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11. 发明授权

US06333430B1 Process for preparing tert-alkyl ester from carboxylic acid 有权
标题翻译：从羧酸制备叔烷基酯的方法
公开(公告)号：US06333430B1
公开(公告)日：2001-12-25
申请号：US09561993
申请日：2000-05-02
申请人： Tetsuya Shintaku , Kiyoshi Sugi , Tadashi Katsura , Nobushige Itaya
发明人： Tetsuya Shintaku , Kiyoshi Sugi , Tadashi Katsura , Nobushige Itaya
IPC分类号： C07C6704
CPC分类号： C07C253/30 , C07C67/04 , C07C69/63 , C07C255/19
摘要： A process for preparing a tert-alkyl carboxylic acid ester represented by the formula (III): wherein R1 is an organic group; and each of R2 and R3 is independently an alkyl group having 1 to 4 carbon atoms, comprising reacting a carboxylic acid represented by the formula (I): R1—COOH (I) wherein R1 is as defined above, with a vinylidene compound represented by the formula (II): wherein R2 and R3 are as defined above, in the presence of a phosphorus halide. The tert-alkyl carboxylic acid ester can be used as intermediates for pharmaceuticals such as antibiotics.
摘要翻译：一种制备由式（III）表示的叔烷基羧酸酯的方法：其中R1是有机基团; 其中R 2和R 3各自独立地为具有1至4个碳原子的烷基，包括使由式（I）表示的羧酸：其中R 1如上定义，与由式（II）表示的亚乙烯基化合物反应：其中R2和R3如上定义，在卤化磷存在下。叔烷基羧酸酯可以用作药物如抗生素的中间体。

12. 发明授权

US5948914A Piperidine derivative and process for preparing the same 失效
标题翻译：哌啶衍生物及其制备方法
公开(公告)号：US5948914A
公开(公告)日：1999-09-07
申请号：US53653
申请日：1998-04-02
申请人： Kiyoshi Sugi , Nobushige Itaya , Tadashi Katsura , Masami Igi , Shigeya Yamazaki , Taro Ishibashi , Teiji Yamaoka , Yoshihiro Kawada , Yayoi Tagami
发明人： Kiyoshi Sugi , Nobushige Itaya , Tadashi Katsura , Masami Igi , Shigeya Yamazaki , Taro Ishibashi , Teiji Yamaoka , Yoshihiro Kawada , Yayoi Tagami
IPC分类号： C07D211/22 , C07D211/60 , C07D211/76 , C07D405/12
CPC分类号： C07D405/12 , C07D211/22 , C07D211/60 , C07D211/76
摘要： A piperidine derivative, which can be used as an intermediate for pharmaceuticals such as paroxetine useful as antidepressants, represented by the general formula (I): ##STR1## wherein R.sup.1 is hydrogen atom, benzyloxycarbonyl group or tert-butoxycarbonyl group; R.sup.2 is hydroxymethyl group, an alkylsulfonyloxymethyl group having an alkyl moiety of 1 to 2 carbon atoms, phenylsulfonyloxymethyl group which may have methyl group at the 4-position, (3,4-methylenedioxyphenyl)oxymethyl group, carboxyl group or --CO.sub.2 R.sup.7 group in which R.sup.7 is an alkyl group having 1 to 5 carbon atoms, and Z is methylene group or carbonyl group.
摘要翻译：哌啶衍生物，其可以用作药物的中间体，例如用作抗抑郁药的帕罗西汀，由通式（I）表示：其中R1是氢原子，苄氧基羰基或叔丁氧基羰基; R2是羟甲基，具有1〜2个碳原子的烷基部分的烷基磺酰氧基甲基，4-位可具有甲基的苯基磺酰氧基甲基，（3,4-亚甲二氧基苯基）氧甲基，羧基或-CO 2 R 7基，其中 R 7为碳原子数为1〜5的烷基，Z为亚甲基或羰基。

