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31. 发明申请

US20010000038A1 Novel intermediates useful for the preparation of antihistaminic piperidine derivatives 失效
标题翻译：用于制备抗组胺型哌啶衍生物的新型中间体
公开(公告)号：US20010000038A1
公开(公告)日：2001-03-15
申请号：US09726625
申请日：2000-12-01
发明人： Richard C. Krauss , Robert M. Strom , Carey L. Scortichini , William J. Kruper , Richard A. Wolf , Weishi W. Wu , Albert A. Carr , David A. Hay , Duane E. Rudisill , Gianbattista Panzone
IPC分类号： C07C069/95 , C07C069/76 , C07D413/00 , C07C233/00 , C07C235/00 , C07C237/00 , C07C239/00 , C07D401/00 , C07D405/00 , C07D409/00
CPC分类号： C07D295/185 , C07C33/46 , C07C45/46 , C07C45/63 , C07C45/65 , C07C45/673 , C07C49/792 , C07C49/798 , C07C49/80 , C07C49/813 , C07C49/82 , C07C49/825 , C07C49/83 , C07C49/835 , C07C49/86 , C07C59/86 , C07C59/88 , C07C69/007 , C07C69/738 , C07C235/78 , C07C255/16 , C07C259/06 , C07C2601/02 , C07D211/22 , C07D401/06 , C07D401/10
摘要： The present invention is related to a novel intermediates and processes which are useful in the preparation of certain antihistaminic piperidine derivatives of the formula 1 wherein W represents nullC(nullO)null or nullCH(OH)null; R1 represents hydrogen or hydroxy; R2 represents hydrogen; R1 and R2 taken together form a second bond between the carbon atoms bearing R1 and R2; n is an integer of from 1 to 5; m is an integer 0 or 1; R3 is nullCOOH or nullCOOalkyl wherein the alkyl moiety has from 1 to 6 carbon atoms and is straight or branched each of A is hydrogen or hydroxy; and pharmaceutically acceptable salts and individual optical isomers thereof, with the proviso that where R1 and R2 are ta to form a second bond between the carbon R1 and R2 or where R1 represented hydrox integer 0.
摘要翻译：本发明涉及可用于制备下式其中W代表-C（= O） - 或-CH（OH） - 的某些抗组氨酸哌啶衍生物的新中间体和方法; R1代表氢或羟基; R2表示氢; R1和R2一起形成带有R1和R2的碳原子之间的第二个键; n为1〜5的整数， m为整数0或1; R3是-COOH或-COO烷基，其中烷基部分具有1至6个碳原子，并且是直链或支链的，每个A是氢或羟基; 以及其药学上可接受的盐和单独的光学异构体，条件是其中R 1和R 2为ta以在碳R 1和R 2之间形成第二个键或其中R 1表示羟基整数0。

32. 发明授权

US6018050A Method of preparing optically active .alpha.-amino acids and .alpha.-amino acid derivatives 失效
标题翻译：制备光学活性α-氨基酸和α-氨基酸衍生物的方法
公开(公告)号：US6018050A
公开(公告)日：2000-01-25
申请号：US43038
申请日：1998-04-30
申请人： Hans-Josef Altenbach , Matthias Kottenhahn , Annegret Vogt , Mike Matthaus , Andreas Grundler , Michael Hahn
发明人： Hans-Josef Altenbach , Matthias Kottenhahn , Annegret Vogt , Mike Matthaus , Andreas Grundler , Michael Hahn
IPC分类号： C07C227/12 , C07C227/32 , C07C229/08 , C07C231/18 , C07C237/04 , C07D235/02 , C07D307/52 , C07D487/10 , C07D498/04 , C07D261/20 , C07C239/00
CPC分类号： C07D235/02 , C07C227/32
摘要： The invention relates to a new process for the preparation of optically active amino acids and amino acid derivatives of the general formula (I), wherein *, X and R.sup.1 to R.sup.4 have the meaning given in the description. Starting from commercially obtainable (-)-menthol or (+)-menthol, the enantiomerically pure compounds of the formula (I) are obtained in high yields. The method is particularly suitable for the preparation of sterically demanding amino acids and amino acid derivatives.
摘要翻译： PCT No.PCT / EP96 / 03984第 371日期：1998年4月30日 102（e）1998年4月30日PCT PCT 1996年9月11日PCT公布。出版物WO97 / 10203 PCT 日期：1997年3月20日本发明涉及制备通式（I）的光学活性氨基酸和氨基酸衍生物的新方法，其中*，X和R1至R4具有说明书中给出的含义。从（ - ） - 薄荷醇或（+） - 薄荷醇开始，以高产率获得式（I）的对映体纯的化合物。该方法特别适用于制备空间要求高的氨基酸和氨基酸衍生物。

