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1. 发明申请

WO2019115404A1 PESTICIDALLY ACTIVE MESOIONIC HETEROCYCLIC COMPOUNDS 审中-公开
公开(公告)号：WO2019115404A1
公开(公告)日：2019-06-20
申请号：PCT/EP2018/084032
申请日：2018-12-07
申请人： SYNGENTA PARTICIPATIONS AG
发明人： JUNG, Pierre, Joseph, Marcel , DUMEUNIER, Raphael , GAGNEPAIN, Julien, Daniel, Henri , STOLLER, André , RENDINE, Stefano
IPC分类号： C07D231/14 , C07D487/04 , C07C15/04 , A01N43/90
CPC分类号： C07D487/04 , C07D231/14
摘要： A compound of formula I, (I), wherein the substituents are as defined in claim (1), and the agrochemically acceptable salts, stereoisomers, enantiomers, tautomers and N-oxides of those compounds, can be used as insecticides.

2. 发明申请

WO2009090038A1 FUNGICIDAL COMPOSITIONS 审中-公开
标题翻译：杀真菌剂
公开(公告)号：WO2009090038A1
公开(公告)日：2009-07-23
申请号：PCT/EP2009/000165
申请日：2009-01-14
申请人： SYNGENTA PARTICIPATIONS AG , GODWIN, Jeremy, R. , TRAH, Stephan , LAMBERTH, Clemens , DUMEUNIER, Raphael , WENDEBORN, Sebastian, Volker , GRASSO, Valeria
发明人： GODWIN, Jeremy, R. , TRAH, Stephan , LAMBERTH, Clemens , DUMEUNIER, Raphael , WENDEBORN, Sebastian, Volker , GRASSO, Valeria
IPC分类号： A01N43/58 , A01P3/00
CPC分类号： A01N43/58 , A01N37/34 , A01N43/54 , A01N43/653 , A01N47/14 , A01N51/00 , A01N2300/00
摘要： A fungicidal composition suitable for control of diseases caused by phytopathogens comprising (A) a compound of formula (I), wherein R 1 is methyl, ethyl or isopropyl; R 2 is 2-chloro-6-fluoro-phenyl, 2,4,6-trifluorophenyl or 2,6-difluoro-4-methoxy-phenyl; R 3 is chloro, fluoro or methoxy; and (B) a compound selected, for example, from the group consisting of (B1) a strobilurin fungicide, (B2) an azole fungicide, (B3) a morpholine fungicide, and (B4) an anilinopyrimidine fungicide.
摘要翻译：一种适于控制由植物病原体引起的疾病的杀真菌组合物，其包含（A）式（I）化合物，其中R 1为甲基，乙基或异丙基; R2是2-氯-6-氟 - 苯基，2,4,6-三氟苯基或2,6-二氟-4-甲氧基 - 苯基; R3是氯，氟或甲氧基; 和（B）选自例如（B1）嗜球果伞素杀真菌剂，（B2）唑类杀真菌剂，（B3）吗啉杀真菌剂和（B4）苯胺基嘧啶杀真菌剂的组合的化合物。

3. 发明申请

WO2011131543A1 PROCESS FOR THE PREPARATION OF PYRAZOLE CARBOXYLIC ACID AMIDES 审中-公开
标题翻译：制备吡唑羧酸酰胺的方法
公开(公告)号：WO2011131543A1
公开(公告)日：2011-10-27
申请号：PCT/EP2011/055869
申请日：2011-04-14
申请人： SYNGENTA PARTICIPATIONS AG , DUMEUNIER, Raphael , TOBLER, Hans
发明人： DUMEUNIER, Raphael , TOBLER, Hans
IPC分类号： C07D231/14 , C07D303/08 , C07D303/36 , C07C211/61
CPC分类号： C07D231/14 , C07D303/08 , C07D303/36
摘要： The invention relates to a process for the preparation of formula (I), which process comprises a) reacting the compound (II), with cyclopentadiene to (III); b) reacting this compound in the presence of an oxidant to the compound of formula (IV); c) hydrogenating this compound in the presence of a metal catalyst and an inert solvent under hydrogen atmosphere to the compound of formula (V); d) reacting this compound in the presence of a Brönsted acid followed by a reducing agent to the compound of formula (VI); e) reacting VI with a compound (VII), in the presence of a base to a compound of formula (VIII); f) converting the compound of formula VIII in the presence of an oxidising agent to the compound of formula (IX); and g) reacting the compound of formula IX in the presence of triphenylphosphane/carbon tetrachloride or riphenylphosphane/bromotrichloromethane to the compound of formula I.
摘要翻译：本发明涉及制备式（I）的方法，该方法包括：a）使化合物（II）与环戊二烯反应至（III）; b）在氧化剂存在下使该化合物与式（Ⅳ）化合物反应; c）在金属催化剂和惰性溶剂的存在下，在氢气氛下将该化合物氢化成式（V）化合物; d）在布朗斯台德酸的存在下将该化合物与式（VI）化合物的还原剂反应; e）使VI与化合物（VII）在碱的存在下与式（VIII）的化合物反应; f）将式VIII化合物在氧化剂存在下转化为式（Ⅸ）化合物; 和g）在三苯基膦/四氯化碳或联苯基膦/溴三氯甲烷存在下将式IX化合物与式I化合物反应。

