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1. 发明申请

US20120238762A1 AZOLE DERIVATIVES AND METHODS FOR PRODUCING THE SAME, INTERMEDIATE COMPOUNDS FOR THE DERIVATIVES AND METHODS FOR PRODUCING THE SAME, AND AGRO-HORTICULTURAL AGENTS AND INDUSTRIAL MATERIAL PROTECTING AGENTS CONTAINING THE DERIVATIVES 审中-公开
标题翻译：衍生物及其制备方法，衍生物的中间体化合物及其制备方法，以及含有衍生物的农业机械和工业材料保护剂
公开(公告)号：US20120238762A1
公开(公告)日：2012-09-20
申请号：US13508337
申请日：2010-11-29
申请人： Keiichi Sudo , Takashi Shimokawara , Eiyu Imai , Nobuyuki Kusano , Hisashi Kanno , Taiji Miyake , Masaru Mori , Toshihide Saishoji
发明人： Keiichi Sudo , Takashi Shimokawara , Eiyu Imai , Nobuyuki Kusano , Hisashi Kanno , Taiji Miyake , Masaru Mori , Toshihide Saishoji
IPC分类号： C07D249/08 , C07D301/02 , C07D303/22 , C07D301/00 , C07D303/04 , C07D303/08
CPC分类号： C07D233/60 , A01N43/50 , A01N43/653 , C07D249/08
摘要： To provide an azole derivative which is contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases. An azole derivative according to the invention is represented by Formula (I), wherein R1 and R2 are same or different, and each denotes a substituted C3-C6 cycloalkyl group or a C1-C4 alkyl group substituted with the substituted C3-C6 cycloalkyl group; and A denotes a nitrogen atom or a methyne group.
摘要翻译：提供在对疾病具有优异控制作用的农业园艺剂中提供作为活性成分含有的唑衍生物。根据本发明的唑衍生物由式（I）表示，其中R 1和R 2相同或不同，并且各自表示取代的C 3 -C 6环烷基或被取代的C 3 -C 6环烷基取代的C 1 -C 4烷基 ; A表示氮原子或甲炔基。

2. 发明授权

US5162356A Azole mycocide and method of treating mycosis 失效
标题翻译：唑类霉菌和治疗真菌病的方法
公开(公告)号：US5162356A
公开(公告)日：1992-11-10
申请号：US666488
申请日：1991-03-06
申请人： Masato Arahira , Toshihide Saishoji , Susumu Ikeda , Satoru Kumazawa
发明人： Masato Arahira , Toshihide Saishoji , Susumu Ikeda , Satoru Kumazawa
IPC分类号： A61K31/415 , A61P31/04 , A61P31/10 , C07D233/60 , C07D233/61 , C07D249/08 , C07D521/00
CPC分类号： C07D231/12 , C07D233/56 , C07D249/08
摘要： Disclosed herein are azole derivatives or the salts thereof which are represented by the general formula (I): ##STR1## wherein X represents a halogen atom, an alkyl group having 1 to 5 carbon atoms, a haloalkyl group, a phenyl group, a cyano group, or a nitro group, Xs being either the same or different from each other; n represents an integer of 1 to 5; A represents a nitrogen atom or CH; and one of R.sub.1 and R.sub.2 represents an alkyl group having 1 to 5 carbon atoms and the other a hydrogen atom or an alkyl group having 1 to 5 carbon atoms, with the proviso that when n is 1 or 2, X does not represent a halogen atom, an alkyl group having 1 to 5 carbon atoms or a phenyl group, and mycocides comprising an effective amount of azole derivative or medically or veterinarily acceptable salt thereof, said azole derivative being represented by the general formula (II): ##STR2## wherein X represents a halogen atom, an alkyl group having 1 to 5 carbon atoms, a haloalkyl group, a phenyl group, a cyano group, or a nitro group, Xs being either the same or different from each other; n represents an integer of 0 to 5; A represents a nitrogen atom or CH; and R.sub.1 and R.sub.2 respectively represent a hydrogen atom or an alkyl group having 1 to 5 carbon atoms, and a diluent or a carrier which is medically or veterinarily acceptable.
摘要翻译：本文公开的是由通式（I）表示的唑衍生物或其盐：其中X表示卤素原子，具有1至5个碳原子的烷基，卤代烷基，苯基，氰基或硝基，Xs彼此相同或不同; n表示1〜5的整数， A表示氮原子或CH; R1和R2之一表示碳原子数为1〜5的烷基，另一个为氢原子或碳原子数为1〜5的烷基，条件是当n为1或2时，X不表示卤素原子，具有1〜5个碳原子的烷基或苯基，以及包含有效量的唑衍生物或其医学上或兽医学上可接受的盐的霉菌，所述唑衍生物由通式（II）表示： II）其中X表示卤素原子，具有1至5个碳原子的烷基，卤代烷基，苯基，氰基或硝基，X可以相同或不同; n表示0〜5的整数， A表示氮原子或CH; R 1和R 2分别表示氢原子或碳原子数1〜5的烷基，以及在医学上或兽医学上可接受的稀释剂或载体。