33. 发明授权

US6013837A Aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides 失效
标题翻译：芳族酰胺，制备方法和含有它们的组合物及其作为农药的用途
公开(公告)号：US6013837A
公开(公告)日：2000-01-11
申请号：US894068
申请日：1997-07-30
申请人： Jacques Demassey , Michel Gohar , Christian Wehrey
发明人： Jacques Demassey , Michel Gohar , Christian Wehrey
IPC分类号： C07D295/18 , A01N37/10 , A01N37/18 , A01N37/22 , A01N37/36 , A01N37/38 , A01N37/44 , A01N37/46 , A01N37/48 , A01N41/10 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/44 , A01N43/713 , A01N43/78 , A01N43/80 , A01N43/84 , A61K31/165 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/4015 , A61K31/42 , A61K31/425 , A61K31/426 , A61K31/44 , A61K31/445 , A61P31/00 , A61P33/00 , C07C51/09 , C07C63/49 , C07C231/02 , C07C233/65 , C07C233/66 , C07C233/75 , C07C235/42 , C07D203/12 , C07D205/12 , C07D207/08 , C07D207/09 , C07D207/14 , C07D207/26 , C07D207/267 , C07D207/27 , C07D211/14 , C07D213/40 , C07D213/61 , C07D213/75 , C07D257/06 , C07D261/08 , C07D261/14 , C07D277/20 , C07D277/28 , C07D277/44 , C07D307/14 , C07D333/20 , C07D333/56 , C07C239/00 , C07C237/00
CPC分类号： C07D207/267 , A01N37/10 , A01N37/18 , A01N37/22 , A01N37/36 , A01N37/38 , A01N37/44 , A01N37/46 , A01N37/48 , A01N41/10 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/44 , A01N43/713 , A01N43/78 , A01N43/80 , A01N43/84 , C07C233/65 , C07C233/75 , C07C235/42 , C07D203/12 , C07D205/12 , C07D207/09 , C07D213/40 , C07D213/61 , C07D257/06 , C07D261/08 , C07D277/28 , C07D307/14 , C07D333/20
摘要： The subject of the invention is the compounds of formula (I):Q(CH.sub.2)a-(X.sub.1).sub.b -Q.sub.1 -Q.sub.2 -C(X.sub.2)--N(R.sub.1)(R.sub.2) (I)in which:Q represents an aryl radical,X.sub.1 represents oxy, thio, sulphinyl or sulphonyl,X.sub.2 represents oxygen or sulphur,Q.sub.1 represents a cyclopropanediyl radical,Q.sub.2 represents an arylene radical,R.sub.1 and R.sub.2 represent:either a hydrogen atom or a hydrocarbon radical or one of the groupsR.sub.3 --C.dbd.X.sub.3, (R.sub.3).sub.2 --P.dbd.X.sub.3, T.sub.2 -R.sub.5 or S(O).sub.j --N(R.sub.6)(R.sub.7)in which X.sub.3 represents an oxygen atom or a sulphur atom, T.sub.2 represents a bivalent oxy, carbonyl or oxycarbonyl group and j is equal to 0, 1 or 2, their preparation process and their use as pesticides.
摘要翻译： PCT No.PCT / FR96 / 00123 Sec。 371日期1997年7月30日 102（e）日期1997年7月30日PCT提交1996年1月25日PCT公布。公开号WO96 / 22965 日期：1996年8月1日本发明的主题是式（I）的化合物：Q（CH 2）a - （X1）b -Q1-Q2-C（X2）-N（R1）（R2）其中：Q表示芳基，X 1表示氧基，硫代，亚磺酰基或磺酰基，X 2表示氧或硫，Q 1表示环丙烷基，Q 2表示亚芳基，R 1和R 2表示：氢原子或烃基或其中X3表示氧原子或硫原子的R3-C = X3，（R3）2-P = X3，T2-R5或S（O）jN（R6）（R7）中的一个，T2表示二价氧，羰基或氧羰基，j等于0,1或2，它们的制备方法及其作为农药的用途。

