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1. 发明授权

US4294606A Novel N-phenyl-substituted N-heterocyclic compounds, their preparation and use in agents for regulating plant growth 失效
标题翻译：新型N-苯基取代的N-杂环化合物，其制备和用于调节植物生长的试剂中
公开(公告)号：US4294606A
公开(公告)日：1981-10-13
申请号：US111552
申请日：1980-01-14
申请人： Hans Tobler , Werner Fory , Rolf Schurter
发明人： Hans Tobler , Werner Fory , Rolf Schurter
IPC分类号： C07D295/12 , A01N43/36 , A01N47/02 , C07D205/08 , C07D207/06 , C07D207/267 , C07D207/27 , C07D207/325 , C07D207/404 , C07D207/452 , C07D211/76 , C07D213/64 , C07D213/80 , C07D213/85 , C07D223/10 , A01N43/40 , A01N43/46
CPC分类号： C07D213/64 , A01N47/02
摘要： The present invention relates to novel active compounds having a plant growth-inhibiting and herbicidal action and their preparation and to agents containing these active ingredients, and their use.The novel active compounds are saturated and unsaturated 4-membered to 7-membered ring nitrogen heterocyclic compounds which are substituted on the nitrogen atom by a phenyl radical which itself carries a trifluoromethanesulphonamido group --NH--SO.sub.2 --CF.sub.3 as a substituent. The phenyl radical can also carry other substituents and the heterocyclic structure can also be substituted. Oxo derivatives of the heterocyclic compound, in which the oxo group is preferably adjacent to the nitrogen atom, form a preferred sub-group of compounds.
摘要翻译：本发明涉及具有植物生长抑制和除草作用的新型活性化合物及其制备方法和含有这些活性成分的试剂及其用途。新型活性化合物是在氮原子上被本身带有三氟甲磺酰氨基-NH-SO 2 -CF 3作为取代基的苯基取代的饱和和不饱和4元至7元环氮杂环化合物。苯基也可以携带其它取代基，杂环结构也可以被取代。其中氧代基优选与氮原子相邻的杂环化合物的氧代衍生物形成优选的化合物亚组。

2. 发明授权

US4208202A N-Phenyl-substituted N-heterocyclic compounds, their preparation and use in agents for regulating plant growth 失效
标题翻译： N-苯基取代的N-杂环化合物，它们的制备和用于调节植物生长的试剂中
公开(公告)号：US4208202A
公开(公告)日：1980-06-17
申请号：US896970
申请日：1978-04-12
申请人： Hans Tobler , Werner Fory , Rolf Schurter
发明人： Hans Tobler , Werner Fory , Rolf Schurter
IPC分类号： C07D295/12 , A01N43/36 , A01N47/02 , C07D205/08 , C07D207/06 , C07D207/267 , C07D207/27 , C07D207/325 , C07D207/404 , C07D207/452 , C07D211/76 , C07D213/64 , C07D213/80 , C07D213/85 , C07D223/10 , A01N9/12
CPC分类号： C07D213/64 , A01N47/02
摘要： The present invention relates to novel active compounds having a plant growth-inhibiting and herbicidal action and their preparation and to agents containing these active ingredients, and their use.The novel active compounds are saturated and unsaturated 4-membered to 7-membered ring nitrogen heterocyclic compounds which are substituted on the nitrogen atom by a phenyl radical which itself carries a trifluoromethanesulphonamido group --NH--SO.sub.2 --CF.sub.3 as a substituent. The phenyl radical can also carry other substituents and the heterocyclic structure can also be substituted. Oxo derivatives of the heterocyclic compound, in which the oxo group is preferably adjacent to the nitrogen atom, form a preferred sub-group of compounds.
摘要翻译：本发明涉及具有植物生长抑制和除草作用的新型活性化合物及其制备方法和含有这些活性成分的试剂及其用途。新型活性化合物是在氮原子上被本身带有三氟甲磺酰氨基-NH-SO 2 -CF 3作为取代基的苯基取代的饱和和不饱和4元至7元环氮杂环化合物。苯基也可以携带其它取代基，杂环结构也可以被取代。其中氧代基优选与氮原子相邻的杂环化合物的氧代衍生物形成优选的化合物亚组。

