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1. 发明授权

US07053082B1 2,3-benzodiazepine derivatives 失效
公开(公告)号：US07053082B1
公开(公告)日：2006-05-30
申请号：US10030436
申请日：2000-07-04
申请人： Zoltan Greff , Geza Szabo , Jozsef Barkoczy , Zoltan Ratkai , Gabor Blasko , Gyula Simig , Gabor Gigler , Bernadett Martonné Marko , György Levay , Karoly Tihanyi , Andras Egyed , Annamaria Simo
发明人： Zoltan Greff , Geza Szabo , Jozsef Barkoczy , Zoltan Ratkai , Gabor Blasko , Gyula Simig , Gabor Gigler , Bernadett Martonné Marko , György Levay , Karoly Tihanyi , Andras Egyed , Annamaria Simo
IPC分类号： A61P25/00 , A61K31/551 , C07D491/04
CPC分类号： C07D491/04
摘要： The invention relates to new 2,3-benzodiazepine derivatives of general Formula (I), (wherein R1 stands for methyl, formyl, carboxy, cyano, —CH═NOH, —CH═NNHCONH2 or —NR5R6, wherein R5 and R6 independently from each other represent hydrogen or lower alkyl or together with the nitrogen atom, they are attached to, form a 5- or 6-membered, saturated or unsaturated heterocyclic ring optionally containing one or more further nitrogen, sulfur and/or oxygen atom(s); R2 is nitro or amino; R3 stands for hydrogen, lower alkanoyl or CO—NR7R8, wherein R7 and R8 independently from each other stand for hydrogen, lower alkoxy, lower alkyl or lower cycloalkyl or together with the nitrogen atom, they are attached to, form a 5- or 6-membered, saturated or unsaturated heterocyclic ring optionally containing one or more further nitrogen, sulfur and/or oxygen atom(s); R4 is hydrogen or lower alkyl; the dotted lines have the following meaning: if R3 and R4 are not present, the bond between positions C8 and C9 is a single bond and the bond between positions C8 and N7 is a double bond; if R3 and R4 are present, the bonds between positions C8 and C9 and between position C8 and N7 are single bonds; and if R3 is present and R4 is missing, the bond between positions C8 and C9 is a double bond and the bond between positions C8 and N7 is a single bond) and salts thereof. The invention compounds have neuroprotective effect.

2. 发明授权

US07960375B2 8-chloro-2,3-benzodiazepine derivatives 失效
标题翻译： 8-氯-2,3-苯并二氮杂衍生物
公开(公告)号：US07960375B2
公开(公告)日：2011-06-14
申请号：US10567598
申请日：2004-07-29
申请人： Jozsef Barkoczy , Istvan Ling , Gyula Simig , Gabor Szenasi , Gabor Gigler , Szabolcs Kertesz , Gyula Szücs , Geza Szabo , Miklos Vegh , Laszlo Gabor Harsing
发明人： Jozsef Barkoczy , Istvan Ling , Gyula Simig , Gabor Szenasi , Gabor Gigler , Szabolcs Kertesz , Gyula Szücs , Geza Szabo , Miklos Vegh , Laszlo Gabor Harsing
IPC分类号： A61P9/10 , A61K31/55 , C07D243/02
CPC分类号： C07D243/02
摘要： The invention relates to new 8-chloro-2,3-benzodiazepine derivatives of the general formula (I), wherein R stands for a lower alkyl group or a group of the general formula —NH—R′, wherein R′ stands for a lower alkyl or a lower cycloalkyl group), and pharmaceutically acceptable acid addition salts thereof. The invention also encompasses a process for the preparation of said compounds, pharmaceutical compositions containing them and new intermediates useful for the preparation of the new 8-chloro-2,3-benzodiazepine derivatives. The compounds according to the invention possess AMPA/kainate receptor inhibiting activity.
摘要翻译：本发明涉及通式（I）的新的8-氯-2,3-苯并二氮杂衍生物，其中R代表低级烷基或通式-NH-R'基团，其中R'代表低级烷基或低级环烷基）及其药学上可接受的酸加成盐。本发明还包括制备所述化合物的方法，含有它们的药物组合物和可用于制备新的8-氯-2,3-苯并二氮杂衍生物的新中间体。根据本发明的化合物具有AMPA /红藻氨酸受体抑制活性。

