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1. 发明授权

US06852734B2 Indole derivatives exhibiting chymase-inhibitory activities and process for preparation thereof 失效
标题翻译：显示糜酶抑制活性的吲哚衍生物及其制备方法
公开(公告)号：US06852734B2
公开(公告)日：2005-02-08
申请号：US10275111
申请日：2001-05-01
申请人： Yasuo Yamamoto , Kenzo Hariyama , Yumiko Yanagisawa , Sojiro Shiokawa , Takumi Takeyasu , Osami Takenouchi , Hidenori Kasai
发明人： Yasuo Yamamoto , Kenzo Hariyama , Yumiko Yanagisawa , Sojiro Shiokawa , Takumi Takeyasu , Osami Takenouchi , Hidenori Kasai
IPC分类号： A61K31/4045 , A61K31/437 , A61K31/4709 , A61K31/5377 , A61P9/00 , A61P9/04 , A61P9/10 , A61P9/12 , A61P11/00 , A61P11/06 , A61P13/12 , A61P17/00 , A61P29/00 , A61P37/08 , A61P43/00 , C07D401/06 , C07D405/06 , C07D405/14 , C07D471/04 , A61K31/47 , C07D209/02 , C07D215/16 , C07D491/02 , C07D515/02
CPC分类号： C07D401/06 , A61K31/4045 , A61K31/437 , A61K31/4709 , A61K31/5377 , C07D405/06 , C07D405/14 , C07D471/04
摘要： According to this invention, there is provided an indole derivative having the general formula (I) wherein A is an oxygen atom or a nitrogen atom which nitrogen atom is optionally substituted with an alkyl group, and (i) R1 and R2 each stand for a hydrogen atom or an alkyl group, independently, or (ii) R1 and R2 as taken together form a cycloalkyl group or an aromatic ring, or (iii) R1 and R2 as taken together form a heterocyclic ring, and R3 is a hydrogen atom, a (C1-C10)alkyl group or others, R4 is a substituted alkyl group and R5 is a hydrogen atom, a halogen atom, an alkyl group or an alkoxy group and so on, as novel compounds by a novel chemical synthetic process. The indole derivative of formula (I) exhibits a useful chymase inhibitory activity.
摘要翻译：根据本发明，提供了具有通式（I）的吲哚衍生物，其中A是氧原子或氮原子，其氮原子任选地被烷基取代，和（i）R 1和R 2，每个代表氢原子或烷基，独立地或（ii）R 1和R 2一起形成环烷基或芳环，或（iii）R 1和R 2 一起形成杂环，R 3为氢原子，（C1-C10）烷基等，R 4为取代烷基，R 5为氢原子，卤素原子，烷基或烷氧基等，作为新化合物，通过新的化学合成方法。式（I）的吲哚衍生物显示出有用的胃促胰酶抑制活性。

2. 发明授权

US08188073B2 Benzoxazines and related nitrogen-containing heterobicyclic compounds useful as mineralocorticoid receptor modulating agents 有权
标题翻译：苯并恶嗪和有用的含氮杂双环化合物可用作盐皮质激素受体调节剂
公开(公告)号：US08188073B2
公开(公告)日：2012-05-29
申请号：US13167986
申请日：2011-06-24
申请人： Toru Iijima , Yasuo Yamamoto , Hidenori Akatsuka , Takayuki Kawaguchi
发明人： Toru Iijima , Yasuo Yamamoto , Hidenori Akatsuka , Takayuki Kawaguchi
IPC分类号： C07D279/16 , A61K31/5415
CPC分类号： C07D265/36 , C07D279/16 , C07D413/04
摘要： The present invention relates to a compound, useful as a mineralocorticoid receptor-modulating agent, of the following formula [I]: wherein Ring A is a benzene ring optionally having a substituent(s) other than R1 etc, R1 is a group of the formula: RaSO2NH— etc, Ra is an alkyl group etc, R2 and R3 are each a hydrogen atom, a phenyl group, an optionally substituted alkyl group etc, X is an oxygen atom etc, Y is a group of the formula: —C(═O)— etc, Ar is an optionally substituted aryl group or an optionally substituted heteroaryl group, Q is a single bond, an alkylene group etc, or a pharmaceutically acceptable salt thereof.
摘要翻译：本发明涉及可用作以下式[I]的盐皮质激素受体调节剂的化合物：其中环A为任选具有除R1等以外的取代基的苯环，R1为式：R a SO 2 NH-等，R a为烷基等，R 2和R 3各自为氢原子，苯基，任意取代的烷基等，X为氧原子等，Y为下式基团-C （= O） - 等，Ar为任选取代的芳基或任选取代的杂芳基，Q为单键，亚烷基等，或其药学上可接受的盐。

