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21. 发明申请

US20080207950A1 Enantioselective Synthesis of a Sterically Hindered Amine 审中-公开
标题翻译：对映选择性合成受阻胺
公开(公告)号：US20080207950A1
公开(公告)日：2008-08-28
申请号：US11792744
申请日：2005-12-12
申请人： Ulrich Berens , Christophe Malan , Hans Jurg Kirner
发明人： Ulrich Berens , Christophe Malan , Hans Jurg Kirner
IPC分类号： C07C209/00 , C07C209/24 , C07C231/00
CPC分类号： C07C231/18 , C07C209/50 , C07C233/13 , C07C2601/04 , C07C211/29
摘要： Compounds of the formula (I) wherein R is phenyl, or phenyl substituted by Cl, Br, C1-C4alkyl or CF3; R1 is H or methyl or ethyl; R2 is H or methyl or acyl; R3 is H or methyl; R′4 is —CH3 or ═CH2; may be obtained in high enantiopurity by hydrogenation of a compound of the formula (II) wherein R and R3 are as in formula (I); A is acyl; and R4 is —CH3 or ═CH2; in the presence of a chiral Rhodium or Ruthenium catalyst. Residues R1 as methyl or ethyl and/or R2 as H or methyl may subsequently be introduced without racemization by deacylation and optional alkylation.
摘要翻译：其中R是苯基的式（I）化合物或被Cl，Br，C 1 -C 4烷基或CF 3取代的苯基， ; R 1是H或甲基或乙基; R 2是H或甲基或酰基; R 3是H或甲基; R'4是-CH 3或-CH 2; 可以通过氢化其中R和R 3如式（I）中的式（II）化合物的高对映体纯度获得; A是酰基; 且R 4为-CH 3或-CH 2 2; 在手性铑或钌催化剂存在下。可以随后引入作为甲基或乙基的残基R 1，和/或作为H或甲基的R 2 2，通过脱酰基和任选的烷基化引入外消旋。

22. 发明授权

US5936109A Ligands for asymmetric catalysis 失效
标题翻译：不对称催化配体
公开(公告)号：US5936109A
公开(公告)日：1999-08-10
申请号：US893105
申请日：1997-07-15
申请人： Ulrich Berens
发明人： Ulrich Berens
IPC分类号： B01J31/24 , C07B53/00 , C07C45/50 , C07F20060101 , C07F9/6568 , C07F15/00 , C07F17/02 , C07F9/02
CPC分类号： C07F17/02 , C07B53/00 , C07C45/505 , C07F15/008 , C07F9/65683
摘要： The subject invention relates to phosphine ligands that are useful for asymmetric reactions, especially as chiral ligands for catalytic asymmetric hydrogenation.
摘要翻译：本发明涉及可用于不对称反应的膦配体，特别是用于催化不对称氢化的手性配体。

23. 发明授权

US08822702B2 Synthesis of amines and intermediates for the synthesis thereof 有权
标题翻译：合成胺及其合成中间体
公开(公告)号：US08822702B2
公开(公告)日：2014-09-02
申请号：US13098535
申请日：2011-05-02
申请人： Ulrich Berens , Oliver Dosenbach , Daniel Sprenger
发明人： Ulrich Berens , Oliver Dosenbach , Daniel Sprenger
IPC分类号： C07D209/12 , C07D209/38
CPC分类号： C07D409/04 , C07D209/16 , C07D209/18 , C07D209/38
摘要： The invention relates in a first embodiment to a method for the manufacture of esters of the formula I, or especially of amides of the formula II, wherein the symbols have the meanings given in the specification, as well as other intermediates and compounds useful in the synthesis of tryptamines and other substances mentioned in the title. The synthesis methods and intermediates are useful in the synthesis of pharmaceuticals.
摘要翻译：本发明在第一个实施方案中涉及制备式I酯，特别是式II的酰胺的方法，其中符号具有说明书中给出的含义，以及其它中间体和化合物标题中提及的色胺和其他物质的合成。合成方法和中间体在药物的合成中是有用的。