3. 发明申请

US20080153814A1 8-Chloro-2,3-Benzodiazepine Derivatives 失效
标题翻译： 8-氯-2,3-苯并二氮杂衍生物
公开(公告)号：US20080153814A1
公开(公告)日：2008-06-26
申请号：US10567598
申请日：2004-07-29
申请人： Jozsef Barkoczy , Istvan Ling , Gyula Simig , Gabor Szenasi , Gabor Gigler , Szabolcs Kertesz , Gyula Szucs , Geza Szabo , Miklos Vegh , Laszio Gabor Harsing
发明人： Jozsef Barkoczy , Istvan Ling , Gyula Simig , Gabor Szenasi , Gabor Gigler , Szabolcs Kertesz , Gyula Szucs , Geza Szabo , Miklos Vegh , Laszio Gabor Harsing
IPC分类号： A61K31/551 , C07D243/02 , A61P25/00
CPC分类号： C07D243/02
摘要： The invention relates to new 8-chloro-2,3-benzodiazepine derivatives of the general formula (I), wherein R stands for a lower alkyl group or a group of the general formula —NH—R′, wherein R′ stands for a lower alkyl or a lower cycloalkyl group), and pharmaceutically acceptable acid addition salts thereof. The invention also encompasses a process for the preparation of said compounds, pharmaceutical compositions containing them and new intermediates useful for the preparation of the new 8-chloro-2,3-benzodiazepine derivatives. The compounds according to the invention possess AMPA/kainate receptor inhibiting activity.
摘要翻译：本发明涉及通式（I）的新的8-氯-2,3-苯并二氮杂衍生物，其中R代表低级烷基或通式-NH-R'基团，其中R'代表低级烷基或低级环烷基）及其药学上可接受的酸加成盐。本发明还包括制备所述化合物的方法，含有它们的药物组合物和可用于制备新的8-氯-2,3-苯并二氮杂衍生物的新中间体。根据本发明的化合物具有AMPA /红藻氨酸盐受体抑制活性。

4. 发明申请

US20090233913A1 OPTICAL ISOMERS OF DIHYDRO-2,3-BENZODIAZEPINES AND THEIR STEREOSELECTIVE SYNTHESIS 审中-公开
标题翻译：二氢-2,3-苯并嗪的光学异构体及其选择性合成
公开(公告)号：US20090233913A1
公开(公告)日：2009-09-17
申请号：US12159251
申请日：2006-12-29
申请人： Istvan Ling , Jozsef Barkoczy , Zoltan Greff , Gabor Szenasi , Gabor Gigler , Szabolcs Kertesz , Gyula Szucs , Mihaly Albert , Gabor Kapus , Geza Szabo , Miklos Vegh , Marta Agoston , Gyorgy Levay , Krisztina Moricz , Laszlo Gabor Harsing
发明人： Istvan Ling , Jozsef Barkoczy , Zoltan Greff , Gabor Szenasi , Gabor Gigler , Szabolcs Kertesz , Gyula Szucs , Mihaly Albert , Gabor Kapus , Geza Szabo , Miklos Vegh , Marta Agoston , Gyorgy Levay , Krisztina Moricz , Laszlo Gabor Harsing
IPC分类号： A61K31/551 , C07D243/02 , C07D311/76 , C07C243/28 , A61P25/08
CPC分类号： C07D243/02 , C07C251/86 , C07C309/66 , C07C309/73 , C07D311/76 , C07D317/58 , C07D403/06 , C07D491/04 , C07D493/04
摘要： The present invention relates to dihydro-2,3-benzodiazepine compounds of high enantiomeric purity according to the general formula (I), which contain an asymmetric centre at the position 4 of the dihydro-2,3-benzodiazepine compound, and the preparation thereof and the used intermediates as well. These compounds have anti-convulsiveA muscle relaxant and neuroprotective effect due their non-competitive AMPA antagonistic properties.
摘要翻译：本发明涉及具有通式（I）的高对映体纯度的二氢-2,3-苯并二氮杂化合物，它在二氢-2,3-苯并二氮杂化合物的4位含有不对称中心，其制备方法和二手中间体。这些化合物由于其非竞争性AMPA拮抗性质而具有抗惊厥性肌松弛剂和神经保护作用。

5. 发明授权

US09825841B2 Method of and network server for detecting data patterns in an input data stream 有权
公开(公告)号：US09825841B2
公开(公告)日：2017-11-21
申请号：US14411547
申请日：2012-06-29
申请人： Geza Szabo , Wesley Davison Braga Melo , Gabor Sandor Enyedi , Stenio Fernandes , Gergely Pongrácz , Djamel Sadok
发明人： Geza Szabo , Wesley Davison Braga Melo , Gabor Sandor Enyedi , Stenio Fernandes , Gergely Pongrácz , Djamel Sadok
IPC分类号： G06F15/16 , H04L12/26 , H04L12/851 , H04L29/06
CPC分类号： H04L43/50 , H04L47/2483 , H04L63/1408
摘要： Computer controlled method, network server (42, 43, 44, 46, 48) and system (40) for detecting data patterns in a data stream (36) received by a computer (30). The data stream (36) comprising a plurality of data symbols. The computer (30) executes a finite automata (10) comprising a plurality of states (11, 12, 13, 14, 15) including a start state (11) and at least one accepting state (15). State transitions (16) are triggered by a data symbol (17a) according to a state transition register (17) and the method comprises the steps of determining (21), by the computer (30), from a data symbol register (18) whether a data symbol of the data stream (36) is comprised in a group of data symbols not resulting in an accepting state (15), and triggering (22), by the computer (30), a transition (16) to the start state (11) for data symbols comprised in the group and a transition (23) to a state (12, 13, 14, 15) according to the state transition register (17) for detecting the data pattern otherwise.

