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1. 发明授权

US3919290A Substituted 14-desoxy-mutilins 失效
标题翻译：取代的14-脱氧菌素
公开(公告)号：US3919290A
公开(公告)日：1975-11-11
申请号：US42751473
申请日：1973-12-26
申请人： SANDOZ LTD
发明人： EGGER HELMUT , REINSHAGEN HELLMUTH
IPC分类号： C07C323/25 , C07D295/088 , C07C143/12
CPC分类号： C07D295/088 , C07C323/25
摘要： WHEREIN EITHER R1 is ethyl or vinyl, N IS AN INTEGER FROM 2 TO 5, X is sulphur, AND PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS AND QUATERNARY SALTS THEREOF. Processes for the preparation of such compounds are described. The compounds are antibiotics with an antibacterial effect.

This invention relates to new pleuromutilins of the formula:
摘要翻译：本发明涉及下式的新型pleuromutilins：

2. 发明授权

US3906041A Oxalic acid derivatives 失效
标题翻译：草酸衍生物
公开(公告)号：US3906041A
公开(公告)日：1975-09-16
申请号：US40533173
申请日：1973-09-07
申请人： SANDOZ LTD
发明人： HOFER KURT , MOESCH RUDOLF , SCHILLI ALFRED , BURDET EVELYNE
IPC分类号： A61K8/42 , A61Q17/04 , C08K5/20 , C08K5/372 , C09K15/22 , C09K15/28 , D06M13/418 , C07C103/30
CPC分类号： A61K8/42 , A61Q17/04 , C08K5/20 , C08K5/3725 , C09K15/22 , C09K15/28 , D06M13/418
摘要： Ultraviolet light absorbers for plastics (for example polyolefins, e.g. polyethylene or polypropylene; polyvinylchloride; or a nitro lacquer), which may be incorporated with or without one or more other known ultraviolet light stabilizers into the plastics, have the formula I

in which each of R1, R2, R3, R4, R5, R6, R7 and R8 represents H, Cl, Br, -CnH2n 1, -CnH2n 1 or -O-CnH2n 1 or an -O-aryl, aryl, aralkyl or alkaryl radical with up to eight carbon atoms, M REPRESENTS A WHOLE NUMBER FROM 1 TO 8 INCLUSIVE, AND N REPRESENTS A WHOLE NUMBER FROM 1 TO 4 INCLUSIVE, WITH THE PROVISO THAT THE RADICALS R1, R2, R3, R4, R5, R6, R7 and R8, within their definition, may be similar or dissimilar and n need not necessarily have the same value in all of the radicals where n occurs, AND THE FORMULA Ia

WHEREIN EACH OF R1'' to R10'', independently of one another, is selected from H, alkyl, aralkyl, alkaryl, alkyl-(OC2H4)n , alkyl-(OC3H6)n , Cl, Br, OH, O-alkyl, O-aryl, S-alkyl, S-aryl, COO-alkyl, COO-aryl, CONH-alkyl, CONH-aryl, NHCO-alkyl, NHCOaryl, alkyl ether radicals and alkyl thioether radicals, with the proviso that at least one of the radicals R''1 to R''10 must be such that at least one -C-S-C- grouping is present in the compound, and N'' REPRESENTS A WHOLE NUMBER OF FROM 1 TO 12 INCLUSIVE.
摘要翻译：可与或不含一种或多种其它已知的紫外光稳定剂一起掺入塑料中的用于塑料的紫外光吸收剂（例如聚烯烃，例如聚乙烯或聚丙烯;聚氯乙烯或硝基漆）具有式I，其中 R1，R2，R3，R4，R5，R6，R7和R8表示H，Cl，Br，-CnH2n + 1，-CnH2n-1或-O-CnH2n + 1或-O-芳基，芳基，芳烷基或烷芳基具有多达8个碳原子的基团，M代表1至8个整数的全部数字，以及N个表示1至4个全部数字，包括R，R2，R3，R4，R5，R6，R7 和R8在其定义中可以是相似的或不相似的，并且n不必在所有发生n的基团中具有相同的值，并且选择彼此独立的每个R 1'至R 10'的式烷基 - （OC 2 H 4）n'，烷基 - （OC 3 H 6）n'，Cl，Br，OH，O-烷基，O-芳基，S-烷基，S-芳基，COO-烷基，COO-芳基，CONH-烷基，CONH-芳基，NHCO-烷基，NHCO-芳基，烷基醚基团和烷基硫醚基团，条件是基团R'1至R'10中的至少一个必须使得至少一个 - 化合物中存在CSC-分组，N'代表从1至12包含的全部数字。

3. 发明授权

US3897421A Organic compounds 失效
标题翻译：有机化合物
公开(公告)号：US3897421A
公开(公告)日：1975-07-29
申请号：US42098773
申请日：1973-12-03
申请人： SANDOZ LTD
发明人： AEBLI HORST , FLECK FRITZ , SCHMID HORST
IPC分类号： C07D249/06 , C07D249/20 , C07D413/10 , C09B23/14
CPC分类号： C07D249/20 , C07D249/06
摘要： The present invention provides novel compounds of the formula:

