专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明授权

US08772266B2 Fungicide pyrazole carboxamides derivates 有权
标题翻译：杀菌剂吡唑甲酰胺衍生物
公开(公告)号：US08772266B2
公开(公告)日：2014-07-08
申请号：US13319614
申请日：2010-05-12
申请人： Guenter Bartels , Angela Becker , Jurgen Benting , Christoph-Andreas Braun , Peter Dahmen , Philippe Desbordes , Christophe Dubost , Stephanie Gary , Ulrich Gorgens , Hiroyuki Hadano , Benoit Hartmann , Thomas Knobloch , Marc Kosten , Norbert Lui , Ruth Meissner , Sergiy Pazenok , Rachel Rama , Arnd Voerste , Ulrike Wachendorff-Neumann
发明人： Guenter Bartels , Angela Becker , Jurgen Benting , Christoph-Andreas Braun , Peter Dahmen , Philippe Desbordes , Christophe Dubost , Stephanie Gary , Ulrich Gorgens , Hiroyuki Hadano , Benoit Hartmann , Thomas Knobloch , Marc Kosten , Norbert Lui , Ruth Meissner , Sergiy Pazenok , Rachel Rama , Arnd Voerste , Ulrike Wachendorff-Neumann
IPC分类号： C07D231/16 , C07D401/12 , A01N55/10 , A01N43/56
CPC分类号： C07D231/16 , A01N43/56 , A01N55/00 , C07D401/12 , C07F7/0812
摘要： The present invention relates to pyrazole carboxamides derivatives of formula (1) wherein Y represents CR5 or N, T represents S or O, X1 and X2 represent a chlorine or a fluorine atom, and Z1 represents a substituted or non-substituted cyclopropyl; Their process of preparation, their use as fungicide, and/or anti-mycotoxin active agents, and/or insecticide, and/or nematicide, particularly in the form of fungicide compositions, and methods for the control of phytopathogenic fungi, notably of plants, using these compounds or compositions.
摘要翻译：本发明涉及式（1）的吡唑甲酰胺衍生物，其中Y表示CR5或N，T表示S或O，X1和X2表示氯或氟原子，Z1表示取代或未取代的环丙基; 其制备方法，它们作为杀真菌剂的用途和/或抗真菌毒素活性剂，和/或杀虫剂和/或杀线虫剂，特别是杀真菌剂组合物的形式，以及用于控制植物病原真菌，特别是植物的方法，使用这些化合物或组合物。

2. 发明申请

US20120065164A1 FUNGICIDE PYRAZOLE CARBOXAMIDES DERIVATES 有权
标题翻译：杀真菌素类吡唑类杀菌剂
公开(公告)号：US20120065164A1
公开(公告)日：2012-03-15
申请号：US13319614
申请日：2010-05-12
申请人： Guenter Bartels , Angela Becker , Juergen Benting , Christoph-Andreas Braun , Peter Dahmen , Philippe Desbordes , Christophe Dubost , Stephanie Gary , Ulrich Gorgens , Hiroyuki Hadano , Benoit Hartmann , Thomas Knobloch , Marc Kosten , Norbert Lui , Ruth Meissner , Sergiy Pazenok , Rachel Rama , Arnd Voerste , Ulrike Wachendorf-Neumann
发明人： Guenter Bartels , Angela Becker , Juergen Benting , Christoph-Andreas Braun , Peter Dahmen , Philippe Desbordes , Christophe Dubost , Stephanie Gary , Ulrich Gorgens , Hiroyuki Hadano , Benoit Hartmann , Thomas Knobloch , Marc Kosten , Norbert Lui , Ruth Meissner , Sergiy Pazenok , Rachel Rama , Arnd Voerste , Ulrike Wachendorf-Neumann
IPC分类号： A01N55/10 , A01N43/56 , C07D401/12 , A01P15/00 , C07D231/14 , A01P5/00 , A01P3/00 , A01N43/40 , C07F5/02
CPC分类号： C07D231/16 , A01N43/56 , A01N55/00 , C07D401/12 , C07F7/0812
摘要： The present invention relates to pyrazole carboxamides derivatives of formula (1) wherein Y represents CR5 or N, T represents S or O, X1 and X2 represent a chlorine or a fluorine atom, and Z1 represents a substituted or non-substituted cyclopropyl; Their process of preparation, their use as fungicide, and/or anti-mycotoxin active agents, and/or insecticide, and/or nematicide, particularly in the form of fungicide compositions, and methods for the control of phytopathogenic fungi, notably of plants, using these compounds or compositions.
摘要翻译：本发明涉及式（1）的吡唑甲酰胺衍生物，其中Y表示CR5或N，T表示S或O，X1和X2表示氯或氟原子，Z1表示取代或未取代的环丙基; 其制备方法，它们作为杀真菌剂的用途和/或抗真菌毒素活性剂，和/或杀虫剂和/或杀线虫剂，特别是杀真菌剂组合物的形式，以及用于控制植物病原真菌，特别是植物的方法，使用这些化合物或组合物。