3. 发明授权

US4394156A Novel N-phenyl-substituted N-heterocyclic compounds, their preparation and use in agents for regulating plant growth 失效
标题翻译：新型N-苯基取代的N-杂环化合物，其制备和用于调节植物生长的试剂中
公开(公告)号：US4394156A
公开(公告)日：1983-07-19
申请号：US314620
申请日：1981-10-26
申请人： Hans Tobler , Werner Fory , Rolf Schurter
发明人： Hans Tobler , Werner Fory , Rolf Schurter
IPC分类号： C07D295/12 , A01N43/36 , A01N47/02 , C07D205/08 , C07D207/06 , C07D207/267 , C07D207/27 , C07D207/325 , C07D207/404 , C07D207/452 , C07D211/76 , C07D213/64 , C07D213/80 , C07D213/85 , C07D223/10 , A01N43/40 , C07D213/68
CPC分类号： C07D213/64 , A01N47/02
摘要： The present invention relates to novel active compounds having a plant growth-inhibiting and herbicidal action and their preparation and to agents containing these active ingredients, and their use.The novel active compounds are saturated and unsaturated 4-membered to 7-membered ring nitrogen heterocyclic compounds which are substituted on the nitrogen atom by a phenyl radical which itself carries a trifluoromethanesulphonamido group -NH-SO.sub.2 -CF.sub.3 as a substituent. The phenyl radical can also carry other substituents and the heterocyclic structure can also be substituted. Oxo derivatives of the heterocyclic compound, in which the oxo group is preferably adjacent to the nitrogen atom, form a preferred sub-group of compounds.
摘要翻译：本发明涉及具有植物生长抑制和除草作用的新型活性化合物及其制备方法和含有这些活性成分的试剂及其用途。新型活性化合物是在氮原子上被本身带有三氟甲磺酰氨基-NH-SO 2 -CF 3作为取代基的苯基取代的饱和和不饱和4元至7元环氮杂环化合物。苯基也可以携带其它取代基，杂环结构也可以被取代。其中氧代基优选与氮原子相邻的杂环化合物的氧代衍生物形成优选的化合物亚组。

4. 发明授权

US4460400A Dihydropyrones, novel starting products used therein, compositions containing the novel dihydropyrones as active ingredients, and the use thereof for combating weeds 失效
标题翻译：二氢呋喃，其中使用的新型起始产物，含有新型二氢吡喃作为活性成分的组合物及其用于防治杂草的用途
公开(公告)号：US4460400A
公开(公告)日：1984-07-17
申请号：US381599
申请日：1982-05-24
申请人： Hans Tobler , Werner Fory
发明人： Hans Tobler , Werner Fory
IPC分类号： A01N43/14 , A01N43/16 , C07D309/32 , C07D309/38 , C07D311/74 , C07D311/94
CPC分类号： C07D311/94 , A01N43/16 , C07D309/32 , C07D311/74
摘要： There are described novel dihydropyrones of the formula I ##STR1## wherein R.sub.1 and R.sub.2 independently of one another are each a C.sub.1 -C.sub.4 -alkyl group, or one of the two substituents is also hydrogen, or R.sub.1 and R.sub.2 jointly form a C.sub.2 -C.sub.6 -alkylene bridge, R.sub.3 is C.sub.1 -C.sub.4 -alkoxy, C.sub.2 -C.sub.6 -alkenyloxy, C.sub.2 -C.sub.4 -alkynyloxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.3 -C.sub.5 -alkoxyalkoxy or hydroxyl, and X, Y and Z independently of one another are each hydrogen, halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -haloalkoxy, --S(O).sub.n -C.sub.1 -C.sub.4 -alkyl, --S(O).sub.n -C.sub.1 -C.sub.4 -haloalkyl, where n is 0, 1 or 2, or they are each C(O)OR.sub.4, where R.sub.4 is hydrogen or C.sub.1 -C.sub.4 -alkyl, or they are each NO.sub.2, CN or NR.sub.5 R.sub.6, where R.sub.5 and R.sub.6 independently of one another are each hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkylcarbonyl, C.sub. 1 -C.sub.4 -haloalkylcarbonyl or C.sub.1 -C.sub.4 -haloalkylsulfonyl, processes for producing them, novel starting products used therein, and the use of the novel dihydropyrones. The active substances of the formula I can be used in the form of agriculturally applicable compositions for combating weeds.
摘要翻译：描述了式I（I）的新型二氢吡咯烷，其中R 1和R 2彼此独立地各自为C 1 -C 4 - 烷基，或者两个取代基中的一个也是氢，或者R 1和R 2共同形成 C 2 -C 6亚烷基桥，R 3为C 1 -C 4 - 烷氧基，C 2 -C 6 - 烯氧基，C 2 -C 4 - 炔氧基，C 1 -C 4 - 卤代烷氧基，C 3 -C 5 - 烷氧基烷氧基或羟基，X，Y和Z独立地为一另一个是氢，卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4卤代烷基，C 1 -C 4 - 卤代烷氧基，-S（O）n -C 1 -C 4烷基， -S（O）n-C 1 -C 4卤代烷基，其中n为0,1或2，或它们各自为C（O）OR 4，其中R 4为氢或C 1 -C 4 - 烷基，或它们各自为NO 2，CN 或NR5R6，其中R5和R6彼此独立地为氢，C1-C4-烷基，C1-C4-烷基羰基，C1-C4-卤代烷基羰基或C1-C4-卤代烷基磺酰基，其制备方法，其中使用的新的起始产物，以及使用新型二氢呋喃。式I的活性物质可以以农业上可用于防治杂草的组合物的形式使用。