4. 发明申请

WO2014210555A1 COMPOUNDS THAT INDUCE ABA RESPONSES 审中-公开
标题翻译：引起ABA反应的化合物
公开(公告)号：WO2014210555A1
公开(公告)日：2014-12-31
申请号：PCT/US2014/044727
申请日：2014-06-27
申请人： THE REGENTS OF THE UNIVERSITY OF CALIFORNIA , SYNGENTA PARTICIPATIONS AG , WENDEBORN, Sebastian, Volker , JUNG, Pierre, Joseph , LACHIA, Mathilde, Denise , DUMEUNIER, Raphael
发明人： WENDEBORN, Sebastian, Volker , JUNG, Pierre, Joseph , LACHIA, Mathilde, Denise , DUMEUNIER, Raphael , CUTLER, Sean, R.
IPC分类号： C07D215/22 , A01N43/42 , A01P15/00
CPC分类号： C07D215/227 , A01N43/42 , C07D215/22
摘要： The present invention provides agonist compounds that active ABA receptors, and agricultural formulations comprising the agonist compounds. The agricultural formulations are useful for inducing ABA responses in plant vegetative tissues, reducing abiotic stress in plants, and inhibiting germination of plant seeds. The compounds are also useful for inducing expression of ABA-responsive genes in cells that express endogenous or heterologous ABA receptors.
摘要翻译：本发明提供了活性ABA受体的激动剂化合物和包含激动剂化合物的农业制剂。农业制剂可用于在植物营养组织中诱导ABA应答，减少植物中的非生物胁迫并抑制植物种子的萌发。该化合物也可用于在表达内源性或异源性ABA受体的细胞中诱导ABA反应基因的表达。

5. 发明申请

WO2014206855A1 PROCESS FOR THE STEREOSELECTIVE PREPARATION OF A PYRAZOLE-CARBOXAMIDE 审中-公开
标题翻译：吡唑酰胺的立体选择性制备方法
公开(公告)号：WO2014206855A1
公开(公告)日：2014-12-31
申请号：PCT/EP2014/062936
申请日：2014-06-19
申请人： SYNGENTA PARTICIPATIONS AG
发明人： DUMEUNIER, Raphael , KESSABI, Jilali , WENDEBORN, Sebastian Volker , NUSSBAUMER, Hannes
IPC分类号： C07D231/14 , C07C239/00
CPC分类号： C07D231/14 , C07C239/20
摘要： The present invention relates to a process for the enantioselective preparation of the compound of formula (lb), which process comprises a) reducing the (E)- or (Z)-form of a compound of formula (II), with an enantioselective reagent to a compound of formula (IlIa), and b) acylating the compound of formula (IlIa) with the compound of formula (IV), or c) coupling the compound of formula (IV) with the compound of formula (II), to give a compound of formula (V)and d) reducing compound of formula (V) in the presence of hydrogen, a catalyst and a chiral ligand, to the compound of formula (lb).
摘要翻译：本发明涉及式（Ib）化合物的对映选择性制备方法，该方法包括a）用对映选择性试剂还原式（II）化合物的（E） - 或（Z）与式（Ⅺa）化合物反应，和b）用式（Ⅳ）化合物酰化式（Ⅺa）化合物，或c）将式（Ⅳ）化合物与式（Ⅳ）化合物偶联至在式（Ⅴ）化合物和式（Ⅴ）化合物的存在下，在氢气，催化剂和手性配体的存在下，得到式（Ⅴ）化合物和d）还原式（Ⅴ）化合物。

6. 发明申请

WO2012084678A1 NOVEL IMIDAZOLES USEFUL AS PLANT FUNGICIDES 审中-公开
标题翻译：新颖的咪达唑作为植物杀真菌剂有用
公开(公告)号：WO2012084678A1
公开(公告)日：2012-06-28
申请号：PCT/EP2011/072880
申请日：2011-12-15
申请人： SYNGENTA PARTICIPATIONS AG , CEDERBAUM, Fredrik , UMARYE, Jayant , DUMEUNIER, Raphael , SONAWANE, Ravindra
发明人： CEDERBAUM, Fredrik , UMARYE, Jayant , DUMEUNIER, Raphael , SONAWANE, Ravindra
IPC分类号： A01N43/50 , C07D401/04 , C07D401/14
CPC分类号： C07D401/04 , A01N43/50 , A01N53/00 , C07D401/14
摘要： Compounds of the general formula (I) wherein the substituents are as defined in claim 1, are useful as fungicides.
摘要翻译：其中取代基如权利要求1中所定义的通式（I）的化合物可用作杀真菌剂。

