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1. 发明申请

US20090062518A1 PROCESS FOR PRODUCTION OF GLUCOPYRANOSYLOXYPYRAZOLE DERIVATIVE 有权
标题翻译：生产葡萄糖酰氧基吡唑衍生物的方法
公开(公告)号：US20090062518A1
公开(公告)日：2009-03-05
申请号：US11908693
申请日：2006-03-16
申请人： Kiyoshi Kasai , Tetsuji Ozawa , Nobuhiko Fushimi , Hidetoshi Isawa , Ken Kikuchi , Masahiro Kobayashi , Junichi Sonehara , Minoru Kubota
发明人： Kiyoshi Kasai , Tetsuji Ozawa , Nobuhiko Fushimi , Hidetoshi Isawa , Ken Kikuchi , Masahiro Kobayashi , Junichi Sonehara , Minoru Kubota
IPC分类号： C07H1/00
CPC分类号： C07H17/02
摘要： The present invention relates to a method for preparing the glucopyranosyloxypyrazole derivatives which are useful as agents for the prevention or treatment of a disease associated with hyperglycemia such as diabetes, diabetic complications, obesity or the like.A glucopyranosyloxypyrazole derivative can be easily and efficiently prepared by allowing a benzylpyrazole derivative represented by the general formula: wherein R1, R2, R3, R4 and R5 may be the same or different, for example each of them is a hydrogen atom, a halogen atom or an alkyl, alkoxy, arylmethyloxy group or the like, R6 is an alkyl group, for example R7 is a hydrogen atom or an alkyl, alkoxy, arylmethyloxy group or the like, to react with a compound represented by the general formula: wherein as an example, PG1 is a pivaloyl group or the like, as an example, X1 is a bromine atom or the like, therefore the present invention is extremely useful as a method for preparing pharmaceutical compounds.
摘要翻译：本发明涉及一种制备吡喃葡萄糖氧吡唑衍生物的方法，其可用作预防或治疗与糖尿病，糖尿病并发症，肥胖症等高血糖相关的疾病的药剂。吡喃葡萄糖氧吡唑衍生物可以容易且有效地制备，其中R 1，R 2，R 3，R 4和R 5可以相同或不同，例如氢原子，卤原子或烷基，烷氧基，芳基甲氧基等，R6是烷基，例如R7是氢原子或烷基，烷氧基，芳基甲氧基等，与通式表示的化合物反应：其中作为作为实例，PG1是新戊酰基等，作为实例，X1是溴原子等，因此本发明作为制备药物化合物的方法是非常有用的。

2. 发明授权

US08022192B2 Process for production of glucopyranosyloxypyrazole derivative 有权
标题翻译：吡喃葡萄糖氧吡唑衍生物的制备方法
公开(公告)号：US08022192B2
公开(公告)日：2011-09-20
申请号：US11908693
申请日：2006-03-16
申请人： Kiyoshi Kasai , Tetsuji Ozawa , Nobuhiko Fushimi , Hidetoshi Isawa , Ken Kikuchi , Masahiro Kobayashi , Junichi Sonehara , Minoru Kubota
发明人： Kiyoshi Kasai , Tetsuji Ozawa , Nobuhiko Fushimi , Hidetoshi Isawa , Ken Kikuchi , Masahiro Kobayashi , Junichi Sonehara , Minoru Kubota
IPC分类号： C07H17/02 , A61K31/7056
CPC分类号： C07H17/02
摘要： The present invention relates to a method for preparing the glucopyranosyloxypyrazole derivatives which are useful as agents for the prevention or treatment of a disease associated with hyperglycemia such as diabetes, diabetic complications, obesity or the like. A glucopyranosyloxypyrazole derivative can be easily and efficiently prepared by allowing a benzylpyrazole derivative represented by the general formula: wherein R1, R2, R3, R4 and R5 may be the same or different, for example each of them is a hydrogen atom, a halogen atom or an alkyl, alkoxy, arylmethyloxy group or the like, R6 is an alkyl group, for example R7 is a hydrogen atom or an alkyl, alkoxy, arylmethyloxy group or the like, to react with a compound represented by the general formula: wherein as an example, PG1 is a pivaloyl group or the like, as an example, X1 is a bromine atom or the like, therefore the present invention is extremely useful as a method for preparing pharmaceutical compounds.
摘要翻译：本发明涉及一种制备吡喃葡萄糖氧吡唑衍生物的方法，其可用作预防或治疗与糖尿病，糖尿病并发症，肥胖症等高血糖相关的疾病的药剂。吡喃葡萄糖氧吡唑衍生物可以容易且有效地制备，其中R 1，R 2，R 3，R 4和R 5可以相同或不同，例如氢原子，卤原子或烷基，烷氧基，芳基甲氧基等，R6是烷基，例如R7是氢原子或烷基，烷氧基，芳基甲氧基等，与通式表示的化合物反应：其中作为作为实例，PG1是新戊酰基等，作为实例，X1是溴原子等，因此本发明作为制备药物化合物的方法是非常有用的。

