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1. 发明授权

US4692527A 2-amino-3,5-di-(halomethyl)-pyrazines and their preparation 失效
标题翻译： 2-氨基-3,5-二（卤代甲基） - 吡嗪及其制备方法
公开(公告)号：US4692527A
公开(公告)日：1987-09-08
申请号：US776460
申请日：1985-09-16
申请人： Hartmut Leininger , Wolfgang Littmann , Joachim Paust , Walter Trautmann
发明人： Hartmut Leininger , Wolfgang Littmann , Joachim Paust , Walter Trautmann
IPC分类号： C07D241/20 , C07D403/04
CPC分类号： C07D403/04 , C07D241/20 , Y02P20/55
摘要： 2-Amino-3,5-di-(halomethyl)-pyrazines of the general formula I ##STR1## where X is either chlorine or bromine, m and n may each be 0, 1, 2 or 3 and R.sup.1 and R.sup.2 are each hydrogen or a protective group or may furthermore be bonded to one another, in particular those compounds of the formula I in which m is 1 and n is 2 and/or R.sup.1 and R.sup.2 together form a phthaloyl radical, are useful intermediates for the pteridine building block of folic acid or folic acid analogs.They are obtained by a method in which a 2-amino-3,5-dimethylpyrazine of the general formula II ##STR2## is treated with a chlorinating or brominating agent and, where R.sup.1 and/or R.sup.2 are protective groups, these are, if desired, eliminated when the chlorination or bromination is complete.
摘要翻译：其中X是氯或溴，m和n的通式I（I）的2-氨基-3,5-二（卤代甲基） - 吡嗪可以各自为0,1,2或3，R1和 R2各自为氢或保护基，或者还可以彼此键合，特别是其中m为1且n为2的式I化合物和/或R 1和R 2一起形成邻苯二甲酰基的有用的中间体叶酸或叶酸类似物的蝶啶结构单元。它们是通过一种方法获得的，其中通式II的2-氨基-3,5-二甲基吡嗪用氯化或溴化剂处理，其中R 1和/或R 2是保护基，这些如果需要，当氯化或溴化完成时，它们被消除。

2. 发明授权

US4725689A Preparation of 2-amino-3-cyano-5-dialkoxymethylpyrazines and intermediates for this method 失效
标题翻译： 2-氨基-3-氰基-5-二烷氧基甲基吡嗪的制备及其制备方法
公开(公告)号：US4725689A
公开(公告)日：1988-02-16
申请号：US776462
申请日：1985-09-16
申请人： Hartmut Leininger , Wolfgang Littmann , Joachim Paust
发明人： Hartmut Leininger , Wolfgang Littmann , Joachim Paust
IPC分类号： C07D241/20 , C07D241/26 , C07D403/04 , C07D475/04
CPC分类号： C07D403/04 , C07D241/20 , C07D241/26 , Y02P20/55
摘要： 2-Amino-3-cyano-5-dialkoxymethylpyrazine derivatives of the general formula III ##STR1## where R.sup.1 and R.sup.2 are each hydrogen or a protective group usually employed for amino groups and R.sup.5 and R.sup.6 are each alkyl of 1 to 4 carbon atoms, or together form an ethylene or propylene radical which is unsubstituted or substituted by methyl, are prepared starting from a novel 3-halomethyl-5-dihalomethyl-2-aminopyrazine derivative of the formula IV ##STR2## where X is Cl or Br, via a novel intermediate of the general formula I ##STR3## where R.sup.3 is --CH.sub.2 --O--CO--CH.sub.3 (a), --CH.sub.2 OH (b), ##STR4## or --C.tbd.N (d) and R.sup.4 is --CHCl.sub.2 or --CHBr.sub.2 or, where R.sup.1 and R.sup.2 are each a protective group, R.sup.4 may furthermore be ##STR5##The compounds according to the invention are useful intermediates for the preparation of folic acid and active compounds derived from this.
摘要翻译：通式III（III）的2-氨基-3-氰基-5-二烷氧基甲基吡嗪衍生物其中R 1和R 2各自为氢或通常用于氨基的保护基，R 5和R 6各自为1-4的烷基碳原子，或一起形成未被取代或被甲基取代的乙烯或丙烯基团，由式IV（IV）的新型3-卤代甲基-5-二卤代甲基-2-氨基吡嗪衍生物制备，其中X为 Cl或Br通过通式I的新型中间体（I），其中R 3是-CH 2 -O-CO-CH 3（a），-CH 2 OH（b），（c）或-C 3 N（d）和R4是-CHCl 2或-CHBr 2，或者其中R 1和R 2各自是保护基，R 4还可以是本发明的化合物是用于制备叶酸和活性化合物的有用中间体由此。

