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71. 发明公开

EP0122533A3 Colour-photographic recording material containing a colour coupler 失效
标题翻译：包含彩色耦合器的彩色摄影记录材料
公开(公告)号：EP0122533A3
公开(公告)日：1987-01-28
申请号：EP84103642
申请日：1984-04-03
申请人： Agfa-Gevaert AG
发明人： Renner, Günter, Dr. , Wolff, Erich, Dr. , Sommer, Friedhelm, Dipl.-Chem. , Stark, Herbert, Dr. , Stieler, Dieter, Dipl.-Phys. , Meier, Egon, Ing. grad.
IPC分类号： G03C07/36 , C07C103/30 , C07C103/38 , C07C147/10 , C07D233/90 , C07D487/04 , C07D235/14 , C07D249/10
CPC分类号： C07D249/12 , C07C43/225 , C07D235/12 , G03C7/30535

72. 发明公开

EP0194764A1 Pesticidal compounds 失效
标题翻译： Pestizide Verbindungen。
公开(公告)号：EP0194764A1
公开(公告)日：1986-09-17
申请号：EP86301074.0
申请日：1986-02-17
申请人： THE WELLCOME FOUNDATION LIMITED
发明人： Blade, Robert John , Black, Malcolm Henry , Weston, John Bernard , Larkin, Patrick , Robinson, John Edward
IPC分类号： C07C103/30 , C07D307/79 , C07D333/24 , C07D333/60 , C07D317/32 , C07D311/74 , C07C121/43 , A01N37/18 , A01N45/00 , A01N43/12 , A01N43/10
CPC分类号： C07D307/79 , A01N37/18 , A01N37/20 , A01N37/26 , A01N37/38 , A01N37/46 , A01N43/06 , A01N43/14 , A01N43/28 , C07C17/2635 , C07C45/29 , C07C47/24 , C07C57/03 , C07C255/00 , C07C2603/26 , C07D311/20 , C07D333/24 , C07C22/08
摘要： Compounds of Formula (I):
wherein:

Ar is phenyl, naphthyl, thienyl, fluorenyl, phenanthrenyl, dibenzo furanyl or a polynuclear group (A):
in which a is 0, 1 or 2; B is (D) b (CH 2 ) c (E) e where each of D and E is oxygen or sulphur, b and e are independently 0 or 1 but not both 1, and c is 0,1, 2 or 3, the sum of a,b,c and e being at least 3, and the ring containing B is wholly or partially saturated; and G is hydrogen or a benzene ring fused to the benzene ring of group (A);
any of the groups Ar may be substituted by one or more of C 1-4 alkyl, halo-(C 1-4 ) alkyl, halo, C 1-4 alkoxy (except 3,4-methylenedioxy) or C 1-4 halo -alkoxy; n is 1 to 8. except that n is 1 to 4 when Ar is phenyl or substituted phenyl;
each of R 2 and R 3 is in each case independently hydrogen, C 1-4 alkyl or halo-(C 1-4 ) alkyl; and R and R' are each selected from hydrogen, alkyl, cycloalkyl, alkenyl or alkoxy (any of which may be substituted by halo, alkenyl, alkyl, cycloalkyl, alkoxy, alkynyl or cyano) are insecticidal and acaricidal.
摘要翻译：式（I）化合物：其中：Ar为苯基，萘基，噻吩基，芴基，菲基，二苯并呋喃基或多核基团（A）。其中a为0,1或2; B是（D）b（CH 2）c（E）e，其中D和E中的每一个是氧或硫，b和e独立地是0或1而不是两者，而c是0,1,2或3， a，b，c和e为至少3，并且含有B的环全部或部分饱和; 和G是氢或与（A）组的苯环稠合的苯环; 卤素 - （C 1-4）烷基，卤代，C 1-4烷氧基（3,4-亚甲基二氧基）或C 1-4卤代 - 烷氧基中的一个或多个取代基中的任何基团Ar可以被一个或多个取代。 n为1至8，当Ar为苯基或取代苯基时，n为1至4; R 2和R 3各自独立地为氢，C 1-4烷基或卤代（C 1-4）烷基; R和R 1各自选自氢，烷基，环烷基，烯基或烷氧基（其中任何一个可被卤素，烯基，烷基，环烷基，烷氧基，炔基或氰基取代）是杀虫和杀螨的。 >

