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1. 发明申请

WO1993013123A1 NOVEL 19-NOR STEROIDS HAVING A THIOCARBON-CONTAINING CHAIN IN THE 11BETA POSITION, A METHOD FOR PREPARING SAME AND INTERMEDIATES THEREFOR, MEDICINAL USES THEREOF AND COMPOSITIONS CONTAINING SAID STEROIDS 审中-公开
标题翻译：具有11BETA位置中的含硫链的新型19-非甾体类抗生素，其制备方法及其中间体，其药物用途及含有STEROIDS的组合物
公开(公告)号：WO1993013123A1
公开(公告)日：1993-07-08
申请号：PCT/FR1992001193
申请日：1992-12-17
申请人： ROUSSEL-UCLAF , CLAUSSNER, André , NIQUE, François , TEUTSCH, Jean-Georges , VAN DE VELDE, Patrick
发明人： ROUSSEL-UCLAF
IPC分类号： C07J43/00
CPC分类号： C07J31/006 , C07J41/0005 , C07J41/0016 , C07J41/0083 , C07J43/003
摘要： Compounds of formula (I), wherein R17 and R'17 are such that: either R17 and R'17 together form ketone, hydrazono, oxime or methylene, or R17 is hydroxyl, hydroxymethyl or acyloxy and R'17 is hydrogen, alkyl or optionally substitued alkenyl or alkynyl; R3 is hydrogen or alkyl; R16 is hydrogen, halogen or alkyl; m is 0, 1 or 2; X, Y and Z are such that: X is methylene, arylene or arylenoxy bonded to the steroid by a carbon atom; Y is a saturated or unsaturated straight or branched aliphatic chain which is optionally interrupted by oxygen; and Z is aryl, arylalkyl or straight or branched alkyl; addition salts thereof, a preparation method therefor, medicinal uses thereof, compositions containing said compounds, and resulting novel intermediates.

2. 发明申请

WO1987005908A1 STEROIDS COMPRISING A SPIRANIC CYCLE IN POSITION 17, PREPARATION PROCESS AND UTILIZATION THEREOF 审中-公开
标题翻译：包含位置17中的SPIRANIC循环的STEROIDS，其制备过程及其利用
公开(公告)号：WO1987005908A1
公开(公告)日：1987-10-08
申请号：PCT/FR1987000096
申请日：1987-03-26
申请人： ROUSSEL-UCLAF , NIQUE, François , NEDELEC, Lucien , PHILIBERT, Daniel , MOGUILEWSKY, Martine
发明人： ROUSSEL-UCLAF
IPC分类号： C07J21/00
CPC分类号： C07J43/003 , C07J31/006 , C07J33/002 , C07J41/0077 , C07J41/0083 , Y10S514/843
摘要： Products having the formula (I) wherein R1 is an aryl or aralkyl, R2 is a hydrocarbonated radical (1-18 carbon atoms), the dotted lines indicate an optional bond, the cycles A, B and C represent (II), (III), (IV), (V), (VI); R' and R'' are H, alkyl (1-4 carbon atoms), Re is H, alkyl (1-6 carbon atoms), acyl, and their salts, their preparation, their application as medicaments, the pharmaceutical compositions containing them and intermediaries.
摘要翻译：具有式（I）的产物，其中R 1是芳基或芳烷基，R 2是烃基（1-18个碳原子），虚线表示任选的键，循环A，B和C表示（II），（III ），（IV），（V），（VI） R'和R“是H，烷基（1-4个碳原子），Re是H，烷基（1-6个碳原子），酰基及其盐，它们的制备，它们作为药物的应用，含有它们的药物组合物和中介。