34. 发明授权

US5725839A Compositions and methods utilizing nitroxides in combination with biocompatible macromolecules for ERI or MRI 失效
标题翻译：使用硝基氧与生物相容性大分子结合用于ERI或MRI的组合物和方法
公开(公告)号：US5725839A
公开(公告)日：1998-03-10
申请号：US482202
申请日：1995-06-07
申请人： Jen-Chang Hsia
发明人： Jen-Chang Hsia
IPC分类号： A61K38/00 , A61K38/38 , A61K38/42 , A61K39/395 , A61K45/06 , A61K47/48 , A61K49/00 , A61K49/20 , C07K14/76 , C07K14/805 , C07K16/00 , A61B5/055 , A01N33/24 , C07C239/00
CPC分类号： A61K38/38 , A61K38/42 , A61K39/395 , A61K45/06 , A61K47/48015 , A61K47/48307 , A61K47/48738 , A61K47/48769 , A61K49/0002 , A61K49/20 , A61K9/127 , B82Y5/00 , C07K14/76 , C07K14/805 , C07K16/00
摘要： Compositions and processes to alleviate free radical toxicity are disclosed based on the use of nitroxides in association with physiologically compatible macromolecules. In particular, hemoglobin-based red cell substitutes are described featuring stable nitroxide free radicals for use in cell-free hemoglobin solutions, encapsulated hemoglobin solutions, stabilized hemoglobin solutions, polymerized hemoglobin solutions, conjugated hemoglobin solutions, nitroxide-labelled albumin, and nitroxide-labelled immunoglobulin. Formulations are described herein that interact with free radicals, acting as antioxidant enzymemimics, which preserve nitroxides in their active form in vivo. Applications are described including blood substitutes, radioprotective agents, imaging agents, agents to protect against ischemia and reperfusion injury, and in vivo enzyme mimics among others.
摘要翻译：基于与生理上相容的大分子结合使用的氮氧化物，公开了减轻自由基毒性的组合物和方法。特别地，描述了基于血红蛋白的红细胞替代物，其特征在于稳定的氮氧自由基用于无细胞血红蛋白溶液，包封的血红蛋白溶液，稳定的血红蛋白溶液，聚合血红蛋白溶液，共轭血红蛋白溶液，氮氧自由基标记的白蛋白和氮氧化物标记免疫球蛋白。本文描述了与自由基相互作用的制剂，其作为抗氧化酶酶学，其在体内保护其活性形式的氮氧化物。描述了应用，包括血液代用品，放射防护剂，成像剂，防止缺血和再灌注损伤的药剂，以及体内酶模拟物等。

