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1. 发明申请

US20060148729A1 Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substitutent in the 4"-or 4'-position 有权
公开(公告)号：US20060148729A1
公开(公告)日：2006-07-06
申请号：US10539274
申请日：2003-12-19
申请人： Peter Maienfisch , Fiona Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Hueter , Pierre Jung
IPC分类号： A01N43/04 , C07H17/08
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula (I): wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —N02, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12 alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)-Z-R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

2. 发明申请

US20080051353A1 Avermectin And Avermectin Monosaccharide Substituted In The 4"- And 4" Position Respectively 有权
标题翻译：阿维菌素和阿维菌素单糖在4“和4”位置分别取代
公开(公告)号：US20080051353A1
公开(公告)日：2008-02-28
申请号：US10599671
申请日：2005-03-09
申请人： Pierre Jung , Thomas Pitterna , Fiona Kessabi , Laura Quaranta , Ottmar Hueter
发明人： Pierre Jung , Thomas Pitterna , Fiona Kessabi , Laura Quaranta , Ottmar Hueter
IPC分类号： C07H19/01 , A01N43/90 , A61K31/7048 , A61P33/00
CPC分类号： A01N43/90 , C07H19/01
摘要： A compound of the formula (I) wherein the bond between carbon atoms 22 and 23 indicated with a broken line is a single or double bond, m is 0 or 1, R1 represents a C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl group, R2 represents a hydrocarbyl group or a substituted hydrocarbyl group, and R3 and R4 represent, independently of each other, hydrogen or a chemical constituent, or either R2 and R3 together or R3 and R4 together represent a three- to seven-membered alkylene or a four- to seven-membered alkenylene bridge, for each of which at least one, preferably a CH2 group may be replaced by O, S or NR6 where R6 represents hydrogen or a hydrocarbyl group or a substituted hydrocarbyl group; or, if appropriate, an E/Z isomer and/or tautomer of the compound of formula (I), in each case in free form or in salt form.
摘要翻译：式（I）的化合物，其中用虚线表示的碳原子22和23之间的键是单键或双键，m是0或1，R 1表示C 1〜 C 1 -C 12烷基，C 3 -C 8 - 环烷基或C 2 -C 3烷基， R 12是链烯基，R 2表示烃基或取代的烃基，R 3和R 4代表独立地是氢或化学成分，或R 2和R 3一起或R 3和R 4 一起代表三至七元亚烷基或四至七元亚烯基桥，其中至少一个，优选CH 2基团可以被O ，S或NR 6，其中R 6表示氢或烃基或取代的烃基; 或者如果合适的话，式（I）化合物的E / Z异构体和/或互变异构体在各种情况下都是游离形式或盐形式。

3. 发明申请

US20060229263A1 Avermectin b1 monosaccharide derivatives 有权
标题翻译：阿维菌素b1单糖衍生物
公开(公告)号：US20060229263A1
公开(公告)日：2006-10-12
申请号：US10560390
申请日：2004-06-15
申请人： Thomas Pitterna , Pierre Jung , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Ottmar Hueter
发明人： Thomas Pitterna , Pierre Jung , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Ottmar Hueter
IPC分类号： A01N43/04 , C07H17/08
CPC分类号： C07H19/01 , C07H17/08
摘要： A compound of formula (I) wherein the bond between carbon atoms 22 and 23 may be a single or a double bond; R1 is C1-C12alkyl, C3-C8cycloalkyl, or C2-C12alkenyl; R2 and R3 are, for example, independently of each other hydrogen, C1-C12alkyl, C3-C12cycloalkyl, C2-C12alkenyl, C2-C12alkynyl, aryl or heteroaryl; and, where applicable, to E/Z isomers, mixtures of E/Z isomers, diastereomers and/or tautomers, in each case in free form or in salt form; pesticidal compositions in which the active ingredient has been selected from those compounds and their tautomers; and a method of controlling pests using those compositions are described.
摘要翻译：式（I）的化合物，其中碳原子22和23之间的键可以是单键或双键; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 1 -C 12烷基，C 3 -C 12烷基，环烷基或C 2 -C 12 - 烯基; R 2和R 3是例如彼此独立的氢，C 1 -C 12烷基 C 3 -C 12环烷基，C 2 -C 12链烯基，C 2 -C 12环烷基，C 2 -C 12亚烷基，炔基，芳基或杂芳基; 在适用的情况下，E / Z异构体，E / Z异构体，非对映异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 其中活性成分选自那些化合物及其互变异构体的杀虫组合物; 并描述了使用这些组合物来控制害虫的方法。