3. 发明申请

US20090030218A1 Method For Producing Aminoalcohol Derivative Having Biphenyl Group 审中-公开
标题翻译：生产具有联苯基团的氨基醇衍生物的方法
公开(公告)号：US20090030218A1
公开(公告)日：2009-01-29
申请号：US11914915
申请日：2006-05-17
申请人： Kiyoshi Kasai , Minoru Kubota , Ritsu Suzuki , Tetsuji Ozawa , Takehiro Ishikawa , Makoto Kobayashi , Junichi Sonehara , Masahiro Kobayashi
发明人： Kiyoshi Kasai , Minoru Kubota , Ritsu Suzuki , Tetsuji Ozawa , Takehiro Ishikawa , Makoto Kobayashi , Junichi Sonehara , Masahiro Kobayashi
IPC分类号： C07D303/40 , C07C69/76 , C07C229/38 , C07C255/00
CPC分类号： C07D303/22 , C07B53/00 , C07C67/08 , C07C67/31 , C07C69/94 , C07C213/06 , C07C253/30 , C07C255/54 , C07C217/22
摘要： The present invention provides an industrial method for preparing aminoalcohol derivatives (I) having a biphenyl group, biphenyloxyacetaldehyde derivatives which are used therefore, preparing methods thereof, and intermediates used for the preparing method.The present invention also provides a preparing method including processes for preparing a 3-substituted biphenylcarboxylic acid derivative represented by the following general formula: by allowing a 3-fluorobiphenylcarboxylic acid derivative prepared from a 3-fluorobiphenylcarbonitrile derivative which can be prepared by allowing a 4-halophenol derivative to react with a 2-fluorobenzonitrile derivative which is substituted by a leaving group at 4-position to react with an organometallic reagent.
摘要翻译：本发明提供了制备具有联苯基的氨基醇衍生物（I）的工业方法，因此使用的联苯氧基乙醛衍生物及其制备方法以及用于制备方法的中间体。本发明还提供了一种制备方法，其包括由以下通式表示的3-取代的联苯基羧酸衍生物的制备方法：通过使由3-氟联苯基腈衍生物制备的3-氟联苯基羧酸衍生物，其可以通过使4- 卤代酚衍生物与在4-位上被离去基团取代的2-氟苄腈衍生物反应，与有机金属试剂反应。