5. 发明授权

US4129573A Compositions for and method of influencing plant growth and novel 1-phenyl-2-oxo-pyrrolidine-4-carboxylic acid derivatives 失效
标题翻译： 1-苯基-2-氧代 - 吡咯烷-4-羧酸衍生物的组合物和影响植物生长的方法
公开(公告)号：US4129573A
公开(公告)日：1978-12-12
申请号：US736656
申请日：1976-10-28
申请人： Daniel Bellus , Werner Fory , Hans Tobler
发明人： Daniel Bellus , Werner Fory , Hans Tobler
IPC分类号： A01N43/36 , C07D207/26 , C07D207/277 , A01N9/22
CPC分类号： C07D207/277
摘要： This invention is directed to compositions for influencing plant growth, especially weed control, growth inhibition and desiccation, containing as active ingredient a 1-phenyl-2-oxo-pyrrolidine-4-carboxylic acid derivative of formula ##STR1## wherein A is --OH, --OR.sub.1, --SR.sub.2 or --CN, R.sub.1 representing a cation or an ester moiety, R.sub.2 an alkyl, benzyl or phenyl group, X being a substituent chosen from alkyl, alkoxy, alkylthio, phenoxy, substituted sulfamoyl or substituted sulfonylamino, Y is hydrogen, halogen, CF.sub.3, alkyl, alkylthio or alkoxy and Z is hydrogen, alkyl, alkylthio or alkoxy.The invention is also concerned with novel compounds of this formula, wherein Y is alkyl, alkylthio, halogen or CF.sub.3.
摘要翻译：本发明涉及用于影响植物生长，特别是杂草控制，生长抑制和干燥的组合物，其包含作为活性成分的式（I）的1-苯基-2-氧代 - 吡咯烷-4-羧酸衍生物，其中A是-OH ，-OR1，-SR2或-CN，R1表示阳离子或酯部分，R2表示烷基，苄基或苯基，X表示选自烷基，烷氧基，烷硫基，苯氧基，取代氨磺酰基或取代磺酰基氨基的取代基，Y表示氢，卤素，CF 3，烷基，烷硫基或烷氧基，Z是氢，烷基，烷硫基或烷氧基。

