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1. 发明申请

WO2008083200A3 SPIROHETEROCYCLIC GLYCOSIDES AND METHODS OF USE 审中-公开
标题翻译：螺环多环糖苷及其使用方法
公开(公告)号：WO2008083200A3
公开(公告)日：2008-10-30
申请号：PCT/US2007088905
申请日：2007-12-27
申请人： THERACOS INC , HADD MICHAEL J , CHEN YUANWEI , FENG YAN , SEN SENGEN , SEED BRIAN
发明人： HADD MICHAEL J , CHEN YUANWEI , FENG YAN , SEN SENGEN , SEED BRIAN
IPC分类号： A01N43/16 , A61K31/35 , A61K31/58
CPC分类号： C07H17/04
摘要： Provided are compounds having an inhibitory effect on sodium-dependent glucose cotransporter SGLT. The invention also provides pharmaceutical compositions, methods of preparing the compounds, synthetic intermediates, and methods of using the compounds, independently or in combination with other therapeutic agents, for treating diseases and conditions which are affected by SGLT inhibition.
摘要翻译：提供了对钠依赖性葡萄糖协同转运蛋白SGLT具有抑制作用的化合物。本发明还提供了药物组合物，制备该化合物的方法，合成中间体以及独立地或与其他治疗剂组合使用该化合物用于治疗受SGLT抑制影响的疾病和病症的方法。

2. 发明申请

WO2007140191A2 GLUCOSE TRANSPORT INHIBITORS AND METHODS OF USE 审中-公开
标题翻译：葡萄糖运输抑制剂及其使用方法
公开(公告)号：WO2007140191A2
公开(公告)日：2007-12-06
申请号：PCT/US2007069487
申请日：2007-05-22
申请人： THERACOS INC , CHEN YUANWEI , FENG YAN , XU BAIHUA , LV BINHUA , DONG JIAJIA , SEED BRIAN , HADD MICHAEL J
发明人： CHEN YUANWEI , FENG YAN , XU BAIHUA , LV BINHUA , DONG JIAJIA , SEED BRIAN , HADD MICHAEL J
IPC分类号： A61K31/70 , A61K31/382 , A61K31/452 , A61K31/453 , A61K31/496 , A61K31/5377
CPC分类号： C07D311/96 , C07D407/12 , C07H7/04 , C07H19/00
摘要： Provided are compounds having an inhibitory effect on sodium-dependent glucose cotransporter SGLT. The invention also provides pharmaceutical compositions, methods of preparing the compounds, synthetic intermediates, and methods of using the compounds, independently or in combination with other therapeutic agents, for treating diseases and conditions which are affected by SGLT inhibition.
摘要翻译：提供对钠依赖性葡萄糖转运蛋白SGLT具有抑制作用的化合物。本发明还提供药物组合物，制备化合物的方法，合成中间体，以及独立地或与其它治疗剂组合使用化合物治疗受SGLT抑制影响的疾病和病症的方法。

3. 发明公开

EP2019679A4 GLUCOSE TRANSPORT INHIBITORS AND METHODS OF USE 有权
标题翻译： GLOBOSETRANSPORTHEMMER UND ANWENDUNGSVERFAHREN
公开(公告)号：EP2019679A4
公开(公告)日：2014-04-23
申请号：EP07784049
申请日：2007-05-22
申请人： THERACOS INC
发明人： CHEN YUANWEI , FENG YAN , XU BAIHUA , LV BINHUA , DONG JIAJIA , SEED BRIAN , HADD MICHAEL J
IPC分类号： C07H7/04 , A61K31/70 , A61P3/04 , A61P3/10 , C07D407/12 , C07H19/01
CPC分类号： C07D311/96 , C07D407/12 , C07H7/04 , C07H19/00
摘要： Provided are compounds having an inhibitory effect on sodium-dependent glucose cotransporter SGLT. The invention also provides pharmaceutical compositions, methods of preparing the compounds, synthetic intermediates, and methods of using the compounds, independently or in combination with other therapeutic agents, for treating diseases and conditions which are affected by SGLT inhibition.
摘要翻译：提供对钠依赖性葡萄糖转运蛋白SGLT具有抑制作用的化合物。本发明还提供药物组合物，制备化合物的方法，合成中间体以及独立地或与其它治疗剂组合使用化合物用于治疗受SGLT抑制影响的疾病和病症的方法。