73. 发明公开

EP0184822A2 Novel anilide derivatives of substituted arylacetic acids 失效
标题翻译： Anilidderivate von substituteierterArylessigsäure。
公开(公告)号：EP0184822A2
公开(公告)日：1986-06-18
申请号：EP85115720.6
申请日：1985-12-10
申请人： SUMITOMO PHARMACEUTICALS COMPANY, LIMITED
发明人： Kawakami, Hajime , Hashimoto, Katsuhiro , Tamoto, Katsumi , Ono, Keiichi , Yamamoto, Michihiro
IPC分类号： C07C103/28 , C07C143/80 , C07C103/30 , C07D213/56 , A61K31/63 , A61K31/165 , A61K31/16 , C07D307/54 , C07D333/24 , A61K31/34
CPC分类号： C07D307/54 , C07D213/56 , C07D333/24
摘要： A compound of the formula I:
wherein Ar is a heterocyclic group or an aromatic hydrocarbon group optionally having one or two substituents selected from the group consisting of halogen, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, nitro, cyano, di(C 1 -C 4 ) alkylamino, benzyloxy, hydroxy, C 1 -C 4 alkylthio, C 1 -C 4 alkylsulfinyl, C 1- C 4 alkylsulfonyl and C 1 -C 4 alkanoylamino, X is a hydroxyl group or either one of the following groups:
(in which R 2 , R 3 , R 4 and R 5 are each independently hydrogen or C 1 -C 4 alkyl or, when R 2 and R 3 or R 4 and R 5 are taken together with the adjacent nitrogen atom to which they are attached, they represent pyrrolidino, piperidino, morpholino, N-(C 1 -C 4 )-alkylpiperazino or N-phenylpipera- zino), R is an aromatic hydrocarbon or heterocyclic group and n is an integer of 1 to 4, or its acid addition salt, which is useful as a cerebral metabolism stimulant or a nootropic agent.
摘要翻译：式I的化合物：其中Ar是杂环基或任选具有一个或两个选自卤素，C 1 -C 4烷基，C 1 -C 4烷氧基，硝基，氰基，二（C 1 -C 4）烷基氨基，苄氧基，羟基，C 1 -C 4烷硫基，C 1 -C 4烷基亚磺酰基，C 1 -C 4烷基磺酰基和C 1 -C 4烷酰氨基，X为羟基或下列基团之一： R 2，R 3，R 4和R 5各自独立地是氢或C 1 -C 4烷基，或者当R 2和R 3或R 4和R 5 它们与相邻的氮原子连在一起，它们代表吡咯烷子基，哌啶子基，吗啉代，N-（C 1 -C 4） - 烷基哌嗪基或N-苯基哌嗪基），R是芳族烃或杂环基，n是 1〜4的整数，或其酸加成盐，其可用作脑代谢兴奋剂或诱发剂。