24. 发明授权

US08758880B2 Ketopyrroles as organic semiconductors 有权
标题翻译：酮基吡咯酮作为有机半导体
公开(公告)号：US08758880B2
公开(公告)日：2014-06-24
申请号：US12680920
申请日：2008-10-16
申请人： Jean-Charles Flores , Ulrich Berens , Frank Bienewald , Hans Jürg Kirner , Mathieu G. R. Turbiez
发明人： Jean-Charles Flores , Ulrich Berens , Frank Bienewald , Hans Jürg Kirner , Mathieu G. R. Turbiez
IPC分类号： H01L35/24
CPC分类号： H01L51/0036 , C08G61/123 , C08G61/124 , H01L51/0043 , H01L51/0545 , Y02E10/549 , Y10T428/24802
摘要： Monomeric or polymeric compounds comprising at least one moiety of the formula (Ia) wherein X is CR, where R is H or a substituent as defined in claim 1, or is another ketopyrrole moiety e.g. of the formula (Ib) or (Ic) with this moiety and all other symbols are as defined in claim 1, show good solubility in organic solvents and excellent film-forming properties. In addition, high efficiency of energy conversion, excellent field-effect mobility, good on/off current ratios and/or excellent stability can be observed, when the polymers according to the invention are used in semiconductor devices or organic photovoltaic (PV) devices (solar cells).
摘要翻译：包含至少一个式（Ia）部分的单体或聚合化合物，其中X是CR，其中R是H或如权利要求1所定义的取代基，或者是另一个酮基吡咯部分。式（Ib）或（Ic）与该部分和所有其它符号如权利要求1中所定义，在有机溶剂中表现出良好的溶解性和优异的成膜性能。此外，当根据本发明的聚合物用于半导体器件或有机光伏（PV）器件时，可以观察到高的能量转换效率，优异的场效应迁移率，良好的导通/截止电流比和/或优异的稳定性太阳能电池）。

25. 发明申请

US20130059723A1 Synthesis of Zeolitic Materials using N,N-Dimethyl Organotemplates 有权
标题翻译：使用N，N-二甲基有机模板合成沸石材料
公开(公告)号：US20130059723A1
公开(公告)日：2013-03-07
申请号：US13605701
申请日：2012-09-06
申请人： Bilge Yilmaz , Ulrich Berens , Vijay Narayanan Swaminathan , Ulrich Müller , Gabriele Iffland , Laszlo Szarvas
发明人： Bilge Yilmaz , Ulrich Berens , Vijay Narayanan Swaminathan , Ulrich Müller , Gabriele Iffland , Laszlo Szarvas
IPC分类号： C01B39/00 , B01D53/94 , C01B39/54 , B01J29/04 , C10G11/05 , C07C1/22
CPC分类号： C10G3/49 , B01D53/9413 , B01D53/9436 , B01D2255/50 , B01J29/70 , B01J29/7015 , B01J29/85 , B01J29/86 , B01J29/87 , B01J2229/183 , C01B39/48 , C01B39/54 , C07C1/20 , C07C2529/70 , C10G11/05 , C10G11/18 , C10G25/03 , C10G2300/405 , Y02C20/10 , C07C11/02
摘要： The present invention relates to a process for the preparation of a zeolitic material having a structure comprising YO2 and optionally comprising X2O3, preferably comprising YO2 and X2O3, wherein said process comprises the steps of (1) providing a mixture comprising one or more ammonium compounds of which the ammonium cation has the formula (I): [R1R2NR3R4]+ (I) and further comprising one or more sources for YO2 and one or more sources for X2O3; (2) crystallizing the mixture provided in (1); wherein Y is a tetravalent element, and X is a trivalent element, and wherein in formula (I) R1 and R2 are independently from one another derivatized or underivatized methyl, and R3 and R4 are independently from one another derivatized or underivatized (C3-C5)alkyl, and wherein the molar ratio of ammonium cation having the formula (I) to Y in the mixture provided in step (1) and crystallized in step (2) is equal to or greater than 0.25.
摘要翻译：本发明涉及一种制备具有包含YO 2和任选地包含X 2 O 3，优选包含YO 2和X 2 O 3的结构的沸石材料的方法，其中所述方法包括以下步骤：（1）提供包含一种或多种铵化合物其中铵阳离子具有式（I）：[R 1 R 2 NR 3 R 4] +（I），并且还包含一种或多种YO源和一种或多种X 2 O 3源; （2）使（1）中提供的混合物结晶; 其中Y是四价元素，X是三价元素，并且其中在式（I）中，R 1和R 2彼此独立地是衍生的或未衍生的甲基，并且R 3和R 4彼此独立地是衍生的或未衍生的（C 3 -C 5 ）烷基，并且其中在步骤（1）中提供并在步骤（2）中结晶的混合物中具有式（I）的铵阳离子与Y的摩尔比等于或大于0.25。

