专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明专利

JPS6165894A Thiazine phosphonic acid derivative, its preparation and insecticide 失效
标题翻译：噻吩磷酸衍生物，其制备和杀虫剂
公开(公告)号：JPS6165894A
公开(公告)日：1986-04-04
申请号：JP18874484
申请日：1984-09-08
申请人： Nippon Chem Ind Co Ltd:The , Shionogi & Co Ltd
发明人： HAYASE YOSHIO , ICHINARI MITSUHIRO , TAGUCHI JUNJI , ISHIGURO TAKEO , TAKAHASHI TOSHIO
IPC分类号： A01N57/32 , C07D279/06 , C07F9/6544
CPC分类号： C07D279/06 , A01N57/32 , C07F9/6544
摘要： NEW MATERIAL:A compound of formula I (R
1 , R
2 are lower alkoxy, lower alkinyloxy, lower alkylthio, arylthio, lower alkylamino; R
3 , R
4 are H, lower alkyl; R
5 is lower alkyl, lower alkoxy, halogen, trifuoromethyl; X is O, S; m is 0W3).
EXAMPLE: 2-Phenylimino-5,5-dimethyl-3,4,5,6-tetrahydro-2H-1,3-thazine-3-thiol phosphonic acid O-methyl S-sec-butyl ester.
USE: Insecticide.
PREPARATION: The reaction between a compound of formula II and another compound of formula III (Y is eliminating group) is conducted, preferably in an inert solvent in the presence of an acid acceptor such as triethylamine at 20W30°C for 2W8hr.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新物质：式I化合物（R 1，R 2）为低级烷氧基，低级烷氧基，低级烷硫基，芳硫基，低级烷基氨基; R 3，R 4为H，低级烷基; 低级烷基，低级烷氧基，卤素，三氟甲基; X为O，S; m为0-3）。实施例：2-苯基亚氨基-5,5-二甲基-3,4,5,6-四氢-2H- 1,3-thazine-3-硫醇膦酸O-甲基S-仲丁酯。用途：杀虫剂。制备：式Ⅱ化合物与另一种式III化合物（Y为取代基）的反应优选在惰性溶剂中，在酸受体如三乙胺存在下，于20-30℃进行反应， 8小时

2. 发明专利

JPS59128306A Fungicide for agricultural purpose 失效
标题翻译：农药用杀真菌剂
公开(公告)号：JPS59128306A
公开(公告)日：1984-07-24
申请号：JP505883
申请日：1983-01-13
申请人： Shionogi & Co Ltd
发明人： MAKIKADO TOKUO , MURABAYASHI AKIRA , WATANABE YOSHIYA , TAKAHASHI TOSHIO
IPC分类号： A01N43/80
摘要： PURPOSE: A fungicide for agricultural purpose that contains one of isoxazole derivatives bearing a halogenoacetamide group, a part of which are novel, as an active ingredient, thus showing powerful fungicidal action against fungi causative crop diseases and being suitable for controlling gray mold in cucumber and other diseases.
CONSTITUTION: A compound of the formula (R
1 is H, alkyl, phenyl which may be substituted, thienyl, furyl; R
2 is H, alkyl, alkoxy, halogen; R
3 is H, alkyl, alkenyl, alkanoyl, phenylalkyl; X is Cl, Br, I), a part of its analogues are novel compounds, is included to give the objective fungicide for agricultural purpose. It is applied to, e.g., seeds, shoots, flower buds, flower bunches, trees, branches, leaves, fruits, soil to control gray mode, Sclerotium, Downy mildew, Anthracnose, powdery mildew or damping-off in cucumber and rice blast.
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：目的：一种用于农业用途的杀真菌剂，其中含有一种具有卤代乙酰胺基团的异恶唑衍生物，其中一部分是新颖的，作为活性成分，因此对真菌致病作物疾病具有强大的杀真菌作用，适用于控制黄瓜中的灰霉病，其他疾病构成：式（R 1）的化合物是H，烷基，可被取代的苯基，噻吩基，呋喃基; R 2是H，烷基，烷氧基，卤素; R 3是H，烷基，烯基，烷酰基，苯基烷基; X是Cl，Br，I），其一部分类似物是新化合物，被包括以提供用于农业目的的客观杀真菌剂。适用于例如种子，芽，花芽，花束，树木，树枝，叶，果实，土壤以控制灰色模式，鳞翅目，霜霉病，炭疽病，黄瓜和稻瘟病中的白粉病或阻滞。

