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31. 发明专利

JPH08253449A SYNTHETIC INTERMEDIATE OF STERILIZER FOR AGRICULTURE AND ITS PRODUCTION 失效
公开(公告)号：JPH08253449A
公开(公告)日：1996-10-01
申请号：JP2270396
申请日：1996-02-08
申请人： SHIONOGI & CO
发明人： HAYASE YOSHIO , KATAOKA TAKAHIRO , TAKENAKA HIDEYUKI , ICHINARI MITSUHIRO , TANIMOTO NORIHIKO , MASUKO MICHIO , TAKAHASHI TOSHIO
IPC分类号： C07C251/50 , A01N37/18 , A01N37/50 , A01N41/04 , A01N41/10 , A01N43/08 , A01N43/16 , A01N43/20 , A01N43/40 , A01N43/42 , A01N43/44 , A01N43/54 , A01N43/78 , A01N55/00 , C07C235/72 , C07C235/78 , C07C249/12 , C07C251/48 , C07C317/44 , C07C317/48 , C07C323/47 , C07C323/60 , C07C323/62 , C07C323/63 , C07D213/64 , C07D215/22 , C07D215/227 , C07D239/34 , C07D277/20 , C07D277/34 , C07D277/68 , C07D303/46 , C07D307/36 , C07D307/40 , C07D307/42 , C07D309/12 , C07D333/24 , C07D521/00 , C07F7/08 , C07F7/10
摘要： PURPOSE: To obtain a synthetic intermediate for agricultural germicides having effect on rice blast, etc. CONSTITUTION: This compound is expressed by formula I (R and R are each independently H, a lower alkyl, etc.; R and R are each independently H, a halogenated lower alkyl, etc.; A is an unsaturated hydrocarbon, a halogenated unsaturated hydrocarbon, etc.; Z is CH2 , CO, etc.). The compound of formula I is obtained by amidating a compound of formula II. The compound of formula I is subjected to alkoximation to provide a compound of formula III [e.g. 2-(2- phenoxyphenyl)-2-methoxyiminoacetic amide].

32. 发明专利

JPH03246268A ALKOXYIMINOACETIC ACID AMIDE COMPOUND AND FUNGICIDE FOR AGRICULTURAL USE 失效
公开(公告)号：JPH03246268A
公开(公告)日：1991-11-01
申请号：JP12744190
申请日：1990-05-17
申请人： SHIONOGI & CO
发明人： HAYASE YOSHIO , KATAOKA TAKAHIRO , TAKENAKA HIDEYUKI , ICHINARI MITSUHIRO , TANIMOTO NORIHIKO , MASUKO MICHIO , TAKAHASHI TOSHIO
IPC分类号： C07C251/50 , A01N37/18 , A01N37/50 , A01N41/04 , A01N41/10 , A01N43/08 , A01N43/16 , A01N43/20 , A01N43/40 , A01N43/42 , A01N43/44 , A01N43/54 , A01N43/78 , A01N55/00 , C07C235/72 , C07C235/78 , C07C249/12 , C07C251/48 , C07C317/44 , C07C317/48 , C07C323/47 , C07C323/60 , C07C323/62 , C07C323/63 , C07D213/64 , C07D215/22 , C07D215/227 , C07D239/34 , C07D277/20 , C07D277/34 , C07D277/68 , C07D303/46 , C07D307/36 , C07D307/40 , C07D307/42 , C07D309/12 , C07D333/24 , C07D521/00 , C07F7/08 , C07F7/10
摘要： NEW MATERIAL:The compound of formula I [R and R are H, alkyl or cycloalkyl; R is alkyl or cycloalkyl; R and R are H, (halogenated) alkyl, alkoxy, alkylsilyl, halogen or NO2; A is (halogenated) unsaturated hydrocarbon group, phenyl or heterocyclic group; Z is CH2, CH(OH), CO, O, S, NR (R is H or alkyl), CH2CH2, CH=CH, group of formula II, CH2O, CH2S, CH2SO, OCH2, SCH2 or SOCH2]. EXAMPLE:2-(2-Phenoxyphenyl)-2-methoxyiminoacetic acid amide. USE:Fungicide for agricultural use. PREPARATION:The objective compound of formula I can be produced e.g. by reacting an oxocarboxylic acid of formula III or its reactive derivative at the carboxyl group with an amine of formula NHR R and reacting the resultant oxocarboxylic acid amide of formula IV with an alkoxylamine of formula H2NOR .