3. 发明授权

US4806686A Preparation of ribitylxylidine 失效
标题翻译：核苷酸的制备
公开(公告)号：US4806686A
公开(公告)日：1989-02-21
申请号：US042823
申请日：1987-04-27
申请人： Hansgeorg Ernst , Hartmut Leininger , Joachim Paust
发明人： Hansgeorg Ernst , Hartmut Leininger , Joachim Paust
IPC分类号： C07B61/00 , B01J25/00 , B01J25/02 , C07C67/00 , C07C213/00 , C07C213/02 , C07C215/10 , C07C215/16 , C07H5/04 , C07C85/02
CPC分类号： C07H5/04
摘要： N-(D)-ribitylxylidine (I) is prepared by reacting (D)-ribose (II) with 3,4-dimethylaniline (III) or 3,4-dimethyl-1-nitrobenzene (IV) in aqueous or aqueous/organic solution or in solution in a water-soluble organic solvent under an elevated hydrogen pressure and in the presence of a hydrogenation catalyst and of a boric acid compound,(a) using the boric acid compound in a catalytic amount of from about 6 to 35 mmol, preferably from 6 to 20 mmol, per mol of ribose,(b) carrying out the reaction under a hydrogen pressure of from 1 to 20, preferably from 2 to 9, bar and(c) carrying out the hydrogenation at from 40.degree. to 80.degree. C. over Raney nickel as hydrogenation catalyst.
摘要翻译：通过（D） - 核糖（II）与3,4-二甲基苯胺（III）或3,4-二甲基-1-硝基苯（IV）的水溶液或水/有机物（I）反应制备N-（D） - 二硫代吗啉溶液或在水溶性有机溶剂中的溶液中，在升高的氢气压力下和在氢化催化剂和硼酸化合物的存在下，（a）使用催化量的约6至35mmol的硼酸化合物，优选6至20mmol，每摩尔核糖，（b）在1至20，优选2至9巴的氢气压力下进行反应，和（c）在40℃至40℃进行氢化 80℃，以阮内镍为加氢催化剂。

4. 发明授权

US4503238A Preparation of dihydro-4,4-dimethylfuran-2,3-dione 失效
标题翻译：二氢-4,4-二甲基呋喃-2,3-二酮的制备
公开(公告)号：US4503238A
公开(公告)日：1985-03-05
申请号：US552389
申请日：1983-11-16
申请人： Joachim Paust , Hartmut Leininger
发明人： Joachim Paust , Hartmut Leininger
IPC分类号： C07D307/33 , C07D307/60
CPC分类号： C07D307/60
摘要： Dihydro-4,4-dimethylfuran-2,3-dione is prepared by oxidation of racemic dihydro-3-hydroxy-4,4-dimethyl-2(3H)-furanone by a process in which the oxidation is carried out by gradually adding powdered calcium oxide to a solution of racemic dihydro-3-hydroxy-4,4-dimethyl-2(3H)-furanone and chlorine in the inert organic solvent.
摘要翻译：通过外消旋二氢-3-羟基-4,4-二甲基-2（3H） - 呋喃酮氧化制备二氢-4,4-二甲基呋喃-2,3-二酮，其中氧化通过逐渐加入将粉末状氧化钙加到外消旋的二氢-3-羟基-4,4-二甲基-2（3H） - 呋喃酮和氯在惰性有机溶剂中的溶液中。

5. 发明申请

US20120114727A1 INSECTICIDAL SHEET-LIKE STRUCTURE FOR PROTECTING HUMANS AND DOMESTIC ANIMALS 审中-公开
标题翻译：用于保护人体和国内动物的杀虫面板结构
公开(公告)号：US20120114727A1
公开(公告)日：2012-05-10
申请号：US13382711
申请日：2010-07-05
申请人： Hartmut Leininger , Susanne Stutz , Ulrich Karl
发明人： Hartmut Leininger , Susanne Stutz , Ulrich Karl
IPC分类号： A01N43/36 , A01P7/04 , A01N25/08
CPC分类号： A01N43/36 , A01N43/56 , A01N53/00 , C08G18/6266 , C08G18/792 , D01F1/10 , D06M13/395 , D06M15/263 , D06M15/285 , D06M15/29 , D06M15/31 , D06M15/643 , D06M16/00 , D21H21/36 , A01N25/34 , A01N2300/00
摘要： A sheet-like structure, in particular a net, finished with an insecticidal mixture comprising a) chlorfenapyr and b) one or more pyrethroids from the group consisting of alpha-cypermethrin (b1), deltamethrin (b2), permethrin (b3) and lambda-cyhalothrin (b4), in an amount of (in each case relative to the sheet-like structure) a) 50 to 150 mg/m2 chlorfenapyr; b1) 50 to 150 mg/m2 alpha-cypermethrin; b2) 15 to 45 mg/m2 deltamethrin; b3) 50 to 750 mg/m2 permethrin; b4) 5 to 30 mg/m2 lambda-cyhalothrin, is suitable for controlling harmful insects in buildings and for protecting humans and domestic animals from such harmful insects and from vector-transmitted diseases which are transmitted by the harmful insects.
摘要翻译：具有杀虫混合物的片状结构，特别是一种杀虫混合物，其包含a）chlorfenapyr和b）一种或多种来自由α-氯氰菊酯（b1），溴氰菊酯（b2），氯菊酯（b3）和λ - 氯沙芬（b4），其量（在每种情况下相对于片状结构）a）50至150mg / m 2氯芬太尼; b1）50〜150mg / m2α-氯氰菊酯; b2）15〜45mg / m2溴氰菊酯; b3）50〜750mg / m2氯菊酯; b4）5〜30mg / m2λ-氯氟氰菊酯，适用于防治建筑物中的有害昆虫，并保护人类和家畜免受有害昆虫和由有害昆虫传播的载体传播疾病。

