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1. 发明授权

US06562810B1 8-substituted-9H-1,3-dioxolo/4,5-h//2,3/benzodiazepine derivatives, as AMPA/kainate receptor inhibitors 失效
标题翻译： 8-取代-9H-1,3-二氧杂环戊烯/ 4,5-h // 2,3 /苯并二氮杂衍生物作为AMPA /红藻氨酸受体抑制剂
公开(公告)号：US06562810B1
公开(公告)日：2003-05-13
申请号：US09485391
申请日：2000-05-19
申请人： László Balázs , József Barkóczy , Imre Domán , András Egyed , Istvän Gacsályi , Gábor Gigler , Zoltán Greff , István Gyertyán , Péter Kótay Nagy , Attila Kovács , György Lávay , Zoltán Rátkai , Péter Seres , Gyula Simig , Annamária Simó , Tamás Szabados , Géza Szabó , Károly Tihanyi , Miklós Végh , Géza Schneider , Judit Cselenyák
发明人： László Balázs , József Barkóczy , Imre Domán , András Egyed , Istvän Gacsályi , Gábor Gigler , Zoltán Greff , István Gyertyán , Péter Kótay Nagy , Attila Kovács , György Lávay , Zoltán Rátkai , Péter Seres , Gyula Simig , Annamária Simó , Tamás Szabados , Géza Szabó , Károly Tihanyi , Miklós Végh , Géza Schneider , Judit Cselenyák
IPC分类号： A61K3155
CPC分类号： C07D491/04
摘要： The disclosure relates to a novel 8-substituted-9H-1,3-dioxolo-[4,5-h][2,3]benzodiazepine compound of formula I and pharmaceutically acceptable quaternary ammonium salts thereof, a process for preparing the same, a pharmaceutical composition containing a 8-substituted-9H-1,3-dioxolo-[4,5-h][2,3]benzodiazepine compound, and a method of treatment using the pharmaceutical composition. A complete description of the compound of formula I is found in the specification. The compounds of the general formula I possess unique competitive AMPA/kainite antagonist properties making them useful in the treatment of diseases where inhibition of the AMPA/kainite receptors may a favorable effect.
摘要翻译：本公开涉及式I的新的8-取代-9,9-1,3-二氧杂 - [4,5-h] [2,3]苯并二氮杂化合物及其药学上可接受的季铵盐，其制备方法，含有8-取代-9,9-1,3-二氧杂 - [4,5-h] [2,3]苯并二氮杂化合物的药物组合物和使用该药物组合物的治疗方法。在说明书中找到了式I化合物的完整描述。通式I的化合物具有独特的竞争性AMPA /卡赛因拮抗剂性质，使其可用于治疗AMPA /卡培酮受体抑制作用的疾病。

2. 发明授权

US07040348B2 Arrangement for a single-grip mixing faucet being operated by turning only 有权
标题翻译：通过转动操作的单把手混合龙头的布置
公开(公告)号：US07040348B2
公开(公告)日：2006-05-09
申请号：US10825222
申请日：2004-04-16
申请人： György Bolgár , Attila Kovács
发明人： György Bolgár , Attila Kovács
IPC分类号： F16K11/074
CPC分类号： F16K11/074 , Y10T137/86823
摘要： The invention relates to a arrangement for single-grip mixing faucets operated by turning only, comprising a fixed inlet disc (11) and a rotating regulation disc (16) arranged above each other forming thereby a plane seal, for regulating the amount and ratio of the cold and hot water flowing through the system. The cold water inlet channel (12) connected to the cold water network and the hot water inlet channel (13) are developed in the fixed inlet disc (11) whereas the cold water flow-through channels (17) and the hot water flow-through channels (18) are developed in the rotating regulation disc (16). The cold water flow-through channel (17) and the hot water flow-through channel (18) are connected to the mixing space (19), which is developed either in the regulation disc (16), or in a turning element (20) being in an operation connection with the regulation disc (16), at the side of the regulation disc (16) opposite to the inlet disc (11). The operating arm (28) is fixed to the turning element (20) at its end opposite to the regulation disc (16).The essence of the arrangement lies in that in the turning element (20) an axial duct (27) is situated leading also through the operating arm (28), one end of which is connected to the mixing space (19), whereas its other end is connected to the duct (30) developed in the armature discharge (29) joined to the turning element (30) above the operating arm (28), which duct (30) is in connection with the discharge outlet (31).
摘要翻译：本发明涉及一种通过仅旋转操作的单把手混合龙头的装置，其包括固定的入口盘（11）和彼此上下布置的旋转调节盘（16），从而形成平面密封件，用于调节冷热水流经系统。连接到冷水网络的冷水入口通道（12）和热水入口通道（13）在固定入口盘（11）中显影，而冷水流通通道（17）和热水流通道通过通道（18）在旋转调节盘（16）中显影。冷水流通通道（17）和热水流通通道（18）连接到在调节盘（16）中或在转动元件（20）中展开的混合空间（19））与调节盘（16）处于与入口盘（11）相对的调节盘（16）侧的操作连接。操作臂（28）在其与调节盘（16）相对的端部处固定到转动元件（20）。该装置的本质在于，在转动元件（20）中，轴向管道（27）也位于通过操作臂（28）的前端，操作臂（28）的一端连接到混合空间（19），而其它的端部连接到与在操作臂（28）上方连接到转动元件（30）的电枢排出口（29）中显影的管道（30）连接，该管道（30）与排出口（31）相连。

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