13. 发明授权

US4266074A Novel insecticidal composition 失效
标题翻译：新型杀虫剂组合物
公开(公告)号：US4266074A
公开(公告)日：1981-05-05
申请号：US596332
申请日：1975-07-16
申请人： Keimei Fujimoto , Nobuo Ohno , Yoshitoshi Okuno , Toshio Mizutani , Isao Ohno , Masachika Hirano , Nobushige Itaya , Takashi Matsuo
发明人： Keimei Fujimoto , Nobuo Ohno , Yoshitoshi Okuno , Toshio Mizutani , Isao Ohno , Masachika Hirano , Nobushige Itaya , Takashi Matsuo
IPC分类号： C07C67/00 , A01N37/00 , A01N37/04 , A01N37/06 , A01N37/10 , A01N37/32 , A01N37/34 , A01N37/38 , A01N37/42 , A01N37/48 , A01N43/06 , A01N43/16 , A01N43/30 , A01N49/00 , C07C43/29 , C07C51/00 , C07C51/08 , C07C57/30 , C07C57/42 , C07C57/58 , C07C57/60 , C07C59/48 , C07C59/56 , C07C59/64 , C07C69/00 , C07C69/612 , C07C69/614 , C07C69/618 , C07C69/635 , C07C69/66 , C07C69/74 , C07C69/743 , C07C69/76 , C07C255/53 , C07C317/00 , C07D209/48 , C07D227/093 , C07D307/34 , C07D307/40 , C07D307/54 , C07D317/48 , C07D317/60 , C07D333/04 , C07D333/16 , C07D333/24 , C07D333/38 , C07D409/06 , A01N41/02 , C07C79/46 , C07C143/67 , C07C147/107 , C07C149/40
CPC分类号： C07D307/54 , C07C323/00 , C07C51/08 , C07C57/42 , C07C59/64 , C07C69/608 , C07C69/612 , C07C69/618 , C07C69/65 , C07C69/734 , C07C69/738 , C07C2101/16 , C07C2102/08 , C07C2102/10
摘要： Substituted acetate compounds represented by the formula ##STR1## which are useful as pesticides and pesticidal composition containing the substituted acetate compounds as active ingredients, as well as processes for preparing the compounds and the compositions are disclosed.
摘要翻译：公开了用作农药和由取代的乙酸酯化合物作为活性成分的杀虫组合物的式“IMAGE”代表的取代的乙酸酯化合物，以及制备化合物和组合物的方法。

14. 发明授权

US4265906A Low mammalian toxic and/or low fish toxic insecticides and/or acaricides 失效
标题翻译：低哺乳动物有毒和/或低毒性杀虫剂和/或杀螨剂
公开(公告)号：US4265906A
公开(公告)日：1981-05-05
申请号：US96212
申请日：1979-11-20
申请人： Kiyoshi Kasamatsu , Tadashi Ohsumi , Nobushige Itaya , Nobuo Ohno , Takashi Kato
发明人： Kiyoshi Kasamatsu , Tadashi Ohsumi , Nobushige Itaya , Nobuo Ohno , Takashi Kato
IPC分类号： C07C253/00 , A01N53/00 , A01N53/08 , C07C67/00 , C07C255/39 , C07C121/75
CPC分类号： A01N53/00
摘要： m-(p-Bromophenoxy)-.alpha.-cyanobenzyl trans- or trans-rich-2,2-dimethyl-3-(2,2-dichlorovinyl)cyclopropanecarboxylate of the formula (I), ##STR1## and their preparation and use as a low fish toxic insecticide and/or acaricide.
摘要翻译：式（I），（I）的间 - （对溴苯氧基）-α-氰基苄基反式或反式 - 富-2,2-二甲基-3-（2,2-二氯乙烯基）环丙烷甲酸酯及其制备并用作低鱼毒杀虫剂和/或杀螨剂。