6. 发明授权

US08514723B2 Traffic monitoring by lowest transmission layer marking 有权
标题翻译：交通监控通过最低传输层标记
公开(公告)号：US08514723B2
公开(公告)日：2013-08-20
申请号：US12996434
申请日：2008-06-05
申请人： Szabolcs Malomsoky , Tamas Borsos , Geza Szabo
发明人： Szabolcs Malomsoky , Tamas Borsos , Geza Szabo
IPC分类号： H04L12/26
CPC分类号： H04L43/026
摘要： A monitoring system is provided for monitoring transport of data through interconnected nodes for processing data packets in a communication system, wherein said data packets conform to a layered transmission protocol, the system comprising: (1) a marking node for marking a packet selected according to a marking rule by placing a monitoring indicator in the lowest protocol layer thereof, said data packet having a first number of protocol layers, (2) at least, one packet processing node for forming a data packet based or the marked packet, such that said formed data packet comprises a second number of protocol layers that is different from said first number of protocol layers and such that said indicator is in the lowest protocol layer of said formed data packet, and (3) a monitoring node for monitoring said transport of data on the basis of the indicators in data packets that have passed through the at least one packet processing node.
摘要翻译：提供了一种监视系统，用于监视通过互连节点的数据传输，以处理通信系统中的数据分组，其中所述数据分组符合分层传输协议，所述系统包括：（1）标记节点，用于标记根据通过将监视指示器放置在其最低协议层中，所述数据分组具有第一数量的协议层，（2）至少一个用于形成数据分组的分组处理节点或标记的分组，使得所述形成的数据分组包括与所述第一协议层数不同的第二数量的协议层，并且使得所述指示符处于所述形成的数据分组的最低协议层，以及（3）用于监视所述数据传输的监视节点基于已经通过至少一个分组处理节点的数据分组中的指示符。

7. 发明授权

US08280956B2 User behavior based mobile broadband user plane traffic generation system and method for real-like measurement generation 有权
标题翻译：基于用户行为的移动宽带用户平面流量生成系统和实时测量生成方法
公开(公告)号：US08280956B2
公开(公告)日：2012-10-02
申请号：US12857684
申请日：2010-08-17
申请人： Geza Szabo , Gergely Pongrácz , Zoltán Richárd Turányi
发明人： Geza Szabo , Gergely Pongrácz , Zoltán Richárd Turányi
IPC分类号： G06F15/16
CPC分类号： H04L67/22 , H04L41/00 , H04L43/00
摘要： A system, a method, and a graphical user interface testing tool are described herein for constructing a validation trace (i.e., high-speed realistic network traffic) using a real network without causing privacy concerns. In one embodiment, the method comprises the steps of: (a) providing a client device which has one or more applications operating thereon and a graphical user interface; (b) recording user interactions on the client device; (c) extracting usage scenarios from real network traffic in the real network; (d) emulating user actions on the client device according to a specific user scenario by utilizing the recorded user interactions and the extracted usage scenarios to generate additional real traffic in the real network; and (e) creating the validation trace based on the generated additional real traffic and the extracted usage scenarios.
摘要翻译：本文描述了一种系统，方法和图形用户界面测试工具，用于使用真实网络构建验证跟踪（即，高速实际网络流量）而不引起隐私问题。在一个实施例中，该方法包括以下步骤：（a）提供在其上操作一个或多个应用的客户端设备和图形用户界面; （b）在客户端设备上记录用户交互; （c）从实际网络中的真实网络流量提取使用场景; （d）通过利用记录的用户交互和所提取的使用场景在实际网络中产生附加的实际业务，根据特定用户场景模拟客户端设备上的用户动作; 和（e）基于生成的附加实际流量和所提取的使用场景来创建验证跟踪。