3. 发明授权

US07919632B2 Method for producing carboxamides 有权
标题翻译：生产甲酰胺的方法
公开(公告)号：US07919632B2
公开(公告)日：2011-04-05
申请号：US11917835
申请日：2006-06-07
申请人： Arnd Neeff , Sergiy Pazenok
发明人： Arnd Neeff , Sergiy Pazenok
IPC分类号： C07D231/16
CPC分类号： C07D231/16
摘要： The present invention relates to a novel process for preparing known fungicidally active 1,3-dimethyl-5-fluoro-1H-pyrazole-4-carboxamides from the corresponding acid fluoride and aniline derivatives in the absence of an acid acceptor.
摘要翻译：本发明涉及在不存在酸受体的情况下，由相应的酰氟和苯胺衍生物制备已知的杀真菌活性1,3-二甲基-5-氟-1H-吡唑-4-甲酰胺的新方法。

4. 发明授权

US07608736B2 Process for preparing acylsulfamoylbenzamides 有权
标题翻译：酰基氨磺酰苯甲酰胺的制备方法
公开(公告)号：US07608736B2
公开(公告)日：2009-10-27
申请号：US10874966
申请日：2004-06-23
申请人： Sergiy Pazenok , Mark James Ford , Günter Schlegel
发明人： Sergiy Pazenok , Mark James Ford , Günter Schlegel
IPC分类号： C07C303/04 , C07C311/04
CPC分类号： C07C303/40 , C07C311/51
摘要： The invention relates to a process for the preparation of a compound of formula (I): Which comprises reaction of a compound of formula (II) with a compound of the formula (III) in the presence of a chlorinating agent, followed by reaction of the resultant compound of the formula (IV) with a compound of formula (V) in the presence of a base: wherein the various symbols are as defined in claim 1.
摘要翻译：本发明涉及一种制备式（I）化合物的方法：其包括式（II）化合物与式（III）化合物在氯化剂存在下反应，随后将所得式（Ⅳ）化合物与式（Ⅴ）化合物在碱存在下反应：其中各种符号如权利要求1所定义。