74. 发明公开

EP0183177A1 Unsaturated fatty acid derivatives and their production 失效
标题翻译： UngesättigteFettsäurederivateund deren Herstellung。
公开(公告)号：EP0183177A1
公开(公告)日：1986-06-04
申请号：EP85114733.0
申请日：1985-11-19
申请人： SUMITOMO PHARMACEUTICALS COMPANY, LIMITED
发明人： Nakamura, Toshio , Muraoka, Masami , Ono, Keiichi , Yamamoto, Michihiro
IPC分类号： C07C103/56 , C07C103/30 , A61K31/16 , C07D295/18 , A61K31/23 , A61K31/19 , C07C69/732 , C07C69/734 , C07C59/42 , C07C59/46
CPC分类号： C07D295/185 , C07C59/42 , C07C59/46 , C07D309/12
摘要： A compound of the formula:
wherein Y is a free or esterified carboxyl group, or a group of the formula:
(wherein R a and R b are each independently a hydrogen atom, a C 1 -C 4 alkyl group, a C 3 -C 7 cycloalkyl group, a benzyl group, a phenyl group, a phenyl group substituted with a halogen atom or a C 1 -C 4 alkyl group, or, when taken together with the adjacent nitrogen atom, they represent a 5 to 7 membered saturated heterocyclic goup); R' is a C 1 -C 12 alkyl group, a C 2 -C 12 alkenyl group, a C 2 -C 12 alkynyl group, a C 3 -C 10 cycloalkyl group, a C 4 -C 10 cycloalkenyl group, a hydroxy C 1 -C 13 alkyl group, an C 1 -C 12 alkyl group substituted with a group of the formula:
(wherein R c and R d are each independently a hydrogen atom, or a C,-C 4 alkyl group), a C 3 -C 10 heterocyclic group, a phenyl group optionally substituted with one to three substituents selected from the group consisting of halogen atom, hydroxyl group, C 1 -C 4 alkyl group, trifluoromethyl group, C 1 -C 4 alkoxy group, and group of the formula:
(wherein R c and R d are as defined above) or a group of the formula:
[wherein A is a C 1 -C 7 alkylene chain and B is a C 3 -C 10 cycloalkyl group, a C 4 -C 10 cycloalkenyl group, a C 1 -C 12 alkoxy group, a C 1 -C 12 alkylthio group, a C 3 -C 10 cycloalkoxy group, a C 4 -C 10 cycloalkenyloxy group, a C 3 -C 10 heterocyclic group, or a phenyl or phenoxy group optionally substituted with one to three substituents selected from the group consisting of halogen atom, hydroxy group, C 1 -C 4 alkyl group, group of the formula:
(wherein R c and R d are as defined above), trifluoromethyl group, C 1 -C 4 alkylthio group and C,-C 4 alkoxy group]; n is 2, 3 or 4; R 2 and R 3 are hydrogen atoms or, when taken together, they mean a single linkage to form a trans double bond between the adjacent carbon atoms, and E is a cis or trans vinylene group; provided that when n is 3 and R' is a n-octyl group, a 2-octenyl group or a 2,5-octadienyl group, R 2 and R 3 are hydrogen atoms, and that when n is 2, E is a trans vinylene group or a non-toxic pharmaceutically acceptable salt thereof. Said compound have potent anti-leucotriene B 4 action, and are useful in the treatment of inflammation and allergy.
摘要翻译：下式的化合物：其中Y是游离或酯化的羧基，或下式的基团：其中R a和R b各自独立地为氢原子，C1- C4烷基，C3-C7环烷基，苄基，苯基，被卤素原子或C1-C4烷基取代的苯基，或者当与相邻的氮原子一起时，它们代表5 至7元饱和杂环苷）; R 1是C 1 -C 12烷基，C 2 -C 12烯基，C 2 -C 12炔基，C 3 -C 10环烷基，C 4 -C 10环烯基，羟基C 1 -C 13烷基，C 1 被下式基团取代的-C 12烷基：其中R c和R d各自独立地为氢原子或C 1 -C 4烷基，C 3 -C 10杂环基，任选被一至三个选自卤素原子，羟基，C 1 -C 4烷基，三氟甲基，C 1 -C 4烷氧基的取代基取代的苯基，和下式基团：其中R c >和R d如上定义）或下式的基团：AB [其中A是C 1 -C 7亚烷基链，B是C 3 -C 10环烷基，C 4 -C 10环烯基，C 1 -C 12 烷氧基，C1-C12烷硫基，C3-C10环烷氧基，C4-C10环烯基氧基，C3-C10杂环基或苯基或苯氧基，任选被一至三个选自由卤素原子，羟基，C 1 -C 4烷基组成的基团，其结构式为：CHEM（其中R c和R d如上所定义），三氟甲基，C 1 -C 4烷硫基和C 1 -C4烷氧基]; n为2,3或4; R 2和R 3是氢原子，或者当它们一起表示单键以在相邻碳原子之间形成反式双键时，E是顺式或反式亚乙烯基; 条件是当n为3且R 1为正辛基，2-辛烯基或2,5-辛二烯基时，R 2和R 3为氢原子，当n为 2，E是反式亚乙烯基或其无毒的药学上可接受的盐。所述化合物具有有效的抗白三烯B4作用，并且可用于治疗炎症和变态反应。