26. 发明授权

US08101776B2 Organic semiconductors and their manufacture 有权
标题翻译：有机半导体及其制造
公开(公告)号：US08101776B2
公开(公告)日：2012-01-24
申请号：US12086157
申请日：2006-12-04
申请人： Ulrich Berens , Frank Bienewald , Hans Jürg Kirner
发明人： Ulrich Berens , Frank Bienewald , Hans Jürg Kirner
IPC分类号： C07D277/60
CPC分类号： H01L51/0071 , C07D471/04 , C07D487/04 , C07D493/04 , C07D495/04 , C07D495/22 , C07D513/04 , C09B5/026 , C09B5/14 , C09B5/60 , C09B57/00 , C09B69/008 , H01L51/0058 , H01L51/0067 , H01L51/0068 , H01L51/0069 , H01L51/0074 , H01L51/0083 , H01L51/0094 , H01L51/0525 , H01L51/0545
摘要： The invention relates to a semiconductor device comprising a compound of the formula I and of the formula XXI, wherein the symbols have the meanings defined in the specification, to the novel compounds of the formula I and XXI and to the use of such a compound as an organic semiconductor for the preparation of an electronic device, and further compounds and devices, as well as other embodiments given in the specification.
摘要翻译：本发明涉及一种半导体器件，其包含式I和式XXI的化合物，其中符号具有本说明书中定义的含义与式I和XXI的新型化合物以及使用这样的化合物用于制备电子器件的有机半导体，以及本说明书中给出的其它化合物和器件以及其它实施方案。

27. 发明授权

US07645886B2 Synthesis of amines and intermediates for the synthesis thereof 有权
标题翻译：合成胺及其合成中间体
公开(公告)号：US07645886B2
公开(公告)日：2010-01-12
申请号：US10539151
申请日：2003-12-12
申请人： Ulrich Berens , Oliver Dosenbach , Daniel Sprenger
发明人： Ulrich Berens , Oliver Dosenbach , Daniel Sprenger
IPC分类号： C07D209/38 , C07D209/18
CPC分类号： C07D409/04 , C07D209/16 , C07D209/18 , C07D209/38
摘要： The invention relates in a first embodiment to a method for the manufacture of esters of the formula (I), or especially of amides of the formula (II), wherein the symbols have the meanings given in the specification, as well as other intermediates and compounds useful in the synthesis of tryptamines and other substances mentioned in the title. The synthesis methods and intermediates are useful in the synthesis of pharmaceuticals.
摘要翻译：本发明在第一个实施方案中涉及一种制备式（I）酯或特别是式（II）的酰胺的酯的方法，其中符号具有说明书中给出的含义以及其它中间体和可用于合成标准物中提及的色胺和其他物质的化合物。合成方法和中间体在药物的合成中是有用的。