IN WHICH R1 signifies hydrogen, fluorine or chlorine atom, a carboxylic or sulphonic acid group or an amide or ester thereof, a cyano group or an alkylsulphonyl or arylsulphonyl group, R2 signifies a hydrogen, fluorine or chlorine atom, a cyano group, a phenyl or alkyl radical which may be substituted, a carboxylic or sulphonic acid group or an amide or ester thereof, an alkylsulphonyl or arylsulphonyl group or a benzoxazole group which may be substituted, R3 and R4 independently signify a hydrogen, fluorine or chlorine atom, an alkyl radical of 1 to 6 carbon atoms which may be substituted, a cyano or carboxy group, a carboxylic acid amide or ester group, and R4 may also signify an aryl radical which may be substituted, and A signifies a hydrogen atom or an alkyl or aryl radical which may be substituted or a group of formula II,
摘要翻译：本发明提供下式的新型化合物：

4. 发明授权

US3896228A Method for treating nephrises 失效
标题翻译：治疗神经病的方法
公开(公告)号：US3896228A
公开(公告)日：1975-07-22
申请号：US49134274
申请日：1974-07-24
申请人： SANDOZ LTD
发明人： RICHARDSON BRIAN PETER
IPC分类号： A61K31/195 , A61K31/48 , A61K27/00
CPC分类号： A61K31/48 , A61K31/195 , Y10S514/869
摘要： This invention concerns a novel method of increasing urine volume and urine pH, which comprises inhibiting prolactin by administering a prolactin inhibiting amount of a prolactininhibitor selected from 2-bromo- Alpha -ergocryptine, ergocornine, 9,10-dihydroergocornine and L-dopa.

5. 发明授权

US3890409A Dicyclic diphosphates and diphosphites 失效
标题翻译：二环磷酸二酯和二亚磷酸酯
公开(公告)号：US3890409A
公开(公告)日：1975-06-17
申请号：US36462973
申请日：1973-05-29
申请人： SANDOZ LTD
发明人： MAYERHOEFER HORST , MUELLER WOLFGANG , SOLIBERGER URS , WOLF RAINER
IPC分类号： C08K5/00 , C07F9/6574 , C08K5/52 , C08K5/527 , C08L7/00 , C08L21/00 , C08L23/00 , C08L33/00 , C08L33/02 , C08L51/00 , C08L51/02 , C08L77/00 , C08L101/00 , C09K21/12 , C07D105/04 , C08F45/58
CPC分类号： C08K5/527 , C07F9/65742 , C07F9/65746
摘要： The present invention relates to phosphorus containing compounds and more specifically to phosphorus and phosphoric acid esters of the formula,

WHEREIN R1 and R2 are each hydrogen or alkyl, N IS AN INTEGER 1 OR 2, AND Y is a mono or divalent aromatic radical. The compounds are useful as flame retardants for, e.g., plastics materials.
摘要翻译：本发明涉及含磷化合物，更具体地涉及下式的磷和磷酸酯，其中R1和R2各自为氢或烷基，N为整数1或2，Y为单价或二价芳族基团。

6. 发明授权

US3884974A 2-Ketoamidines 失效
标题翻译： 2-酮酰胺
公开(公告)号：US3884974A
公开(公告)日：1975-05-20
申请号：US42671473
申请日：1973-12-13
申请人： SANDOZ LTD
发明人： HEFFE WILHELM
IPC分类号： C07D263/04 , C07D295/28 , C07C123/00
CPC分类号： C07D263/04 , C07D295/28 , Y10S514/866
摘要： The present invention relates to amidino ketones of the formula

WHEREIN R1 is alkyl of 1 to 4 carbon atoms, phenyl or substituted phenyl, and R2 is alkyl of 1 to 4 carbon atoms, or R1 and R2 together are -(CH2)n-, wherein n is an integer from 2 to 7, AND R3 is alkyl of 1 to 4 carbon atoms, or R1, R2 and R3 together with the carbon atom to which they are bound form the adamantyl radical, R4 is alkyl of 1 to 8 carbon atoms, alkenyl of 2 to 8 carbon atoms, alkoxyalkyl of 2 to 8 carbon atoms in the aggregate thereof, cyanoalkyl wherein the alkyl radical is of 1 to 5 carbon atoms, or a group of formula