15. 发明授权

US4212829A Preparation of m-(p-bromophenoxy)benzaldehyde 失效
标题翻译：制备m-（对溴苯氧基）苯甲醛
公开(公告)号：US4212829A
公开(公告)日：1980-07-15
申请号：US5170
申请日：1979-01-22
申请人： Tadashi Ohsumi , Nobushige Itaya
发明人： Tadashi Ohsumi , Nobushige Itaya
IPC分类号： C07C45/00 , C07C45/63 , C07C47/575 , C07C67/00
CPC分类号： C07C47/575 , C07C45/63
摘要： A process for preparing m-(p-bromophenoxy)benzaldehyde of the formula, ##STR1## characterized by brominating m-phenoxybenzaldehyde with bromine or bromine chloride as a brominating agent.
摘要翻译：一种制备下式的对 - （对溴苯氧基）苯甲醛的方法，其特征在于用溴或氯化溴作为溴化剂溴化间苯氧基苯甲醛。

16. 发明授权

US4176189A Insecticidal and acaricidal hydantoin N-methylol esters 失效
标题翻译：杀虫剂和杀螨剂乙内酰脲N-羟甲基酯
公开(公告)号：US4176189A
公开(公告)日：1979-11-27
申请号：US909107
申请日：1978-05-24
申请人： Nobushige Itaya , Masachika Hirano
发明人： Nobushige Itaya , Masachika Hirano
IPC分类号： A01N43/50 , A01N53/00 , A01N53/04 , A01N53/10 , C07D233/72 , A61K31/415 , C07D405/12
CPC分类号： C07D233/72 , A01N43/50 , A01N53/00
摘要： Hydantoin N-methylol esters of the formula, ##STR1## wherein one of X and Y is a carbonyl group and the other is a methylene, ethylidene or propylidene group, R.sub.1 is a lower alkyl, lower alkenyl or lower alkynyl having up to 3 carbon atoms, R.sub.2 is a group represented by the formula, ##STR2## in which R.sub.3 is a hydrogen atom or a methyl group; when R.sub.3 is a hydrogen atom, R.sub.4 is a methoxyiminomethyl or 2,2-disubstituted vinyl group in which the substituents can be selected from the group consisting of methyl, vinyl, fluorine, chlorine and bromine, or both of the substituents may form tetramethylene chain; when R.sub.3 is a methyl group, R.sub.4 is a methyl group; R.sub.5 is a methyl, methoxy, fluorine, chlorine, bromine or 3,4-methylenedioxy group; and n is 1 or 2, a process for producing the same, insecticides and acaricides containing the same as an active ingredient, and novel intermediate compounds.
摘要翻译：乙酰头孢菌素N-羟甲基酯，其中X和Y中的一个是羰基，另一个是亚甲基，亚乙基或亚丙基，R 1是具有至多3个碳的低级烷基，低级链烯基或低级炔基原子，R 2是由下式表示的基团，其中R 3是氢原子或甲基; 当R3为氢原子时，R4为甲氧基亚氨基甲基或2,2-二取代的乙烯基，其中取代基可以选自甲基，乙烯基，氟，氯和溴，或两者均可形成四亚甲基链 ; 当R 3为甲基时，R 4为甲基; R5是甲基，甲氧基，氟，氯，溴或3,4-亚甲二氧基; n为1或2，其制造方法为含有与活性成分相同的杀虫剂和杀螨剂，以及新型中间体化合物。

17. 发明授权

US4062968A Insecticidal substituted acetate compounds 失效
公开(公告)号：US4062968A
公开(公告)日：1977-12-13
申请号：US596334
申请日：1975-07-16
申请人： Keimei Fujimoto , Nobuo Ohno , Yoshitoshi Okuno , Toshio Mizutani , Isao Ohno , Masachika Hirano , Nobushige Itaya , Takashi Matsuo
发明人： Keimei Fujimoto , Nobuo Ohno , Yoshitoshi Okuno , Toshio Mizutani , Isao Ohno , Masachika Hirano , Nobushige Itaya , Takashi Matsuo
IPC分类号： A01N37/36 , A01N43/06 , C07D307/54 , A01N9/00
CPC分类号： C07D307/54 , C07C323/00
摘要： Substituted acetate compounds represented by the formula ##STR1## which are useful as pesticides and pesticidal composition containing the substituted acetate compounds as active ingredients, as well as processes for preparing the compounds and the compositions are disclosed.