35. 发明授权

US5488150A Crystals of N-(trans-4-isopropylcyclohexycarbonyl)-D-phenylalanine and methods for preparing them 失效
标题翻译： N-（反式-4-异丙基环己基羰基）-D-苯丙氨酸的晶体及其制备方法
公开(公告)号：US5488150A
公开(公告)日：1996-01-30
申请号：US166144
申请日：1993-12-14
申请人： Michito Sumikawa , Yoshihito Koguchi , Takao Ohgane , Yasuo Irie , Satoji Takahashi
发明人： Michito Sumikawa , Yoshihito Koguchi , Takao Ohgane , Yasuo Irie , Satoji Takahashi
IPC分类号： C07C231/24 , A61K31/13 , A61K31/195 , C07C211/43 , C07C231/22 , C07C233/63 , C07C239/00
CPC分类号： C07C231/22 , C07C233/63
摘要： Stable crystals of N-(trans-4-isopropylcyclohexylcarbonyl)-D-phenylalanine may be produced by treating this compound with a solvent at a temperature of at least 10.degree. C. and forming crystals in the solvent at a temperature of at least 10.degree. C. For example, crystals may be formed by crystallization out of solution, or may be formed from solid particles of the compound suspended in a solvent. Crystals formed in this way have different melting point, infra red spectrum and X-ray diffraction patterns from previously known forms of the compound and have enhanced processability, eg. stability to grinding.
摘要翻译： N-（反式-4-异丙基环己基羰基）-D-苯丙氨酸的稳定晶体可以通过在至少10℃的温度下用溶剂处理该化合物并在溶剂中在至少10℃的温度下形成晶体来制备例如，可以通过从溶液中结晶而形成晶体，或者可以由悬浮在溶剂中的化合物的固体颗粒形成晶体。以这种方式形成的晶体具有来自先前已知形式的化合物的不同的熔点，红外光谱和X射线衍射图，并具有增强的可加工性，例如。稳定磨削。

36. 发明授权

US5318994A N-[2-(7-lower-alkoxynaphth-1-yl)ethyl]benzamides 失效
标题翻译： N- [2-（7-低级 - 烷氧基萘-1-基）乙基]苯甲酰胺
公开(公告)号：US5318994A
公开(公告)日：1994-06-07
申请号：US970578
申请日：1992-11-03
申请人： Jean Andrieux , Raymond Houssin , Said Yous , Beatrice Guardiola , Daniel Lesieur
发明人： Jean Andrieux , Raymond Houssin , Said Yous , Beatrice Guardiola , Daniel Lesieur
IPC分类号： A61K31/165 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/4015 , A61K31/403 , A61K31/404 , A61K31/415 , A61K31/4409 , A61K31/445 , A61K31/495 , A61K31/535 , A61K31/5375 , A61P17/00 , A61P25/00 , A61P25/18 , A61P25/28 , A61P35/00 , C07C217/60 , C07C233/17 , C07C233/22 , C07C233/60 , C07C233/73 , C07C237/08 , C07D207/12 , C07D207/27 , C07D209/42 , C07D213/81 , C07D233/60 , C07D241/44 , C07D295/14 , C07D295/15 , C07D333/38 , C07C235/00 , A61K31/15 , A61K31/16 , C07C233/00 , C07C237/00 , C07C239/00
CPC分类号： C07D295/15 , C07C217/60 , C07C233/22 , C07C233/60 , C07C233/73 , C07C237/08 , C07D207/12 , C07C2101/02 , C07C2101/04 , C07C2101/08 , C07C2101/14
摘要： Compounds of the formula: ##STR1## in which: A represents ##STR2## R represents linear or branched lower alkyl, R.sub.1 represents hydrogen or linear or branched lower alkyl, andR.sub.2 represents aryl or lower arylalkyl or aryl or lower arylalkyl substituted by lower alkyl, lower alkoxy, trifluoromethyl, or halogen, aryl means phenyl or naphthyl, as well as optical isomers, epimers and diastereoisomers and addition salts thereof with a pharmaceutically-acceptable acid, lower alkyl and lower alkoxy having 1 to 6 carbon atoms inclusive, andmedicaments containing the same which are useful for the treatment of disorders of the melatoninergic system.
摘要翻译：下式的化合物：其中：A表示直链或支链的低级烷基，R 1表示氢或直链或支链的低级烷基，R 2表示芳基或低级芳烷基或被低级烷基取代的芳基或低级芳烷基，低级烷氧基，三氟甲基或卤素，芳基是指苯基或萘基，以及光学异构体，差向异构体和非对映异构体及其与药学上可接受的酸，低级烷基和含1-6个碳原子的低级烷氧基的加成盐，以及药物含有相同的，可用于治疗褪黑激素系统的病症。