6. 发明申请

US20110089075A1 METHOD FOR COATING GLASS, POLYETHYLENE OR POLYESTER CONTAINERS, AND SUITABLE AQUEOUS FORMULATIONS FOR SAID COATING METHOD 审中-公开
标题翻译：用于涂覆玻璃，聚乙烯或聚酯容器的方法，以及用于涂覆方法的适用的水性配方
公开(公告)号：US20110089075A1
公开(公告)日：2011-04-21
申请号：US12992391
申请日：2009-05-11
申请人： Heike Pfistner , Hartmut Leininger , Bernd Düttra , Petra Neumann , Nicole Klöden
发明人： Heike Pfistner , Hartmut Leininger , Bernd Düttra , Petra Neumann , Nicole Klöden
IPC分类号： B65D79/00 , B05D1/18 , B05D1/02 , B32B1/02 , C09D191/06
CPC分类号： C09D123/0884 , C08K5/17 , C08K5/5205 , C08K5/521 , C09D123/0869 , Y10T428/1352 , C08L2666/02
摘要： A method of coating containers made of glass, polyethylene or polyester by treatment with a substantially paraffin-free aqueous formulation comprising (A) at least one acid-functional waxy copolymer selected from (A1) partially oxidized polyethylene waxes having an acid number in the range from 10 to 100 mg KOH/g, determined in accordance with DIN 53402, with (A2) copolymers having a melt flow rate (MFR) in the range from 1 to 50 g/10 min, measured at 160° C. under a load of 325 g in accordance with EN ISO 1133, which in copolymerized form comprise (a) 60% to 88% by weight of ethylene, (b) 12% to 40% by weight of at least one ethylenically unsaturated carboxylic acid, and which are at least partially neutralized with alkali metal or amine, (B) if desired, at least one nonionic or anionic surfactant, (C) if desired, at least one defoamer, (D) if desired, at least one organic amine, (E) if desired, at least one organic solvent.
摘要翻译：一种涂覆由玻璃，聚乙烯或聚酯制成的容器的方法，用基本上无石蜡的水性制剂处理，其包含（A）至少一种选自（A1）部分氧化的聚乙烯蜡的酸官能的蜡质共聚物，其酸值在该范围内根据DIN 53402测定的10至100mg KOH / g，其中（A2）共聚物的熔体流动速率（MFR）在1至50g / 10min的范围内，在160℃下在负载下测量根据EN ISO 1133，其共聚形式包含（a）60重量％至88重量％的乙烯，（b）12重量％至40重量％的至少一种烯键式不饱和羧酸，其为至少部分用碱金属或胺中和，（B）如果需要，至少一种非离子或阴离子表面活性剂，（C）如果需要，至少一种消泡剂，（D）如果需要，至少一种有机胺，（E）如果需要，至少一种有机溶剂。

7. 发明授权

US09288978B2 Insecticide-impregnated nets and use thereof for protecting against pests 有权
标题翻译：杀虫剂浸渍网及其用于防止害虫的用途
公开(公告)号：US09288978B2
公开(公告)日：2016-03-22
申请号：US13055555
申请日：2009-07-27
申请人： Ulrich Karl , Susanne Stutz , Hartmut Leininger , Claus Kaiser
发明人： Ulrich Karl , Susanne Stutz , Hartmut Leininger , Claus Kaiser
IPC分类号： A01G13/02 , A01N25/34
CPC分类号： A01N25/34 , Y10T29/49826 , A01N53/00 , A01N2300/00
摘要： Insecticide-impregnated nets made of textile fibers, which nets have a small mesh size, and their use for the protection against pests.
摘要翻译：由网织物尺寸小的纺织纤维制成的杀虫剂浸渍网及其用于防止害虫的用途。