18. 发明授权

US4058622A Substituted phenyl acetate, insecticidal composition and method of use 失效
标题翻译：取代的乙酸苯酯，杀虫剂组合物和使用方法
公开(公告)号：US4058622A
公开(公告)日：1977-11-15
申请号：US557694
申请日：1975-03-12
申请人： Keimei Fujimoto , Nobuo Ohno , Yoshitoshi Okuno , Toshio Mizutani , Isao Ohno , Masachika Hirano , Nobushige Itaya , Takashi Matsuo
发明人： Keimei Fujimoto , Nobuo Ohno , Yoshitoshi Okuno , Toshio Mizutani , Isao Ohno , Masachika Hirano , Nobushige Itaya , Takashi Matsuo
IPC分类号： C07C69/612 , C07D307/54 , A01N9/24 , C07C69/76
CPC分类号： C07D307/54 , C07C323/00
摘要： Substituted acetate compounds represented by the formula ##STR1## which are useful as pesticides and pesticidal compositions containing the substituted acetate compounds as active ingredients, as well as processes for preparing the compounds and the compositions are disclosed.
摘要翻译：公开了用作农药和由取代的乙酸酯化合物作为活性成分的杀虫组合物的式“IMAGE”代表的取代的乙酸酯化合物，以及制备化合物和组合物的方法。

19. 发明授权

US4039680A Insecticidal substituted acetate compounds 失效
标题翻译：杀虫剂取代的乙酸酯化合物
公开(公告)号：US4039680A
公开(公告)日：1977-08-02
申请号：US596335
申请日：1975-07-16
申请人： Keimei Fujimoto , Nobuo Ohno , Yoshitoshi Okuno , Toshio Mizutani , Isao Ohno , Masachika Hirano , Nobushige Itaya , Takashi Matsuo
发明人： Keimei Fujimoto , Nobuo Ohno , Yoshitoshi Okuno , Toshio Mizutani , Isao Ohno , Masachika Hirano , Nobushige Itaya , Takashi Matsuo
IPC分类号： A01N37/08 , A01N37/36 , A01N43/06 , C07D307/54 , A01N9/00
CPC分类号： C07D307/54 , C07C323/00
摘要： Substituted acetate compounds represented by the formula ##STR1## which are useful as pesticides and pesticidal composition containing the substituted acetate compounds as active ingredients, as well as processes for preparing the compounds and the compositions are disclosed.

20. 发明申请

US20090118534A1 METHOD OF PRODUCING OPTICALLY ACTIVE (S)-7-HYDROXY-6-METHYLHEPTAN-2-ONE AND PRECURSOR THEREOF 失效
标题翻译：生产光学活性（S）-7-羟基-6-甲基硫脲-2-酮的方法及其前体
公开(公告)号：US20090118534A1
公开(公告)日：2009-05-07
申请号：US12294051
申请日：2007-03-22
申请人： Nobushige Itaya , Hiroshi Maeda , Yuki Sato
发明人： Nobushige Itaya , Hiroshi Maeda , Yuki Sato
IPC分类号： C07C69/66 , C12P7/62
CPC分类号： C07C323/52 , C07B2200/07 , C07C67/31 , C07C69/708 , C12P7/26 , C12P7/62 , C12P41/005
摘要： Provided is a method capable of industrially producing optically active (S)-7-hydroxy-6-methylheptan-2-one and its precursor simply and efficiently. The production method, allows a R-body preferentially hydrolyzable Aspergillus microorganism-derived esterase to act on a 2-methyl-6-oxoheptanoate (II), to produce an optically active (S)-2-methyl-6-oxoheptanoate (III).
摘要翻译：本发明提供能够简单有效地工业生产光学活性（S）-7-羟基-6-甲基庚-2-酮及其前体的方法。制备方法允许R体优先水解的曲霉微生物衍生的酯酶作用于2-甲基-6-氧代庚酸酯（II），以产生光学活性的（S）-2-甲基-6-氧代庚酸酯（III）。

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