37. 发明授权

US5103010A Diphenylethylene derivatives, pharmaceutical compositions containing same and treatment method 失效
标题翻译：二氯乙烯衍生物，含有该药物的药物组合物和治疗方法
公开(公告)号：US5103010A
公开(公告)日：1992-04-07
申请号：US612829
申请日：1990-11-13
申请人： Youji Yamagishi , Kozo Akasaka , Takeshi Suzuki , Mitsuaki Miyamoto , Kouji Nakamoto , Kazuo Okano , Shinya Abe , Hironori Ikuta , Kenji Hayashi , Hiroyuki Yoshimura , Tohru Fujimori , Koukichi Harada , Isao Yamatsu
发明人： Youji Yamagishi , Kozo Akasaka , Takeshi Suzuki , Mitsuaki Miyamoto , Kouji Nakamoto , Kazuo Okano , Shinya Abe , Hironori Ikuta , Kenji Hayashi , Hiroyuki Yoshimura , Tohru Fujimori , Koukichi Harada , Isao Yamatsu
IPC分类号： C07C57/42 , A61K31/15 , A61K31/165 , A61K31/18 , A61K31/19 , A61K31/215 , A61K31/22 , A61K31/275 , A61K31/277 , A61K31/33 , A61P7/02 , A61P9/08 , A61P9/10 , C07C51/00 , C07C59/64 , C07C67/00 , C07C69/618 , C07C231/00 , C07C231/02 , C07C233/01 , C07C233/02 , C07C233/11 , C07C235/14 , C07C235/34 , C07C237/20 , C07C239/00 , C07C241/00 , C07C251/40 , C07C251/60 , C07C253/00 , C07C253/30 , C07C255/04 , C07C255/32 , C07C255/34 , C07C255/37 , C07C255/41 , C07C255/61 , C07C255/62 , C07C257/04 , C07C257/06 , C07C257/10 , C07C257/18 , C07C301/00 , C07C303/38 , C07C311/00 , C07C311/13 , C07C311/15 , C07C311/17 , C07C325/00 , C07C327/00 , C07C327/58 , C07D207/46 , C07D213/40 , C07D213/72 , C07D213/75 , C07D249/12 , C07D257/04 , C07D339/08 , C07D521/00
CPC分类号： C07D257/04 , C07C235/14 , C07C235/34 , C07C251/40 , C07C251/60 , C07C255/00 , C07C255/41 , C07C255/62 , C07C257/06 , C07C257/18 , C07C311/13 , C07C311/17 , C07C327/58 , C07C59/64 , C07D207/46 , C07D213/40 , C07D213/75 , C07D231/12 , C07D233/56 , C07D249/08 , C07D339/08
摘要： A new diphenyl-methane derivative is useful to inhibit agglomeration of blood and is defined by the formula, including a diphenylethylene derivative and a benzophenone oxime ether derivative. ##STR1## in which R1 and R2 each are hydrogen, hydroxyl or a lower alkoxy, U is .dbd.CXY or .dbd.N--O--W,X is hydrogen, cyano or --COR6, R6 being hydroxyl or an amino, Y is --R10--COOR3, R3 being hydrogen or a lower alkoxy, R10 being an alkylene having 1 to 3 carbon atoms, straight or branched, --CO--NR4R5, R4 and R5 each being hydrogen, a lower alkyl or a lower arylalkyl, --CH2--NHSO2--C6H5 or --C(R8).dbd.NR7, R7 being a lower alkoxy or an aryl, R8 is --VR9, V being oxygen, sulfur or nitrogen, R9 being an alkyl or an aryl,W is --CH2--CO--CH2--COOR13, R13 being hydrogen or a lower alkyl, --CH2--C(.dbd.NOR14)--CH2--COOR15, R15 being hydrogen or a lower alkyl, R14 being a lower alkyl, --CH(CN)--(CH2)q--COOR16, R16 being hydrogen or a lower alkyl, q being an integer of 1 to 3, or --(CH2)p--Z, Z being --SH, --SCN or a monovalent group derived from a five- or six-membered ring which may be substituted by a ring having one or more sulfur atoms in the ring, p being 1 or 2.
摘要翻译：二苯基甲烷衍生物。式（I）为新的（其中R 1和R 2各自为H，OH或低级烷氧基; U = -C XY或= NOW; X = H，CN或-COR 6; R 6 = OH或NH 2; Y = COOR 3，-CONR 4 R 5，-CH 2 NHSO 2 -C 6 H 5或-C（R 8）= NR 7; R 3 = H或低级烷氧基; R 10 =支链1-3C亚烷基; R 4和R 5各自为H，低级烷基或低级芳基烷基; 低级烷氧基或芳基; R8 = -VR9; V = O，S或N; R9 =烷基或芳基; W = -CH2-CO-CH2-COOR13，-CH2-C（= NOR14）-CH2-COOR15，-CH （CN） - （CH 2）q -COOR 16或 - （CH 2）pZ; R 13 = H或低级烷基; R 14 =低级烷基; R 15 = H或低级烷基; R 16 = H或低级烷基; q = = -SH，-SCN或衍生自5-或6-元环选择的单价gp，通过环中具有1个或更多个S的环; p = 1或2。

