer , Peter Sch{umlaut over (a)}fer
发明人： Gerhard Hamprecht , Joachim Gebhardt , Heinz Isak , Michael Rack , Joachim Rheinheimer , Peter Sch{umlaut over (a)}fer
IPC分类号： C02D2472
CPC分类号： C07D213/62
摘要： A process for preparing substituted phenylpyridines of the formula I comprises reacting substituted pyridines of the formula II with an aryl compound of the formula III.
摘要翻译：制备式I取代的苯基吡啶的方法包括使式II的取代的吡啶与式III的芳基化合物反应。

57. 发明授权

US5750705A Substituted trifluoromethylpyridines 失效
标题翻译：取代的三氟甲基吡啶
公开(公告)号：US5750705A
公开(公告)日：1998-05-12
申请号：US695475
申请日：1996-08-12
申请人： Gerhard Hamprecht , Elisabeth Heistracher , Ralf Klintz , Peter Schafer , Cyrill Zagar
发明人： Gerhard Hamprecht , Elisabeth Heistracher , Ralf Klintz , Peter Schafer , Cyrill Zagar
IPC分类号： A01N43/56 , C07D213/64 , C07D213/73 , C07D213/74 , C07D213/77 , C07D401/04 , A01N43/40 , A61K31/44
CPC分类号： C07D213/77 , C07D213/64 , C07D213/73
摘要： Substituted trifluoromethylpyridines of the general formula Ia or Ib ##STR1## where the substituents have the following meanings: R.sup.1 is amino or hydrazino, in the case of Ib additionally chlorine or fluorine; R.sup.2 is halogen; and R.sup.3 is C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl or C.sub.2 -C.sub.6 -alkynyl, it being possible for these groups to have attached to them up to 6 halogen atoms, C.sub.3 -C.sub.6 -cycloalkyl which can have attached to it up to 3 C.sub.1 -C.sub.3 -alkyl radicals, C.sub.1 -C.sub.6 -cyanoalkyl, C.sub.1 -C.sub.4 -alkoxy-C.sub.2 -C.sub.6 -alkyl, 3-oxetanyl, carboxyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxycarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkoxy-C.sub.2 -C.sub.4 -alkoxycarbonyl-C.sub.1 -C.sub.6 -alkyl, aminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -dialkylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.4 -alkenylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.4 -alkynylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkyl-C.sub.3 -C.sub.4 -alkenylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkyl-C.sub.3 -C.sub.4 -alkynylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -(.alpha.-alkylalkylidene)iminoxy-C.sub.2 -C.sub.6 -alkyl, cyclopropylmethyl, C.sub.1 -C.sub.6 -alkylamino, C.sub.1 -C.sub.6 -dialkylamino, C.sub.1 -C.sub.6 -alkylideneimino- or .alpha.-(C.sub.1 -C.sub.4 -alkyl) -C.sub.2 -C.sub.6 -alkylideneimino; and halogen is fluorine, chlorine, bromine or iodine, and processes for their preparation.
摘要翻译：取代基具有以下含义的取代的三氟甲基吡啶，其中R 1是氨基或肼基，在Ib的情况下另外是氯或氟; R2是卤素; 并且R 3是C 1 -C 6 - 烷基，C 2 -C 6 - 烯基或C 2 -C 6 - 炔基，这些基团可以连接至多达6个卤素原子，可以连接到其上的C 3 -C 6环烷基至3个C 1 -C 3 - 烷基，C 1 -C 6 - 氰基烷基，C 1 -C 4 - 烷氧基-C 2 -C 6 - 烷基，3-氧杂环丁烷基，羧基-C 1 -C 6烷基，C 1 -C 6 - 烷氧基羰基-C 1 -C 6烷基，C 1 -C 4 - 烷氧基-C 2 -C 4 - 烷氧基羰基-C 1 -C 6烷基，氨基羰基-C 1 -C 6 - 烷基，C 1 -C 4 - 烷基氨基羰基-C 1 -C 6烷基，C 1 -C 4 - 二烷基氨基羰基-C 1 -C 6烷基，C 2 -C 4 - 链烯基氨基羰基-C 1 -C 6烷基，C 3 -C 4 - 炔基氨基羰基-C 1 -C 6 - 烷基，C 1 -C 4烷基-C 3 -C 4链烯基氨基羰基-C 1 -C 6 - 烷基，C 1 -C 4烷基-C 3 C 1-4 - 炔基氨基羰基-C 1 -C 6烷基，C 3 -C 6 - （α-烷基亚烷基）亚氨基-C 2 -C 6 - 烷基，环丙基甲基，C 1 -C 6烷基氨基，C 1 -C 6 - 二烷基氨基，C 1 -C 6亚烷基亚氨基或α- - （C 1 -C 4 - 烷基）-C 2 -C 6亚烷基亚氨基; 并且卤素是氟，氯，溴或碘，并且其制备方法。

