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11. 发明申请

US20030176363A1 Novel compounds and methods 失效
标题翻译：新型化合物和方法
公开(公告)号：US20030176363A1
公开(公告)日：2003-09-18
申请号：US10338679
申请日：2003-01-09
申请人： PharmAxis Pty Ltd.
发明人： William Butler Cowden , Bart Michael Eschler , Darren Ray March , Douglas John Francis , Sendaba Gerba , Gavin James Bartell , Brett Charlton
IPC分类号： A61K031/7024 , C07H005/06
CPC分类号： C07H11/04 , C07F9/6552 , C07F9/65586
摘要： The present invention provides phosphotetrahydropyran compounds and the use thereof in treating diseases or conditions that are dependent on T-lymphocyte migration, as well as compositions containing said compounds.
摘要翻译：本发明提供磷酸四氢吡喃化合物及其在治疗依赖于T淋巴细胞迁移的疾病或病症中的用途，以及含有所述化合物的组合物。

12. 发明申请

US20030114392A1 Process for preparing pseudoephedrine tannate 失效
标题翻译：制备假麻黄碱的方法
公开(公告)号：US20030114392A1
公开(公告)日：2003-06-19
申请号：US10326361
申请日：2002-12-20
申请人： Jame Fine Chemicals, Inc.
发明人： Sham N. Redkar , James R. Schleck , Vilas M. Chopdekar
IPC分类号： A61K031/7024 , C07H013/02
CPC分类号： A61K45/06 , A61K31/137 , A61K31/44 , A61K31/7024 , Y10S514/849 , A61K2300/00
摘要： The invention pertains to a method for preparing pseudoephedrine tannate by reacting pseudoephedrine free base at a temperature of about 70 to about 110null C. with tannic acid neat or as an aqueous slurry containing about 5 to about 30 wt. % water.
摘要翻译：本发明涉及一种通过在约70至约110℃的温度下将无麻黄碱游离碱与纯鞣酸或作为含约5至约30重量％的鞣酸的含水浆液反应来制备鞣酸假麻黄碱的方法。％水。

13. 发明申请

US20030040491A1 Use of pentosan polysulfate to treat certain conditions of the prostate 失效
公开(公告)号：US20030040491A1
公开(公告)日：2003-02-27
申请号：US10209331
申请日：2002-07-30
申请人： The U.S. of America, as represented by the Secretary, Dept. of Health & Human Services
发明人： Gary E. Striker
IPC分类号： A61K031/7024
CPC分类号： A61K31/715 , A61K31/737
摘要： The invention relates to the field of pharmacology. More particularly, the invention relates to the treatment of prostate conditions, such as BPH. The invention provides new therapeutic compositions and methods for treating BPH, as well as chronic prostatitis, prostadynia, and irritative bladder conditions, other than interstitial cystitis. The compositions and methods according to the invention, which may be administered orally, efficaciously and safely treat the designated conditions by causing regression of established lesions and reduction of bladder irritation. In particular, the compositions and methods of the invention treat BPH by reducing the size of the prostate gland and decreasing the associated obstructive symptoms.

14. 发明申请

US20030032602A1 Methods and compositions for collagen homeostasis 审中-公开
标题翻译：胶原体内稳态的方法和组合物
公开(公告)号：US20030032602A1
公开(公告)日：2003-02-13
申请号：US09927764
申请日：2001-08-09
发明人： Dusan Miljkovic
IPC分类号： A61K031/7024 , A61K009/127
CPC分类号： A61K8/60 , A61K8/14 , A61K8/19 , A61K8/44 , A61K8/676 , A61K2800/782 , A61Q19/00 , A61Q19/08
摘要： Methods and compositions are directed to a cosmetic preparation comprising a collagenase inhibitor at a concentration effective to reduce a collagenase activity in a skin, wherein the inhibitor comprises boron. Particularly contemplated compositions are topically applied to the skin, and may further comprise a skin penetration enhancer and/or have the collagenase inhibitor formulated in a liposome formulation.
摘要翻译：方法和组合物涉及包含胶原酶抑制剂的化妆品制剂，其浓度有效降低皮肤中的胶原酶活性，其中抑制剂包含硼。特别考虑的组合物局部施用于皮肤，并且还可以包含皮肤渗透增强剂和/或配制在脂质体制剂中的胶原酶抑制剂。