8. 发明申请

US20120114726A1 INSECTICIDE-COATED SUBSTRATE FOR PROTECTING HUMANS AND PETS 审中-公开
标题翻译：用于保护人体和皮肤的杀虫剂涂层基材
公开(公告)号：US20120114726A1
公开(公告)日：2012-05-10
申请号：US13382694
申请日：2010-07-05
申请人： Hartmut Leininger , Susanne Stutz , Ulrich Karl
发明人： Hartmut Leininger , Susanne Stutz , Ulrich Karl
IPC分类号： A01N43/36 , A01N25/08 , A01P7/04
CPC分类号： D06M16/00 , A01N25/10 , A01N25/34 , A01N53/00 , D06M15/263 , D06M15/285 , A01N43/36 , A01N2300/00
摘要： A substrate treated with a composition comprising a pyrethroid, chlorfenapyr and a special acrylate binder is suitable for controlling harmful insects in buildings, for protecting humans and domestic animals from such harmful insects and for protecting humans and domestic animals from vector-transmitted diseases which are transmitted by the harmful insects.
摘要翻译：用包含拟除虫菊酯，chlorfenapyr和特殊丙烯酸酯粘合剂的组合物处理的底物适于控制建筑物中的有害昆虫，用于保护人类和家畜免受这种有害昆虫的伤害，并保护人和家畜免受所传播的传染病由有害昆虫。

9. 发明申请

US20080194706A1 Modified Open-Cell Foams and Method for Production Thereof 审中-公开
标题翻译：改性开孔泡沫及其制备方法
公开(公告)号：US20080194706A1
公开(公告)日：2008-08-14
申请号：US11720289
申请日：2005-11-26
申请人： Ulrich Karl , Stefan Frenzel , Volker Schwendemann , Ulrich Steinbrenner , Hartmut Leininger
发明人： Ulrich Karl , Stefan Frenzel , Volker Schwendemann , Ulrich Steinbrenner , Hartmut Leininger
IPC分类号： C08J9/30 , A01P1/00 , A61K8/72 , C11D3/37
CPC分类号： C08J9/40 , C08J9/405 , C08J2205/05
摘要： Modified open-cell foams and method for the production thereofProcess for production of modified open-cell foams, which comprises bringing the following materials into contact (a) open-cell foams with density in the range from 5 to 500 kg/m3 and average pore diameter in the range from 1 μm to 1 mm, and (b) aqueous formulation of at least one compound having at least one hemiaminal or aminal group per molecule, or at least one copolymer comprising at least one copolymerized OH-containing or β-dicarbonyl-containing or epoxy-containing comonomer.
摘要翻译：改性开孔泡沫及其制备方法生产改性开孔泡沫的方法，其包括使以下材料接触（a）密度为5至500kg / m 2的开孔泡沫 > 3和平均孔径在1μm至1mm的范围内，和（b）每分子具有至少一个半缩醛基或亚胺基的至少一种化合物的水性制剂，或至少一种共聚物，至少包含一种共聚的含OH或含二羰基或含环氧基的共聚单体。

10. 发明授权

US08653004B2 Actives-comprising polymer networks, processes for producing them, and their use 失效
标题翻译：含活性剂的聚合物网络，其生产方法及其用途
公开(公告)号：US08653004B2
公开(公告)日：2014-02-18
申请号：US12671613
申请日：2008-07-25
申请人： Alexandre Terrenoire , Hartmut Leininger , James Bullock , Mohammed Shoaib Qureshi , Hans-Werner Schmidt , Reiner Giesa , Meik Ranft , Oscar Lafuente Cerda
发明人： Alexandre Terrenoire , Hartmut Leininger , James Bullock , Mohammed Shoaib Qureshi , Hans-Werner Schmidt , Reiner Giesa , Meik Ranft , Oscar Lafuente Cerda
IPC分类号： A01N25/10 , A01N25/00 , A61K9/14
CPC分类号： A61L9/042 , A01N25/10 , A61L9/12 , A01N25/12 , A01N25/18 , A01N37/40 , A01N43/70 , A01N61/00
摘要： Process for producing actives-comprising polymeric networks from oligomers containing (meth)acrylate groups, optionally from further monomers, and from actives, the polymeric networks obtainable by the process, and the use of the networks for various purposes, more particularly for protecting materials or in crop protection.
摘要翻译：从含有（甲基）丙烯酸酯基团的寡聚物，任选地由其它单体和活性成分制备含活性成分的聚合物网络的方法，可通过该方法获得的聚合物网络，以及网络用于各种目的，尤其用于保护材料或在作物保护。

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