3. 发明授权

US5010206A Novel azole derivative and agricultural/horticultural fungicide containing said derivative as active ingredient 失效
标题翻译：含有所述衍生物的新型唑衍生物和农/园艺杀真菌剂作为活性成分
公开(公告)号：US5010206A
公开(公告)日：1991-04-23
申请号：US560754
申请日：1990-07-31
申请人： Hiroyuki Enari , Satoru Kumazawa , Susumu Shimizu , Atsushi Ito , Nobuo Sato , Toshihide Saishoji
发明人： Hiroyuki Enari , Satoru Kumazawa , Susumu Shimizu , Atsushi Ito , Nobuo Sato , Toshihide Saishoji
IPC分类号： A01N43/50 , A01N43/653 , C07D233/58 , C07D233/60 , C07D249/08 , C07D521/00
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要： An azole derivative represented by the formula ##STR1## wherein X and Y independently represent a halogen atom, a phenyl group or a hydrogen atom, providing that at least one of X and Y is not a hydrogen atom, n represents an integer of 0, 1 or 2, and A represents a nitrogen atom or CH, and an agricultural/horticultural fungicide comprising the azole derivative as an active ingredient are disclosed.The azole derivative exhibits an excellent effect in preventing and curing a wide spectrum of plant diseases and possesses low toxicity to mammals.

4. 发明授权

US5099029A Azole derivative and agrucultural/horticultural fungicide containing said derivative as active ingredient active ingredient 失效
标题翻译：含有衍生物的农药/农药/杀真菌剂作为主动成分活性成分
公开(公告)号：US5099029A
公开(公告)日：1992-03-24
申请号：US648043
申请日：1991-01-30
申请人： Hiroyuki Enari , Satoru Kumazawa , Susumu Shimizu , Atsushi Ito , Nobuo Sato , Toshihide Saishoji
发明人： Hiroyuki Enari , Satoru Kumazawa , Susumu Shimizu , Atsushi Ito , Nobuo Sato , Toshihide Saishoji
IPC分类号： A01N43/50 , A01N43/653 , C07D233/58 , C07D233/60 , C07D249/08 , C07D521/00
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要： An azole derivative represented by the formula (I): ##STR1## wherein X and Y independently represent a halogen atom, a phenyl group or a hydrogen atom, providing that at least one of X and Y is not a hydrogen atom, n represents an integer of 0, 1 or 2, and A represents a nitrogen atom or CH, and an agricultural/horticultural fungicide comprising the azole derivative as an active ingredient are disclosed.The azole derivative exhibits an excellent effect in preventing and curing a wide spectrum of plant diseases and possesses low toxicity to mammals.

5. 发明授权

US5264450A Imidazole substituted cycloalkanol derivatives and fungicidal compositions containing same 失效
标题翻译：咪唑取代的环烷醇衍生物和含有它的杀真菌组合物
公开(公告)号：US5264450A
公开(公告)日：1993-11-23
申请号：US863007
申请日：1992-04-06
申请人： Atsushi Ito , Toshihide Saishoji , Satoru Kumazawa
发明人： Atsushi Ito , Toshihide Saishoji , Satoru Kumazawa
IPC分类号： A01N43/50 , A01N43/653 , C07C25/18 , C07C45/67 , C07C49/697 , C07C69/757 , C07D303/08 , C07D521/00 , C07D233/60
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07C25/18 , C07C45/676 , C07C49/697 , C07C69/757 , C07D233/56 , C07D249/08 , C07D303/08 , C07C2101/14 , C07C2101/18
摘要： The present invention discloses an azole-substituted cycloalkanol derivative represented by the formula (I) available for agricultural and horticultural fungicide and a process for preparing the same: ##STR1## wherein R.sup.1 represents a lower alkyl group, R.sup.2 represents a hydrogen atom or a lower alkyl group, n is an integer of 1 or 2 and A represents a nitrogen atom or a CH group.
摘要翻译：本发明公开了可用于农业和园艺杀真菌剂的式（I）表示的唑取代的环烷醇衍生物及其制备方法：其中R 1表示低级烷基，R 2表示氢原子或低级烷基，n为1或2的整数，A表示氮原子或CH基。