15. 发明申请

US20020107208A1 Gabapentin prodrugs and formulations 失效
标题翻译：加巴喷丁前药和制剂
公开(公告)号：US20020107208A1
公开(公告)日：2002-08-08
申请号：US10040251
申请日：2001-10-23
发明人： Chih-Ming Chen , Jane Chen
IPC分类号： A61K031/7024 , A61K031/195 , A61K031/215
CPC分类号： C07C229/28 , A61K9/0004 , A61K31/221 , C07C2601/14
摘要： The present invention relates to novel prodrugs of gabapentin and to pharmaceutical formulations and sustained release formulations containing the prodrugs.
摘要翻译：本发明涉及加巴喷丁的新型前药和含有前体药物的药物制剂和持续释放制剂。

16. 发明申请

US20020094960A1 Anticonvulsant derivatives useful for the treatment of depression 失效
标题翻译：用于治疗抑郁症的抗惊厥药物
公开(公告)号：US20020094960A1
公开(公告)日：2002-07-18
申请号：US09916742
申请日：2001-07-27
发明人： Carlos R. Plata-Salaman , Josue Bacaltchuk , Pedro A.S. Prado-Lima
IPC分类号： A61K031/7024 , A61K031/35 , A61K031/357 , A61K031/255
CPC分类号： A61K31/7048 , A61K31/255 , A61K31/35 , A61K31/357 , A61K31/7024
摘要： Anticonvulsant derivatives useful for treating depression as monotherapy or combination therapy are disclosed.
摘要翻译：公开了用于治疗抑郁症作为单一疗法或组合疗法的抗惊厥药物。

17. 发明申请

US20020082222A1 Treatments for neurogenetic disorders, impulse control disorder, and wound healing 审中-公开
标题翻译：治疗神经源性疾病，冲动控制障碍和伤口愈合
公开(公告)号：US20020082222A1
公开(公告)日：2002-06-27
申请号：US09997447
申请日：2001-11-30
发明人： Nathan Andrew Shapira , Mary Catherine Lessig , Daniel John Driscoll
IPC分类号： A61K031/7024 , A61K031/351 , A61K031/255
CPC分类号： A61K31/00 , A61K31/18 , A61K31/255 , A61K31/35 , A61K31/351 , A61K31/357 , A61K31/7024
摘要： The subject invention provides methods and compositions for the treatment of neurogenetic disorders, particularly DSM-IV impulse control disorders such as intermittent explosive disorder, kleptomania, pyromania, pathologic gambling, trichotillomania, and other impulse control disorders such as compulsive buying and problematic Internet use. In a preferred embodiment, the subject invention provides methods for treating or controlling symptoms associated with ADHD or PWS comprising the administration of therapeutically effective amounts of compositions containing compounds of the formulas I-V. In another embodiment, the subject invention provides for methods of promoting wound healing comprising the administration of a therapeutically effective amount of a composition comprising the compounds of formulas I-V. Compositions may administered to a wound site via a salve, ointment, or as a component of a bandage or bioadhesive applied to the site of injury. The invention also provides therapeutically effective compositions comprising one or more of the compounds of formulas I-V.
摘要翻译：本发明提供了用于治疗神经源性疾病，特别是DSM-IV脉冲控制障碍（例如间歇性爆发性疾病，克雷帕托尼亚，pyromania，病理性赌博，拔毛病等）和诸如强迫性购买和有问题的因特网使用的其它冲动控制障碍的方法和组合物。在一个优选的实施方案中，本发明提供了治疗或控制与ADHD或PWS相关的症状的方法，包括施用治疗有效量的含有式I-V化合物的组合物。在另一个实施方案中，本发明提供促进伤口愈合的方法，包括施用治疗有效量的包含式I-V化合物的组合物。组合物可以通过药膏，软膏或作为施用于损伤部位的绷带或生物粘合剂的组分施用于伤口部位。本发明还提供包含一种或多种式I-V化合物的治疗有效组合物。