7. 发明申请

WO2009127615A1 NOVEL IMIDAZOLE DERIVATIVES HAVING MICROBIOCIDAL ACTIVITY 审中-公开
标题翻译：具有微生物活性的新咪唑烷衍生物
公开(公告)号：WO2009127615A1
公开(公告)日：2009-10-22
申请号：PCT/EP2009/054389
申请日：2009-04-14
申请人： SYNGENTA PARTICIPATIONS AG , DUMEUNIER, Raphael , LAMBERTH, Clemens , TRAH, Stephan
发明人： DUMEUNIER, Raphael , LAMBERTH, Clemens , TRAH, Stephan
IPC分类号： C07D233/60 , C07D233/68 , C07D403/12 , A01N43/50 , A61K31/4489 , A61P35/00
CPC分类号： C07D233/68 , C07D233/60 , C07D403/12
摘要： The present invention relates to novel imidazole derivatives of formula I as active ingredients which have microbiocidal activity, in particular fungicidal activity wherein (I) wherein R 1 is halogen, C 1 -C 4 alkyl or C 1 -C 4 haloalkyl, R 2 is an optionally substituted aryl, R 3 is halogen or OR 7 , R 4 and R 5 are, independently of each other, hydrogen, halogen or OR 7 , R 6 is halogen or C 1 -C 4 alkyl, and R 7 is hydrogen, C 1 -C 6 alkyl, C 3 -C 7 cycloalkyl, C 3 -C 10 cycloalkylalkyl, C 1 -C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C3-C7 cycloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 2 -C 6 alkyloxyalkyl, C 3 -C 8 dialkylaminoalkyl, C 4 -C 10 cycloalkylaminoalkyl or C4-C10 heterocyclylalkyl, or an agrochemically usable salt form thereof, provided that when R 3 is halogen, at least one of R 4 or R 5 is OR 7 , or when R 3 is OR7, at least one of R 4 or R 5 is OR 7 or halogen
摘要翻译：本发明涉及式I的新型咪唑衍生物，其具有杀微生物活性，特别是杀真菌活性的活性成分，其中（I）其中R1是卤素，C1-C4烷基或C1-C4卤代烷基，R2是任选取代的芳基，R3是卤素或OR7，R4和R5彼此独立地为氢，卤素或OR7，R6为卤素或C1-C4烷基，R7为氢，C1-C6烷基，C3-C7环烷基，C3-C10环烷基烷基，C1- C 6卤代烷基，C 2 -C 6烯基，C 2 -C 6卤代烯基，C 3 -C 7环烯基，C 2 -C 6炔基，C 2 -C 6卤代炔基，C 2 -C 6烷氧基烷基，C 3 -C 8二烷基氨基烷基，C 4 -C 10环烷基氨基烷基或C 4 -C 10杂环基烷基，条件是当R 3为卤素时，R 4或R 5中的至少一个为OR 7，或者当R 3为OR 7时，R 4或R 5中的至少一个为OR 7或卤素

8. 发明申请

WO2009127612A1 NOVEL PYRAZOLE DERIVATIVES 审中-公开
标题翻译：新型吡咯衍生物
公开(公告)号：WO2009127612A1
公开(公告)日：2009-10-22
申请号：PCT/EP2009/054386
申请日：2009-04-14
申请人： SYNGENTA PARTICIPATIONS AG , DUMEUNIER, Raphael , LAMBERTH, Clemens , TRAH, Stephan
发明人： DUMEUNIER, Raphael , LAMBERTH, Clemens , TRAH, Stephan
IPC分类号： C07D231/16 , A61K31/33 , A61P35/00 , A01N43/00
CPC分类号： C07D231/16 , A01N43/56
摘要： The present invention relates tonovel pyrazolederivatives of Formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R 1 is C 1 -C 4 alkyl or C 1 -C haloalkyl; R 2 is an optionally substituted aryl or heteroaryl; R 3 is halogen; R 4 is hydrogen, halogen, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, cyano or OR 6 ; R 5 is hydrogen, halogen, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, cyano or OR 6 ; R 6 is hydrogen, C 1 -C 6 alkyl, C 3 -C 7 cycloalkyl, C 3 -C 10 alkylcycloalkyl, C 1 -C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C haloalkenyl, C 3 -C 7 cycloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 2 -C 6 alkyloxyalkyl; R 7 is halogen or OR 6 ; X is N or C-R 4 ; or an agrochemically usablesalt form thereof.
摘要翻译：本发明涉及具有杀微生物活性，特别是杀真菌活性的作为活性成分的式（I）的次级吡唑衍生物，其中R1是C1-C4烷基或C1-C卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢，卤素，C1-C4烷基，C1-C4卤代烷基，氰基或OR6; R5是氢，卤素，C1-C4烷基，C1-C4卤代烷基，氰基或OR6; R6是氢，C1-C6烷基，C3-C7环烷基，C3-C10烷基环烷基，C1-C6卤代烷基，C2-C6烯基，C2-C卤代烯基，C3-C7环烯基，C2-C6炔基，C2-C6卤代炔基，C2 -C 6烷氧基烷基; R7为卤素或OR6; X为N或C-R4; 或其农业化学用途形式。