75. 发明公开

EP0171146A1 13-Aza-14-oxo-txa2 analogues 失效
标题翻译： 13氮杂-14-氧代 - TXA2类似物。
公开(公告)号：EP0171146A1
公开(公告)日：1986-02-12
申请号：EP85304148.1
申请日：1985-06-12
申请人： ONO PHARMACEUTICAL CO., LTD.
发明人： Miyake, Hajimu , Okegawa, Tadao , Kawasaki, Akiyoshi
IPC分类号： C07C103/38 , C07C103/42 , C07C103/30 , C07C103/46 , C07C149/32 , C07C149/26 , C07C125/065 , C07C127/15 , C07C177/00 , C07C103/00 , A61K31/00
CPC分类号： C07D209/18 , C07C33/14 , C07C51/367 , C07C59/11 , C07C405/0091
摘要： A novel 13-aza-14-oxo-TXA 2 analogue of general formula:
[wherein symbol A represents

(i) a group of general formula: -CH 2 CH 2 -(CH 2 ) m -,
(ii)) a group of general formula: cis-CH=CH-(CH 2 ) 17 ,
(iii) a group of general formula: -CH 2 O-(CH 2 ) m -,
(iv) a group of general formula: -S-(CH 2 ) m -(wherein m represents an integer of from 1 to 6) or
(v) a group of general formula: -

R 1 represents a hydrogen atom or a straight or branched alkyl group of from 1 to 12 carbon atom(s);
R 2 represents a bond or a straight or branched alkylene or alkylene group of from 1 to 10 carbon atom(s) unsubstituted or substituted by at least one of hydroxy group, amino group, halogen atom or phenylthio group;
R 3 represents
(i) a phenyl, phenoxy or phenylthio group unsubstituted or substituted by at least one of straight or branched alkyl or alkoxy group of from 1 to 6 carbon atom(s), halogen atom or hydroxy group,
(ii) a straight or branched alkyl, alkenyl or alkynyl group of from 1 to 6 carbon atom(s) unsubstituted or substituted by at least one of halogen atom or hydroxy group,
(iii) a cycloalkyl, cycloalkyloxy or cycloalkylthio group of from 4 to 7 carbon atoms unsubstituted or substituted by at least one of straight or branched alkyl group of from 1 to 6 carbon atom(s), halogen atom or hydroxy group,
(iv) a naphthyl, indolyl or indanyl group, or
(v) an amino group unsubstituted or substituted by at least one of straight or branched alkyl group of from 1 to 6 carbon atom(s); and
R 4 represents a hydrogen atom or a methyl group.
With proviso that, the carbon atom neighbored with R 3 in R 2 should have no substituents, when R 3 represents a phenyloxy, phenylthio, cycloalkyloxy or cycloalkylthio group unsubstituted or substituted.]
and cyclodextrin clathrates thereof and non-toxic salts thereof wherein R' represents a hydrogen atom possess an antagonistic activity on TXA 2 , in particular, inhibit blood platelet aggregation and contraction of artery, and are, therefore, useful for prevention and/or treatment of inflammation, hypertension, thrombus, cerebral apoplexy, asthma, cardiac infarction, angina pectoris, cerebral infarction and death by acute cardiac diseases in mammals, in particular in humans, which are induced by thromboxane A 2 .

76. 发明公开

EP0156644A1 Process and intermediates for 4-acetylimidazoles 失效
标题翻译： Verfahren und Zwischenproduktefür4-乙酰基咪唑。
公开(公告)号：EP0156644A1
公开(公告)日：1985-10-02
申请号：EP85302066.7
申请日：1985-03-26
申请人： PFIZER INC.
发明人： Reiter, Lawrence Alan
IPC分类号： C07D233/64 , C07C103/30
CPC分类号： C07D233/64 , C07D261/14
摘要： This invention provides a two-step process for the preparation of 4-acetylimidazoles. In the first step, a 4-acylamino-5-methylisoxazole is subjected to catalytic hydrogenolysis to give a 4-amino-3-acyl-amino-3-buten-2-one. In the second step, the intermediate 3-buten-2-one compound is cyclized to a 4-acetylimidazole by treatment with a basic agent. The 4-acetylimidazoles are chemical intermediates for preparing known antisecretory agents and histamine H 2 antagonists, useful for the treatment of gastric hyperacidity and peptic ulcers.
摘要翻译：本发明提供了制备4-乙酰基咪唑的两步法。在第一步中，将4-酰基氨基-5-甲基异恶唑进行催化氢解，得到4-氨基-3-酰基 - 氨基-3-丁烯-2-酮。在第二步中，通过用碱性试剂处理将中间体3-丁烯-2-酮化合物环化成4-乙酰基咪唑。 4-乙酰咪唑是制备已知的抗分泌剂和组胺H2拮抗剂的化学中间体，可用于治疗胃酸过多和消化性溃疡。

