专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明授权

US4328216A Novel organosilicon compounds and anti-tumor agents containing the same 失效
标题翻译：新型有机硅化合物和含有相同的抗肿瘤剂
公开(公告)号：US4328216A
公开(公告)日：1982-05-04
申请号：US102225
申请日：1979-12-10
申请人： Shigeshi Toyoshima , Ryuichi Sato , Koichi Ito , Toshio Shinohara , Yasushi Yamamoto , Shoji Ichinohe
发明人： Shigeshi Toyoshima , Ryuichi Sato , Koichi Ito , Toshio Shinohara , Yasushi Yamamoto , Shoji Ichinohe
IPC分类号： A61K31/695 , A61P35/00 , C07F7/08 , C07F7/10
CPC分类号： C07F7/0818
摘要： The invention provides a novel anti-tumor agent highly effective for inhibiting growth of several tumor or cancer cells with low toxicity. The active ingredient contained in the anti-tumor agent is an .omega.-triorganosilyl-substituted linear alkanoic acid anilide which is a hitherto unknown novel compound prepared by the reaction of corresponding acid chloride and aniline.
摘要翻译：本发明提供了用于抑制几种具有低毒性的肿瘤或癌细胞生长的新型抗肿瘤剂。包含在抗肿瘤剂中的活性成分是ω-三有机甲硅烷基取代的直链烷酸酰苯胺，它是迄今未知的通过相应的酰氯和苯胺反应制备的新化合物。

2. 发明授权

US4278666A Novel organosilicon compounds and anti-transplanted tumor agents containing the same 失效
标题翻译：新型有机硅化合物和含有其的抗移植肿瘤剂
公开(公告)号：US4278666A
公开(公告)日：1981-07-14
申请号：US124957
申请日：1980-02-26
申请人： Shigeshi Toyoshima , Ryuichi Sato , Koichi Ito , Toshio Shinohara , Yasushi Yamamoto
发明人： Shigeshi Toyoshima , Ryuichi Sato , Koichi Ito , Toshio Shinohara , Yasushi Yamamoto
IPC分类号： A61K31/695 , A61P35/00 , C07F7/08 , C07F7/10 , A61K31/725 , A01N55/00
CPC分类号： C07F7/0818
摘要： The invention provides a novel class of organosilicon compounds and a method for the preparation thereof as well as an anti-tumor agent containing the compound having very remarkable anti-tumor activity but with very low toxicity. The inventive compound is a (trihydrocarbylsilylmethyloxyimino)alkane, which is a silicon-containing oxime compound hitherto not described in any prior art literatures, represented by the general formula R.sup.1.sub.3 Si--CH.sub.2 --O--N.dbd.Y, R.sup.1 is a substituted or unsubstituted monovalent hydrocarbon group having from 1 to 10 carbon atoms and Y is a divalent hydrocarbon group denoted by .dbd.CR.sup.2 R.sup.3 or .dbd.CR.sup.4, R.sup.2 and R.sup.3, which may be identical or different, having the same meaning as R.sup.1 defined above and R.sup.4 being an alkylene group to form a ring structure jointly with the carbon atom directly bonded to the nitrogen atom. Typical examples of the compounds are: 2-(trimethylsilylmethyloxyimino) butane, 2-(trimethylsilylmethyloxyimino)propane, 2-(dimethylphenylsilylmethyloxyimino) butane and trimethylsilylmethyloxyiminocyclohexane.
摘要翻译：本发明提供了一类新颖的有机硅化合物及其制备方法以及含有非常显着的抗肿瘤活性但毒性非常低的化合物的抗肿瘤剂。本发明化合物是一种（三烃基甲硅烷基甲氧基亚氨基）烷烃，其是迄今尚未在任何现有技术文献中描述的含硅肟化合物，由通式R 13 Si-CH 2 -ON A = Y表示，R 1是取代或未取代的单价烃基， 1至10个碳原子，Y是由= CR 2 R 3或= CR 4，R 2和R 3表示的二价烃基，其可以相同或不同，具有与上述R 1相同的含义，R 4为形成环的亚烷基与与氮原子直接键合的碳原子结合。化合物的典型实例是：2-（三甲基甲硅烷基甲氧基亚氨基）丁烷，2-（三甲基甲硅烷基甲氧基亚氨基）丙烷，2-（二甲基苯基甲硅烷基甲氧基亚氨基）丁烷和三甲基甲硅烷基甲氧基亚氨基环己烷。