18. 发明申请

US20020034558A1 Compositions in the form of water-in-oil emulsions and their use as cosmetics 审中-公开
标题翻译：油包水乳液形式的组合物及其作为化妆品的用途
公开(公告)号：US20020034558A1
公开(公告)日：2002-03-21
申请号：US09848412
申请日：2001-05-04
申请人： L' OREAL
发明人： Odile Sonneville-Aubrun , Jean-Thierry Simonnet
IPC分类号： A61K035/78 , A61K031/7024
CPC分类号： A61Q19/00 , A61K8/064 , A61K8/31 , A61K8/585 , A61K8/602 , A61K8/92 , A61Q19/007
摘要： The invention relates to a composition in the form of a water-in-oil emulsion containing at least 80% of aqueous phase and at least one glycoglyceride. The glycoglyceride may be obtained by synthesis or by extraction, and it may be, in particular, a galactolipid such as, for example, digalactosyl diglyceride or monogalactosyl diglyceride. The composition according to the invention provides a great sensation of freshness when applied to the skin, and may be used in particular in cosmetics and/or dermatology.
摘要翻译：本发明涉及含有至少80％的水相和至少一种甘油三酯的油包水乳液形式的组合物。甘油酸甘油酯可以通过合成或提取获得，特别可以是半乳糖脂，例如双乳糖二甘油二酯或单半乳糖基甘油二酯。当应用于皮肤时，根据本发明的组合物提供了很大的新鲜感，并且可以特别用于化妆品和/或皮肤病学。

19. 发明申请

US20020032164A1 Antimicrobial compounds and methods for their use 审中-公开
标题翻译：抗菌化合物及其使用方法
公开(公告)号：US20020032164A1
公开(公告)日：2002-03-14
申请号：US09847654
申请日：2001-05-03
发明人： Roderic M. K. Dale , Steven L. Gatton , Amy Arrow , Terry Thompson
IPC分类号： A61K048/00 , A61K031/7068 , A61K031/7076 , A61K031/7024 , A61K031/675
CPC分类号： A61K31/66 , A01N57/12 , A01N57/16 , A61K9/0014 , A61K31/70
摘要： The present invention provides protonated compounds having antimicrobial activity. The invention also provides antimicrobial compositions comprising protonated compounds of the invention. The protonated compounds of the invention provide efficacious antimicrobial activity against resistant strains of bacteria and opportunistic fungi.
摘要翻译：本发明提供具有抗微生物活性的质子化化合物。本发明还提供包含本发明的质子化化合物的抗微生物组合物。本发明的质子化化合物为细菌和机会真菌的抗性菌株提供有效的抗微生物活性。

20. 发明申请

US20040258773A1 Composition and methods for treating subjects with hyperglycemia 审中-公开
标题翻译：用于治疗高血糖患者的组合物和方法
公开(公告)号：US20040258773A1
公开(公告)日：2004-12-23
申请号：US10487904
申请日：2004-07-30
发明人： Xiaozhuo Chen , Fang Liu , Yungsheng Li , Jing Li
IPC分类号： A61K035/78 , A61K031/7024
CPC分类号： A61K31/7024 , A61K36/185
摘要： A partially purified plant extract for treating subjects who are hyperglycemic is provided. The partially-purified plant extract comprises a plurality of water soluble compounds having a molecular weight greater than 800 and less than 1500 grams/mole. One of the compounds in the partially-purified plant extract is the hydrolysable gallotannin known as penta-O-galloyl-D-glucose. The partially-purified plant extract is substantially free of triterpenoids, including corosolic acid and high molecular weight ellagitannins, i.e., ellagitannins having a molecular weight of greater than 1500 grams/mole. In a highly preferred embodiment, the partially purified plant extract is derived from the tropical plant Lagerstroemia Speciosa. L, which is also known as banaba. The present invention also relates to a method of using the present partially-purified extract to treat subjects who are hyperglycemic.
摘要翻译：提供了用于治疗高血糖患者的部分纯化的植物提取物。部分纯化的植物提取物包含分子量大于800且小于1500克/摩尔的多种水溶性化合物。部分纯化的植物提取物中的一种化合物是称为五-O-酰基-D-葡萄糖的可水解的gal单宁。部分纯化的植物提取物基本上不含三萜类化合物，包括科罗索酸和高分子量鞣花素，即分子量大于1500克/摩尔的鞣花素。在非常优选的实施方案中，部分纯化的植物提取物衍生自热带植物紫薇。 L，也被称为banaba。本发明还涉及使用本发明部分纯化的提取物来治疗高血糖患者的方法。

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