3. 发明申请

WO1988007856A1 BUTYL HYDROXYANISOLES FOR THE TREATMENT OF RETROVIRAL DISEASES 审中-公开
标题翻译：用于治疗退行性疾病的丁基羟肟酸酯
公开(公告)号：WO1988007856A1
公开(公告)日：1988-10-20
申请号：PCT/FR1988000173
申请日：1988-04-08
申请人： ROUSSEL-UCLAF , MARCEL, Georges
发明人： ROUSSEL-UCLAF
IPC分类号： A61K31/085
CPC分类号： A61K31/085
摘要： The invention concerns chemical compounds consisting of the buty hydroxyanisoles and their salts for use in a method of therapeutic treatment of the human or animal body, in particular for use in a method of prophylactic or curative treatment of retroviral diseases, such as AIDS.
摘要翻译：本发明涉及由用于人或动物体的治疗性治疗方法的丁基羟基茴香醚及其盐组成的化合物，特别是用于预防或治疗性治疗逆转录病毒疾病如AIDS的方法。

4. 发明申请

WO1983003756A1 ORAL FORM OF CLOMETACIN AND PREPARATION THEREOF 审中-公开
标题翻译：甲壳胺的口服形式及其制备
公开(公告)号：WO1983003756A1
公开(公告)日：1983-11-10
申请号：PCT/FR1983000073
申请日：1983-04-20
申请人： ROUSSEL-UCLAF
发明人： ROUSSEL-UCLAF , HERCELIN, Bernard , MARY, Irène , NUNG, Vien, Nghia
IPC分类号： A61K09/16
CPC分类号： A61K31/405 , A61K9/1605 , A61K9/1611 , A61K9/5047 , Y10S514/962
摘要： New oral pharmaceutical form of clometacin consisting of pellets obtained by extrusion, containing 50 to 70 % of clometacin, 5 to 20 % of alkaline carbonate and an anhydrous granulation excipient, by wet process.
摘要翻译：新的口服药物形式的clometacin由通过挤出获得的颗粒组成，通过湿法包含50-70％的clometacin，5〜20％的碱性碳酸盐和无水造粒赋形剂。

5. 发明申请

WO1983002545A1 APPLICATION AS GROWTH FACTORS OF VEGETABLES OF HYDROXYLAMINE DERIVATIVES 审中-公开
标题翻译：作为羟基胺衍生物蔬菜生长因子的应用
公开(公告)号：WO1983002545A1
公开(公告)日：1983-08-04
申请号：PCT/FR1983000019
申请日：1983-01-26
申请人： ROUSSEL-UCLAF
发明人： ROUSSEL-UCLAF , VAN ASSCHE, Charles, Jacques , HERVE, Jean-Jacques , CARLES, Pierre, Marius
IPC分类号： A01N33/24
CPC分类号： A01N33/24
摘要： Application as growth factors of vegetables of compounds having the formula (I): wherein - either R1 is hydrogen, and R2 is hydrogen and R3 is hydrogen, methyl in position 2, 3 or 4, a chlorine in 3 or 4, a bromine or CF3 in 4 or NO2 in position 2, or else R2 is nitro in position 2 and R3 is nitro or CF3 in position 4; -or R1 is nitro in 2 and R2 is nitro in 4 and R4 is nitro in 6, or R2 is nitro in 6 and R3 is CF3 in 4, as well as their addition salts with the organic and mineral acids. The invention also relates to compositions used as growth factors of vegetables, containing as an active principle, at least one of the compounds of formula (I) or of their salts.
摘要翻译：作为具有式（I）的化合物的蔬菜的生长因子的应用：其中 - R1是氢，R2是氢，R3是氢，2,3或4位的甲基，3或4的氯，位置2中的4或NO 2中的溴或CF 3，或者R 2在位置2是硝基，R 3是位置4的硝基或CF 3; 或者R1为硝基，R2为硝基，R6为硝基，R6为硝基，R6为R3，R3为CF3，以及它们与有机酸和无机酸的加成盐。本发明还涉及用作蔬菜生长因子的组合物，其含有作为活性成分的至少一种式（I）化合物或其盐。