5. 发明授权

US06541640B2 Process for the preparation of 4-haloalkylnicotinonitriles 失效
标题翻译：制备4-卤代烷基硝基腈的方法
公开(公告)号：US06541640B2
公开(公告)日：2003-04-01
申请号：US10013470
申请日：2001-12-13
申请人： Sergiy Pazenok , Henricus Maria Martinus Bastiaans
发明人： Sergiy Pazenok , Henricus Maria Martinus Bastiaans
IPC分类号： C07D21312
CPC分类号： C07C255/24 , C07C255/27 , C07C255/30 , C07D211/78 , C07D211/90 , C07D213/85
摘要： 4-Haloalkylnicotinonitriles having the formula (I) which are suitable as intermediates in the preparation of pesticides, are obtained by: (a) reacting a 3-amino-1-haloalkyl-2-propen-1-one RF—C(O)—CH═CH—NH2 (II) in a condensation reaction with a compound of the formula (III) to (VII), (R1Z)CH═CH—CN (III) (R1Z)2CH—CH2—CN (IV) Hal-CH═CH—CN (V) Hal2CH—CH2CN (VI) HC≡C—CN (VII), to give a compound of the formula (VIII), (IX) and/or (X), RF—C(O)—CH═CH—NH—CH═CH—CN (VIII) RF—C(O)—CH═CH—NH—CH(ZR1)—CH2—CN (IX) RF—C(O)—CH═CH—NH—CH(Hal)—CH2—CN (X) wherein RF is (C1-C4)-haloalkyl, R1 is alkyl, Hal is Cl or Br and each Z, independently, is O, S, NR or OCO; and (b) subjecting the reaction product to a ring closure reaction.
摘要翻译：通过以下方法获得具有式（I）的适合作为制备农药中间体的式（I）的4-卤代烷基硝基腈：（a）使缩合反应中的3-氨基-1-卤代烷基-2-丙烯-1-酮与得到式（VIII），（IX）和/或（X）的化合物，其中RF是（C 1 -C 4） - 卤代烷基，R 1是烷基，Hal是 Cl或Br，每个Z独立地是O，S，NR或OCO; 和（b）使反应产物进行闭环反应。

6. 发明申请

US20090306401A1 Method For The Production of 5-Fluoro-1,3-Dialkyl-1H-Pyrazol-4-Carbonyl Fluorides 有权
标题翻译： 5-氟-1,3-二烷基-1H-吡唑-4-羰基氟化物的制备方法
公开(公告)号：US20090306401A1
公开(公告)日：2009-12-10
申请号：US12066377
申请日：2006-09-05
申请人： Arnd Neeff , Sergiy Pazenok
发明人： Arnd Neeff , Sergiy Pazenok
IPC分类号： C07D231/14
CPC分类号： C07D231/16 , B01J31/0237 , B01J31/0251 , B01J31/0268 , B01J31/0271
摘要： The present invention relates to a novel process for preparing known 5-fluoro-1,3-dialkyl-1H-pyrazole-4-carbonyl fluorides which can be used as starting materials for active fungicidal ingredients by a halex reaction.
摘要翻译：本发明涉及一种制备已知的5-氟-1,3-二烷基-1H-吡唑-4-羰基氟化物的新方法，其可以通过halex反应用作活性杀真菌成分的起始原料。

7. 发明授权

US07501527B2 Method for the production of fluoromethyl-substituted heterocycles 有权
标题翻译：制备氟甲基取代的杂环的方法
公开(公告)号：US07501527B2
公开(公告)日：2009-03-10
申请号：US10576742
申请日：2004-10-19
申请人： Reinhard Lantzsch , Sergiy Pazenok , Frank Memmel
发明人： Reinhard Lantzsch , Sergiy Pazenok , Frank Memmel
IPC分类号： C07D231/12
CPC分类号： C07D263/34 , C07D231/14 , C07D277/30
摘要： The present invention relates to a process for preparing fluoromethyl-substituted heterocycles of the formula (I) in which R1, R2, R3 and A are each as defined in the disclosure, by fluorinating the corresponding chloromethyl-substituted precursors.
摘要翻译：本发明涉及通过氟化相应的氯甲基取代的前体制备式（I）的氟甲基取代的杂环的方法，其中R 1，R 2，R 3和A各自如本公开所定义。