4. 发明申请

US20060140997A1 Avermectin and avermectin monosaccharide derivatives substituted in the 4"-or 4'-position having pesticidal properties 有权
公开(公告)号：US20060140997A1
公开(公告)日：2006-06-29
申请号：US10543637
申请日：2004-01-30
申请人： Thomas Pitterna , Fiona Kessabi , Peter Maienfisch , Jerome Cassayre , Pierre Jung , Laura Quaranta
发明人： Thomas Pitterna , Fiona Kessabi , Peter Maienfisch , Jerome Cassayre , Pierre Jung , Laura Quaranta
IPC分类号： A01N25/00 , A01N43/04 , C07H17/08
CPC分类号： A01N43/90 , C07H17/08
摘要： What is described are a compound of the formula (I) Wherein U is —N(R2)OR3 or —N+(O−)═C(RE)RZ); n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 are, for example; independently from each other, -Q, —C(═O)-Z-Q or —CN; RZ and RE are, independently from each other, -Q, —C(═O)-Z-Q or —CN; or RZ and RE together are a three- to seven membered alkylene or alkenylene bridge, which is unsubstituted or mono- to tri-substituted; Z is a bond, O or —NR4—; Q is H, C1-C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12-Cycloalkyl, C5-C12-cycloalkenyl, aryl, or heterocyclyl, which are unsubstituted or mono- to pentasubstituted; R4 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl or C2-C8alkenyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions.

5. 发明申请

US20060154879A1 Avermectins substituted in the 4" and 4'-positions having pesticidal properties 有权
标题翻译：在4“和4”位取代的阿维菌素具有杀虫特性
公开(公告)号：US20060154879A1
公开(公告)日：2006-07-13
申请号：US10544274
申请日：2004-02-03
申请人： Jerome Cassayre , Hans Tobler , Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Laura Quaranta , Ottmar Hueter
发明人： Jerome Cassayre , Hans Tobler , Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Laura Quaranta , Ottmar Hueter
IPC分类号： A01N43/04 , C07H17/08
CPC分类号： C07H17/08
摘要： What is described are a compound of the formula (I) Wherein A-B is —CH═CH— or —CH2—CH2—; n is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 for instance are either, (i) independently from each other for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; or (ii) together form with the nitrogen atom to which they are bound a three- to seven-membered ring, (iii) together are ═C(R4)R5; R4 and R5 are, independently from each other, for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; Y is O or S; Q is for instance H or unsubstituted or mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions.
摘要翻译：描述的是式（I）的化合物，其中A-B是-CH-CH-或-CH 2 -CH 2 - 。 n为0或1; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 3 -C 12烷基，C 3 -C 12烷基，C 3 -C 12烷基， >环烷基或C 2 -C 12 - 烯基; 例如，R 2和R 3是（i）彼此独立地例如-Q，-C（-Y）-Q或-C（ - Y）-OQ; 或（ii）与其结合的氮原子一起形成三至七元环，（iii）一起为-C（R 4）R 5 >; R 4和R 5各自独立地为例如-Q，-C（-Y）-Q或-C（-Y）-O-Q; Y为O或S; Q是例如H或未被取代或单取代或未取代的C 1 -C 12烷基; 或者，如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体; 制备这些化合物，其异构体和互变异构体的方法以及这些化合物，其异构体和互变异构体的用途; 活性化合物选自这些化合物及其互变异构体的杀虫组合物; 用于制备所述式（I）化合物的中间体，式（I）化合物的制备方法和使用这些组合物来控制害虫的方法。

6. 发明申请

US20110230429A1 AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4"-OR 4'-POSITION 有权
标题翻译：在4“-OR 4'-位置具有烷氧基取代基的AVERMECTIN B1和AVERMECTIN B1单糖衍生物
公开(公告)号：US20110230429A1
公开(公告)日：2011-09-22
申请号：US13117292
申请日：2011-05-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jérôme Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jérôme Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A01N43/22 , C07H17/08 , A01P7/00
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