4. 发明授权

US08952428B2 Element isolation structure of a solid-state pickup device 有权
标题翻译：固体拾取装置的元件隔离结构
公开(公告)号：US08952428B2
公开(公告)日：2015-02-10
申请号：US13360356
申请日：2012-01-27
申请人： Masahiro Kobayashi
发明人： Masahiro Kobayashi
IPC分类号： H01L27/148 , H01L27/146
CPC分类号： H01L27/14641 , H01L27/14607 , H01L27/1461 , H01L27/14616
摘要： An N-type semiconductor region and a floating diffusion region are disposed in an active region. A transfer gate electrode for transferring charges from a PD to an FD is disposed on a semiconductor substrate through an insulator. A part of the N-type semiconductor region constituting the PD and a part of the transfer gate electrode are overlapped with each other. A P-type semiconductor region is disposed in the active region. The P-type semiconductor region and the portion overlapped with the transfer gate electrode of the N-type semiconductor region are disposed adjacent to each other in the direction parallel to the interface of the semiconductor substrate and the insulator. The position of the impurity concentration peak of the N-type semiconductor region and the position of the impurity concentration peak of the P-type semiconductor region are different from each other in depth.
摘要翻译： N型半导体区域和浮动扩散区域设置在有源区域中。用于将电荷从PD转移到FD的转移栅电极通过绝缘体设置在半导体衬底上。构成PD的N型半导体区域的一部分和传输栅电极的一部分重叠。 P型半导体区域设置在有源区域中。 P型半导体区域和与N型半导体区域的传输栅电极重叠的部分在与半导体衬底和绝缘体的界面平行的方向上彼此相邻配置。 N型半导体区域的杂质浓度峰的位置和P型半导体区域的杂质浓度峰的位置的深度彼此不同。

5. 发明申请

US20140324310A1 PARKING ASSIST CONTROL APPARATUS AND CONTROL METHOD 有权
标题翻译：停车辅助控制装置和控制方法
公开(公告)号：US20140324310A1
公开(公告)日：2014-10-30
申请号：US13806051
申请日：2011-06-09
申请人： Masahiro Kobayashi , Takuya Inoue , Youji Hamaguchi
发明人： Masahiro Kobayashi , Takuya Inoue , Youji Hamaguchi
IPC分类号： B60W30/06 , B60W30/09
CPC分类号： B62D15/027 , B60K26/021 , B62D15/0285
摘要： A parking assist control apparatus includes an obstacle detector that detects an obstacle around a vehicle; a parking operation assist unit that executes a parking operation assist for preventing a close approach between the obstacle and the vehicle when judges that a distance of the obstacle to the vehicle becomes equal-to or shorter-than a predetermined control start distance; a parking start judgment unit that judges a parking operation; a parking progress judgment unit that judges a parking progress degree during the parking operation judged by the parking start judgment unit; and a parking progress computing unit that reduces an assist control amount by the parking operation assist unit according to the parking progress degree judged by the parking progress judgment unit. According to the parking assist control apparatus, the parking operation assist for the obstacle around the vehicle can be executed more adequately.
摘要翻译：一种停车辅助控制装置，包括：检测车辆周围的障碍物的障碍物检测器; 停车操作辅助单元，当判定所述障碍物与所述车辆的距离变得等于或短于预定控制开始距离时，执行用于防止所述障碍物与所述车辆之间的紧密接近的停车操作辅助; 判断停车操作的停车开始判断单元; 停车进入判断单元，其判断由所述停车开始判断单元判断的停车动作期间的停车进位度; 以及停车进度计算单元，其根据由停车进行判断单元判断的停车进度，减少由停车操作辅助单元进行的辅助控制量。根据停车辅助控制装置，可以更充分地执行对车辆周围的障碍物的驻车操作辅助。