3. 发明专利

JPS5978168A Stabilized imidazole complex and agricultural fungicide containing the same 失效
标题翻译：稳定的咪唑复合物和含有其的农业化合物
公开(公告)号：JPS5978168A
公开(公告)日：1984-05-04
申请号：JP19059982
申请日：1982-10-28
申请人： Shionogi & Co Ltd
发明人： OGATA HIDE , TAKAHASHI TETSUYA , WATANABE YOSHIHISA , TAKAHASHI TOSHIO
IPC分类号： C07D233/60 , A01N43/50
摘要： NEW MATERIAL:The stabilized imidazole complex obtained by treating the compound of formula I (R
1 is alkyl or phenylalkyl which may have 1W5 substituent groups selected from alkyl, alkoxy, halogen and CF
3 on benzene ring; R
2 is alkylidene; X is H, alkyl, alkoxy or halogen; n is integer of 1W4) with an acid or metallic salt capable of forming a stabilized complex therewith.
EXAMPLE: The (1:1) complex of phenolphthalin and compound of formula II.
USE: An agricultural fungicide relatively stable to light as an aqueous solution, and having long residual activity and low phytotoxicity to crops.
PROCESS: The stabilized imidazole complex can be prepared by treating the compound of formula I with an acid such as phenolphthalin, pamoic acid, etc. or a metallic salt such as cupric chloride, zinc chloride, nickel chloride, etc. capable of forming a stable complex with the compound of formula I .
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新材料：通过处理式I化合物（R 1是在苯环上可以具有1-5个选自烷基，烷氧基，卤素和CF 3的取代基的烷基或苯基烷基）得到的稳定的咪唑络合物; R 2是亚烷基; X为H，烷基，烷氧基或卤素; n为1-4的整数）与能与其形成稳定化络合物的酸或金属盐。实施例：酚酞和式II化合物的（1:1）络合物。用途：农药杀菌剂作为水溶液与光相对稳定，残留活性长，作物植物毒性低。方法：稳定的咪唑络合物可以通过用酸，如苯酚酞，双羟萘酸等处理式I化合物或能形成稳定的氯化铜，氯化锌，氯化镍等金属盐，与式I的化合物络合。

4. 发明专利

JPS5973575A Propynylaminoisoxazole derivative 失效
标题翻译：丙烯胺氧基唑衍生物
公开(公告)号：JPS5973575A
公开(公告)日：1984-04-25
申请号：JP17676282
申请日：1982-10-05
申请人： Shionogi & Co Ltd
发明人： MAKIKADO TOKUO , MURABAYASHI AKIRA , TAWARA KATSUYA , WATANABE YOSHIYA , TAKAHASHI TOSHIO , KONISHI TAKAO
IPC分类号： A01N43/80 , A61K31/42 , A61P31/04 , A61P31/10 , A61P33/02 , C07D261/14 , C07D413/04 , C07D413/06 , C07D413/12 , C07D521/00
CPC分类号： C07D231/12 , A01N43/80 , C07D233/56 , C07D249/08 , C07D261/14 , C07D413/04
摘要： NEW MATERIAL:A compound of formula I [R
1 and R
2 are H, alkyl, alkoxyl, cycloalkyl, R
5 -Y-, R
6 , R
6 -Y- or R
6 -Y-O-(R
5 is alkoxyl, alkylamino, etc.; Y is alkylene; R
6 is phenyl or aromatic heterocyclic ring residue containing N, O or S), R
1 and R
2 may link to form an alkylene; R
3 and R
4 are H or alkyl; X is H or I].
EXAMPLE: 3-Ethyl-4-chloro-5-(N-methyl-N-3-iodo-2-propynyl)aminoisoxazole.
USE: An antimycotic agent and agricultural germicide.
PROCESS: A desired group R
3 is introduced into the amino group in a compound of formula II as a raw material, and 2-propynyl group is then introduced into the resultant mono-substituted amino group to give the aimed substance. The R
3 and 2-propynyl groups are introduced into the compound of formula II by using the corresponding halide or dialkyl sulfate.
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新物质：式I化合物[R 1和R 2为H，烷基，烷氧基，环烷基，R 5 -Y-，R 6，R 6 -Y-或R“ （R 5是烷氧基，烷基氨基等; Y是亚烷基; R 6是含有N，O或S的苯基或芳族杂环残基），R 1和R 2是可以连接形成亚烷基; R 3和R 4是H或烷基; X为H或I]。实施例：3-乙基-4-氯-5-（N-甲基-N-3-碘-2-丙炔基）氨基异恶唑。用途：抗真菌剂和农业杀菌剂。方法：将所需基团R 3引入作为原料的式II化合物中的氨基，然后将2-丙炔基引入所得单取代的氨基中，得到目标物质。通过使用相应的卤化物或二烷基硫酸盐将R 3和2-丙炔基引入式II化合物。