33. 发明专利

JPH03218355A NITROGEN-CONTAINING HETEROCYCLIC OXYPHENOXYACETIC ACID DERIVATIVE AND USE AS HERBICIDE 失效
公开(公告)号：JPH03218355A
公开(公告)日：1991-09-25
申请号：JP30143790
申请日：1990-11-06
申请人： SHIONOGI & CO , NIPPON CHEMICAL IND
发明人： HAYASE YOSHIO , MATSUMOTO KOHEI , KAMEI KAZUO , IDE KINYA , TAKAHASHI TOSHIO
IPC分类号： C07D241/44 , A01N43/40 , A01N43/60 , C07D213/64 , C07D213/643 , C07D401/12 , C07D403/12 , C07D405/12 , C07D413/12
摘要： NEW MATERIAL:A nitrogen-containing heterocyclic oxyphenoxyacetic acid derivative of formula I (R is pyridyl or quinoxalinyl which may be substituted with one or two halogen atoms or halogeno lower alkyl groups; R , R are H, lower alkyl; R is formula II, NHR , etc.; R , R are H, lower alkyl or both may be combined with the adjacent N to five or six membered saturated nitrogen-containing heterocyclic ring group which may further contain an atom selected from N, S and O hetero atoms; R is lower cycloalkyl, allyl, etc.) or a salt thereof. EXAMPLE:N-Methoxycarbonylmethoxy-2-[4-(3,5-dichloro-2-pyridyloxy) phenoxy]propionamide. USE:Useful as a herbicide. The compound of formula I does not cause chemical injuries on broad-leaved crops and exhibits intergenetic selectivity on monocotyledon plants. PREPARATION:The compound of formula I is prepared by the reaction equation shown in this caption.

34. 发明专利

JPH03218312A PREVENTIVE AND TREATING AGENT OF MICROBISM FOR ANIMAL 失效
公开(公告)号：JPH03218312A
公开(公告)日：1991-09-25
申请号：JP31957990
申请日：1990-11-21
申请人： SHIONOGI & CO
发明人： IMOSE JUN , TOBITAKA SHIGETADA , OGATA HIDE , KATAOKA TAKAHIRO , UEDA KAZUO , TAKAHASHI TOSHIO
IPC分类号： C07D401/04 , A61K31/435 , A61K31/47 , A61K31/535 , A61P31/04 , C07D471/04 , C07D498/06
摘要： PURPOSE:To obtain the title preventive and treating agent effective especially for animal respiratory infectious diseases, comprising a specific pyridonecarboxylic acid compound as an active ingredient. CONSTITUTION:The title preventive and treating agent comprising a compound shown by formula I [R is (halo) alkyl, cycloalkyl or (substituted) phenyl; R and R are H, OH, alkoxy, halogen or CH2N (R ) R (R and R are H, alkyl, alkenyl, etc.); R is H, oxo, alkoxy, halogen, or CH2N (R ) R (R and R are H or alkyl); X is H or halogen; Y is CQ (Q is H or halogen), N or Y is bonded to R to form group shown by formula II (R is H or alkyl); Z is H or NH2; (l) and (n) are 1 or 2; (m) is 0 or 1] or a salt thereof as an active ingredient. The preventive and treating agent is effective against mycoplasma infectious diseases and infectious KORIZA infectious diseases of domestic fowl, swine mycoplasma infectious diseases and haemophilus pleuropneumonia, bovine mycoplasma pneumonia, etc.

35. 发明专利

JPS62228089A ORGANIC PHOSPHORUS COMPOUND, PRODUCTION THEREOF AND INSECTICIDAL AND MITICIDAL AGENT CONTAINING SAME 失效
公开(公告)号：JPS62228089A
公开(公告)日：1987-10-06
申请号：JP29096786
申请日：1986-12-06
申请人： SHIONOGI & CO , NIPPON CHEMICAL IND
发明人： HAYASE YOSHIO , ICHINARI MITSUHIRO , KAMEI KAZUO , TAGUCHI JUNJI , OBA KATSUAKI , TAKAHASHI TOSHIO
IPC分类号： C07F9/24 , A01N57/32 , C07F9/6539
摘要： NEW MATERIAL:The compound of formula I (R and R are 1-5C alkoxy or 1-5C alkylthio; R -R are H or 1-5C alkyl; R -R are H, 1-5C alkyl or halogen; X is O or S). EXAMPLE:2-Phenylimino-1,3-thiazolidine-3-thiolphosphonic acid O-methyl S-sec- butyl ester. USE:Insecticidal and miticidal agent. PREPARATION:The compound of formula II (e.g. 2-phenylimino-1,3-thiazolidine) is made to react with the compound of formula III (Y is eliminable group) (e.g. monochlorothiolphosphoric acid O-methyl S-sec-butyl ester).

