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1. 发明授权

US4963582A Macrolide compounds, their preparation and their use 失效
标题翻译：大环内酯类化合物，其制备及其用途
公开(公告)号：US4963582A
公开(公告)日：1990-10-16
申请号：US30217
申请日：1987-03-24
申请人： Kazuo Sato , Toshiaki Yanai , Takao Kinoto , Keiji Tanaka , Akira Nishida , Toshimitsu Toyama , Bruno Frei , Anthony O'Sullivan
发明人： Kazuo Sato , Toshiaki Yanai , Takao Kinoto , Keiji Tanaka , Akira Nishida , Toshimitsu Toyama , Bruno Frei , Anthony O'Sullivan
IPC分类号： A01N43/90 , A01N47/06 , A01P5/00 , A01P7/02 , A01P7/04 , A61K31/365 , C07D493/22 , C07H19/01
CPC分类号： C07D493/22 , A01N43/90 , A01N47/06 , C07H19/01
摘要： Compounds having a 16-membered macrolide ring, and related to the milbemycins and avermectins, with substituents at positions 5, 13, 25 and optionally also 23, have acaricidal, insecticidal and anthelmintic properties. They are useful for treating various pests in plants and animals.

2. 发明授权

US5405867A Macrolide compounds, their preparation and their use 失效
标题翻译：大环内酯类化合物，其制备及其用途
公开(公告)号：US5405867A
公开(公告)日：1995-04-11
申请号：US133776
申请日：1993-10-08
申请人： Kazuo Sato , Toshiaki Yanai , Takao Kinoto , Keiji Tanaka , Akira Nishida , Toshimitsu Toyama , Bruno Frei , Anthony O'Sullivan
发明人： Kazuo Sato , Toshiaki Yanai , Takao Kinoto , Keiji Tanaka , Akira Nishida , Toshimitsu Toyama , Bruno Frei , Anthony O'Sullivan
IPC分类号： A01N43/90 , A01N47/06 , A01P5/00 , A01P7/02 , A01P7/04 , A61K31/365 , C07D493/22 , C07H19/01 , C07D313/00
CPC分类号： C07D493/22 , A01N43/90 , A01N47/06 , C07H19/01
摘要： Compounds having a 16-membered macrolide ring, and related to the milbemycins and avermectins, with substituents at positions 5.13, 25 and optionally also 23, have acaricidal, insecticidal and anthelmintic properties. They are useful for treating various pests in plants and animals.
摘要翻译：具有16位大环内酯环，与米尔倍霉素和阿凡曼菌素相关的化合物，其具有位置5.13,25和任选地23的取代基具有杀螨，杀虫和驱虫性质。它们可用于处理植物和动物中的各种害虫。

3. 发明授权

US4945105A 13-Halomilbemycin derivatives, their preparation and compositions containing them 失效
标题翻译： 13-哈美列霉素衍生物，其制备方法和含有它们的组合物
公开(公告)号：US4945105A
公开(公告)日：1990-07-31
申请号：US290835
申请日：1988-12-28
申请人： Kazuo Sato , Toshiaki Yanai , Noritoshi Kitano , Akira Nishida , Bruno Frei , Anthony O'Sullivan
发明人： Kazuo Sato , Toshiaki Yanai , Noritoshi Kitano , Akira Nishida , Bruno Frei , Anthony O'Sullivan
IPC分类号： C07D493/22 , A01N43/90 , A01P5/00 , A01P7/02 , A01P7/04 , A61K31/365 , A61P33/10 , C07D307/00 , C07D309/00 , C07H19/01
CPC分类号： C07H19/01 , A01N43/90
摘要： Derivatives of milbemycins D, A.sub.3 and A.sub.4 and of the corresponding sec-butyl compound have a halogen atom at the 13-position; at the 5-position, they have an oxygen (keto) atom, an oxime group or a substituted oxime group. They may be prepared from known compounds by any appropriate combination of halogenation, ketonization and oximation.
摘要翻译：米尔倍霉素D，A3和A4及相应的仲丁基化合物的衍生物在13位具有卤素原子; 在5位，它们具有氧（酮）原子，肟基或取代的肟基。它们可以通过卤化，酮化和肟化的任何适当组合由已知化合物制备。