7. 发明申请

US20080300134A1 Derivatives of Avermectin, Avermectin Monosaccharide and Avermectin Aglycone 有权
标题翻译：阿维菌素，阿维菌素单糖和阿维菌素糖苷配基的衍生物
公开(公告)号：US20080300134A1
公开(公告)日：2008-12-04
申请号：US11574588
申请日：2005-08-19
申请人： Ottmar Franz Hueter , Thomas Pitterna , Pierre Jung , Fiona Murphy Kessabi , Laura Quaranta
发明人： Ottmar Franz Hueter , Thomas Pitterna , Pierre Jung , Fiona Murphy Kessabi , Laura Quaranta
IPC分类号： C07H17/08 , A01N43/90 , C07D313/00
CPC分类号： C07H17/08 , A01N43/90
摘要： A compound of the formula (I) wherein the bond between carbon atoms 22 and 23 indicated with a broken line is a single or double bond, n is 0, 1 or 2, R1 represents, for instance, a C1-C12alkyl group, R2 represents, for instance, R15 group, R3 represents, for instance, R2 group, R4 represents, for instance, a chemical constituent, R5 represents, for instance, hydrogen, and R6 represents, for instance, R16 group; wherein R15 represents, for instance, unsubstituted or mono- to pentasubstituted C1-C6alkyl group, and R16 represent, for instance, hydrogen, or R15; and if appropriate, an E/Z isomer and/or diastereoisomer and/or tautomer of the compound of formula (I), in each case in free form or in salt form. Such compounds have been found to have pesticidal properties.
摘要翻译：式（I）的化合物，其中用虚线表示的碳原子22和23之间的键是单键或双键，n是0,1或2，R1表示例如C1-C12烷基，R2 表示例如R 15基，R 3表示例如R 2基，R 4表示例如化学成分，R 5表示例如氢，R 6表示例如R 16基; 其中R 15表示例如未取代或单价至五价取代的C 1 -C 6烷基，R 16表示例如氢或R 15; 并且如果合适的话，式（I）化合物的E / Z异构体和/或非对映异构体和/或互变异构体在各种情况下均为游离形式或盐形式。已经发现这些化合物具有杀虫性质。

8. 发明授权

US08017589B2 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position 有权
标题翻译：在4“ - 或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物
公开(公告)号：US08017589B2
公开(公告)日：2011-09-13
申请号：US12768280
申请日：2010-04-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A61K31/70 , C07H17/04
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

9. 发明申请

US20100210574A1 AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4"-OR 4'-POSITION 有权
标题翻译：在4“-OR 4'-位置具有烷氧基取代基的AVERMECTIN B1和AVERMECTIN B1单糖衍生物
公开(公告)号：US20100210574A1
公开(公告)日：2010-08-19
申请号：US12768280
申请日：2010-04-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A01N43/16 , C07H17/08 , A01P17/00
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

10. 发明授权

US07632820B2 Avermectin and avemectin monosaccharide derivatives substituted in the 4″- or 4′-position having pesticidal properties 有权
标题翻译：在4“或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物
公开(公告)号：US07632820B2
公开(公告)日：2009-12-15
申请号：US10543638
申请日：2004-01-30
申请人： Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Pierre Jung
发明人： Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Pierre Jung
IPC分类号： A01N43/04 , A61K31/40 , A61K31/335 , A61K31/70 , A61K31/397 , A61K31/445 , A61K31/44 , A01N43/38
CPC分类号： A01N43/90 , C07H17/08
摘要： Disclosed are compounds of the formulain which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —SO2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.
摘要翻译：公开了n为0或1的甲醛化合物; X-Y是-CH-CH-或-CH 2 -CH 2 - ; Z是-C（-O） - ， - C（-S） - 或-SO 2 - ; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R2为R3-Z-，R3-O-Z-，R4或-Z-N（R6）（R7）; Q是O或-N-R5; R 3和R 4例如是H，C 1 -C 12烷基，C 2 -C 12烯基，C 2 -C 12炔基，C 3 -C 12环烷基，C 5 -C 12环烯基，芳基或杂环基; R5是例如H，C1-C8烷基，羟基-C1-C8烷基，C3-C8环烷基，C2-C8链烯基，C2-C8炔基，苯基或苄基; R 6和R 7为例如未取代的或未被取代的一价或五价取代的C 1 -C 12烷基，未被取代的或一至五取代的C 2 -C 12链烯基或（如果合适的话）E / Z异构体，E / Z异构体混合物和/或其互变异构体，在每种情况下以游离形式或盐形式，都可用作农药。

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