9. 发明申请

WO2010046215A2 DIAZA-INDOLE DERIVATIVES AND THEIR USE AS FUNGICIDES 审中-公开
标题翻译： DIAZA-INDOLE DORIVATIVES及其作为FUNGICIDES的用途
公开(公告)号：WO2010046215A2
公开(公告)日：2010-04-29
申请号：PCT/EP2009/062673
申请日：2009-09-30
申请人： SYNGENTA PARTICIPATIONS AG , SELLES, Patrice , SRINIVAS, Nityakalyani , DUMEUNIER, Raphael , CEDERBAUM, Frederik , UMARYE, Jayant
发明人： SELLES, Patrice , SRINIVAS, Nityakalyani , DUMEUNIER, Raphael , CEDERBAUM, Frederik , UMARYE, Jayant
CPC分类号： A01N43/90 , C07D471/04 , C07D487/04
摘要： The present invention relates to novel compounds of the formula (I) in which any one of G 1 , G 2 and G 3 is N and the other two of G 1 , G 2 and G 3 are CR 8 , CR 1 or CR 2 , such that when G 1 is not N, G 1 is CR 8 ; when G 2 is not N, G 2 is CR 1 ; when G 3 is not N, G 3 is CR 2 ; and X 1 , X 2 , R 1 , R 2 , R 3 , R 4 , R 6 , R 7 , and R 8 are as defined in the claims. In particular, the invention relates to use of these compounds in methods for the control and/or prevention of fungal infection in plants. The invention also relates to compositions containing these compounds as well as methods for preparing these compounds.
摘要翻译：本发明涉及式（I）的新化合物，其中，G1，G2和G3中的任一个为N，而G1，G2和G3中的任一个为CR8，CR1或CR2，使得当G1不为N时， G1是CR8; 当G2不是N时，G2是CR1; 当G3不为N时，G3为CR2; 并且X 1，X 2，R 1，R 2，R 3，R 4，R 6，R 7和R 8如权利要求中所定义。特别地，本发明涉及这些化合物在控制和/或预防植物真菌感染的方法中的用途。本发明还涉及含有这些化合物的组合物以及制备这些化合物的方法。

10. 发明申请

WO2009090039A1 PYRIDAZINE FUNGICIDES 审中-公开
标题翻译：吡咯烷类杀真菌剂
公开(公告)号：WO2009090039A1
公开(公告)日：2009-07-23
申请号：PCT/EP2009/000166
申请日：2009-01-14
申请人： SYNGENTA PARTICIPATIONS AG , TRAH, Stephan , LAMBERTH, Clemens , DUMEUNIER, Raphael , WENDEBORN, Sebastian, Volker
发明人： TRAH, Stephan , LAMBERTH, Clemens , DUMEUNIER, Raphael , WENDEBORN, Sebastian, Volker
IPC分类号： C07D401/04 , A01N43/58 , A61P35/00
CPC分类号： C07D401/04
摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R 1 is methyl, ethyl or isopropyl; R 2 is chloro, fluoro, hydroxy or C 1 -C 2 alkoxy; R 3 is H, chloro, fluoro, methoxy or C 1 -C 3 alkyl; R 4 is chloro, fluoro or bromo; and R 5 is H, fluoro or methoxy; or an agrochemically usable salt form thereof; with the proviso that when R 1 is methyl, R 2 is chloro and R 3 is H, then R 4 or R 5 is different from fluoro.
摘要翻译：本发明涉及式（I）的新的哒嗪衍生物作为具有杀微生物活性的活性成分，特别是杀真菌活性：其中R1是甲基，乙基或异丙基; R2是氯，氟，羟基或C1-C2烷氧基; R3是H，氯，氟，甲氧基或C1-C3烷基; R4是氯，氟或溴; R5为H，氟或甲氧基; 或其农业化学可用的盐形式; 条件是当R 1为甲基时，R 2为氯且R 3为H，则R 4或R 5不同于氟。

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