6. 发明授权

US08655549B2 Vehicle driving control apparatus and vehicle driving control method 有权
标题翻译：车辆驾驶控制装置和车辆驾驶控制方法
公开(公告)号：US08655549B2
公开(公告)日：2014-02-18
申请号：US12497787
申请日：2009-07-06
申请人： Yasuhisa Hayakawa , Masahiro Kobayashi , Ko Sato , Shuhei Nishimaki
发明人： Yasuhisa Hayakawa , Masahiro Kobayashi , Ko Sato , Shuhei Nishimaki
IPC分类号： B62D6/00
CPC分类号： B60W30/12 , B60T8/17557 , B60T2201/08 , B60T2201/087 , B60W30/08
摘要： A vehicle driving control apparatus is provided with a lane detecting device, a future position estimating device and a vehicle control device. The lane detecting device detects a lane marker of a lane. The future position estimating device estimates a future transverse position of a host vehicle after a prescribed amount of time. The vehicle control device executes a vehicle control such that a yaw moment is imparted to the host vehicle toward a middle of the lane. The yaw moment is imparted upon determining that the future transverse position is positioned laterally farther toward an outside of the lane from the middle of the lane than a prescribed widthwise lane position that is determined in advance using the lane marker as a reference. The vehicle control device suppresses an impartation of the yaw moment device when a recognition degree of the lane marker is lower than a prescribed value.
摘要翻译：车辆行驶控制装置具备车道检测装置，未来位置估计装置和车辆控制装置。车道检测装置检测车道的车道标记。未来位置估计装置在规定的时间量之后估计本车辆的未来横向位置。车辆控制装置执行车辆控制，使得向主车辆向车道的中心施加横摆力矩。在确定未来横向位置比从预先使用车道标记作为参考确定的规定的宽度方向车道位置横向更远离车道中部的车道中间位置时，赋予偏航力矩。当车道标记的识别度低于规定值时，车辆控制装置抑制偏航力矩装置的赋予。

7. 发明授权

US08577515B2 Vehicle driving assistant and vehicle driving assisting method 有权
标题翻译：车辆驾驶助理和车辆驾驶辅助方法
公开(公告)号：US08577515B2
公开(公告)日：2013-11-05
申请号：US13384017
申请日：2010-07-15
申请人： Masahiro Kobayashi , Yasuhisa Hayakawa , Kou Sato
发明人： Masahiro Kobayashi , Yasuhisa Hayakawa , Kou Sato
IPC分类号： G05D1/00 , G05D3/00 , G06F7/00 , G06F17/00
CPC分类号： B60T8/17558 , B60K2350/1084 , B60T7/22 , B60T2201/08 , B60T2210/32 , B60W30/08 , B60W2550/10 , G08G1/166 , G08G1/167
摘要： A driving assisting system for a vehicle comprises a side obstacle detector configured to detect an obstacle present in an obstacle detection area; an obstacle approach prevention controller configured to implement an obstacle approach prevention control which assists an approach prevention for preventing the vehicle from approaching an obstacle detected by the side obstacle detector; an overtaking state detector configured to detect an overtaking state which is at least one of a first state where the vehicle is overtaking the obstacle detected by the side obstacle detector and a second state where the vehicle is estimated to overtake the obstacle. The overtaking state detector is configured to detect the overtaking state based at least on (i) a distance between the vehicle and the obstacle, (ii) a speed of the vehicle relative to the obstacle, and (iii) a detection angle of the obstacle relative to the vehicle.
摘要翻译：一种用于车辆的驾驶辅助系统，包括：侧障碍物检测器，被配置为检测障碍物检测区域中存在的障碍物; 障碍物进近防止控制器，被配置为实现障碍物进近防止控制，其辅助防止车辆接近由侧面障碍物检测器检测到的障碍物的防止接近; 超车状态检测器，被配置为检测超车状态，所述超车状态是车辆超越侧障碍物检测器检测到的障碍物的第一状态和估计车辆超过障碍物的第二状态中的至少一个。超车状态检测器被配置为至少基于（i）车辆与障碍物之间的距离，（ii）车辆相对于障碍物的速度，以及（iii）障碍物的检测角度来检测超车状态相对于车辆。

8. 发明授权

US08552353B2 Photoelectric conversion apparatus and imaging system using the same 有权
标题翻译：光电转换装置及使用其的成像系统
公开(公告)号：US08552353B2
公开(公告)日：2013-10-08
申请号：US12989556
申请日：2009-05-07
申请人： Masahiro Kobayashi , Yuichiro Yamashita
发明人： Masahiro Kobayashi , Yuichiro Yamashita
IPC分类号： H01L27/146 , H04N5/335
CPC分类号： H01L27/1463 , H01L27/14603 , H01L27/14609 , H01L27/14612 , H01L27/14623 , H04N5/37452 , H04N5/37457
摘要： In a photoelectric conversion apparatus including charge storing portions in its imaging region, isolation regions for the charge storing portions include first isolation portion each having a PN junction, and second isolation portions each having an insulator. A second isolation portion is arranged between a charge storing portion and at least a part of a plurality of transistors.
摘要翻译：在其成像区域中包括电荷存储部分的光电转换装置中，用于电荷存储部分的隔离区域包括每个具有PN结的第一隔离部分和分别具有绝缘体的第二隔离部分。第二隔离部分布置在电荷存储部分和多个晶体管的至少一部分之间。

