会员体验
专利管家(专利管理)
工作空间(专利管理)
风险监控(情报监控)
数据分析(专利分析)
侵权分析(诉讼无效)
联系我们
交流群
官方交流:
QQ群: 891211   
微信请扫码    >>>
现在联系顾问~
热词
    • 3. 发明专利
    • BR0214997A
    • 2004-12-07
    • BR0214997
    • 2002-11-25
    • SYNGENTA LTDSYNGENTA PARTICIPATIONS AG
    • WHITTINGHAM WILLIAM GUYLAWSON KEVIN ROBERTWORTHINGTON PAUL ANTHONYRUSSELL CHARLES ADAMSALMON ROGERMAY LESLIE FRANCISJORG MARIOPACHLATKO JOHANNES PAUL
    • A01N25/02A01N25/08A01N43/40C07D213/65C07D213/68C07D213/70C07D213/79C07D213/80C07D213/81C07D213/82C07D213/84C07D213/85
    • Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
    • 4. 发明专利
    • DE60218213T2
    • 2007-11-08
    • DE60218213
    • 2002-11-25
    • SYNGENTA LTDSYNGENTA PARTICIPATIONS AG
    • WHITTINGHAM WILLIAM GUYLAWSON KEVIN ROBERTWORTHINGTON PAUL ANTHONYRUSSELL CHARLES ADAMSALMON ROGERMAY LESLIE FRANCISJORG MARIOPACHLATKO JOHANNES
    • C07D213/65A01N25/02A01N25/08A01N43/40C07D213/68C07D213/70C07D213/79C07D213/80C07D213/81C07D213/82C07D213/84C07D213/85
    • Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
    • 5. 发明专利
    • PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES
    • CA2467527A1
    • 2003-06-12
    • CA2467527
    • 2002-11-25
    • SYNGENTA PARTICIPATIONS AGSYNGENTA LTD
    • JORG MARIOPACHLATKO JOHANNES PAULWHITTINGHAM WILLIAM GUYSALMON ROGERRUSSELL CHARLES ADAMLAWSON KEVIN ROBERTMAY LESLIE FRANCISWORTHINGTON PAUL ANTHONY
    • A01N25/02A01N25/08A01N43/40C07D213/65C07D213/68C07D213/70C07D213/79C07D213/80C07D213/81C07D213/82C07D213/84C07D213/85
    • Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C1-8 alkyl, C3-6 cycloalkyl, C2-8 alkenyl, C2-8 alkynyl, C1-8 alkoxy, C1-8 alkylthio, nitro, amino, mono- or di-(C1- 6)alkylamino, mono- or di-(C2-6)alkenylamino, mono- or di-(C2-6)alkynylamino , formylamino, C1-4 alkyl(formyl)amino, C1-4 alkylcarbonylamino, C1-4 alkyl(C1 -4 alkylcarbonyl)amino, cyano, formyl, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C1-4)alkylaminocarbonyl, carboxy, C1-4 alkylcarbonyloxy, aryl(C1-4)alkylcarbonyloxy, C1-4 alkylsulphinyl, C1-4 alkylsulphonyl, C1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R1 is phenyl, cyano, C1-4 alkyl, C2-4 alkenyl or C2- 4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C1-4 alkylcarbonyl group, with a C1-4 alkoxycarbonyl group or with a hydroxy group, or R1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the tota l number of carbon atoms is 2 or 3; R2 is H, C1-4 alkyl, C1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C1-4 alkoxy; R3 and R4 are independently H, C1-3 alkyl, C2- 3 alkenyl or C2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R3 a nd R4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C1-4 alkyl; and R5 is halo, C1-4 alkyl o r C3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C1-6 alkoxy, C1-6 alkylthio, cyano, C1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C1-4)alkylaminocarbonyloxy, or tri(C1-4)alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
    • 6. 发明专利
    • PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES
    • PL370740A1
    • 2005-05-30
    • PL37074002
    • 2002-11-25
    • SYNGENTA LTDSYNGENTA PARTICIPATIONS AG
    • WHITTINGHAM WILLIAM GUYLAWSON KEVIN ROBERTWORTHINGTON PAUL ANTHONYRUSSELL CHARLES ADAMSALMON ROGERMAY LESLIE FRANCISJORG MARIOPACHLATKO JOHANNES PAUL
    • A01N25/02A01N25/08A01N43/40C07D213/65C07D213/68C07D213/70C07D213/79C07D213/80C07D213/81C07D213/82C07D213/84C07D213/85
    • Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
    • 7. 发明专利
    • PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES
    • AU2002365647A1
    • 2003-06-17
    • AU2002365647
    • 2002-11-25
    • SYNGENTA LTDSYNGENTA PARTICIPATIONS AG
    • JORG MARIOPACHLATKO JOHANNES PAULWHITTINGHAM WILLIAM GUYLAWSON KEVIN ROBERTWORTHINGTON PAUL ANTHONYRUSSELL CHARLES ADAMSALMON ROGERMAY LESLIE FRANCIS
    • A01N25/02A01N25/08A01N43/40C07D213/65C07D213/68C07D213/70C07D213/79C07D213/80C07D213/81C07D213/82C07D213/84C07D213/85
    • Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
    • 8. 发明专利
    • DERIVADOS DE AMIDAS DE ACIDOS PIRIDILOXIALCANOICOS UTILES COMO FUNGICIDAS.