6. 发明授权

US08536089B2 Fungicidal compositions 有权
标题翻译：杀真菌剂
公开(公告)号：US08536089B2
公开(公告)日：2013-09-17
申请号：US11573277
申请日：2005-08-11
申请人： Harald Walter , Urs Neuenschwander , Ronald Zeun , Josef Ehrenfreund , Hans Tobler , Camilla Corsi , Clemens Lamberth
发明人： Harald Walter , Urs Neuenschwander , Ronald Zeun , Josef Ehrenfreund , Hans Tobler , Camilla Corsi , Clemens Lamberth
IPC分类号： A01N43/56 , A01N43/00 , A01N43/36 , A01N43/40 , A01N43/54 , A01N63/00
CPC分类号： A01N43/56 , A01N43/36 , A01N43/653 , A01N43/707 , A01N43/90 , A01N2300/00
摘要： The invention relates to fungicidal compositions comprising as active ingredient a combination of components A) and B) as defined in the patent claims, to a method of controlling phytopathogenic diseases on crop plants using such a compositions and to a method of protecting natural substances of vegetable and/or animal origin and/or their processed forms using such a composition.
摘要翻译：本发明涉及杀真菌组合物，其包含作为活性成分的组合物A）和B）如专利权利要求中所定义的组合，使用这种组合物控制作物植物病原性疾病的方法和保护植物天然物质的方法和/或动物来源和/或其加工形式。

7. 发明授权

US08207207B2 Heterocyclic a amide derivatives useful as microbiocides 有权
标题翻译：杂环酰胺衍生物可用作杀微生物剂
公开(公告)号：US08207207B2
公开(公告)日：2012-06-26
申请号：US12765942
申请日：2010-04-23
申请人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi
发明人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi
IPC分类号： A01N43/78 , A01P1/00
CPC分类号： C07C205/06 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/647 , A01N43/76 , A01N43/78 , C07C205/11 , C07C205/12 , C07C205/37 , C07C205/45 , C07C211/61 , C07C2603/66 , C07D207/34 , C07D207/46 , C07D213/89 , C07D231/14 , C07D249/04 , C07D263/34 , C07D277/56 , C07D327/06
摘要： The invention relates to a fungicidally active compound of formula (I): as defined in claim 1; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：如权利要求1所定义; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

8. 发明授权

US08183416B2 Heterocyclic amide derivatives useful as microbiocides 有权
标题翻译：用作杀微生物剂的杂环酰胺衍生物
公开(公告)号：US08183416B2
公开(公告)日：2012-05-22
申请号：US12765929
申请日：2010-04-23
申请人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi
发明人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi
IPC分类号： C07C205/06
CPC分类号： C07C205/06 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/647 , A01N43/76 , A01N43/78 , C07C205/11 , C07C205/12 , C07C205/37 , C07C205/45 , C07C211/61 , C07C2603/66 , C07D207/34 , C07D207/46 , C07D213/89 , C07D231/14 , C07D249/04 , C07D263/34 , C07D277/56 , C07D327/06
摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R6, R7 and R8; R1 is hydrogen, C1-4 alkyl, C1-4 haloalkyl, C1-4alkoxy, C1-4haloalkoxy, CH2C≡CR9, CH2CR10═CHR11, CH═C═CH2 or COR12; R2 and R3 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl or C1-4 haloalkoxy; R4 and R5 are each independently selected from halo, cyano and nitro; or one of R4 and R5 is hydrogen and the other is selected from halo, cyano and nitro; R6, R7 and R8 are each, independently, hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4haloalkoxy(C1-4)alkyl or C1-4haloalkoxy, provided that at least one of R6, R7 and R8 is not hydrogen; R9, R10 and R11 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 haloalkyl or C1-4 alkoxy(C1-4)alkyl; and R12 is hydrogen, C1-6 alkyl, C1-6haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4 alkylthio(C1-4)-alkyl, C1-4 alkoxy or aryl; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被R6基团取代，R7和R8; R 1是氢，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基，CH 2C≡CR9，CH 2 CR 10 = CHR 11，CH = C = CH 2或COR 12; R 2和R 3各自独立地为氢，卤素，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基或C 1-4卤代烷氧基; R4和R5各自独立地选自卤素，氰基和硝基; 或者R 4和R 5中的一个是氢，另一个选自卤素，氰基和硝基; R 6，R 7和R 8各自独立地为氢，卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4卤代烷氧基（C 1-4）烷基或C 1 -4卤代烷氧基，条件是R 6，R 7和R 8中的至少一个不是氢; R 9，R 10和R 11各自独立地为氢，卤素，C 1-4烷基，C 1-4卤代烷基或C 1-4烷氧基（C 1-4）烷基; 并且R 12是氢，C 1-6烷基，C 1-6卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4烷硫基（C 1-4） - 烷基，C 1-4烷氧基或芳基; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

