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1. 发明授权

US4692461A Fungicidal thienylurea derivatives 失效
标题翻译：杀真菌噻吩脲衍生物
公开(公告)号：US4692461A
公开(公告)日：1987-09-08
申请号：US933492
申请日：1986-11-21
申请人： Werner Hallenbach , Hans Lindel , Wilhelm Brandes
发明人： Werner Hallenbach , Hans Lindel , Wilhelm Brandes
IPC分类号： C07D333/36 , A01N47/36 , C07D333/38 , C07D333/66 , C07D333/68 , C07D333/78 , C07D333/80 , A01N43/02 , C07D333/56
CPC分类号： C07D333/68 , A01N47/36 , C07D333/38 , C07D333/78 , C07D333/80
摘要： Fungicidally active novel thienylurea derivatives of the formula ##STR1## in which X represents oxygen or sulphur,R represents cyano, hydroxycarbonyl or alkoxycarbonyl,R.sup.1 represents hydrogen or alkyl,R.sup.2 represents hydrogen or alkyl,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl,R.sup.4 represents hydrogen, alkyl or optionally substituted aryl,R.sup.5 represents hydrogen, alkyl or optionally substituted aryl, orR.sup.4 and R.sup.5 together represent the radical --(CH.sub.2).sub.n --, andn represents the numbers 3, 4, 5 or 6,or acid addition salts thereof.
摘要翻译：式“IMAGE”的杀真菌活性新型噻吩脲衍生物，其中X表示氧或硫，R表示氰基，羟基羰基或烷氧基羰基，R1表示氢或烷基，R2表示氢或烷基，R3表示氢，烷基或任选取代的芳基，R4 表示氢，烷基或任选取代的芳基，R 5表示氢，烷基或任选取代的芳基，或者R 4和R 5一起代表基团 - （CH 2）n - ，n代表数字3,4,5或6或酸加成的盐。

2. 发明授权

US4737515A Use of tetrahydrobenzothienylurea derivatives as fungicides 失效
标题翻译：四氢苯并噻吩脲衍生物用作杀真菌剂
公开(公告)号：US4737515A
公开(公告)日：1988-04-12
申请号：US931295
申请日：1986-11-14
申请人： Werner Hallenbach , Hans Lindel , Wilhelm Brandes
发明人： Werner Hallenbach , Hans Lindel , Wilhelm Brandes
IPC分类号： A01N47/36 , C07D333/70 , C07D333/78 , A01N43/12
CPC分类号： C07D333/78 , A01N47/36 , C07D333/70
摘要： A method of combating fungi which comprises applying to such fungi or to a fungus habitat a fungicidally effective amount of a tetrahydrobenzothienylurea derivative of the formula ##STR1## in which n is 3, 4, 5 or 6,X is oxygen or sulphur,R is C.sub.1-4 -alkoxy or hydroxyl, andR.sup.1 is C.sub.1-4 -alkyl.
摘要翻译：一种防治真菌的方法，其包括将杀真菌有效量的式“IMAGE”的四氢苯并噻吩脲衍生物施用于这种真菌或真菌栖息地，其中n为3,4,5或6，X为氧或硫，R为 C 1-4 - 烷氧基或羟基，R 1是C 1-4 - 烷基。

3. 发明授权

US4740520A Use of thienylurea derivatives as selective fungicides 失效
标题翻译：使用噻吩脲衍生物作为选择性杀真菌剂
公开(公告)号：US4740520A
公开(公告)日：1988-04-26
申请号：US931293
申请日：1986-11-14
申请人： Werner Hallenbach , Hans Lindel , Wilhelm Brandes
发明人： Werner Hallenbach , Hans Lindel , Wilhelm Brandes
IPC分类号： A01N47/36 , C07D333/38 , A01N43/06
CPC分类号： A01N47/36 , C07D333/38
摘要： A method of combating fungi which comprises applying to such fungi or to a fungus habitat a fungicidally effective amount of a thienylurea derivative of the formula ##STR1## in which X is oxygen or sulphur,R is C.sub.1 -C.sub.4 -alkoxy,R.sup.1 is C.sub.3 -C.sub.4 -alkyl, andR.sup.2 and R.sup.3 each independently is C.sub.1 -C.sub.4 -alkyl and one of them may also be hydrogen.
摘要翻译：一种防治真菌的方法，其包括将杀真菌有效量的式（I）的噻吩基脲衍生物（其中X为氧或硫），R为C1-C4-烷氧基，R1为C3- C 4 - 烷基，R 2和R 3各自独立地为C 1 -C 4 - 烷基，并且它们之一也可以是氢。