4. 发明公开

EP2187742A4 BENZYLBENZENE DERIVATIVES AND METHODS OF USE 有权转让
标题翻译：苄基苯并呋喃衍生物及其使用方法
公开(公告)号：EP2187742A4
公开(公告)日：2012-10-03
申请号：EP08798514
申请日：2008-08-22
申请人： THERACOS INC
发明人： SONG YANLI , CHEN YUANWEI , CHENG HUAWEI , LI SHENGBIN , WU YUELIN , FENG YAN , LV BINHUA , XU BAIHUA , SEED BRIAN , HADD MICHAEL J , DU JIYAN , WANG CONGNA , ROBERGE JACQUES Y
IPC分类号： C07D407/12 , A61K31/351 , A61P3/10 , C07D309/10
CPC分类号： C07H7/04 , C07D309/10 , C07D407/12

5. 发明公开

EP2064222A4 BENZYLIC GLYCOSIDE DERIVATIVES AND METHODS OF USE 有权
标题翻译： VERFAHREN ZU IHRER VERWENDUNG BENZYLISCHE GLYCOSIDDERIVATE
公开(公告)号：EP2064222A4
公开(公告)日：2011-12-14
申请号：EP08744883
申请日：2008-04-01
申请人： THERACOS INC
发明人： CHEN YUANWEI , FENG YAN , XU BAIHUA , LV BINHUA , SEED BRIAN , HADD MICHAEL J , CHENG HUAWEI , SHENG ZELIN , XU MIN , WANG CONGNA , DU JIYAN , ZHANG LILI , XU GE , WU YUELIN
IPC分类号： C07G3/00
CPC分类号： C07H7/04 , A61K38/00 , C07D309/10

6. 发明专利

BRPI0815708A2 未知
公开(公告)号：BRPI0815708A2
公开(公告)日：2014-09-30
申请号：BRPI0815708
申请日：2008-08-22
申请人： THERACOS INC
发明人： CHEN YUANWEI , CHENG HUAWEI , LI SHENGBIN , WU YUELIN , FENG YAN , LV BINHUA , SEED BRIAN , HADD MICHAEL J , DU JIYAN , WANG CONGNA , ROBERGE JACQUES Y , SONG YANLI
IPC分类号： A01N43/04 , A61K31/70
摘要： Provided are compounds having an inhibitory effect on sodium-dependent glucose cotransporter SGLT. The invention also provides pharmaceutical compositions, methods of preparing the compounds, synthetic intermediates, and methods of using the compounds, independently or in combination with other therapeutic agents, for treating diseases and conditions which are affected by SGLT inhibition, such as diabetes mellitus. The compounds have formula IA below.