3. 发明申请

US20110251185A1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS 有权
标题翻译：苯并噻唑类和相关的含氮杂环化合物作为矿物质受体调节剂有用
公开(公告)号：US20110251185A1
公开(公告)日：2011-10-13
申请号：US13167986
申请日：2011-06-24
申请人： Toru IIJIMA , Yasuo Yamamoto , Hidenori Akatsuka , Takayuki Kawaguchi
发明人： Toru IIJIMA , Yasuo Yamamoto , Hidenori Akatsuka , Takayuki Kawaguchi
IPC分类号： A61K31/5415 , A61K31/538 , A61P5/00 , C07D279/16 , A61P9/00 , A61P9/12 , C07D413/04 , C07D265/36
CPC分类号： C07D265/36 , C07D279/16 , C07D413/04
摘要： The present invention relates to a compound, useful as a mineralocorticoid receptor-modulating agent, of the following formula [I]: wherein Ring A is a benzene ring optionally having a substituent(s) other than R1 etc, R1 is a group of the formula: RaSO2NH— etc, Ra is an alkyl group etc, R2 and R3 are each a hydrogen atom, a phenyl group, an optionally substituted alkyl group etc, X is an oxygen atom etc, Y is a group of the formula: —C(═O)— etc, Ar is an optionally substituted aryl group or an optionally substituted heteroaryl group, Q is a single bond, an alkylene group etc, or a pharmaceutically acceptable salt thereof.
摘要翻译：本发明涉及可用作以下式[I]的盐皮质激素受体调节剂的化合物：其中环A为任选具有除R1等以外的取代基的苯环，R1为式：R a SO 2 NH-等，R a为烷基等，R 2和R 3各自为氢原子，苯基，任意取代的烷基等，X为氧原子等，Y为下式基团-C （= O） - 等，Ar为任选取代的芳基或任选取代的杂芳基，Q为单键，亚烷基等，或其药学上可接受的盐。

4. 发明授权

US07965438B2 Display method and display device 有权
标题翻译：显示方式和显示设备
公开(公告)号：US07965438B2
公开(公告)日：2011-06-21
申请号：US11599409
申请日：2006-11-15
申请人： Jun Kawahara , Satoshi Tatsuura , Kei Shimotani , Yasuo Yamamoto
发明人： Jun Kawahara , Satoshi Tatsuura , Kei Shimotani , Yasuo Yamamoto
IPC分类号： G02B26/00 , G02F1/03 , G02F1/07 , G02F1/15
CPC分类号： G02F1/1506 , G02F2001/1517 , G02F2203/02
摘要： The invention provides a display method for displaying an image by deposition of metal fine particles. The display method includes at least depositing metal fine particles, from an electrolytic solution that has at least a metal ion of the metal particles and that is provided between a pair of substrates having at least one translucent substrate, onto a surface of any one of the pair of substrates by imparting one stimulus. A concentration of the metal ion of the metal fine particles in the electrolytic solution after imparting the stimulus is about 200 mmol/l or less. The invention further provides a display device which uses the display method.
摘要翻译：本发明提供了一种通过沉积金属微粒显示图像的显示方法。所述显示方法至少包含从至少具有所述金属粒子的金属离子的电解液沉积金属微粒并且设置在具有至少一个透光性基板的一对基板之间的金属微粒的表面上通过赋予一个刺激物对一对底物。赋予刺激后的电解液中的金属微粒的金属离子浓度为约200mmol / l以下。本发明还提供一种使用显示方法的显示装置。