4. 发明授权

US5086181A 4-bromo-6-chloro-5-amino-2-substituted pyridyl compounds 失效
标题翻译： 4-溴-6-氯代-5-氨基-2-取代的吡啶化合物
公开(公告)号：US5086181A
公开(公告)日：1992-02-04
申请号：US581815
申请日：1990-09-13
申请人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Gernot Klotz , Heinrich A. Greife
发明人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Gernot Klotz , Heinrich A. Greife
IPC分类号： A23K1/16 , C07D213/73 , C07D213/74 , C07D213/75
CPC分类号： C07D213/73 , C07D213/75
摘要： A pyridine derivative of the formula ##STR1## in which A stands for ##STR2## is useful in the preparation of 4-bromo-6-chloro-5-amino-2-pyridyl-ethanolamines, their physiologically tolerated salts and their N-oxides. The 4-bromo-6-chloro-5-amino-2-pyridyl-ethanolamines are useful as yield promoters in animals and as feedstuff additives to achieve higher increases in weight and improved feed utilization.

5. 发明授权

US5149822A Preparation of 2,3-dichloro-5-acetylpyridine 失效
标题翻译：制备2,3-二氯-5-乙酰基吡啶
公开(公告)号：US5149822A
公开(公告)日：1992-09-22
申请号：US336969
申请日：1989-04-12
申请人： Hans Lindel , Werner Hallenbach , Bernd Gallenkamp
发明人： Hans Lindel , Werner Hallenbach , Bernd Gallenkamp
IPC分类号： C07D213/50 , C07D213/61
CPC分类号： C07D213/61
摘要： A process for the preparation of 2,3-dichloro-5-acetylpyridine of the formula ##STR1## comprising decarboxylating a compound of the formula ##STR2## in which R.sup.1 stands for methyl or ethyl,in a mixture of water and a water miscible aprotic solvent.
摘要翻译：制备式（I）的2,3-二氯-5-乙酰基吡啶的方法包括使式（Ⅳ）化合物（Ⅳ）脱羧，其中R1代表甲基或乙基，以水和水混溶的非质子溶剂。

6. 发明授权

US4845262A Novel arylethanolamines for promoting livestock production 失效
标题翻译：用于促进畜牧生产的新型芳基乙醇胺
公开(公告)号：US4845262A
公开(公告)日：1989-07-04
申请号：US89691
申请日：1987-08-25
申请人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Anno de Jong , Martin Scheer
发明人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Anno de Jong , Martin Scheer
IPC分类号： A23K1/16 , A61K31/135 , A61K31/275 , A61P3/00 , C07C67/00 , C07C255/58 , C07C255/59 , C07C313/00 , C07C315/04 , C07C317/48 , C07C317/50
CPC分类号： C07C255/00 , A23K20/111
摘要： The growth of livestock is promoted by the novel arylethanolamines of the formula ##STR1## in which R.sup.1 represents cyano,R.sup.2 represents amino, alkylamino or acylamino,R.sup.3 represents hydrogen, halogen, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, hydroxymethyl, nitro or methylsulphonylmethyl,R.sup.4 represents hydrogen, alkyl or acyl,R.sup.5 represents hydrogen or alkyl,R.sup.6 represents alkyl,n represents 1, 2 or 3,R.sup.7 represents the radicals --COR.sup.9, --O-alkylene-COR.sup.9, -alkylene-R.sup.10 or --O-alkylene-R.sup.10,R.sup.8 represents hydrogen, alkyl or halogen,R.sup.9 represents hydroxyl, alkoxy or the radical --NR.sup.11 R.sup.12,R.sup.10 represents hydroxyl, alkoxy or the radical NR.sup.11 R.sup.12,R.sup.11 represents hydrogen or alkyl, andR.sup.12 represents hydrogen or alkyl,and the physiologically acceptable salts thereof.
摘要翻译：通过式（I）的新型芳基乙醇胺促进家畜的生长，其中R1代表氰基，R2代表氨基，烷基氨基或酰氨基，R3代表氢，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，羟基甲基，硝基或甲基磺酰基甲基，R 4表示氢，烷基或酰基，R 5表示氢或烷基，R 6表示烷基，n表示1,2或3，R 7表示基团-COR 9，-O-亚烷基-CON 9， - 亚烷基-R 10或-O - 亚烷基-R 10，R 8表示氢，烷基或卤素，R 9表示羟基，烷氧基或基团-NR 11 R 12，R 10表示羟基，烷氧基或基团NR 11 R 12，R 11表示氢或烷基，R 12表示氢或烷基，其可接受的盐。