8. 发明申请

US20090054661A1 Method for Producing Carboxamides 有权
标题翻译：生产甲酰胺的方法
公开(公告)号：US20090054661A1
公开(公告)日：2009-02-26
申请号：US11917865
申请日：2006-06-06
申请人： Arnd Neeff , Sergiy Pazenok
发明人： Arnd Neeff , Sergiy Pazenok
IPC分类号： C07D231/16
CPC分类号： C07D231/16
摘要： The present invention relates to a novel process for preparing known fungicidally active 1,3-dimethyl-5-fluoro-1H-pyrazole-4-carboxamides from the corresponding acid fluoride and aniline derivatives in the presence of alkylpyridine derivatives as an acid acceptor.
摘要翻译：本发明涉及在烷基吡啶衍生物作为酸受体存在下，由相应的酰氟和苯胺衍生物制备已知的杀真菌活性的1,3-二甲基-5-氟-1H-吡唑-4-甲酰胺的新方法。

9. 发明申请

US20090054660A1 METHOD FOR PRODUCING CARBOXAMIDES 有权
标题翻译：生产碳酰胺的方法
公开(公告)号：US20090054660A1
公开(公告)日：2009-02-26
申请号：US11917835
申请日：2006-06-07
申请人： Arnd Neeff , Sergiy Pazenok
发明人： Arnd Neeff , Sergiy Pazenok
IPC分类号： C07D231/16
CPC分类号： C07D231/16
摘要： The present invention relates to a novel process for preparing known fungicidally active 1,3-dimethyl-5-fluoro-1H-pyrazole-4-carboxamides from the corresponding acid fluoride and aniline derivatives in the absence of an acid acceptor.
摘要翻译：本发明涉及在不存在酸受体的情况下，由相应的酰氟和苯胺衍生物制备已知的杀真菌活性1,3-二甲基-5-氟-1H-吡唑-4-甲酰胺的新方法。

10. 发明授权

US07317105B2 Preparation of 4-haloalkylnicotinamides 失效
标题翻译：制备4-卤代烷基烟酰胺
公开(公告)号：US07317105B2
公开(公告)日：2008-01-08
申请号：US10515507
申请日：2003-05-09
申请人： Sergiy Pazenok
发明人： Sergiy Pazenok
IPC分类号： C07D213/08
CPC分类号： C07D213/82
摘要： The invention relates to a method for producing 4-haloalkylnicotinamides having the formula (I): wherein R1 is (C1-C4)haloalky, comprising subjecting one or more 3-((C1-C4)haloalkyl-3-oxo-1-alkenylamino)nitriles of the formula (II), (III) or (IV): R1—C(O)—CH═CH—NH—CH═CH—CN (II) R1—C(O)—CH═CH—NH—CH(ZR2)—CH2—CN (III) R1—C(O)—CH═CH—NH—CH(Hal)—CH2—CN (IV) where R1 is as defined above, R2 is the same or different and is (C1-C6)-alkyl and Z is the same or different and is O, S or NR1, to a ring-closing reaction and simultaneous hydrolysis in the presence of a strong acid.
摘要翻译：本发明涉及一种制备具有式（I）的4-卤代烷基烟酰胺的方法：其中R 1是（C 1 -C 4 - ）包括使式（II）的一种或多种3 - （（C 1 -C 4 -C 4）卤代烷基-3-氧代-1-烯基氨基）腈，（ III）或（IV）：<？in-line-formula description =“In-line Formulas”end =“lead”？> R 1 -C（O）-CH-CH-NH- CH-CH-CN（II）<？in-line-formula description =“In-line Formulas”end =“tail”？> <？in-line-formula description =“In-line Formulas”end =“lead” （O）-CH-CH-NH-CH（ZR 2） - CH 2 -CN（III） <？in-line-formula description =“In-line Formulas”end =“tail”？> <？in-line-formula description =“In-line Formulas”end =“lead”？> R < -C（O）-CH-CH-NH-CH（Hal）-CH 2 -CN（IV）<β在线公式描述=“在线式”末端 =“尾”→其中R 1如上所定义，R 2相同或不同，为（C 1 -C 3 - C 1-6烷基，Z相同或不同并且为O，S或NR 1至闭环反应，并在强酸存在下同时水解。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式