WHEREIN R7 and R8 are the same or different and each is alkyl of 1 to 4 carbon atoms, or R7 and R8 together with the nitrogen atom are a heterocyclic ring, or a heterocyclic ring having a ring oxygen atom, and R5 and R6 are the same or different and each is alkyl of 1 to 8 carbon atoms, alkenyl of 2 to 8 carbon atoms, alkoxyalkyl of 2 to 8 carbon atoms in the aggregate thereof or cyanoalkyl wherein the alkyl is of 1 to 5 carbon atoms, or one of R4, R5 and R6 is phenyl or substituted phenyl and the others of R4, R5 and R6 are as defined above, useful as hypoglycaemic agents.
摘要翻译：本发明涉及下式的脒基酮：其中R 1为1至4个碳原子的烷基，苯基或取代的苯基，R 2为1至4个碳原子的烷基，或者R 1和R 2一起为 - （CH 2）n - 其中n是2至7的整数，并且R 3是1至4个碳原子的烷基，或者R 1，R 2和R 3与它们所连接的碳原子一起形成金刚烷基，R4是1至8个碳原子的烷基 2〜8个碳原子的链烯基，2〜8个碳原子的烷氧基烷基，其中烷基为1〜5个碳原子的氰基烷基，或式WHEREIN R7和R8的基团相同或不同，各自为1至4个碳原子的烷基，或者R 7和R 8与氮原子一起为杂环，或具有环氧原子的杂环，R 5和R 6相同或不同，分别为1〜 8个碳原子，2至8个碳原子的链烯基，2至8个碳原子的烷氧基烷基或氰基烷基w 此处烷基为1至5个碳原子，或者R4，R5和R6中的一个为苯基或取代的苯基，R4，R5和R6中的其它基团如上定义，可用作低血糖药。

7. 发明授权

US3875233A Bis-P-hydroxy-phenethyl amines 失效
标题翻译：双-P-羟基 - 苯乙胺
公开(公告)号：US3875233A
公开(公告)日：1975-04-01
申请号：US32587773
申请日：1973-01-22
申请人： SANDOZ LTD
发明人： BASTIAN JEAN-MICHEL , HASSPACHER KLAUS
IPC分类号： C07C311/08 , A61K20060101 , C07C20060101 , C07C67/00 , C07C217/20 , C07C301/00 , C07C303/40 , C07C87/28
CPC分类号： C07C233/12
摘要： The invention concerns novel compounds of the formula:

WHEREIN R1 is hydroxyl, hydroxymethyl or
摘要翻译：本发明涉及下式的新型化合物：

8. 发明授权

US3865604A Flame-retardant regenerated cellulose 失效
标题翻译：阻燃再生纤维素
公开(公告)号：US3865604A
公开(公告)日：1975-02-11
申请号：US34672273
申请日：1973-04-02
申请人： SANDOZ LTD
发明人： RIEDEL MANFRED , WOLF RAINER
IPC分类号： C08L1/00 , C08L1/22 , D01F2/00 , D01F2/08 , C08B21/20 , C08B27/52
CPC分类号： C08B16/00 , C08K5/0066 , C08K5/5399 , D01F2/10 , C08L1/22
摘要： The products of the reaction between (NPCl2 n, where n is at least 3, and a glycol are used as flame retardants in the production of regenerated cellulose materials of reduced flammability. Production of regenerated cellulose materials of reduced flammability is effected by precipitating the cellulose from a solution containing the above mentioned products.
摘要翻译：在生产具有降低的可燃性的再生纤维素材料的（NPCl2 n，其中n至少为3）和二醇之间的反应的产物被用作阻燃剂。通过沉淀纤维素从包含上述产品的解决方案。

9. 发明授权

US3865571A Method for selective herbicidal treatment of cereal and carrot cultures 失效
标题翻译：谷物和胡萝卜培养物的选择性除草方法
公开(公告)号：US3865571A
公开(公告)日：1975-02-11
申请号：US27550672
申请日：1972-07-27
申请人： SANDOZ LTD
发明人： SCHULER MAX
IPC分类号： B43M7/00 , C07C273/18 , C07C275/34 , A01M21/04
CPC分类号： C07C273/1845 , C07C273/1827 , C07C275/34
摘要： N-(3-chloro-4-methoxyphenyl)-N'',N''-dimethylurea of the formula:

IS DISCLOSED AS POSSESSING A SURPRISING SELECTIVE HERBICIDAL ACTIVITY. A method is disclosed for selectively combating weeds in a cereal locus and a carrot locus, which comprises applying to the locus to be protected from weeds, a dosage of from 2 to 10 kilograms per hectare of the above compound.
摘要翻译：具有下式的N-（3-氯-4-甲氧基苯基）-N'，N'-二甲基脲：

10. 发明授权

US3853915A 9-or 10-halo-4h-benzo{8 4,5{9 cyclo-hepta{8 1,2-b{9 thiophen-4-ones 失效
标题翻译： 9-OR 10-HALO-4H-BENZO {8} 4,5 {9环己基-β-{8,12-B {9-噻吩-4-酮
公开(公告)号：US3853915A
公开(公告)日：1974-12-10
申请号：US27873872
申请日：1972-08-08
申请人： SANDOZ LTD
发明人： BOURQUIN J , SCHWARB G , WALDVOGEL E
IPC分类号： C07D333/24 , C07D333/80 , C07D63/18
CPC分类号： C07D333/24 , C07D333/80 , Y10S514/885
摘要： The present invention concerns novel compounds of the formula,

WHEREIN R1 is hydrogen, halogen, or alkoxy of 1 to 4 carbon atoms, and Y is chlorine or bromine in the 9 or 10 position. The compounds are intermediates for the production of pharmacologically active compounds, particularly for compounds which are histaminolytics.
摘要翻译：本发明涉及下式的新型化合物，其中R1是氢，卤素或1-4个碳原子的烷氧基，Y是9或10位的氯或溴。

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