7. 发明授权

US5028617A Heteroarylethanol-pyridylalkylamines for controlling animal growth 失效
标题翻译：用于控制动物生长的杂芳基乙醇 - 吡啶基烷基胺
公开(公告)号：US5028617A
公开(公告)日：1991-07-02
申请号：US467593
申请日：1990-01-19
申请人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Heinrich A. Greife , Gernot Klotz
发明人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Heinrich A. Greife , Gernot Klotz
IPC分类号： A23K1/16 , A61K31/44 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61P3/04 , C07D213/38 , C07D213/61 , C07D213/64 , C07D213/65 , C07D213/73 , C07D213/80
CPC分类号： C07D213/64 , C07D213/38 , C07D213/61 , C07D213/65 , C07D213/73 , C07D213/80
摘要： A compound for promoting livestock production and for controlling obesity in humans and animals, of the formula ##STR1## in which A represents .dbd.CH-- or .dbd.N--,R.sup.0 represents hydrogen or methyl,R.sup.1 and R.sup.3 each independently represents hydrogen, hydroxyl, halogen, cyano, alkyl, halogenoalkyl, hydroxyalkyl, alkoxycarbonyl, aminocarbonyl, mono- and dialkylaminocarbonyl, alkoxy, halogenoalkoxy, halogenoalkylthio, NHSO.sub.2 -alkyl,R.sup.2 represents hydrogen, hydroxyl, alkoxy or the radical --NR.sup.5 R.sup.6,R.sup.4 represents hydrogen, C.sub.1 -C.sub.10 -alkyl which is optionally substituted by hydroxyl, halogen, alkoxy, acyloxy or the radical --NH.sup.7 R.sup.8, or represents the radical COR.sup.9 or the radical --O--Z--R.sup.10,Z represents C.sub.1 -C.sub.10 -alkylene, -alkenylene or alkynylene,R.sup.5 represents hydrogen or alkyl,R.sup.6 represents hydrogen, alkyl, halogenoalkyl or acyl, or R.sup.5 and R.sup.6 together with the adjoining N atom form a saturated or unsaturated heterocyclic 4-, 5- or 6-membered ring,R.sup.7 and R.sup.8 each independently represents hydrogen, optionally substituted alkyl, optionally substituted aryl,R.sup.9 represents hydroxyl, alkoxy or the radical --NR.sup.7 R.sup.8,R.sup.10 represents hydroxyl, alkoxy, acyloxy, optionally substituted aryloxy or aralkyloxy,with the substituent R.sup.4 and the alkylamino group in the pyridyl ring of the formula I being in the p position with respect to one another, or a physiologically tolerated salt thereof, or, if A represents nitrogen, optionally the N-oxide thereof.
摘要翻译：一种用于促进家畜生产和控制人和动物肥胖的化合物，其中A表示= CH-或= N-，R0表示氢或甲基，R1和R3各自独立地表示氢，羟基，卤素，氰基，烷基，卤代烷基，羟基烷基，烷氧基羰基，氨基羰基，一烷基氨基羰基和二烷基氨基羰基，烷氧基，卤代烷氧基，卤代烷硫基，NHSO2-烷基，R2代表氢，羟基，烷氧基或基-NR5R6，R4代表氢，C1- 任选被羟基，卤素，烷氧基，酰氧基或基团-NH 7 R 8取代的C 10 - 烷基，或表示基团COR 9或基团-OZ-R 10，Z表示C 1 -C 10 - 亚烷基， - 亚烯基或亚炔基，R 5表示氢或烷基，R 6表示氢，烷基，卤代烷基或酰基，或R 5和R 6与相邻的N原子一起形成饱和或不饱和的4-，5-或6-元环，R 7和R 8各自独立地表示氢，取代的烷基，任选取代的芳基，R 9表示羟基，烷氧基或基团-NR 7 R 8，R 10表示羟基，烷氧基，酰氧基，任选取代的芳氧基或芳烷氧基，式I的吡啶环中的取代基R4和烷基氨基在相对于彼此的p位置或其生理上耐受的盐，或者如果A表示氮，则任选地其N-氧化物。