36. 发明专利

JPS6229594A THIAZINE RING-CONTAINING ORGANIC PHOSPHOROUS COMPOUND 失效
公开(公告)号：JPS6229594A
公开(公告)日：1987-02-07
申请号：JP17050785
申请日：1985-07-31
申请人： SHIONOGI & CO , NIPPON CHEMICAL IND
发明人： HAYASE YOSHIO , ICHINARI MITSUHIRO , TAGUCHI JUNJI , ISHIGURO TAKEO , TAKAHASHI TOSHIO
IPC分类号： C07F9/6558 , A01N57/32
摘要： NEW MATERIAL:A compound shown by the formula I (R and R are lower alkoxy, lower alkynyloxy, lower alkylthio or arylthio; R and R are H or lower alkyl; R -R are H, lower alkyl, halogen or CF3; Y is methine or N; n is 1 or 2). EXAMPLE:2-( 2,4-Dichlorobenzylimino )-5,5-dimethyl-3,4,5,6-tetrahydro-2H -1,3-thia zine-3-thiolphosphonic acid O-methyl,S-iso-butyl ester. USE:An insecticide. PREPARATION:A compound shown by the formula II is reacted with a compound (e.g., O-methyl S-iso-butylthiophosphoric acid chloride, etc.,) shown by the formula III (Z is eliminable group) preferably in a solvent (e.g., toluene, etc.,) in the presence of a base (e.g., triethylamine, etc.,) at 20-80 deg.C for 2-8hr.

37. 发明专利

JPS59112978A Propynylaminothiazole derivative 失效
标题翻译：丙烯酰胺唑衍生物
公开(公告)号：JPS59112978A
公开(公告)日：1984-06-29
申请号：JP22527182
申请日：1982-12-21
申请人： Shionogi & Co Ltd
发明人： MAKIKADO TOKUO , MURABAYASHI AKIRA , TAWARA KATSUYA , WATANABE YOSHIYA , TAKAHASHI TOSHIO
IPC分类号： A01N43/78 , A61K31/425 , A61K31/426 , A61K31/428 , A61P31/04 , A61P31/10 , C07D277/20 , C07D277/42 , C07D277/56 , C07D277/82
CPC分类号： C07D277/82 , C07D277/42 , C07D277/56
摘要： NEW MATERIAL:A compound of formula I [R
1 is H, alkyl, carboxy, alkoxycarbonyl, formula II (R
4 is H or alkyl; R
5 is alkyl, carboxyalkyl, etc.), formyl, phenyl, etc.; R
2 is H, alkyl, alkoxycarbonyl or halogen; R
1 and R
2 together with the carbon atoms to which they are linked form a condensed benzene ring; R
3 is H or alkyl; X is H or I ].
EXAMPLE: 2-(N-Methyl-2-propynylamino)-5-methylthiazole.
USE: With powerful antifungal action and low toxicity, and capable of exhibiting a germicidal or fungistatic effect not only on fungi infecting humans and cattle therewith but also on pathogenic germs of agricultural and forestry and horticultural crops.
PROCESS: A 2-aminothiazole derivative of formula III is reacted with a 2-propynyl halide in an inert solvent in the presence of a base to afford the compound of formula I (X is H).
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新物质：式I化合物[R 1]为H，烷基，羧基，烷氧基羰基，式II（R 4为H或烷基; R 5为烷基，羧基烷基等），甲酰基，苯基等等 R 2是H，烷基，烷氧基羰基或卤素; R 1和R 2与它们所连接的碳原子一起形成稠合苯环; R 3是H或烷基; X为H或I]。实施例：2-（N-甲基-2-丙炔基氨基）-5-甲基噻唑。用途：具有强大的抗真菌作用和低毒性，并且能够不仅对感染人和牛的真菌表现出杀菌或抑菌作用，而且对农业和林业和园艺作物的病原菌也具有杀菌或抑菌作用。方法：将式III的2-氨基噻唑衍生物与2-丙炔基卤化物在惰性溶剂中在碱的存在下反应，得到式I化合物（X为H）。

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