5. 发明授权

US07688496B2 Display medium, display device and display method 有权
标题翻译：显示介质，显示设备和显示方式
公开(公告)号：US07688496B2
公开(公告)日：2010-03-30
申请号：US11438743
申请日：2006-05-22
申请人： Hiroaki Moriyama , Yasuo Yamamoto , Jun Kawahara , Masaaki Abe
发明人： Hiroaki Moriyama , Yasuo Yamamoto , Jun Kawahara , Masaaki Abe
IPC分类号： G02B26/00
CPC分类号： G02F1/167 , G09G3/344 , G09G2320/0626
摘要： The invention provides a display medium having a dimmer layer which comprises at least two kinds of charged mobile fine particles. Each of the at least two kinds of the charged mobile fine particles respectively has different coloration and a different mobility, and the charged mobile fine particles of at least one kind of the at least two kinds show coloration when in a dispersed state. The invention further provides a display device having an electric field forming unit and the dimmer layer. The invention further provides a display method which uses the display medium and includes putting the charged mobile fine particles of at least one of the kinds being dispersed while having other charged mobile fine particles not being dispersed.
摘要翻译：本发明提供了一种显示介质，其具有包含至少两种带电移动细颗粒的调光层。所述至少两种所述带电移动微粒分别具有不同的着色和不同的迁移率，并且当处于分散状态时，所述至少两种至少一种的带电移动细颗粒显示着色。本发明还提供一种具有电场形成单元和调光器层的显示装置。本发明还提供了一种显示方法，其使用显示介质，并且包括将具有分散的至少一种的带电移动细颗粒放置在不分散其它带电移动微粒的同时。

6. 发明授权

US07616373B2 Display device particles, process for producing the same, image-display medium, and image-forming device 失效
标题翻译：显示装置颗粒，其制造方法，图像显示介质和图像形成装置
公开(公告)号：US07616373B2
公开(公告)日：2009-11-10
申请号：US10863390
申请日：2004-06-09
申请人： Hidehiko Soyama , Satoshi Hiraoka , Yasuo Yamamoto
发明人： Hidehiko Soyama , Satoshi Hiraoka , Yasuo Yamamoto
IPC分类号： G02B26/00 , G09G3/34
CPC分类号： G02F1/167 , G03G5/00 , G09F9/372
摘要： The present invention provides display device particles that have positive or negative chargeability and have color and are produced using at least a calcium compound, in which a concentration of the calcium compound in the display device particle is 0.05% by weight or less in terms of a calcium element content, a process for producing the display device particles, as well as an image-display medium and an image-forming device each using the display device particles.
摘要翻译：本发明提供具有正或负带电性并具有颜色并且至少使用钙化合物制成的显示装置颗粒，其中显示装置颗粒中的钙化合物的浓度为0.05重量％以下钙元素含量，制造显示装置颗粒的方法，以及使用显示装置颗粒的图像显示介质和图像形成装置。

7. 发明申请

US20090258921A1 INDOLE DERIVATIVES 有权
标题翻译： INDOLE DORIVATIVES
公开(公告)号：US20090258921A1
公开(公告)日：2009-10-15
申请号：US12487264
申请日：2009-06-18
申请人： Sumihiro NOMURA , Yasuo Yamamoto
发明人： Sumihiro NOMURA , Yasuo Yamamoto
IPC分类号： A61K31/404 , C07D209/04 , A61P3/10
CPC分类号： C07D401/14 , C07D405/04 , C07D405/14 , C07D409/14 , C07H19/044 , C07H19/22
摘要： Novel indole derivatives of formula (I) or a pharmaceutically acceptable salt thereof: wherein R1 is halogen, or alkyl, R2 is hydrogen, or halogen, Ar is phenyl, or thienyl, which may be substituted with halogen, alkyl, alkoxy, alkylthio, etc.
摘要翻译：式（I）的新型吲哚衍生物或其药学上可接受的盐：其中R1是卤素，或烷基，R2是氢或卤素，Ar是苯基或噻吩基，其可以被卤素，烷基，烷氧基，烷硫基，等等