38. 发明授权

US5100987A Monoethylenically unsaturated compounds whose polymers are useful as photoinitiators 失效
标题翻译：聚合物作为光敏剂有用的单一不饱和化合物
公开(公告)号：US5100987A
公开(公告)日：1992-03-31
申请号：US603092
申请日：1990-10-25
申请人： Kevin B. Hatton , Edward Irving , Josephine M. A. Walshe , Anne Mallaband
发明人： Kevin B. Hatton , Edward Irving , Josephine M. A. Walshe , Anne Mallaband
IPC分类号： C07C67/00 , C07C69/54 , C07C69/738 , C07C235/74 , C07C235/78 , C07C237/08 , C07C239/00 , C07C271/16 , C07C323/12 , C07C323/22 , C07C323/36 , C07D295/10 , C07D295/108 , C07F9/40 , C07F9/44 , C08F20/00 , C08F20/10 , C08F20/26 , C08F20/30 , C08F20/34 , C08F20/36 , C08F30/02
CPC分类号： C07D295/108 , C07F9/4056 , Y10S430/136 , Y10S522/904 , Y10S522/905
摘要： Monethylenically unsaturated compounds whose polymers are useful as polymeric photoinitiators are of formula Ar.sup.1 COC(R.sup.1)(R.sup.2)R.sup.3 where R.sup.1 is C.sub.1 -C.sub.10 alkyl or alkoxy, R.sup.2 is C.sub.1 -C.sub.10 alkyl, --X--O--R.sup.4 --OCOC(R.sup.5).dbd.CH.sub.2 (II) --X--NH--R.sup.6 --OCOC(R.sup.5).dbd.CH.sub.2 (III), or --CH.sub.2 [OCH.sub.2 CH(OH)CH.sub.2 ].sub.a OCOC(R.sup.5).dbd.CH.sub.2 (IIIA) or R.sup.1 and R.sup.2, together with the attached carbon, denote C.sub.4 -C.sub.8 cycloalkyl, R.sup.3 is a C.sub.6 -C.sub.20 aromatic group, OH, tert.amino, --OCOC(R.sup.5).dbd.CH.sub.2 (VI) or --OCH.sub.2 CH(OH)CH.sub.2 OCOC(R.sup.5).dbd.CH.sub.2 (VIA), R.sup.4 is C.sub.1 -C.sub.4 alkylene, which may be substituted by --OH or by C.sub.2 -C.sub.20 acyloxy, R.sup.5 is H or C.sub.1 -C.sub.4 alkyl, R.sup.6 is C.sub.1 to C.sub.4 alkylene, X is a group of formula R.sup.7 CO-- or ##STR1## where R.sup.7 is C.sub.1 -C.sub.4 alkylene, R.sup.8 is C.sub.1 to C.sub.4 alkyl, and is 0 or 1, Ar.sup.1 is a C.sub.6 -C.sub.20 aromatic group, with the provisos that (i) R.sup.2, R.sup.3 or Ar.sup.1 contains a group (VI), (ii) where R.sup.1 and R.sup.2 together with the attached carbon atom denote cycloalkyl, R.sup.3 is --OH, tert.amino or a group VI or VIA (iii) when R.sup.2 is a group II, a is 0, (iv) when R.sup.2 is a group III a is 1, (v) when R.sup.2 denotes a group IIIA, R.sup.3 denotes said monovalent aromatic group (vi) when R.sup.3 denotes a group VI, R.sup.1 and R.sup.2 together with the attached carbon denote C.sub.4 -C.sub.8 cycloalkyl, (vii) when Ar.sup.1 contains a group VI R.sup.1 is --CH.sub.3 and R.sup.3 is --OH, R.sup.2 is C.sub.2 -C.sub.10 alkyl, and (viii) when Ar.sup.1 contains a group VI, R.sup.1 and R.sup.2 are each alkyl and R.sup.3 is --OH, the group VI is linked to an aromatic C atom in Ar.sup.1 through a group --YR.sup.10 OR.sup.9 -- or --YR.sup.10 OCONHR.sup.6 --, Y being attached to an aromatic C atom, where Y is O or S, R.sup.9 is 2-hydroxypropylene or 2-(C.sub.2 -C.sub.20 acyloxy)propylene and R.sup.10 is C.sub.1 -C.sub.4 alkylene.