    • ES2282518T3
    • 2007-10-16
    • ES02804256
    • 2002-11-25
    • SYNGENTA LTDSYNGENTA PARTICIPATIONS AG
    • WHITTINGHAM WILLIAM GUYLAWSON KEVIN ROBERTWORTHINGTON PAUL ANTHONY SYNGERUSSELL CHARLES ADAMSALMON ROGERMAY LESLIE FRANCIS
    • C07D213/65A01N25/02A01N25/08A01N43/40C07D213/68C07D213/70C07D213/79C07D213/80C07D213/81C07D213/82C07D213/84C07D213/85
    • Un compuesto de fórmula general (I): en donde X e Y son independientemente H, halo, alquilo 1-8C, cicloalquilo 3-6C, alquenilo 2-8C, alquinilo 2-8C, alcoxi 1-8C, alquil(1-8C)tio, nitro, amino, mono- o di-alquil(1-6C)amino, mono- o di-alquenil(2-6C)amino, mono- o di-alquinil(2-6C)amino, formilamino, alquil(1-4C)(formil)amino, alquil(1-4C)carbonilamino, alquil(1-4C)(alquil(1-4C)carbonil)amino, ciano, formilo, alquil(1-4C)carbonilo, alcoxi(1-4C)carbonilo, aminocarbonilo, mono- o di-alquil(1-4C)aminocarbonilo, alcoxi, alquil(1-4C)carboniloxi, arilalquil(1-4C)carboniloxi, alquil(1-4C)sulfinilo, alquil(1-4C)sulfonilo, alquil(1-4C)sulfoniloxi, arilo, heteroarilo, ariloxi, ariltio, heteroariloxi o heteroariltio en donde cualquiera de los anteriores grupos o mitades alquilo, cicloalquilo, alquenilo, alquinilo, arilo, heteroarilo están opcionalmente sustituidos; R1 es fenilo, ciano, alquilo 1-4C, alquenilo 2-4C o alquinilo 2-4C en donde los grupos alquilo, alquenilo y alquinilo están opcionalmente sustituidos en su átomo de carbono terminado con 1, 2 o 3 átomos de halógeno (por ejemplo, 2-fluormetilo, 2-cloroetilo, 2, 2-difluoretilo y 2, 2, 2-trifluoretilo), con un grupo ciano (por ejemplo, cianometilo), con un grupo alquil(1-4C)carbonilo (por ejemplo, acetilmetilo), con un grupo alcoxi(1-4C)carbonilo (por ejemplo, metoxicarbonilmetilo y metoxicarboniletilo) o con un grupo hidroxi (por ejemplo, hidroximetilo), o R1 es alcoxialquilo, alquiltioalquilo, alquilsulfinilalquilo o alquilsulfonilalquilo en donde el número total de átomos de carbono es 2 o 3 (por ejemplo, metoximetilo, metiltiometilo, etoximetilo, 1-metoxietilo y 2-metoxietilo); R2 es H, alquilo 1-4C, alcoxi(1-4C)metilo o benciloximetilo en donde el anillo fenilo de la mitad bencilo está opcionalmente sustituido con alcoxi 1-4C; R3 y R4 son independientemente H, alquilo 1-3C, alquenilo 2-3C o alquinilo 2-3C siempre que ambos no sean H y siempre que cuando ambos son distintos de H su total combinado de átomos de carbono no excede de 4, o R3 y R4 junto con el átomo de carbono al cual están unidos forman un anillo carbocíclico de 3 o 4 miembros que contiene opcionalmente un átomo de O, S o N y opcionalmente sustituido con halo o alquilo 1-4C; y R5 es halo, alquilo 1-4C, cicloalquilo 3-6C en donde el grupo alquilo o cicloalquilo está opcionalmente sustituido con halo, hidroxi, alcoxi 1-6C, alquil(1-6C)tio, ciano, alquil(1-4C)carboniloxi, aminocarboniloxi, mono- o di-alquil(1-4C)aminocarboniloxi o tri-alquil(1-4C)sililoxi.
    • 9. 发明专利
    • DE60218213D1
    • 2007-03-29
    • DE60218213
    • 2002-11-25
    • SYNGENTA LTDSYNGENTA PARTICIPATIONS AG
    • WHITTINGHAM WILLIAM GUYLAWSON KEVIN ROBERTWORTHINGTON PAUL ANTHONYRUSSELL CHARLES ADAMSALMON ROGERMAY LESLIE FRANCISJORG MARIOPACHLATKO PAUL
    • C07D213/65A01N25/02A01N25/08A01N43/40C07D213/68C07D213/70C07D213/79C07D213/80C07D213/81C07D213/82C07D213/84C07D213/85
    • Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
    • 10. 发明专利
    • AT353878T
    • 2007-03-15
    • AT02804256
    • 2002-11-25
    • SYNGENTA LTDSYNGENTA PARTICIPATIONS AG
    • WHITTINGHAM WILLIAM GUYLAWSON KEVIN ROBERTWORTHINGTON PAUL ANTHONYRUSSELL CHARLES ADAMSALMON ROGERMAY LESLIE FRANCISJORG MARIOPACHLATKO JOHANNES PAUL
    • A01N25/02A01N25/08A01N43/40C07D213/65C07D213/68C07D213/70C07D213/79C07D213/80C07D213/81C07D213/82C07D213/84C07D213/85
    • Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.