6. 发明申请

WO1991018604A1 USE OF TETRAHYDROISOQUINOLINE DERIVATIVES FOR PREPARING ANTITUMORAL DRUGS 审中-公开
标题翻译：四氢喹啉衍生物用于制备抗肿瘤药物的应用
公开(公告)号：WO1991018604A1
公开(公告)日：1991-12-12
申请号：PCT/FR1991000448
申请日：1991-06-06
申请人： ROUSSEL-UCLAF , FRECHET, Daniel , MARCHANDEAU, Christian , CZECH, Jörg , SEDLACEK, Hans, Harald
发明人： ROUSSEL-UCLAF
IPC分类号： A61K31/47
CPC分类号： A61K31/47 , A61K31/475
摘要： The substances of formula (I), wherein A) either Y = H and X = (a) and Ar = (b) or (c); or B) X = H and Y = benzyl and Ar = (d); R2 and R3 = H or C1-4 alkyl; R1 = H or CH3; and the salts thereof, are used for preparing an anti-tumoral drug.

7. 发明申请

WO1991009833A1 USE OF 9,10-DIHYDROPHENANTHRENE DERIVATIVES TO PREPARE AN ANTITUMORAL DRUG, AND NOVEL DERIVATIVES THEREOF 审中-公开
标题翻译：使用9,10-二氢萘衍生物来制备抗肿瘤药物及其新型衍生物
公开(公告)号：WO1991009833A1
公开(公告)日：1991-07-11
申请号：PCT/FR1990000952
申请日：1990-12-27
申请人： ROUSSEL-UCLAF , CZECH, Jörg , SEDLACEK, Hans, Harald , NEDELEC, Lucien , GUILLAUME, Jacques , MARCHANDEAU, Christian
发明人： ROUSSEL-UCLAF
IPC分类号： C07C211/42
CPC分类号： C07C211/42 , A61K31/13 , C07C2603/26
摘要： The use of products of formula (I) is described, wherein X and Y represent hydrogen, hydroxy or alkoxy; and R1 and R2 represent H, alkyl, alkenyl or alkynyl, arylalkyl, acyl or R1 and R2 together with nitrogen form a heterocycle for preparing an antitumoral drug.
摘要翻译：描述了使用式（I）的产物，其中X和Y表示氢，羟基或烷氧基; 并且R 1和R 2表示H，烷基，烯基或炔基，芳烷基，酰基或R 1和R 2与氮一起形成用于制备抗肿瘤药物的杂环。

8. 发明申请

WO1989008096A1 NEW PYRETHRINOID ESTERS CARRYING AN INDANYL RING, PREPARATION METHOD AND APPLICATION AS PESTICIDES 审中-公开
标题翻译：作为农药的新型吡咯啉酯，制备方法和应用
公开(公告)号：WO1989008096A1
公开(公告)日：1989-09-08
申请号：PCT/FR1989000087
申请日：1989-03-03
申请人： ROUSSEL-UCLAF , BABIN, Didier , DEMOUTE, Jean-Pierre , TESSIER, Jean
发明人： ROUSSEL-UCLAF
IPC分类号： C07C69/74
CPC分类号： C07C35/50 , A01N53/00 , C07C255/53 , C07C2602/08
摘要： The invention relates to compounds having the formula (I) wherein the radical A is represented by the formula (II) wherein D is hydrogen, halogen, alkoxyl, G is oxygen or sulphur, J is alkyl, aryl or a heterocycle optionally substituted, Z is hydrogen, halogen, alkyl, aryl or a keto group, n is 1, 2 or 3; Y is hydrogen, halogen, CF3, CN, alkyl, aryl, m being 1 or 2; W is either one of the values indicated for Y, or NO2, OCH3, N3, N(R4)2 or SnR5, R4 and R5 representing hydrogen or alkyl, p being 1 or 2. The compounds (I) have interesting pesticidal properties.
摘要翻译：本发明涉及具有式（I）的化合物，其中基团A由式（II）表示，其中D为氢，卤素，烷氧基，G为氧或硫，J为烷基，芳基或任选取代的杂环，Z 是氢，卤素，烷基，芳基或酮基，n是1,2或3; Y是氢，卤素，CF 3，CN，烷基，芳基，m是1或2; W是Y表示的值之一，或NO2，OCH3，N3，N（R4）2或SnR5，R4和R5表示氢或烷基，p为1或2.化合物（I）具有有趣的农药性质。