8. 发明申请

US20090103207A1 ROTOR HUB, SPINDLE MOTOR AND HARD DISK DRIVE 有权
标题翻译：转子集线器，主轴电机和硬盘驱动器
公开(公告)号：US20090103207A1
公开(公告)日：2009-04-23
申请号：US12256597
申请日：2008-10-23
申请人： Toshiaki Miyauchi , Yasuo Yamamoto
发明人： Toshiaki Miyauchi , Yasuo Yamamoto
IPC分类号： G11B17/02 , G11B33/00
CPC分类号： G11B19/2009 , B21J1/025 , B21J1/04 , B21K1/32 , Y10T29/49025
摘要： In a method for manufacturing a rotor hub for use in a spindle motor, free-cutting stainless steel is used as a material of the rotor hub. A slug of free-cutting stainless steel is subjected to a plastic working to form a disk mounting portion and a cylindrical surface positioned radially inwardly of the disk mounting portion. Then, a cylindrical disk fitting surface is formed by machining substantially the entirety of the cylindrical surface. The rotor hub contains A-type inclusions appearing in a cross section taken along a center axis of the disk mounting portion. The A-type inclusions are oriented in directions different than the center axis.
摘要翻译：在制造用于主轴电动机的转子轮毂的方法中，使用自由切削不锈钢作为转子轮毂的材料。一块自由切削不锈钢经过塑性加工，以形成圆盘安装部分和位于圆盘安装部分径向内侧的圆柱形表面。然后，通过对基本上整个圆柱形表面进行加工来形成圆柱形盘装配表面。转子毂包含沿着盘安装部的中心轴线截取的横截面中的A型夹杂物。 A型夹杂物的取向方向与中心轴不同。

9. 发明申请

US20080076917A1 Intermediates of 2-Substituted Carbapenem Derivatives and Process for Production Thereof 失效
标题翻译： 2-取代的碳青霉烯衍生物的中间体及其制备方法
公开(公告)号：US20080076917A1
公开(公告)日：2008-03-27
申请号：US10538466
申请日：2003-12-15
申请人： Toshiro Sasaki , Takashi Ando , Yasuo Yamamoto , Takahiro Imai , Dai Kubota , Katsuhiko Noguchi , Nobuyuki Hori , Eiki Shitara , Kunio Atsumi , Shohei Yasuda
发明人： Toshiro Sasaki , Takashi Ando , Yasuo Yamamoto , Takahiro Imai , Dai Kubota , Katsuhiko Noguchi , Nobuyuki Hori , Eiki Shitara , Kunio Atsumi , Shohei Yasuda
IPC分类号： C07D205/00 , C07D487/00
CPC分类号： C07D513/04 , C07F9/6561 , Y02P20/55
摘要： The present invention relates to compounds represented by formula (1) and a process for producing the same. The use of these compounds can realize the production of carbapenem derivatives having potent antimicrobial activity and a wide antimicrobial spectrum in a safe and cost-effective manner.
摘要翻译：本发明涉及由式（1）表示的化合物及其制备方法。这些化合物的使用可以以安全和成本有效的方式实现具有有效抗微生物活性和广谱抗菌谱的碳青霉烯衍生物的生产。

10. 发明授权

US07288144B2 Non-aqueous ink-jet ink composition 有权
标题翻译：非水性喷墨油墨组合物
公开(公告)号：US07288144B2
公开(公告)日：2007-10-30
申请号：US11101769
申请日：2005-04-08
申请人： Shunsuke Uozumi , Yasuo Yamamoto
发明人： Shunsuke Uozumi , Yasuo Yamamoto
IPC分类号： C09D11/02
CPC分类号： C09D11/36
摘要： A non-aqueous ink-jet ink composition contains at least a pigment, a solvent, and a dispersing agent. The non-aqueous ink-jet ink composition further contains a chelating agent, which is soluble in the solvent. The chelating agent may be a crown ether and/or a cryptand, which acts as a neutral carrier. Alternatively, the chelating agent may be at least one chelating agent acting as an ionic carrier, which is selected from the group consisting of GEDTA, BAPTA, and DTPA. The non-aqueous ink-jet ink composition has good storage stability and good jetting-out performance through suppression of occurrence of sediments due to a change with the passage of time.
摘要翻译：非水性喷墨油墨组合物至少含有颜料，溶剂和分散剂。非水性喷墨油墨组合物还含有可溶于溶剂的螯合剂。螯合剂可以是作为中性载体的冠醚和/或穴状物。或者，螯合剂可以是作为离子载体的至少一种螯合剂，其选自GEDTA，BAPTA和DTPA。非水性喷墨油墨组合物通过抑制随时间的变化而产生的沉积物，具有良好的储存稳定性和良好的喷出性能。

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