6. 发明授权

US5159118A Cyclopentanone derivatives 失效
标题翻译：环戊酮衍生物
公开(公告)号：US5159118A
公开(公告)日：1992-10-27
申请号：US691406
申请日：1991-04-25
申请人： Satoru Kumazawa , Susumu Shimizu , Hiroyuki Enari , Atsushi Ito , Susumu Ikeda , Nobuo Sato , Toshihide Saishoji
发明人： Satoru Kumazawa , Susumu Shimizu , Hiroyuki Enari , Atsushi Ito , Susumu Ikeda , Nobuo Sato , Toshihide Saishoji
IPC分类号： A01N43/50 , A01N43/653 , C07C1/00 , C07C13/28 , C07C17/00 , C07C17/26 , C07C25/18 , C07C45/00 , C07C45/67 , C07C49/657 , C07C49/697 , C07C67/00 , C07C69/716 , C07D233/60 , C07D249/08 , C07D303/04 , C07D303/08 , C07D521/00
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07C13/28 , C07C25/18 , C07C45/676 , C07C49/657 , C07C49/697 , C07D233/56 , C07D249/08 , C07D303/04 , C07D303/08
摘要： Disclosed herein are an azole derivative represented by the formula(I): ##STR1## wherein R.sup.1 and R.sup.2 respectively represent a (C.sub.1 -C.sub.5) alkyl group or a hydrogen atom; X represents a halogen atom, a (C.sub.1 -C.sub.5) alkyl group or a phenyl group; n represents an integer of from 0 to 2 and A represents a nitrogen atom or a CH, provided that R.sup.1 is not a hydrogen atom when R.sup.2 is a hydrogen atom, a process for producing the azole derivative represented by the formula(I), and an agricultural and horticultural composition containing the azole derivative represented by the formula(I).
摘要翻译：本文公开的是由式（I）表示的唑衍生物：其中R 1和R 2分别表示（C 1 -C 5）烷基或氢原子; X表示卤素原子，（C1-C5）烷基或苯基; n表示0〜2的整数，A表示氮原子或CH，条件是当R 2为氢原子时，R 1不为氢原子，由式（I）表示的唑衍生物的制造方法，以及含有由式（I）表示的唑衍生物的农业和园艺组合物。

7. 发明授权

US5124345A Triazole substituted cycloalkanol derivative and an agriculturally and horticulturally fungicidal composition comprising the derivatives 失效
标题翻译：三唑取代的环烷醇衍生物和包含衍生物的农业和农业的杀真菌组合物
公开(公告)号：US5124345A
公开(公告)日：1992-06-23
申请号：US550836
申请日：1990-07-10
申请人： Atsushi Ito , Toshihide Saishoji , Satoru Kumazawa
发明人： Atsushi Ito , Toshihide Saishoji , Satoru Kumazawa
IPC分类号： A01N43/50 , A01N43/653 , C07C17/26 , C07C25/06 , C07C25/18 , C07C45/65 , C07C45/67 , C07C49/105 , C07C49/697 , C07C65/24 , C07C69/757 , C07D233/60 , C07D249/08 , C07D303/08 , C07D521/00
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07C25/18 , C07C45/676 , C07C49/697 , C07C69/757 , C07D233/56 , C07D249/08 , C07D303/08 , C07C2101/14 , C07C2101/18
摘要： The present invention discloses an azole-substituted cycloalkanol derivative represented by the formula (I) available for agricultural and horticultural fungicide and a process for preparing the same: ##STR1## wherein R.sup.1 represents a lower alkyl group, R.sup.2 represents a hydrogen atom or a lower alkyl group, n is an integer of 1 or 2 and A represents a nitrogen atom or a CH group.