8. 发明授权

US4895950A 5-halogeno-6-amino-nicotinic acid halides 失效
标题翻译： 5-卤代-6-氨基烟酰卤
公开(公告)号：US4895950A
公开(公告)日：1990-01-23
申请号：US216047
申请日：1988-07-07
申请人： Hans Lindel , Werner Hallenbach
发明人： Hans Lindel , Werner Hallenbach
IPC分类号： C07D213/75 , C07D213/73 , C07D213/74 , C07D213/78 , C07D401/04
CPC分类号： C07D213/73 , C07D213/78
摘要： Novel 5-halogeno-6-amino-nicotinic acid halides of the formula ##STR1## in which R represents hydrogen or alkyl,R.sup.1 represents hydrogen, alkyl or acyl orR and R.sup.1, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical,R.sup.2 represents halogen andHal represents halogen,are prepared by halogenating the corresponding nicotinic acids. The Co Hal moiety is converted to CH.sub.3 by reaction withR.sup.3 OMgCR.sup.4 (COOR.sup.3).sub.2 (IV)in whichR.sup.3 represents C.sub.1-3 alkyl andR.sup.4 represents hydrogen or C.sub.1 -C.sub.2 -alkyl,and then hydrolyzing and decarboxylating the product.
摘要翻译：式（I）的新的5-卤代-6-氨基烟碱酰卤，其中R表示氢或烷基，R 1表示氢，烷基或酰基或R和R 1与它们所在的氮原子一起表示任选取代的杂环基，R2表示卤素，Hal表示卤素，通过卤化相应的烟酸制备。通过与R 3表示C 1-3烷基和R 4表示氢或C 1 -C 2 - 烷基的R 3 OMgCR 4（COOR 3）2（Ⅳ）反应将Co Hal部分转化成CH3，然后水解和脱羧产物。