9. 发明申请

US20120065239A1 PROCESS FOR THE PRODUCTION OF AMIDES 有权
标题翻译：生产助剂的方法
公开(公告)号：US20120065239A1
公开(公告)日：2012-03-15
申请号：US13198739
申请日：2011-08-05
申请人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi , Fanny Giordano , Martin Zeller , Gottfried Seifert , Shailesh Shah , Neil George , Ian Kevin Jones , Paul Edward Bonnett
发明人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi , Fanny Giordano , Martin Zeller , Gottfried Seifert , Shailesh Shah , Neil George , Ian Kevin Jones , Paul Edward Bonnett
IPC分类号： A01N43/56 , A01P3/00 , C07D231/14
CPC分类号： C07C211/61 , A01N43/56 , C07C205/06 , C07C209/325 , C07C209/70 , C07C2603/66 , C07D231/14
摘要： The present invention relates to a process for the preparation of compounds of formula I wherein R1 and R2 are each independently of the other hydrogen or C1-C5alkyl and R3 is CF3 or CF2H, by a) reaction of a compound of formula II wherein R1 and R2 are as defined for formula I, with at least one reducing agent to form a compound of formula wherein R1 and R2 are as defined for formula I, and b) reaction of that compound with at least one reducing agent to form a compound of formula IV wherein R1 and R2 are as defined for formula I, and (c) reaction of that compound with a compound of formula V wherein Q is chlorine, fluorine, bromine, iodine, hydroxy or C1-C6alkoxy and R3 is as defined for formula I, to form the compound of formula I; and to novel intermediates for use in that process.
摘要翻译：本发明涉及一种制备式Ⅰ化合物的方法，其中R1和R2分别独立地为氢或C1-C5烷基，R3为CF3或CF2H，通过a）式II化合物的反应其中R 1和 R 2如式I所定义，与至少一种还原剂形成下式化合物，其中R 1和R 2如式I所定义，和b）该化合物与至少一种还原剂的反应形成式 IV其中R1和R2如式I所定义，和（c）该化合物与式V化合物的反应，其中Q是氯，氟，溴，碘，羟基或C 1 -C 6烷氧基，R 3如式I所定义，形成式I化合物; 以及用于该过程的新型中间体。

10. 发明授权

US07820830B2 Process for the production of carboxanilides 有权
标题翻译：生产甲酰苯胺的方法
公开(公告)号：US07820830B2
公开(公告)日：2010-10-26
申请号：US12093619
申请日：2006-11-13
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Hans Tobler
IPC分类号： C07D231/14
CPC分类号： C07D231/14
摘要： The present invention relates to a novel process for the preparation of a compound of general formula (I): wherein R1 is H or C1-4 alkyl and R2 is difluoromethyl or trifluoromethyl, which comprises reacting a compound of general formula (II): wherein R1 has the meaning given above and X is chloro or bromo, with a compound of general formula (III): wherein R2 has the meaning given above, in the presence of a base, a palladium catalyst and a ferrocenyl biphoshine ligand of the Josiphos type, the reaction being carried out in an ether solvent at a reflux temperature of at least 100° C.
摘要翻译：本发明涉及一种制备通式（I）化合物的新方法：其中R1是H或C1-4烷基，R2是二氟甲基或三氟甲基，其包括使通式（II）的化合物：其中 R1具有上面给出的含义，X是氯或溴，与通式（III）的化合物：其中R 2具有上面给出的含义，在碱存在下，钯催化剂和Josiphos型的二茂铁基二膦配体，反应在乙醚溶剂中在至少100℃的回流温度下进行。

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