9. 发明授权

US08525655B2 Vehicle control system 失效
标题翻译：车辆控制系统
公开(公告)号：US08525655B2
公开(公告)日：2013-09-03
申请号：US13056442
申请日：2009-06-04
申请人： Masahiro Kobayashi , Youji Hamaguchi , Takuya Inoue
发明人： Masahiro Kobayashi , Youji Hamaguchi , Takuya Inoue
IPC分类号： B60Q1/00 , G08G1/00 , G01C22/00
CPC分类号： B60T7/22 , B60W30/06 , B60W30/09 , B60W30/095 , B60W30/18036 , B60W50/08 , B60W50/16 , B60W2050/143 , B60W2520/06 , B60W2550/308 , B62D15/0285 , F02D11/04 , G08G1/166
摘要： In the case that a vehicle 1 is making a reverse movement, a control section 4 sets a braking control operation distance according to an angle formed by the vehicle 1's proceeding direction and an extending direction of a road on which an approaching vehicle is traveling. With this, a braking control is implemented at a delayed timing in a scene where the following possibility is high: the driver wishes to end the reverse movement operation as early as possible when a space for allowing the approaching vehicle to pass by is not present at the back of the vehicle 1. Thereby, the cumbersomeness or discomfort which may be felt by the driver with respect to the braking control can be decreased.
摘要翻译：在车辆1进行倒车的情况下，控制部4根据由车辆1的前进方向和接近的车辆行驶的道路的延伸方向形成的角度来设定制动控制操作距离。由此，在以下可能性高的场景中，以延迟的定时进行制动控制：当允许接近的车辆通过的空间不存在时，驾驶员希望尽可能早地结束反向运动操作因此，可以减少驾驶员相对于制动控制可能感觉到的麻烦或不适。

10. 发明授权

US08497654B2 Single phase AC synchronized motor 有权
标题翻译：单相交流同步电动机
公开(公告)号：US08497654B2
公开(公告)日：2013-07-30
申请号：US13105480
申请日：2011-05-11
申请人： Takahiro Sakaguchi , Masahiro Kobayashi
发明人： Takahiro Sakaguchi , Masahiro Kobayashi
IPC分类号： H02P1/46 , H02P6/00
CPC分类号： H02P1/50 , H02P1/465 , H02P6/181 , H02P6/22 , H02P6/26
摘要： There is provided a single-phase AC synchronized motor that does not need smooth of rectifier waves but stably performs shift from a starting operation to a synchronized operation. In the motor, based on detected signals of a position sensor, rectified current is reciprocally flowed to each direction of a single-phase coil which starts the motor. The motor includes a start-up operation circuit with a sensor starting period that increases a rotational speed until reaching to a first predetermined rotational speed; and a control device that controls operation of the motor as that shift to synchronized operation is performed when a rotational speed of a permanent magnetic rotor is reached to a second predetermined rotational speed nearby a synchronized rotational speed but not exceeding the synchronized rotational speed, and when the rise and fall of detected signals of the position sensor and the zero-cross point of AC current are approximately correspondent to each other.
摘要翻译：提供了单相AC同步电动机，其不需要整流波的平滑，而是稳定地执行从启动操作到同步操作的移位。在电动机中，基于位置传感器的检测信号，整流电流往复地流向启动电动机的单相线圈的各个方向。电动机包括具有传感器启动时段的启动操作电路，其增加转速直到达到第一预定转速; 以及当永磁转子的转速达到同步转速附近的第二预定转速而不超过同步转速时，执行转向同步操作的电动机的操作的控制装置，何时位置传感器的检测信号和交流电流的过零点的上升和下降大致对应。

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