3. 发明授权

US4349682A 2-(3-Trimethylsilylpropyl)benzothiazole 失效
标题翻译： 2-（3-三甲基甲硅烷基丙基）苯并噻唑
公开(公告)号：US4349682A
公开(公告)日：1982-09-14
申请号：US186211
申请日：1980-09-11
申请人： Shigeshi Toyoshima , Ryuichi Sato , Koichi Ito , Toshio Shinohara , Yasushi Yamamoto
发明人： Shigeshi Toyoshima , Ryuichi Sato , Koichi Ito , Toshio Shinohara , Yasushi Yamamoto
IPC分类号： A61K31/695 , A61P35/00 , C07F7/08 , C07F7/10 , A61K31/425
CPC分类号： C07F7/0812
摘要： The invention provides a novel compound 2-(3-trimethylsilylpropyl)benzothiazole having remarkable anti-tumor effects or, in particular, inhibiting growth of melanoma cells in test animals. The compound is synthesized by the ring-closing intramolecular dehydration condensation of 2-mercapto-(.gamma.-trimethylsilyl)butyroanilide which in turn is obtained by the dehydrochlorination condensation of 2-aminothiophenol and .gamma.-trimethylsilylbutyryl chloride in a polar solvent in the presence of an acid acceptor.
摘要翻译：本发明提供了具有显着的抗肿瘤作用或特别是抑制试验动物中黑素瘤细胞生长的新型化合物2-（3-三甲基甲硅烷基丙基）苯并噻唑。通过2-巯基 - （γ-三甲基甲硅烷基）丁酰苯胺的闭环分子内脱水缩合合成化合物，其通过2-苯基硫酚和γ-三甲基甲硅烷基丁酰氯在极性溶剂中的脱氯化氢缩合获得，酸受体。

4. 发明授权

US4336251A Medicaments containing an organosilicon compound 失效
标题翻译：含有机硅化合物的药物
公开(公告)号：US4336251A
公开(公告)日：1982-06-22
申请号：US178359
申请日：1980-08-15
申请人： Shigeshi Toyoshima , Ryuichi Sato , Koichi Ito , Toshio Shinohara , Yasushi Yamamoto , Shoji Ichinohe
发明人： Shigeshi Toyoshima , Ryuichi Sato , Koichi Ito , Toshio Shinohara , Yasushi Yamamoto , Shoji Ichinohe
IPC分类号： A61K31/695 , A61P9/12 , A61P35/00 , C07F7/08
CPC分类号： A61K31/695 , C07F7/0818
摘要： A novel medicament which is effective as an antihypertensive agent is proposed which contains, as its effective ingredient, an organosilicon compound represented by the general formulaR.sub.3 Si(CH.sub.2).sub.n COOH,where R denotes an alkyl group having from 1 to 6 carbon atoms and n is an integer from 1 to 5 inclusive, or a therapeutically acceptable salt thereof such as a salt with an alkali metal, e.g. sodium or potassium. The effectiveness of the compound, for example, 3-trimethylsilyl butyric acid as well as the sodium and potassium salts thereof is established by the animal test undertaken with hypertensive rats.
摘要翻译：提出作为抗高血压药有效的新型药物，其含有作为其有效成分的由通式R 3 Si（CH 2）n COOH表示的有机硅化合物，其中R表示具有1至6个碳原子的烷基，n为 1〜5的整数，或其治疗上可接受的盐，例如与碱金属的盐，例如，钠或钾。化合物，例如3-三甲基甲硅烷基丁酸及其钠盐和钾盐的有效性是通过用高血压大鼠进行的动物试验建立的。

5. 发明授权

US4320172A Organopolysiloxane resin compositions for release papers 失效
标题翻译：用于剥离纸的有机聚硅氧烷树脂组合物
公开(公告)号：US4320172A
公开(公告)日：1982-03-16
申请号：US165148
申请日：1980-07-01
申请人： Minoru Takamizawa , Toshio Shinohara , Yasushi Yamamoto , Tasuku Tanino , Kiyoyuki Takano , Fumiaki Mori
发明人： Minoru Takamizawa , Toshio Shinohara , Yasushi Yamamoto , Tasuku Tanino , Kiyoyuki Takano , Fumiaki Mori
IPC分类号： C08L33/06 , D21H27/00 , C08L31/02 , C08L67/06 , C08L83/10
CPC分类号： D21H27/001 , C08L33/06 , Y10T428/31663
摘要： The invention provides a novel in-process release paper, i.e. a release paper used as a backing paper in the manufacturing of, e.g. a synthetic leather with a polyurethane resin. The releasing resin composition with which the release paper is coated is novel as comprising (a) a base resin selected from the group consisting of alkyd resins and acrylic resins modified with an organopolysiloxane, of which from 15 to 50% by moles of the organic groups directly bonded to the silicon atoms in a molecule are phenyl groups, having at least one hydroxy-substituted organic group directly bonded to the silicon atom in a molecule, (b) an alkanol-modified amino resin and (c) an acidic catalyst. The inventive in-process release paper is very superior to the conventional ones in the very much reduced peeling resistance, increased surface gloss and durability in repeated use.
摘要翻译：本发明提供了一种新颖的过程中的脱模纸，即在例如制造中用作背纸的剥离纸。具有聚氨酯树脂的合成革。包含剥离纸的释放树脂组合物是新颖的，包括（a）选自醇酸树脂和用有机聚硅氧烷改性的丙烯酸树脂的基础树脂，其中15至50摩尔％的有机基团与分子中的硅原子直接键合的苯基具有至少一个羟基取代的有机基团，其分子中直接与硅原子键合，（b）链烷醇改性的氨基树脂和（c）酸性催化剂。本发明的在制脱模纸非常优于常规剥离纸，在非常降低的抗剥离性，增加的表面光泽度和重复使用中的耐久性。