7. 发明专利

ES2466672T3 Derivados de glicósido bencílico y métodos de uso 未知
公开(公告)号：ES2466672T3
公开(公告)日：2014-06-10
申请号：ES08744883
申请日：2008-04-01
申请人： THERACOS INC
发明人： CHEN YUANWEI , FENG YAN , XU BAIHUA , LV BINHUA , SEED BRIAN , HADD MICHAEL J , CHENG HUAWEI , SHENG ZELIN , XU MIN , WANG CONGNA , DU JIYAN , ZHANG LILI , XU GE , WU YUELIN
IPC分类号： C07D309/10
摘要： Un compuesto que tiene la fórmula: donde V es oxígeno o un enlace sencillo; W es alquileno C1-C6 ; X es oxígeno o azufre; Y es un miembro seleccionado entre el grupo que consiste en haloalquilo C1-C6, hidroxialquilo C1-C6, alquenilo C2-C6, alquinilo C2-C6, cicloalquilo C3-C10, cicloalquenilo C5-C10, (alquiloxi C1-C4)alquilo C1-C3, (alqueniloxi C2-C4)alquilo C1-C3 y (cicloalquiloxi C3- C10)alquilo C1-C3; donde los grupos o porciones alquilo, alquenilo, alquinilo, cicloalquilo y cicloalquenilo de Y opcionalmente están parcial o completamente fluorados y opcionalmente están mono- o disustituidos con sustituyentes idénticos o diferentes seleccionados entre cloro, hidroxi, alquilo C1-C3 y alcoxi C1-C3, y en los grupos o porciones cicloalquilo y cicloalquenilo de Y, opcionalmente uno o dos grupos metileno están reemplazados independientemente el uno del otro con O, S, CO, SO, SO2 o NRb, y opcionalmente uno o dos grupos metino están reemplazados con N, donde el heterociclo formado mediante dicho reemplazo opcional es distinto de heteroarilo; R1 se selecciona entre el grupo que consiste en hidrógeno, halo, alquilo C1-C6 y cicloalquilo C3-C10; R3 se selecciona entre el grupo que consiste en hidrógeno, halo, hidroxi, alquilo C1-C6, alquiloxi C1-C6, alquenilo C2-C6, alquinilo C2-C6, cicloalquilo C3-C10 y cicloalquiloxi C3-C10, donde los grupos o porciones alquilo y cicloalquilo de R3 opcionalmente están parcial o completamente fluorados, y en los grupos cicloalquilo de R3 un grupo metileno está opcionalmente reemplazado con O, S, CO, SO o SO2; y cada Rb es un miembro seleccionado independientemente entre el grupo que consiste en H, alquilo C1-C4 y (alquil C1-C4)carbonilo, donde los grupos o porciones alquilo de Rb opcionalmente están parcial o completamente fluorados; o una sal farmacéuticamente aceptable del mismo.

8. 发明专利

CA2697349C BENZYLBENZENE DERIVATIVES AND METHODS OF USE 未知
公开(公告)号：CA2697349C
公开(公告)日：2012-04-24
申请号：CA2697349
申请日：2008-08-22
申请人： THERACOS INC
发明人： SONG YANLI , CHEN YUANWEI , CHENG HUAWEI , LI SHENGBIN , WU YUELIN , FENG YAN , LV BINHUA , XU BAIHUA , SEED BRIAN , HADD MICHAEL J , DU JIYAN , WANG CONGNA , ROBERGE JACQUES Y
IPC分类号： C07D309/10 , A61K31/351 , A61P3/10 , C07D405/12 , C07D407/12
摘要： Provided are compounds having an inhibitory effect on sodium-dependent glucose cotransporter SGLT. The invention also provides pharmaceutical compositions, methods of preparing the compounds, synthetic intermediates, and methods of using the compounds, independently or in combination with other therapeutic agents, for treating diseases and conditions which are affected by SGLT inhibition.

9. 发明专利

DK2064222T3 Benzyliske glycosid-derivater og fremgangsmåder til anvendelse deraf 未知
公开(公告)号：DK2064222T3
公开(公告)日：2014-07-21
申请号：DK08744883
申请日：2008-04-01
申请人： THERACOS INC
发明人： CHEN YUANWEI , XU BAIHUA , LV BINHUA , CHENG HUAWEI , SHENG ZELIN , XU MIN , WANG CONGNA , DU JIYAN , ZHANG LILI , XU GE , WU YUELIN , FENG YAN , SEED BRIAN , HADD MICHAEL J
IPC分类号： C07D309/10

10. 发明专利

AU2008232419B2 Benzylic glycoside derivatives and methods of use 未知
公开(公告)号：AU2008232419B2
公开(公告)日：2013-06-20
申请号：AU2008232419
申请日：2008-04-01
申请人： THERACOS INC
发明人： WU YUELIN , LV BINHUA , FENG YAN , WANG CONGNA , CHENG HUAWEI , DU JIYAN , XU MIN , CHEN YUANWEI , HADD MICHAEL J , ZHANG LILI , SHENG ZELIN , XU BAIHUA , SEED BRIAN , XU GE
IPC分类号： C07G3/00
摘要： Provided are compounds having an inhibitory effect on sodium-dependent glucose cotransporter SGLT. The invention also provides pharmaceutical compositions, methods of preparing the compounds, synthetic intermediates, and methods of using the compounds, independently or in combination with other therapeutic agents, for treating diseases and conditions which are affected by SGLT inhibition.

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