9. 发明授权

US5216170A (2-aminopropyl) pyridines useful as intermediates 失效
标题翻译：（2-氨基丙基）吡啶可用作中间体
公开(公告)号：US5216170A
公开(公告)日：1993-06-01
申请号：US677020
申请日：1991-03-28
申请人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Heinrich A. Greife , Gernot Klotz
发明人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Heinrich A. Greife , Gernot Klotz
IPC分类号： C07D213/38 , C07D213/61 , C07D213/64 , C07D213/65 , C07D213/73 , C07D213/80
CPC分类号： C07D213/64 , C07D213/38 , C07D213/61 , C07D213/65 , C07D213/73 , C07D213/80
摘要： A compound for promoting livestock production and for controlling obesity in humans and animals, of the formula ##STR1## in which A represents .dbd.CH-- or .dbd.N--,R.sup.0 represents hydrogen or methyl,R.sup.1 and R.sup.3 each independently represents hydrogen, hydroxyl, halogen, cyano, alkyl, halogenoalkyl, hydroxyalkyl, alkoxycarbonyl, aminocarbonyl, mono- and dialkylaminocarbonyl, alkoxy, halogenoalkoxy, halogenoalkylthio, NHSO.sub.2 -alkyl,R.sup.2 represents hydrogen, hydroxyl, alkoxy or the radical --NR.sup.5 R.sup.6,R.sup.4 represents hydrogen, C.sub.1 -C.sub.10 -alkyl which is optionally substituted by hydroxyl, halogen, alkoxy, acyloxy or the radical --NR.sup.7 R.sup.8, or represents the radical COR.sup.9 or the radical --O--Z--R.sup.10,Z represents C.sub.1 -C.sub.10 -alkylene, -alkenylene or alkynylene,R.sup.5 represents hydrogen or alkyl,R.sup.6 represents hydrogen, alkyl, halogenoalkyl or acyl, or R.sup.5 and R.sup.6 together with the adjoining N atom form a saturated or unsaturated heterocyclic 4-, 5- or 6-membered ring,R.sup.7 and R.sup.8 each independently represents hydrogen, optionally substituted alkyl, optionally substituted aryl,R.sup.9 represents hydroxyl, alkoxy or the radical --NR.sup.7 R.sup.8,R.sup.10 represents hydroxyl, alkoxy, acyloxy, optionally substituted aryloxy or aralkyloxy,with the substituent R.sup.4 and the alkylamino group in the pyridyl ring of the formula I being in the p position with respect to one another,or a physiologically tolerated salt thereof, or, if A represents nitrogen, optionally the N-oxide thereof.
摘要翻译：一种用于促进家畜生产和控制人和动物肥胖的化合物，其中A表示= CH-或= N-，R0表示氢或甲基，R1和R3各自独立地表示氢，羟基，卤素，氰基，烷基，卤代烷基，羟基烷基，烷氧基羰基，氨基羰基，一烷基氨基羰基和二烷基氨基羰基，烷氧基，卤代烷氧基，卤代烷硫基，NHSO2-烷基，R2代表氢，羟基，烷氧基或基-NR5R6，R4代表氢，C1- 任选被羟基，卤素，烷氧基，酰氧基或基团-NR 7 R 8取代的C 10 - 烷基，或表示基团COR 9或基团-OZ-R 10，Z表示C 1 -C 10亚烷基， - 亚烯基或亚炔基，R 5表示氢或烷基，R 6表示氢，烷基，卤代烷基或酰基，或R 5和R 6与相邻的N原子一起形成饱和或不饱和的4-，5-或6-元环，R 7和R 8各自独立地表示氢，取代的烷基，任选取代的芳基，R 9表示羟基，烷氧基或基团-NR 7 R 8，R 10表示羟基，烷氧基，酰氧基，任选取代的芳氧基或芳烷氧基，式I的吡啶环中的取代基R4和烷基氨基在相对于彼此的p位置或其生理上耐受的盐，或者如果A表示氮，则任选地其N-氧化物。

10. 发明授权

US4988694A 4-bromo-6-chloro-5-amino-2-pyridyl-ethanolamines and their use as yield promoters 失效
标题翻译： 4-溴-6-氯-5-氨基-2-吡啶基 - 乙醇胺及其作为产率促进剂的用途
公开(公告)号：US4988694A
公开(公告)日：1991-01-29
申请号：US340936
申请日：1989-04-20
申请人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Gernot Klotz , Heinrich A. Greife
发明人： Hans Lindel , Werner Hallenbach , Friedrich Berschauer , Gernot Klotz , Heinrich A. Greife
IPC分类号： A23K1/16 , C07D213/73 , C07D213/74 , C07D213/75
CPC分类号： C07D213/73 , C07D213/75
摘要： 4-Bromo-6-chloro-5-amino-2-pyridyl-ethanolamines, intermediates for preparation thereof and their use as yield promoters for animals and as feedstuff additives to achieve higher increases in weight and improved feed utilization of the formula ##STR1## in which R.sup.1 stands for hydrogen, alkyl, acyl or substituted silyl,R.sup.2 stands for hydrogen or alkyl,R.sup.3 stands for hydrogen, alkyl, cycloalkyl, substituted alkyl, optionally substituted aralkyl, aryl or heterocyclyl, orR.sup.2 and R.sup.3, together with the nitrogen atom to which they are bonded, can stand for an optionally substituted heterocyclic radical,R.sup.4 stands for hydrogen or alkyl andR.sup.5 stands for hydrogen, alkyl, halogenoalkyl or acyl, and their physiologically tolerated salts and their N-oxides have been found.
摘要翻译： 4-溴-6-氯-5-氨基-2-吡啶基 - 乙醇胺，其制备的中间体及其作为动物产率促进剂和作为饲料添加剂的用途，以实现更高的重量增加和改善饲料利用的方法。其中R1代表氢，烷基，酰基或取代的甲硅烷基，R2代表氢或烷基，R3代表氢，烷基，环烷基，取代烷基，任选取代的芳烷基，芳基或杂环基，或R 2和R 3与氮可以代表任意取代的杂环基，R4代表氢或烷基，R5代表氢，烷基，卤代烷基或酰基，并且已经发现它们的生理上耐受的盐和它们的N-氧化物。

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