58. 发明授权

US5849920A Substituted trifluoromethylpyridines 失效
标题翻译：取代的三氟甲基吡啶
公开(公告)号：US5849920A
公开(公告)日：1998-12-15
申请号：US891967
申请日：1997-07-14
申请人： Gerhard Hamprecht , Elisabeth Heistracher , Ralf Klintz , Peter Schafer , Cyrill Zagar
发明人： Gerhard Hamprecht , Elisabeth Heistracher , Ralf Klintz , Peter Schafer , Cyrill Zagar
IPC分类号： A01N43/56 , C07D213/64 , C07D213/73 , C07D213/74 , C07D213/77 , C07D401/04 , A01N43/40 , C07D213/82
CPC分类号： C07D213/77 , C07D213/64 , C07D213/73
摘要： A trifluoromethylpyridine of the formula Ib ##STR1## where the substituents have the following meanings: R.sup.1 is chlorine or fluorine; R.sup.2 is halogen; and R.sup.3 is C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl or C.sub.2 -C.sub.6 -alkynyl, said groups being optionally substituted with 1 to 6 halogen atoms, C.sub.3 -C.sub.6 -cycloalkyl which is optionally substituted with 1 to 3 C.sub.1 -C.sub.3 -alkyl radicals, C.sub.1 -C.sub.6 -cyanoalkyl, C.sub.1 -C.sub.4 -alkoxy-C.sub.2 -C.sub.6 -alkyl, 3-oxetanyl, carboxyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxycarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkoxy-C.sub.2 -C.sub.4 -alkoxycarbonyl-C.sub.1 -C.sub.6 -alkyl, aminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -dialkylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.4 -alkenylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.4 -alkynylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkyl-C.sub.3 -C.sub.4 -alkenylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkyl-C.sub.3 -C.sub.4 -alkynylaminocarbonyl-C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -(.alpha.-alkylalkylidene)iminoxy-C.sub.2 -C.sub.6 -alkyl, cyclopropylmethyl, C.sub.1 -C.sub.6 -alkylamino, C.sub.1 -C.sub.6 -dialkylamino, C.sub.1 -C.sub.6 -alkylideneimino or .alpha.-(C.sub.1 -C.sub.4 -alkyl)-C.sub.2 -C.sub.6 -alkylideneimino; and halogen is fluorine, chlorine, bromine or iodine.
摘要翻译：式Ib的三氟甲基吡啶（ib）其中取代基具有以下含义：R 1是氯或氟; R2是卤素; 并且R 3为C 1 -C 6 - 烷基，C 2 -C 6 - 烯基或C 2 -C 6 - 炔基，所述基团任选被1至6个卤素原子取代，任选被1至3个C 1 -C 3 - 烷基，C 1 -C 6 - 氰基烷基，C 1 -C 4 - 烷氧基-C 2 -C 6 - 烷基，3-氧杂环丁烷基，羧基-C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基羰基-C 1 -C 6烷基，C 1 -C 4烷氧基 C 2 -C 4烷氧基羰基-C 1 -C 6烷基，氨基羰基-C 1 -C 6烷基，C 1 -C 4烷基氨基羰基-C 1 -C 6烷基，C 1 -C 4二烷基氨基羰基-C 1 -C 6烷基，C 2 -C 4链烯基氨基羰基 C 1 -C 6 - 烷基，C 3 -C 4 - 炔基氨基羰基-C 1 -C 6 - 烷基，C 1 -C 4烷基-C 3 -C 4 - 烯基氨基羰基-C 1 -C 6烷基，C 1 -C 4烷基-C 3 -C 4 - 炔基氨基羰基-C 1 C 1-6 - 烷基，C 3 -C 6 - （α-烷基亚烷基）亚氨基-C 2 -C 6 - 烷基，环丙基甲基，C 1 -C 6烷基氨基，C 1 -C 6 - 二烷基氨基，C 1 -C 6亚烷基亚氨基或α- ）-C2-C6-亚烷基亚氨基; 卤素是氟，氯，溴或碘。