6. 发明授权

US09606517B2 Actuator control method and actuator control device 有权
公开(公告)号：US09606517B2
公开(公告)日：2017-03-28
申请号：US14241366
申请日：2012-08-10
申请人： Yasushi Yamamoto
发明人： Yasushi Yamamoto
IPC分类号： G06F7/70 , G05B13/02 , G05B19/416 , G05B19/23 , G05B19/29 , G05B19/35
CPC分类号： G05B13/02 , G05B19/23 , G05B19/29 , G05B19/35 , G05B19/416 , G05B2219/34311 , G05B2219/43045 , G05B2219/43064
摘要： An actuator control method and an actuator control device that perform energy evaluation control that compares kinetic energy of a controlled object and work that can be done by braking and switches driving to braking at a point of time at which the kinetic energy of the controlled object and the work become equal, and also repeatedly makes a comparison between the kinetic energy of the controlled object and the work at each preset time, as a new control method that replaces PID control in mechanics for effectively utilizing vehicle energy to improve vehicle fuel consumption and control methods thereof, a control result is obtained by a simpler method.

7. 发明授权

US09522857B2 3,3′,4,4′-tetraalkyl cyclohexylbenzene and method for producing same 有权
标题翻译： 3,3'，4,4'-四烷基环己基苯及其制备方法
公开(公告)号：US09522857B2
公开(公告)日：2016-12-20
申请号：US14118190
申请日：2012-05-18
申请人： Yasushi Yamamoto , Hikaru Yatabe
发明人： Yasushi Yamamoto , Hikaru Yatabe
IPC分类号： C07C13/38 , C07C15/14 , C07C2/76 , B01J23/44 , B01J23/46 , B01J29/08 , C07C13/28 , C07D407/04 , C07C2/74 , C07C5/367
CPC分类号： C07C2/76 , B01J23/44 , B01J23/462 , B01J29/088 , C07C2/74 , C07C5/367 , C07C13/28 , C07C2521/04 , C07C2521/08 , C07C2521/12 , C07C2521/16 , C07C2521/18 , C07C2523/44 , C07C2523/63 , C07C2529/08 , C07C2529/18 , C07C2529/40 , C07C2529/50 , C07C2529/70 , C07C2601/14 , C07D407/04 , Y02P20/52 , C07C15/14
摘要： A 3,3′,4,4′-tetraalkyl cyclohexylbenzene represented by the general formula (1): in which R represents an alkyl group having 1 to 4 carbon atoms, which may be easily converted into a 3,3′,4,4′-biphenyltetracarboxylic acid and a 3,3′,4,4′-biphenyltetracarboxylic dianhydride thereof, which are starting materials for a polyimide, via a 3,3′,4,4′-tetraalkylbiphenyl; and a method for producing the same.