77. 发明公开

EP0150709A3 7-oxabicycloheptane prostaglandin analogs 失效
标题翻译： 7-氧杂二环庚烷前列腺素类似物
公开(公告)号：EP0150709A3
公开(公告)日：1985-10-02
申请号：EP85100040
申请日：1985-01-02
申请人： E.R. Squibb & Sons, Inc.
发明人： Nakane, Masami
IPC分类号： C07D493/08 , A61K31/34 , C07C103/30 , C07D307/00
CPC分类号： C07D493/08
摘要： 7-0xabicycloheptane substituted oxamide prostaglandin analogs are provided having the structural formula
and including all stereoisomers thereof. The compounds are cardiovascular agents useful, for example, in the treatment of thrombolytic disease.
摘要翻译：提供7-0x-二环庚烷取代的草酰胺前列腺素类似物，其具有结构式并且包括其所有立体异构体。这些化合物是有用的心血管药剂，例如，用于溶解血栓疾病的治疗。

78. 发明公开

EP0144844A2 Fluorine-containing compounds 失效
标题翻译：荧光黄酮
公开(公告)号：EP0144844A2
公开(公告)日：1985-06-19
申请号：EP84113916.5
申请日：1984-11-16
申请人： DAIKIN INDUSTRIES, LIMITED
发明人： Hisamoto, Iwao , Yamana, Masayuki
IPC分类号： C07C103/30 , C07C91/12 , C07C103/44 , C07C143/74 , C07C143/63 , C07C87/30 , C07C93/02
CPC分类号： B01F17/0064 , B01D19/0413 , B01F17/0042 , B01F17/0057 , B01D19/0418 , B01D19/0422 , B01D19/0427
摘要： A fluorine-containing compound of the formula:
wherein

R, is a C 3 -C 21 fluorinated hydrocarbon group or a C 3 -C 2 , fluorinated oxyhydrocarbon group;
X' is a C 1 -C 11 hydrocarbon group;
X 2 , X 3 and X 4 are each a C 2 -C 6 hydrocarbon group;
Y 1 is a group of the formula:

Y 2 is a group of the formula:

W 1 is a group of the formula:

W 2 is a C 1 -C 10 hydrocarbon group optionally having -OH or -COOH or a amide group in the backbone;
Z 1 is halogen or a group of the formula:

Z 2 is a group of the formula:

Z 3 is a group of the formula:

R 1 is hydrogen or a C 1 -C 5 hydrocarbon group;
R 2 is hydrogen or a C 2 -C 4 acyl group;
R 3 is hydrogen or a group of the formula: -(X 1 O) q H or -R 7 Z 3 ;
R 4 is a group of the formula: -(X 1 O) q H or -R 7 Z 3 ;
R 5 and R 6 are each a C 1 -C 20 hydrocarbon group or a group of the formula:
-(X 1 O) q H, -X 1 k COOM, -R, or -Y 1 X 1 k R f ;
R 7 is a C 1 -C 20 hydrocarbon group or a group of the formula: -(CH 2 CH 2 OCH 2 CH 2 ) r -;
R 8 , R 9 and R 10 are each a C 1 -C 20 hydrocarbon group or a group of the formula:
-(X 1 O) q H, -R f or -Y 1 X 1 k R f ;
R" is C 2 -C 6 alkylene group optionally having one or two oxygen or sulfur atoms;
R 12 is hydrogen, a C 1 -C 20 hydrocarbon group or a C 2 -C 20 acyl group;
R 13 is hydrogen or a C 1 -C 20 hydrocarbon group;
M is hydrogen, an alkali metal, an alkaline earth metal or a NH 4 group;
k is zero or one;
m is an integer of 1 to 50;
n is an integer of 1 to 5;
q is an integer of 1 to 20; and
r is an integer of 1 to 5.
摘要翻译：一种下式的含氟化合物：其中R f为C 3 -C 21氟化烃基或C 3 -C 21氟代羟基烃基; X 1是C 1 -C 11烃基; X 2，X 3和X 4各自为C 2 -C 6烃基; Y 1是下式的基团：CH 2 CH 2是下式的基团： W 1是下式的基团： W 2是C 1 -C 10烃基在骨架中任选具有-OH或-COOH或酰胺基; Z 1是卤素或下式的基团：CHEM> Z 2是下式的基团：CH 2 CH 3 Z 3是下式的基团： -COOM，-SO 3 M，-OSO 3 M，-O（OM）2或CHEM R 1是氢或C 1 -C 5烃基; R 2是氢或C 2 -C 4酰基; R 3是氢或下式的基团： - （X 1 O）q H或-R 7 Z 3; R 4是下式的基团： - （X 1 O）q H或-R 7 Z 3; R 5和R 6各自为C 1 -C 20烃基或下式基团： - （X 1 O）q H，-X 1 kCOOM，-R f或-Y 1 X 1 kR f; R 7是C 1 -C 20烃基或下式的基团： - （CH 2 CH 2 OCH 2 CH 2）r - ; R 8，R 9和R 1各自为C 1 -C 20烃基或下式基团： - （X 1 O）q H，-R f或-Y 1 X <1>的KrF; R 1是任选具有一个或两个氧或硫原子的C 2 -C 6亚烷基; R 1是氢，C 1 -C 20烃基或C 2 -C 20酰基; R 1是氢或C 1 -C 20烃基; M是氢，碱金属，碱土金属或NH 4基; k为零或一; m为1〜50的整数。 n为1〜5的整数， q为1〜20的整数， r为1〜5的整数