5. 发明专利

JPS6147471A Triazine derivative and herbicide 失效
标题翻译： TRIAZINE衍生物和除草剂
公开(公告)号：JPS6147471A
公开(公告)日：1986-03-07
申请号：JP17013184
申请日：1984-08-15
申请人： Shionogi & Co Ltd
发明人： HAYASE YOSHIO , MORITA KOICHI , IDE KINYA , TAKAHASHI TOSHIO
IPC分类号： C07D251/26 , A01N43/70 , C07D251/52
CPC分类号： C07D251/52 , A01N43/70
摘要： NEW MATERIAL:The triazine derivative of formula I [R
1 , R
2 , R
3 and R
4 are H, aliphatic hydrocarbon residue, lower alkoxy(lower)alkyl, cyano(lower)alkyl, aryl(lower)alkyl, or R
1 and R
2 , or R
3 and R
4 together form a lower alkylene].
EXAMPLE: 2,4-Bis(ethylamino)-6-difluoromethyl-1,3,5-triazine.
USE: Herbicide effective to the weed in cultivated field such as plowed land, paddy field, orchard, tea plantation, mulberry plantation, disused land, etc., and uncultivated land such as railway, road, lawn, industrial site, river bed, building land, etc. It is effective to the weeds in plowed land and paddy field, such as large crab-grass, green foxtail, barnyard grass, wheat, etc. Harmless to man, animal and bird. It has high safety.
PREPARATION: The compound of formula I can be prepared by reacting the compound of formula II (X is eliminable group) with the compound of formula IIIin a solvent preferably in the presence of a base.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新物质：式I [R 1，R 2，R 3和R 4]的三嗪衍生物是H，脂族烃残基，低级烷氧基（低级）烷基，氰基（低级）烷基，芳基（低级）烷基，或R 1和R 2，或R 3和R 4一起形成低级亚烷基]。实施例：2,4-双（乙基氨基）-6-二氟甲基-1,3,5-三嗪。用途：除草剂，耕地，水田，果园，茶园，桑树种植园，废弃土地等耕地的除草剂，以及铁路，公路，草坪，工地，河床，建筑物等未耕地土地等，对ab草，绿草，稗草，小麦等耕地，水田等杂草有效。对人，动，禽无害。安全性高。制备：式I化合物可以通过使式II化合物（X是可消除基团）与式III化合物在溶剂中，优选在碱存在下反应来制备。

6. 发明专利

JPS59112978A Propynylaminothiazole derivative 失效
标题翻译：丙烯酰胺唑衍生物
公开(公告)号：JPS59112978A
公开(公告)日：1984-06-29
申请号：JP22527182
申请日：1982-12-21
申请人： Shionogi & Co Ltd
发明人： MAKIKADO TOKUO , MURABAYASHI AKIRA , TAWARA KATSUYA , WATANABE YOSHIYA , TAKAHASHI TOSHIO
IPC分类号： A01N43/78 , A61K31/425 , A61K31/426 , A61K31/428 , A61P31/04 , A61P31/10 , C07D277/20 , C07D277/42 , C07D277/56 , C07D277/82
CPC分类号： C07D277/82 , C07D277/42 , C07D277/56
摘要： NEW MATERIAL:A compound of formula I [R
1 is H, alkyl, carboxy, alkoxycarbonyl, formula II (R
4 is H or alkyl; R
5 is alkyl, carboxyalkyl, etc.), formyl, phenyl, etc.; R
2 is H, alkyl, alkoxycarbonyl or halogen; R
1 and R
2 together with the carbon atoms to which they are linked form a condensed benzene ring; R
3 is H or alkyl; X is H or I ].
EXAMPLE: 2-(N-Methyl-2-propynylamino)-5-methylthiazole.
USE: With powerful antifungal action and low toxicity, and capable of exhibiting a germicidal or fungistatic effect not only on fungi infecting humans and cattle therewith but also on pathogenic germs of agricultural and forestry and horticultural crops.
PROCESS: A 2-aminothiazole derivative of formula III is reacted with a 2-propynyl halide in an inert solvent in the presence of a base to afford the compound of formula I (X is H).
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新物质：式I化合物[R 1]为H，烷基，羧基，烷氧基羰基，式II（R 4为H或烷基; R 5为烷基，羧基烷基等），甲酰基，苯基等等 R 2是H，烷基，烷氧基羰基或卤素; R 1和R 2与它们所连接的碳原子一起形成稠合苯环; R 3是H或烷基; X为H或I]。实施例：2-（N-甲基-2-丙炔基氨基）-5-甲基噻唑。用途：具有强大的抗真菌作用和低毒性，并且能够不仅对感染人和牛的真菌表现出杀菌或抑菌作用，而且对农业和林业和园艺作物的病原菌也具有杀菌或抑菌作用。方法：将式III的2-氨基噻唑衍生物与2-丙炔基卤化物在惰性溶剂中在碱的存在下反应，得到式I化合物（X为H）。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式