9. 发明申请

WO1993007750A1 CONTROL OF INSECTS 审中-公开
标题翻译：管理控制
公开(公告)号：WO1993007750A1
公开(公告)日：1993-04-29
申请号：PCT/EP1992002345
申请日：1992-10-12
申请人： ROUSSEL-UCLAF , MARTIN, Robert , CAYLEY, George, R. , THACKER, J., Richard, M. , HALL, Franklin, R.
发明人： ROUSSEL-UCLAF
IPC分类号： A01N53/00
CPC分类号： A01N53/00 , A01N25/04 , A01N2300/00
摘要： A method of controlling insects on plants which comprises the application to the plant of an effective amount of an aqueous formulation that contains a pyrethroid insecticide as active ingredient, an evaporation retardant and an emulsifier, optionally together with a carrier or solvent for the active ingredient, which the formulation satisfies the formula: mass of oil phase/mass of retardant )]]/C] where L is less than or equal to 15, A = 700376, B = -1.51, C = 0.8472, Moil is the weighted average relative molar mass of the oil phase, Mretardant is the average molar mass of the retardant, and X = Moil / Y where Y is the molar solubility ratio of the formulation, defined as the minimum number of moles of oil phase which will dissolve the retardant, divided by the number of moles of retardant, provided that, in the formula above, any solvent which has no liquid phase at 27 DEG C at atmospheric pressure is excluded.
摘要翻译：一种控制植物昆虫的方法，其包括向植物施用有效量的含有拟除虫菊酯杀虫剂作为活性成分的水性制剂，蒸发阻燃剂和乳化剂，任选地与活性成分的载体或溶剂一起使用，该配方满足以下公式：油相质量/阻燃剂质量/摩尔/摩擦剂。 X Exp [[ln（L / 4）+ [C x ln（AX B）]] / C]其中L小于或等于15，A = 700376，B = -1.51，C = 0.8472，是油相的加权平均相对摩尔质量，Mretardant是阻燃剂的平均摩尔质量，X = Moil <1.8> / Y，其中Y是制剂的摩尔溶解度比，定义为最小摩尔数将阻燃剂溶解的油相除以阻燃剂的摩尔数，条件是在上式中，排除了在27℃下在大气压下没有液相的任何溶剂。

10. 发明申请

WO1992013950A2 NUCLEOTIDIC SEQUENCES CODING FOR VARIABLE REGIONS OF 'beta' CHAINS OF HUMAN T LYMPHOCYTE RECEPTORS, CORRESPONDING PEPTIDIC SEGMENTS AND DIAGNOSTIC AND THERAPEUTIC APPLICATIONS 审中-公开
标题翻译：人类淋巴细胞受体β链可变区的核苷酸序列编码，相应的部分和诊断和治疗应用
公开(公告)号：WO1992013950A2
公开(公告)日：1992-08-20
申请号：PCT/FR1992000130
申请日：1992-02-12
申请人： ROUSSEL-UCLAF , HERCEND, Thierry , TRIEBEL, Frédéric , ROMAN-ROMAN, Sergio , FERRADINI, Laurent
发明人： ROUSSEL-UCLAF
IPC分类号： C12N15/12
CPC分类号： C12N15/1138 , A61K38/00 , C07K14/7051 , C07K16/2809
摘要： The invention relates to new nucleotidic sequences coding for variable regions of beta chains of human T lymphocyte receptors, the corresponding peptidic segments and the diagnostic and therapeutic applications.
摘要翻译：本发明涉及编码人类T淋巴细胞受体β链的可变区的新的核苷酸序列，相应的肽段以及诊断和治疗应用。

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