79. 发明公开

EP0120321A1 Acrylsäureamide, ihre Herstellung und Verwendung 失效
标题翻译：丙烯酰胺，其制备方法和用途。
公开(公告)号：EP0120321A1
公开(公告)日：1984-10-03
申请号：EP84102012.6
申请日：1984-02-27
申请人： Shell Agrar GmbH & Co. KG
发明人： Nickl, Josef, Dr. Dipl.-Chem. , Pieper, Helmut, Dr. Dipl.-Chem. , Curtze, Jürgen, Dr. Dipl.-Chem. , Drandarevski, Christo, Dr. , Lust, Sigmund, Dr.
IPC分类号： C07D295/18 , C07C103/30 , C07D265/30 , C07D317/60 , C07D213/56 , C07D307/54 , C07D333/24 , C07D295/22
CPC分类号： C07D295/185 , A01N37/10 , A01N37/34 , A01N37/38 , A01N37/44 , A01N37/46 , A01N37/48 , C07C45/46 , C07C59/64 , C07C205/45 , C07D213/56 , C07D295/194 , C07D295/32 , C07D307/54 , C07D317/60 , C07D333/24 , C07C49/84
摘要： Die Verbindungen der Formel Doppelkeg
in der A für die Gruppe
B für die Gruppe
Q für eine der Gruppen
und
X für 0, 5 oder NH, für einen gegebenenfalls substituierten Rest aus der Gruppe Alkyl-Alkenyl, -Cycloalkyl, -Cycloalkenyl, Pyridyl, Furyl,
Thienyl, α-und β-Naphthyl; oder zusammen mit der Gruppe CR 5 für einen
cycloaliphatischen Rest, an den ein Benzolring ankondensiert sein kann; oder für den Rest
steht, wobei

k die Zahlen 0, 1 oder 2,
m die Zahlen 1, 2, 3 oder 4,
n die Zahlen 0 oder 1,
R, Wasserstoff, C 1 -C 5 -Alkyl, Cyano und, wenn k gleich 0 ist, auch Chlor, Brom oder Jod,
R 2 und R 11 Wasserstoff, Halogen, Nitro, gegebenenfalls substituiertes -Alkyl oder -Alkoxy, -Alkinyloxy, Amino, NH( -Alkyl), N( -Alkyl) 2 , Cyano, Phenyl, -Cycloalkyl, -Alkenyloxy, Hydroxy( -Alkyl), NH COR 6 , CO 2 R 6 , CON-R 7 R 8 , durch Sauerstoff unterbrochenes -Alkyl oder