8. 发明申请

US20110019574A1 TECHNIQUE FOR CLASSIFYING NETWORK TRAFFIC AND FOR VALIDATING A MECHANISM FOR CLASSIFYING NETWORK TRAFFIC 审中-公开
标题翻译：分类网络交通和验证分类网络交通机制的技术
公开(公告)号：US20110019574A1
公开(公告)日：2011-01-27
申请号：US12922019
申请日：2008-03-10
申请人： Szabolcs Malomsoky , Daniel Orincsay , Geza Szabo
发明人： Szabolcs Malomsoky , Daniel Orincsay , Geza Szabo
IPC分类号： H04L12/26
CPC分类号： H04L47/10 , H04L41/5022 , H04L47/2441 , H04L47/2475
摘要： A technique for classifying network traffic in the form of data packets generated by multiple applications installed on a device (400) is provided. A method implementation of this technique performed by the device (400) comprises the steps of receiving data packets belonging to one or more data flows, wherein each data flow includes the data packets generated by a specific one of the multiple applications, analyzing the received data packets to identify the application associated with each analyzed data packet, and classifying at least one data flow by including an application identifier in at least one of the analyzed data packets of this data flow.
摘要翻译：提供了一种以设备（400）上安装的多个应用程序生成的数据包形式对网络流量进行分类的技术。由该设备（400）执行的该技术的方法实现包括以下步骤：接收属于一个或多个数据流的数据分组，其中每个数据流包括由多个应用中的特定应用产生的数据分组，分析所接收的数据分组，以识别与每个分析的数据分组相关联的应用，并且通过在该数据流的所分析的数据分组中的至少一个中包括应用标识符来对至少一个数据流进行分类。

9. 发明授权

US09124528B2 Method and arrangement for data clustering 有权
标题翻译：数据聚类的方法和布置
公开(公告)号：US09124528B2
公开(公告)日：2015-09-01
申请号：US13658031
申请日：2012-10-23
申请人： Geza Szabo , Gergely Pongrácz , Zoltán Richárd Turányi
发明人： Geza Szabo , Gergely Pongrácz , Zoltán Richárd Turányi
IPC分类号： H04L12/24 , H04L12/26 , H04L12/715 , H04L12/851
CPC分类号： H04L45/46 , H04L41/145 , H04L43/0882 , H04L43/16 , H04L47/2441
摘要： This disclosure relates a method within a network node and a corresponding network node for determining input information for creation of a data traffic clustering model. The method comprises obtaining data descriptors of data flows, wherein the data descriptors describe data of the data flows, and obtaining flow information of the data flows. In addition, the method comprises determining clustering model input information based on the obtained data descriptors and the obtained flow information. One exemplary advantage of the present disclosure is that it allows traffic clustering based solely on packet header information, making the present disclosure appropriate for handling encrypted traffic.
摘要翻译：本公开涉及网络节点和对应的网络节点中的方法，用于确定用于创建数据业务聚类模型的输入信息。该方法包括获取数据流的数据描述符，其中数据描述符描述数据流的数据，并获得数据流的流信息。另外，该方法包括基于所获得的数据描述符和获得的流信息来确定聚类模型输入信息。本公开的一个示例性优点是其仅允许基于分组报头信息的业务聚类，使得本公开适合于处理加密业务。

10. 发明申请

US20130194930A1 Application Identification Through Data Traffic Analysis 审中-公开
标题翻译：应用程序识别通过数据流量分析
公开(公告)号：US20130194930A1
公开(公告)日：2013-08-01
申请号：US13876288
申请日：2010-10-14
申请人： Geza Szabo , Zoltán Richárd Turányi
发明人： Geza Szabo , Zoltán Richárd Turányi
IPC分类号： H04L12/26
CPC分类号： H04L43/0876 , H04L41/0213 , H04L41/142 , H04L43/026 , H04L43/18
摘要： There is provided a method of processing, analysing or profiling traffic in a packet switched telecommunications network. During a first phase (S1 to S4), for each of a plurality of applications, traffic generated by the application is analysed (S2) to identify a collection of one or more characteristic bit sequences for the application, or at least such a plurality of collections is provided. During a second phase (S5 to S11), traffic is received from the network (S5), and the following steps are performed for each of at least one of the plurality of collections: (i) for each of at least one of the characteristic bit sequences in the collection: a sequence alignment process (S8) is performed on the received traffic against the characteristic bit sequence to derive a per-sequence score; and (ii) a per-collection score is assigned to the collection (S10) based on the per-sequence scores for the collection, the per-collection score being indicative of a likelihood that the traffic was generated by the application associated with the collection.
摘要翻译：提供了在分组交换电信网络中处理，分析或分析业务的方法。在第一阶段（S1至S4）期间，对于多个应用中的每一个应用，分析由应用产生的业务（S2）以识别用于该应用的一个或多个特征位序列的集合，或至少这样的多个提供集合。在第二阶段（S5至S11）期间，从网络（S5）接收业务，并且对多个集合中的至少一个集合中的每一个执行以下步骤：（i）对于以下各项中的至少一个：集合中的比特序列：针对特征比特序列对所接收的流量执行序列比对过程（S8）以导出每序列得分; 和（ii）基于收集的每序列得分将收集分数分配给收集（S10），每收集分数指示与收集相关联的应用程序生成的流量的可能性。

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