39. 发明授权

US5085975A Radiation sensitive composition utilizing ethylenically unsaturated perfluoroalkyl group-containing compounds and reproduction layers produced therefrom 失效
标题翻译：辐射敏感组合物利用乙烯基不饱和全氟烷基基团的化合物和生产的复合物
公开(公告)号：US5085975A
公开(公告)日：1992-02-04
申请号：US426490
申请日：1989-10-23
申请人： Werner H. Mueller
发明人： Werner H. Mueller
IPC分类号： G03F7/038 , C07C67/00 , C07C69/54 , C07C69/62 , C07C69/76 , C07C233/20 , C07C239/00 , C08F20/24 , G03F7/00 , G03F7/004
CPC分类号： C08F20/24 , G03F7/0046
摘要： Polymerizable compounds comprising perfluoroalkyl groups, reproduction layers containing these compounds, and use of the reproduction layers for waterless offset printing. The novel polymerizable compounds comprise at least two acryloyl or methacryloyl groups and at least one perfluoroalkyl group which is linked to the molecule through a functional group, in particular, an ester or amide function. The compounds can be prepared, for example, from hydroxyl group-containing acrylates or methacrylates and perfluoroalkyl group-containing carboxylic acid chlorides, in the presence of an amine or from perfluoroalkyl group-containing carboxylic acid derivatives and reactive acryloyloxy or methacryloyloxy compounds. Oligomeric compounds can additionally be synthesized from the above-mentioned compounds by linking, for example, with diisocyanates. The compounds are particularly used in radiation-sensitive reproduction layers which also contain at least one photoinitiator and, optionally, at least one organic polymeric binder. Reproduction layers of this kind are applied as radiation-sensitive coatings to support materials for printing plates used in waterless offset printing.
摘要翻译：包含全氟烷基的可聚合化合物，含有这些化合物的再生层，以及再生层用于无水胶印的用途。新型可聚合化合物包含至少两个丙烯酰基或甲基丙烯酰基和至少一个通过官能团，特别是酯或酰胺官能团与分子连接的全氟烷基。化合物可以由例如含羟基的丙烯酸酯或甲基丙烯酸酯和含全氟烷基的羧酸氯化物在胺或含全氟烷基的羧酸衍生物和反应性丙烯酰氧基或甲基丙烯酰氧基化合物的存在下制备。另外从上述化合物可以通过例如与二异氰酸酯连接来合成低聚化合物。这些化合物特别用于还含有至少一种光引发剂和任选的至少一种有机聚合物粘合剂的辐射敏感繁殖层中。这种复制层被用作辐射敏感涂层，以支持无水胶版印刷中使用的印版的材料。