R 3 , R 4 , R 12 und R 13 Wasserstoff, Halogen, -Alkyl, -Alkoxy, (-Alkyl) -S(0)p (p = 0,1 oder 2), Hydroxy oder (-Acyl)oxy, R 3 /R 4 und R 12 =/R 13 jeweils gemeinsam auch Methylendioxy oder Ethylendioxy, gebunden an zwei Benachbarte Atome des Phenykings,
R 3 und R 4 Wasserstoff oder -Alkyl, R 5 außerdem, zusammen mit dem C-Atom, an das es gebunden ist, und Y einen cycloaliphatischen Rest, an den ein Benzolring ankondensiert sein kann
R 7 und R. -Alkyl, -Cycoalkyl, Phenyl, Benzyl, Furfuryl, Tetrahydrofurfuryl oder-Alkenyl, gemeinsam außerdem auch eine -Alkylentette. die durch 0, NR., S(0)q (mit q = 0, 1 oder 2) unterbrochen sein kann, R 7 außerdem Wasserstoff.
R. und R 16 , die nur vorliegen, wenn R 7 und R 3 gemeinsam eine Kette darstellen, Wasserstoff oder -Alkyl bedeuten, sowie gegebenenfalls die Säureadditionssalze der vorstehend defineirten Verbindungen, haben insbesondere fungizide Wirkung gegen phytopathogene Pilze.

Die Herstellung und Formulierung der Verbindungen erfolgt nach konventionellen Methoden.
摘要翻译：式Doppelkeg 其中A是该组的组 B的化合物Y-（CR5 = CR6）K（III）中，Q表示的基团之一 X是0，5或NH用于任选被取代的选自烷基烯基，环烷基，环烯基，吡啶基，呋喃基，噻吩基，α和β萘基; 或与CR5组为一个环族基团一起形成一个苯环可以稠合; 或表示基团其中，k是数字0,1或2，M的数字1，2，3或4，n中的号码0或1，R1是氢，C1-CA-烷基氰基和，如果k 等于0，也氯，溴或碘，R 2和R 11是氢，卤素，硝基，任选取代的烷基或烷氧基，炔氧基，氨基，NH（烷基），N（烷基）2，氰基，苯基，环烷基，链烯基，羟基（烷基），NH COR6，O2R6，CON-R7-R8，被氧烷基或 R3，R4，R12和R13是氢，卤素，烷基，烷氧基，（中断烷基）-S（O）p（p = 0时，1或2），羟基或（酰基）氧基，R3 / R4和R12 / R13在每一种情况下一起是可替换地亚甲二氧基或亚乙二氧基，连接到苯环，R 5的两个相邻原子并且R6是氢或烷基，R 5还连同碳原子其所连接，并且Y是环脂族基，向其中苯环可以稠合。 R7和R8是烷基，环烷基，苯基，苄基，糠基，四氢糠基或链烯基，也一起由0，NR 6，S（0）将被中断的亚烷基链Q（其中q = 0,1或2）也可以是氢，R9和R10，仅当R7和R8一起代表一个链，代表氢或烷基，和任选的上述defineirten化合物的酸加成盐具有抗植物病原性真菌特别是杀真菌活性发生R7。该化合物的制备和制剂根据常规方法进行。

80. 发明授权

EP0019745B1 2-Aminopropanalacetale, deren Herstellung, sie enthaltende Fungizide, deren Herstellung und Verfahren zur Bekämpfung von Pilzen 失效
标题翻译： 2-氨基壬酸乙酯，其制剂，含有它们的杀真菌配方，其制备和处理真菌的方法
公开(公告)号：EP0019745B1
公开(公告)日：1982-07-28
申请号：EP80102417.5
申请日：1980-05-05
申请人： BASF Aktiengesellschaft
发明人： Ammermann, Eberhard, Dr. , Zeeh, Bernd, Dr. , Thym, Sabine, Dr. , Plath, Peter, Dr. , Rentzea, Costin, Dr. , Eicken, Karl, Dr. , Goetz, Norbert, Dr. , Pommer, Ernst-Heinrich, Dr.
IPC分类号： A01N53/00 , A01N37/22 , A01N43/00 , A01N47/08 , C07C103/30 , C07C125/065 , C07C125/067 , C07C127/19 , C07C155/02 , C07D521/00
CPC分类号： C07D213/81 , A01N43/653 , C07D231/06 , C07D231/12 , C07D233/56 , C07D249/08 , C07D261/18 , C07D307/32 , C07D307/68 , C07D309/28 , C07D333/38

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