4. 发明申请

US20060105970A1 Avermectins substituted in the 4"-position having pesticidal properties 有权
标题翻译：在4“位置取代的阿维菌素具有杀虫特性
公开(公告)号：US20060105970A1
公开(公告)日：2006-05-18
申请号：US11319686
申请日：2005-12-28
申请人： Thomas Pitterna , Anthony O'Sullivan , William Lutz
发明人： Thomas Pitterna , Anthony O'Sullivan , William Lutz
IPC分类号： A01N43/04 , C07H17/08
CPC分类号： C07H19/01 , A01N43/90 , A01N47/12 , A01N47/14 , A01N47/28 , A01N47/30 , A01N47/32
摘要： What is described are a compound of the formula in which R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 is H, unsubstituted or mono- to pentasubstituted C1-C12alkyl or unsubstituted or mono-to pentasubstituted C1-C12alkenyl; R3 is C2-C12alkyl, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C1-C6alkoxy-C1-C6alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl, C2-C12alkenyl, C2-C12alkynyl; or R2 and R3 together are an alkylene or alkenylene bridge; with the proviso that R1 is not sec-butyl or isopropyl if R2 is H and R3 is 2-hydroxyethyl, isopropyl, n-octyl or benzyl;or, if appropriate, in E/Z isomer, an E/Z isomer mixture and/or a tautomer thereof; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中R 1是C 1 -C 12 -C 12烷基，C 3〜 C 1 -C 8环烷基或C 2 -C 12 - 烯基; R 2是H，未取代的或一至五取代的C 1 -C 12烷基或未被取代的或单取代或单取代的C 1 C 12 -C 12烯基; R 3是C 2 -C 12烷基，一至五取代C 1 -C 12烷基，C 1 -C 12烷基，C 1 -C 12烷基，未取代的或一至五取代的C 1 -C 6烷氧基-C 1 -C 6烷基，未取代的或一至五取代的C 3 -C 12环烷基，C 2 -C 12烷基，烯基，C 2 -C 12炔基; 或R 2和R 3一起是亚烷基或亚烯基桥; 条件是R 1不是仲丁基或异丙基，如果R 2是H，R 3是2-羟乙基，异丙基，n 辛基或苄基;或如果合适，在E / Z异构体中，E / Z异构体混合物和/或其互变异构体; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

5. 发明申请

US20080076920A1 PREPARATION OF THIAZOLES 失效
标题翻译：制备THIAZOLES
公开(公告)号：US20080076920A1
公开(公告)日：2008-03-27
申请号：US11947891
申请日：2007-11-30
申请人： Thomas Pitterna , Henry Szczepanski , Peter Maienfisch , Ottmar Huter , Thomas Rapold , Marcel Senn , Thomas Gobel , Anthony O'Sullivan
发明人： Thomas Pitterna , Henry Szczepanski , Peter Maienfisch , Ottmar Huter , Thomas Rapold , Marcel Senn , Thomas Gobel , Anthony O'Sullivan
IPC分类号： C07D417/02 , C07D277/36 , C07D417/14
CPC分类号： C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74
摘要： The present disclosure is directed to a process for the preparation of a compound having the formula: wherein R is unsubstituted or substituted C1-C12alkyl, unsubstituted or substituted C2-C4alkenyl, unsubstituted or substituted C2-C4alkynyl, unsubstituted or substituted C3-C6cycloalkyl, unsubstituted or substituted aryl, unsubstituted or substituted heteroaryl, or —SR1; R1 is unsubstituted or substituted C1-C12alkyl, unsubstituted or substituted C2-C4alkenyl, unsubstituted or substituted C2-C4alkynyl, unsubstituted or substituted cycloalkyl, unsubstituted or substituted aryl or unsubstituted or substituted heteroaryl; and X is a selected leaving group that is not halogen, and may specifically be methylsulfonate, trifluoromethylsulfonate, and p-toluenesulfonate. These compounds are valuable intermediates useful in the synthesis of compounds having pesticidal activity. Generally, the process includes reacting a water-removing reagent, with a compound having the formula Water-removing agents that may be used include thionyl chloride (SOCl2), thionyl bromide (SOBr2), phosphorus oxychloride (POCl3), phosphorus oxybromide (POBr3), phosphorus pentachloride or a sulfonic acid chloride or bromide.
摘要翻译：本公开涉及制备具有下式的化合物的方法：其中R是未取代或取代的C 1 -C 12烷基，未取代或取代的C 1 -C 12烷基，未取代或取代的C 2 -C 4炔基，未取代或取代的C 1 -C 4烷基， 3个C 6环烷基，未取代或取代的芳基，未取代或取代的杂芳基或-SR 1 N; R 1是未取代或取代的C 1 -C 12烷基，未取代或取代的C 2 -C 3 未取代或取代的C 2 -C 4炔基，未取代或取代的环烷基，未取代或取代的芳基或未取代或取代的杂芳基; X是不是卤素的选择的离去基团，可以具体为甲基磺酸酯，三氟甲基磺酸酯和对甲苯磺酸酯。这些化合物是有用的合成具有杀虫活性的化合物的中间体。通常，该方法包括使除水试剂与具有式的化合物反应可以使用的除水剂包括亚硫酰氯（SOCl 2/2），亚硫酰溴（SO 2 R 2）（POCl 3 3），三溴氧化磷（POBr 3 N），五氯化磷或磺酰氯或溴化物。