40. 发明授权

US5073184A Fungicidal thienyl propenoates 失效
标题翻译：杀真菌三烯丙酸酯
公开(公告)号：US5073184A
公开(公告)日：1991-12-17
申请号：US506152
申请日：1990-04-09
申请人： Vivienne M. Anthony , John M. Clough , Paul deFraine , Christopher R. A. Godfrey , Kevin Beautement
发明人： Vivienne M. Anthony , John M. Clough , Paul deFraine , Christopher R. A. Godfrey , Kevin Beautement
IPC分类号： C07C241/00 , A01N37/36 , A01N37/42 , A01N37/44 , A01N37/48 , A01N43/06 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/38 , A01N43/58 , C07C67/00 , C07C69/734 , C07C201/00 , C07C205/56 , C07C229/64 , C07C233/58 , C07C239/00 , C07C245/06 , C07C251/02 , C07C251/44 , C07C253/00 , C07C255/57 , C07C255/59 , C07C309/63 , C07C313/00 , C07C323/54 , C07D207/32 , C07D207/337 , C07D207/34 , C07D209/18 , C07D307/42 , C07D307/54 , C07D307/79 , C07D333/24 , C07D333/32 , C07D333/34 , C07D333/38 , C07D333/60 , C07F7/18
CPC分类号： C07D207/337 , A01N43/06 , A01N43/36 , A01N43/38 , A01N43/58 , C07D209/18 , C07D307/54 , C07D307/79 , C07D333/24 , C07D333/60
摘要： Compounds of formula (I): ##STR1## and stereoisomers thereof, wherein W is R.sup.1 O.sub.2 C--C.dbd.CH--ZR.sup.2, wherein R.sup.1 and R.sup.2, which are the same or different, are alkyl or fluoroalkyl groups, and Z is either an oxygen or sulphur atom; A is an oxygen or sulphur atom, --NR.sup.3 --, or --CR.sup.4 R.sup.5 --; X, Y and Z.sup.1, which are the same or different, are hydrogen or halogen atoms, or hydroxy, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl, optionally substituted aralkyl, optionally substituted heteroarylalkyl, optionally substituted aryloxyalkyl, optionally substituted heteroaryloxyalkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted alkoxy, optionally substituted arylalkoxy, optionally substituted aryloxy, optionally substituted heteraryloxy, optionally substituted acyloxy, optionally substituted amino, optionally substituted acylamino, optionally substituted arylazo, nitro, cyano, --CO.sub.2 R.sup.6, --CONR.sup.7 R.sup.8, --COR.sup.9 --CR.dbd.NR.sup.10, --CR.dbd.NOR.sup.10 or --N.dbd.CR.sup.11 R.sup.12 groups; or the groups X and Y, when they are in adjacent positions on the ring, optionally join to form a fused ring, either aromatic or aliphatic, optionally containing one or more heteroatoms; and R, R.sup.3, R.sup.4, R.sup.5, R.sup.6, R.sup.7, R.sup.8, R.sup.9, R.sup.10, R.sup.11 and R.sup.12, which are the same or different, are hydrogen atoms (provided that R.sup.4 and R.sup.5 are not hydrogen) or optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl, optionally substituted aralkyl, optionally substituted heterarylalkyl, optionally substituted aryloxyalkyl, optionally substituted heteroaryloxyalkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted aryl or optionally substituted heteroaryl groups; and metal compelxes thereof.The compounds are useful in agriculture, especially as fungicides but also as insecticides and plant growth regulators.

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