8. 发明授权

US09519275B2 Actuator control method and actuator control device 有权
标题翻译：执行器控制方式和执行器控制装置
公开(公告)号：US09519275B2
公开(公告)日：2016-12-13
申请号：US14345167
申请日：2012-08-10
申请人： Yasushi Yamamoto
发明人： Yasushi Yamamoto
IPC分类号： G05B11/01 , G05B13/02 , G05B19/416 , G05B11/16 , G05B11/36 , G05B19/23 , G05B19/29 , G05B19/35
CPC分类号： G05B13/02 , G05B11/16 , G05B11/36 , G05B13/021 , G05B19/23 , G05B19/29 , G05B19/35 , G05B19/416 , G05B2219/41086 , G05B2219/41087 , G05B2219/41414 , G05B2219/43034 , G05B2219/43062
摘要： In an actuator control method and an actuator control device, time optimal control is used, and a switching time at which an acceleration output is switched to a deceleration output, and an end time of the deceleration output are calculated using a maximum acceleration and a maximum deceleration at the time of a maximum output of a control force. A control force of an actuator is set as a maximum acceleration output from a calculation time to the switching time, the control force of the actuator is set as a maximum deceleration output from the switching time to the end time, output of the control force is ended at the end time, and the switching time and the end time are repeatedly calculated, and updated for each preset time. The control output is reduced along with decrease of residual energy, which is a sum of remaining work and kinetic energy of a control system. From this, an element of feedback control is incorporated in the time optimal control, and the control output is converged after the end of the control.
摘要翻译：在致动器控制方法和致动器控制装置中，使用时间优化控制，将加速度输出切换为减速输出的切换时间，并且使用最大加速度和最大值来计算减速输出的结束时间控制力最大输出时减速。将致动器的控制力设定为从计算时间到切换时间的最大加速度输出，将致动器的控制力设定为从切换时间到结束时间的最大减速度输出，控制力的输出为在结束时间结束，并重复计算切换时间和结束时间，并针对每个预设时间更新。控制输出随着剩余能量的减少而减小，剩余能量是控制系统的剩余功率和动能之和。由此，在时间最优控制中并入反馈控制的要素，控制输出在控制结束后收敛。

9. 发明授权

US08951158B2 Planetary friction gear continuously variable transmission 有权
标题翻译：行星摩擦齿轮无级变速器
公开(公告)号：US08951158B2
公开(公告)日：2015-02-10
申请号：US14114331
申请日：2012-04-27
申请人： Shou Ozaki , Yasushi Yamamoto , Hirotsugu Yabe
发明人： Shou Ozaki , Yasushi Yamamoto , Hirotsugu Yabe
IPC分类号： F16H15/48 , F16H13/06 , F16H15/50 , F16H15/52
CPC分类号： F16H15/50 , F16H15/52
摘要： Planetary friction gear continuously variable transmission including an input shaft; a carrier; a planetary friction gear having a tapered roller at an inclined rotating shaft; an input-side support section, formed by notching a portion of an outer periphery of a carrier bottom section, rotatably supports an input side of the shaft; a sun roller provided on a same line as the shaft; a ring roller which is rotated by contacting a roller of the gear; an output shaft spaced from the ring roller; a loading section having a rolling body which presses the ring roller and the output shaft in an axial direction when a torque differential arises; and a transmission ring which contacts the tapered roller and allows the gear to spin.
摘要翻译：行星摩擦齿轮无级变速器，包括输入轴; 承运人具有在倾斜旋转轴上的圆锥滚子的行星摩擦齿轮; 通过切割载体底部的外周的一部分而形成的输入侧支撑部，可旋转地支撑轴的输入侧; 设置在与轴相同的线上的太阳辊; 环形滚筒，其通过与齿轮的辊接触而旋转; 与环形滚筒间隔开的输出轴; 具有滚动体的装载部，当产生扭矩差时，滚动体在轴向上按压环形滚筒和输出轴; 以及与圆锥滚子接触并允许齿轮旋转的传动环。

10. 发明授权

US08938863B2 Fastener stringer and slide fastener 有权
标题翻译：紧固件纵梁和拉链
公开(公告)号：US08938863B2
公开(公告)日：2015-01-27
申请号：US13639493
申请日：2010-04-06
申请人： Yoshimichi Yamakita , Masamichi Hasegawa , Yasushi Yamamoto , Nobuhiro Murai
发明人： Yoshimichi Yamakita , Masamichi Hasegawa , Yasushi Yamamoto , Nobuhiro Murai
IPC分类号： A44B19/08 , A44B19/06
CPC分类号： A44B19/06 , Y10T24/25 , Y10T24/2543 , Y10T24/2589
摘要： Disclosed is a fastener stringer where at least one surface of each of the fastener elements is colored. A plurality of fine fixing spaces is disposed on at least one surface of the fastener element which is colored. Accordingly, when a slide fastener is colored through an inkjet method, ink droplets ejected to the fastener element may be received by a plurality of fixing spaces and stably fixed onto a surface of the element. Consequently, a desired pattern or color can be continuously given to a fastener tape or the fastener element, and the contour of the pattern or color can be formed clearly and neatly.
摘要翻译：公开了一种紧固件纵梁，其中每个紧固件元件的至少一个表面是着色的。多个精细固定空间设置在着色的紧固件元件的至少一个表面上。因此，当通过喷墨方法着色拉链时，喷射到拉链件的墨滴可以被多个固定空间容纳并稳定地固定在元件的表面上。因此，可以连续地对拉链带或拉链件施加期望的图案或颜色，并且可以清楚和整齐地形成图案或颜色的轮廓。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式