28. 发明授权

US07407910B2 Ligands for asymmetric reactions 失效
标题翻译：不对称反应配体
公开(公告)号：US07407910B2
公开(公告)日：2008-08-05
申请号：US11473035
申请日：2006-06-23
申请人： Ulrich Berens
发明人： Ulrich Berens
IPC分类号： B01J27/00 , C07D233/00
CPC分类号： C07F15/008 , B01J31/1845 , B01J31/1865 , B01J31/187 , B01J31/226 , B01J31/2471 , B01J2231/321 , B01J2231/323 , B01J2231/52 , B01J2231/643 , B01J2531/80 , B01J2531/821 , B01J2531/822 , B01J2531/824 , B01J2531/827 , B01J2531/828 , B01J2531/845 , B01J2531/847 , C07B53/00 , C07C45/505 , C07F9/6506 , C07F9/65517 , C07F9/655354 , C07F9/65683 , C07F9/65719 , C07F15/00 , C07F15/0073
摘要： The invention relates to a process for the manufacture of bidentate ligands of the formula IA and IIA, characterized in that N,N-(optionally substituted) dialkylamino phosphines bound to an aromatic carbon are lithiated in ortho-position and the lithiated compounds are further converted to said bidentate ligands: wherein X1 is NR, O or S; X2 is CHR1 or CR1; X3 is CHR2 or NR2 or, if X2 is CR1, X3 is CR2 or N; and R, R1 and R2 are radicals such as alkyl groups or R1 and R2 together form an annealed ring; Y1*, Y2* and Y1′* are, independently of each other, an element of the fifth group of the periodic table of elements as such or in thioxo or oxo form; Z1*, Z2*, Z3*, Z4*, Z1′*, Z2′* are, independently of each other, for example halogen, hydrogen, or an unsubstituted or substituted moiety selected from radicals such as alkyl groups; the substituents have otherwise the meanings given in the specification; and the ligands are capable of forming metal complexes, which can be used as catalysts in stereoselective synthesis, especially hydrogenation, of various organic molecules.
摘要翻译：本发明涉及制备式IA和IIA的二齿配体的方法，其特征在于与邻位连接的与芳族碳键合的N，N-（任选取代的）二烷基氨基膦进一步转化，并且锂化合物进一步转化所述二齿配体：其中X 1是NR，O或S; X 2是CHR 1或CR 1; X 3是CHR 2或NR 2 2，或者如果X 2是CR 1，则 >，X 3是CR 2 N或N; 和R 1，R 1和R 2是基团，例如烷基或R 1和R 2共同形成退火环; Y 1 *，Y 2 *和Y 1 *彼此独立地是元素周期表第五组元素元素，或硫代或氧代形式; Z 1，Z 2，Z 3，Z 4，Z 1，Z 3， Z 2是独立的，例如卤素，氢或选自基团如烷基的未取代或取代的部分; 取代基另有说明书中给出的含义; 并且配体能够形成金属络合物，其可以用作各种有机分子的立体选择性合成，特别是氢化中的催化剂。

29. 发明申请

US20070173536A1 Crystalline forms of zolmitriptan 审中-公开
标题翻译：唑来曲坦的结晶形式
公开(公告)号：US20070173536A1
公开(公告)日：2007-07-26
申请号：US10588176
申请日：2005-01-28
申请人： Paul Van Der Schaaf , Fritz Blatter , Martin Szelagiewicz , Ulrich Berens , Susan De Paul
发明人： Paul Van Der Schaaf , Fritz Blatter , Martin Szelagiewicz , Ulrich Berens , Susan De Paul
IPC分类号： A61K31/422 , C07D413/02
CPC分类号： C07D413/06
摘要： The present invention is directed to a novel crystalline form of Zolmitriptan, herein designated as Form A, and several novel solvates of Zolmitriptan, herein designated as Form B, C, D, E, F, and G, processes for the preparation thereof and pharmaceutical compositions comprising these crystalline forms.
摘要翻译：本发明涉及Zolmitriptan的新型结晶形式，本文命名为A型，以及佐米曲坦的几种新型溶剂合物，本文命名为B型，C，D，E，F和G型，其制备方法和药物包含这些结晶形式的组合物。

30. 发明申请

US20060058367A1 Synthesis of amines and intermediates for the synthesis thereof 有权
标题翻译：合成胺及其合成中间体
公开(公告)号：US20060058367A1
公开(公告)日：2006-03-16
申请号：US10539151
申请日：2003-12-12
申请人： Ulrich Berens , Oliver Dosenbach , Daniel Sprenger
发明人： Ulrich Berens , Oliver Dosenbach , Daniel Sprenger
IPC分类号： A61K31/405 , A61K31/407 , C07D209/36 , C07D209/18
CPC分类号： C07D409/04 , C07D209/16 , C07D209/18 , C07D209/38
摘要： The invention relates in a first embodiment to a method for the manufacture of esters of the formula (I), or especially of amides of the formula (II), wherein the symbols have the meanings given in the specification, as well as other intermediates and compounds useful in the synthesis of tryptamines and other substances mentioned in the title. The synthesis methods and intermediates are useful in the synthesis of pharmaceuticals.
摘要翻译：本发明在第一个实施方案中涉及一种制备式（I）酯或特别是式（II）的酰胺的酯的方法，其中符号具有说明书中给出的含义以及其它中间体和可用于合成标准物中提及的色胺和其他物质的化合物。合成方法和中间体在药物的合成中是有用的。

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