8. 发明授权

US5095028A 2-(4-chlorobenzyl)-1-(1H-imidazole-1-ylmethyl)-1-cyclohexanol and cycloheptanol 失效
标题翻译： 2-（4-氯苄基）-1-（1H-咪唑-1-基甲基）-1-环己醇和环庚醇
公开(公告)号：US5095028A
公开(公告)日：1992-03-10
申请号：US479436
申请日：1990-02-14
申请人： Atsushi Ito , Satori Kamazawa , Nobuo Sato , Toshihide Saishoji
发明人： Atsushi Ito , Satori Kamazawa , Nobuo Sato , Toshihide Saishoji
IPC分类号： C07D233/60 , C07D521/00
CPC分类号： C07D231/12 , C07D233/56 , C07D249/08
摘要： Disclosed herein are (1) a novel azole-substituted cycloalkanol derivative represented by the formula (I): ##STR1## wherein n is an integer of 1 or 2 and A represents a nitrogen atom or a CH group, (2) an agricultural and horticultural fungicide having said cycloalkanol derivative as an active ingredient, (3) a process for producing said cycloalkanol derivative and (4) several novel intermediate compounds to produce said cycloalkanol derivative.
摘要翻译：本文公开了（1）由式（I）表示的新型唑衍生的环烷醇衍生物：其中n为1或2的整数，A表示氮原子或CH基团，（2）具有所述环烷醇衍生物作为活性成分的农业和园艺杀真菌剂，（3）制备所述环烷醇衍生物的方法和（4）几种新的中间体化合物以制备所述环烷醇衍生物。

9. 发明授权

US4902702A Novel azole derivative and agricultural/horticultural fungicide containing said derivative as active ingredient 失效
标题翻译：含有所述衍生物的新型唑衍生物和农/园艺杀真菌剂作为活性成分
公开(公告)号：US4902702A
公开(公告)日：1990-02-20
申请号：US129629
申请日：1987-12-07
申请人： Hiroyuki Enari , Satoru Kumazawa , Susumu Shimizu , Atsushi Ito , Nobuo Sato , Toshihide Saishoji
发明人： Hiroyuki Enari , Satoru Kumazawa , Susumu Shimizu , Atsushi Ito , Nobuo Sato , Toshihide Saishoji
IPC分类号： A01N43/50 , A01N43/653 , C07D233/58 , C07D233/60 , C07D249/08 , C07D521/00
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要： An azole derivative represented by the formula (I): ##STR1## wherein X and Y independently represent a halogen atom, a phenyl group or a hydrogen atom, providing that at least one of X and Y is not a hydrogen atom, n represents an integer of 0, 1 or 2, and A represents a nitrogen atom or CH, and an agricultural/horticultural fungicide comprising the azole derivative as an active ingredient are disclosed.The azole derivative exhibits an excellent effect in preventing and curing a wide spectrum of plant diseases and possesses low toxicity to mammals.

10. 发明授权

US5504096A Biocidal compositions for industrial materials 失效
标题翻译：用于工业材料的杀生物组合物
公开(公告)号：US5504096A
公开(公告)日：1996-04-02
申请号：US143023
申请日：1993-10-29
申请人： Masato Arahira , Toshihide Saishoji , Katsuhisa Ohsugi , Satoru Kumazawa
发明人： Masato Arahira , Toshihide Saishoji , Katsuhisa Ohsugi , Satoru Kumazawa
IPC分类号： A01N43/50 , A01N43/653 , B27K3/34 , C07D521/00 , C08K5/3445 , C08K5/3472 , C14C9/00 , D21H17/07 , D21H21/36 , A61K31/415
CPC分类号： A01N43/50 , A01N43/653 , C07D231/12 , C07D233/56 , C07D249/08 , C08K5/3445 , C08K5/3472 , C14C9/00 , D21H17/07 , D21H21/36 , B27K3/343 , B27K3/38
摘要： Disclosed herein is a method for preventing deterioration of an industrial material by using an azole derivative represented by the following formula ##STR1## wherein X means a halogen atom or a C.sub.1 -C.sub.5 alkyl, haloalkyl, phenyl, cyano or nitro group, n stands for 0 or an integer of 1-5, A denotes a nitrogen atom or CH, R.sub.1 and R.sub.2 mean individually a hydrogen atom or a C.sub.1 -C.sub.5 alkyl group, R.sub.3 denotes a hydrogen atom or a C.sub.1 -C.sub.3 alkyl group, and when n is an integer of 2-5, Xs may be the same or different. A biocidal composition for the method is also disclosed.
摘要翻译：本文公开了通过使用由下式（I）表示的唑衍生物来防止工业材料劣化的方法：其中X表示卤素原子或C 1 -C 5烷基，卤代烷基，苯基，氰基或硝基，n代表0或1-5的整数，A表示氮原子或CH，R 1和R 2分别表示氢原子或C 1 -C 5烷基，R 3表示氢原子或C 1 -C 3 烷基，当n为2-5的整数时，X可以相同或不同。还公开了该方法的杀生物剂组合物。

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