6. 发明授权

US07601743B2 Cyano anthranilamide insecticides 失效
标题翻译：氰基邻氨基苯甲酰胺杀虫剂
公开(公告)号：US07601743B2
公开(公告)日：2009-10-13
申请号：US11911887
申请日：2006-04-18
申请人： Andre Jeanguenat , Anthony O'Sullivan , Michael Muehlebach , Stephan Trah , Roger Graham Hall
发明人： Andre Jeanguenat , Anthony O'Sullivan , Michael Muehlebach , Stephan Trah , Roger Graham Hall
IPC分类号： C07D401/04 , A61K31/4439
CPC分类号： A01N43/56 , C07D401/04
摘要： Compounds of formula (I) wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula I can be used as agrochemical active ingredients and can be prepared in a manner known per se.
摘要翻译：其中取代基如权利要求1中所定义的式（I）化合物和式I化合物的农业化学可接受的盐和所有立体异构体和互变异构体形式可用作农业化学活性成分，并且可以以本身已知的方式制备。

7. 发明授权

US07323564B2 Preparation of thiazoles 失效
标题翻译：噻唑的制备
公开(公告)号：US07323564B2
公开(公告)日：2008-01-29
申请号：US11552255
申请日：2006-10-24
申请人： Thomas Pitterna , Henry Szczepanski , Peter Maienfisch , Ottmar Franz Huter , Thomas Rapold , Marcel Senn , Thomas Gobel , Anthony O'Sullivan
发明人： Thomas Pitterna , Henry Szczepanski , Peter Maienfisch , Ottmar Franz Huter , Thomas Rapold , Marcel Senn , Thomas Gobel , Anthony O'Sullivan
IPC分类号： C07D413/14 , C07D277/74 , C07D277/36
CPC分类号： C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74
摘要： The present invention is directed to a process for preparing a compound having the formula: wherein R is a range of organic groups and X is a leaving group. The process may include reacting a compound of the formula with a water-removing reagent. Also, when X is a halogen, the process may include reacting a compound of the formula with a halogenating agent or a sulfonylating agent. Alternatively, when X is a halogen, the process may be carried out by reacting a compound of the formula IV where R2 and R3 are defined organic groups with a compound of the formula halogen-C(—O)—O—C1 -C8alkyl, halogen-C(—O)—O-aryl or halogen-C(—O)—O-benzyl.
摘要翻译：本发明涉及制备具有下式的化合物的方法：其中R是有机基团的范围，X是离去基团。该方法可以包括使式的化合物与除水试剂反应。此外，当X是卤素时，该方法可以包括使式的化合物与卤化剂或磺酰化剂反应。或者，当X是卤素时，该方法可以通过使式IV化合物（其中R 2和R 3定义为有机基团）与化合物式中卤素-C（-O）-O-C 1 -C 8烷基，卤素-C（-O）-O-芳基或卤素-C（ - ） - O-苄基。