59. 发明授权

US07687435B2 Benzoyl-substituted phenylalanineamides 有权
标题翻译：苯甲酰取代的苯丙氨酰胺
公开(公告)号：US07687435B2
公开(公告)日：2010-03-30
申请号：US10581444
申请日：2004-12-17
申请人： Matthias Witschel , Michael Puhl , Gerhard Hamprecht , Liliana Parra Rapado , Ulf Misslitz , CyrilL Zagar , Peter Plath , Robert Reinhard , Bernd Sievernich , Rex Liebl
发明人： Matthias Witschel , Michael Puhl , Gerhard Hamprecht , Liliana Parra Rapado , Ulf Misslitz , CyrilL Zagar , Peter Plath , Robert Reinhard , Bernd Sievernich , Rex Liebl
IPC分类号： A01N37/18 , C07C237/42
CPC分类号： C07D213/54 , A01N37/48 , A01N41/04 , A01N47/06 , A01N47/12 , C07C233/87 , C07C237/22 , C07C255/60 , C07C271/12 , C07C271/28 , C07C275/24 , C07C275/42 , C07C309/66 , C07C311/06 , C07C311/08 , C07C311/09 , C07C311/53 , C07C311/55 , C07C323/52 , C07C323/60 , C07C323/62 , C07C323/63 , C07D213/80 , C07D231/12 , C07D239/60 , C07D249/08 , C07D309/08 , C07D317/32 , C07D333/24 , C07F7/1804
摘要： The present invention relates to benzoyl-substituted phenylalanineamides of the formula I in which the variables R1 to R15 are as defined in the description, and to their agriculturally useful salts, to processes and intermediates for their preparation and to the use of these compounds or of compositions comprising these compounds for controlling unwanted plants.
摘要翻译：本发明涉及式I的苯甲酰基取代的苯丙氨酰胺，其中变量R1至R15如说明书中所定义，以及其农业上有用的盐，其制备方法和中间体以及这些化合物的使用或包含这些化合物以控制不想要的植物的组合物。

60. 发明授权

US06888003B2 Method for producing 7-(pyrazole-3-yl) benzoxazoles 失效
标题翻译： 7-（吡唑-3-基）苯并恶唑的制备方法
公开(公告)号：US06888003B2
公开(公告)日：2005-05-03
申请号：US10221206
申请日：2001-03-15
申请人： Cyrill Zagar , Robert Reinhard , Michael Puhl , Thorsten Volk , Norbert Götz , Gerhard Hamprecht , Olaf Menke , Ingo Sagasser
发明人： Cyrill Zagar , Robert Reinhard , Michael Puhl , Thorsten Volk , Norbert Götz , Gerhard Hamprecht , Olaf Menke , Ingo Sagasser
IPC分类号： C07D231/12 , A01N43/56 , A01N43/76 , C07B61/00 , C07D231/16 , C07D231/18 , C07D413/04 , C07D413/14 , C07D498/00
CPC分类号： C07D413/04 , A01N43/56
摘要： A process for preparing 7-(pyrazol-3-yl)benzoxazoles of the formula I in which the variables R1-R6 are as defined in claim 1, which process is characterized in that a 2-halo-3-(pyrazol-3-yl)anilide of the formula II, in which X is bromine or iodine is reacted with a base in the presence of a transition metal compound of subgroup VIIa, VIIIa or Ib of the Periodic Table of the Elements, is disclosed.
摘要翻译：制备其中变量R 1〜6的定义的式I的7-（吡唑-3-基）苯并恶唑的方法如权利要求1所定义，该方法其特征在于式Ⅱ的2-卤代-3-（吡唑-3-基）酰苯胺，其中X是溴或碘，在Ⅶa族，Ⅷa族或Ⅷa族过渡金属化合物存在下与碱反应公开了元素周期表的Ib。

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