8. 发明申请

US20080182750A1 Cyano Anthranilamide Insecticides 失效
标题翻译：氰基邻氨基苯甲酰胺杀虫剂
公开(公告)号：US20080182750A1
公开(公告)日：2008-07-31
申请号：US11911887
申请日：2006-04-18
申请人： Andre Jeanguenat , Anthony O'Sullivan , Michel Muehlebach , Stephan Trah , Roger Graham Hall
发明人： Andre Jeanguenat , Anthony O'Sullivan , Michel Muehlebach , Stephan Trah , Roger Graham Hall
IPC分类号： A01N43/40 , C07D401/04 , A01P7/04
CPC分类号： A01N43/56 , C07D401/04
摘要： Compounds of formula (I) wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula I can be used as agrochemical active ingredients and can be prepared in a manner known per se.
摘要翻译：其中取代基如权利要求1中所定义的式（I）化合物和式I化合物的农业化学可接受的盐和所有立体异构体和互变异构体形式可用作农业化学活性成分，并且可以以本身已知的方式制备。

9. 发明申请

US20070055063A1 PREPARATION OF THIAZOLES 失效
标题翻译：制备THIAZOLES
公开(公告)号：US20070055063A1
公开(公告)日：2007-03-08
申请号：US11552255
申请日：2006-10-24
申请人： Thomas Pitterna , Henry Szczepanski , Peter Maienfisch , Ottmar Huter , Thomas Rapold , Marcel Senn , Thomas Gobel , Anthony O'Sullivan
发明人： Thomas Pitterna , Henry Szczepanski , Peter Maienfisch , Ottmar Huter , Thomas Rapold , Marcel Senn , Thomas Gobel , Anthony O'Sullivan
IPC分类号： C07D417/02
CPC分类号： C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74
摘要： A process for the preparation of a compound of the formula and, where applicable, its E/Z-isomers, mixtures of E/Z-isomers and/or tautomers and acid addition products thereof, in each case in free form or in salt form, wherein: R is unsubstituted or substituted C1-C12alkyl, unsubstituted or substituted C2-C4alkenyl, unsubstituted or substituted C2-C4alkynyl, unsubstituted or substituted C3-C6cycloalkyl, unsubstituted or substituted aryl, unsubstituted or substituted heteroaryl, or —SR1; R1 is unsubstituted or substituted C1-C12alkyl, unsubstituted or substituted C2-C4alkenyl, unsubstituted or substituted C2-C4alkynyl, unsubstituted or substituted cycloalkyl, unsubstituted or substituted aryl or unsubstituted or substituted heteroaryl; and X is a leaving group; The process comprises reacting a compound of the formula: with a halogenating agent or a sulfonylating agent. Alternatively, when X is a selected halogen, the process can comprise reacting a compound of the formula with a compound having a formula selected from the group consisting of halogen-C(═O)—O—C1-C8alkyl; halogen-C(═O)—O-aryl; and halogen-C(═O)—O-benzyl.
摘要翻译：制备下式化合物及其E / Z-异构体的方法，E / Z-异构体和/或互变异构体的混合物及其酸加成产物，各自为游离形式或盐形式，其中：R是未取代或取代的C 1 -C 12烷基，未取代或取代的C 2 -C 4 烯基，未取代或取代的C 2 -C 4炔基，未取代或取代的C 3 -C 6环烷基，未取代或取代的芳基，未取代或取代的杂芳基或-SR 1 N; R 1是未取代或取代的C 1 -C 12烷基，未取代或取代的C 2 -C 3 未取代或取代的C 2 -C 4炔基，未取代或取代的环烷基，未取代或取代的芳基或未取代或取代的杂芳基; X为离去群; 该方法包括使下式化合物与卤化剂或磺酰化剂反应。或者，当X是选择的卤素时，该方法可以包括使下式的化合物与具有选自以下的式的化合物反应：卤素-C（ - ） - O-C 1 -C 烷基; 卤素-C（ - ） - O-芳基; 和卤素-C（ - ） - O-苄基。

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