专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明申请

US20060128965A1 Novel substituted 1H-dihydropyrazoles, their preparation and use 失效
标题翻译：新型取代的1H-二氢吡唑，其制备和用途
公开(公告)号：US20060128965A1
公开(公告)日：2006-06-15
申请号：US11352805
申请日：2006-02-13
申请人： Gary Annis , George Lahm , Thomas Selby , Thomas Stevenson
发明人： Gary Annis , George Lahm , Thomas Selby , Thomas Stevenson
IPC分类号： C07D403/04 , C07F7/02 , C07D231/32
CPC分类号： C07D213/77 , A01N43/56 , C07C251/76 , C07C255/66 , C07D231/08 , C07D231/14 , C07D231/16 , C07D401/04 , C07D403/04 , C07D413/04 , C07D413/14
摘要： This invention provides compounds of Formula I, methods for their preparation and use for preparing compounds of Formula II wherein R1, R2, R3, R5, R6, X and n are as defined in the disclosure. This invention also discloses preparation of compounds of Formula III wherein R1, R2, R7, R8, R9 and n are as defined in the disclosure. This invention also pertains to certain compounds of Formula 4 and 6 used to prepare compounds of Formula I. wherein R1, R2, R5, X and n are as defined in the disclosure.
摘要翻译：本发明提供式I的化合物，其制备方法和用于制备式II化合物的方法，其中R 1，R 2，R 3， R 5，R 6，X和n如本公开所定义。本发明还公开了式III化合物的制备，其中R 1，R 2，R 7，R 8， R 9和n如本公开所定义。本发明还涉及用于制备式I化合物的某些式4和6化合物，其中R 1，R 2，R 5，，X和n如本公开中所定义。

2. 发明申请

US20060205748A1 Heterocyclic diamide invertebrate pest control agents 失效
标题翻译：杂环二酰胺无脊椎害虫防治剂
公开(公告)号：US20060205748A1
公开(公告)日：2006-09-14
申请号：US11158200
申请日：2005-06-21
申请人： Gary Annis , Bruce Finkelstein
发明人： Gary Annis , Bruce Finkelstein
IPC分类号： A01N43/54 , C07D49/02 , A01N43/56
CPC分类号： C07D213/81 , A01N43/10 , A01N43/40 , A01N43/54 , A01N43/80 , C07D213/82 , C07D231/40 , C07D333/38
摘要： This invention provides compounds of Formula (I), N-oxides and suitable salts thereof, wherein A and B are independently O or S; each J is independently a phenyl ring, a naphthyl ring system, a 5- or 6-membered heteroaromatic ring or an aromatic 8-, 9- or 10-membered fused heterobicyclic ring system wherein each ring or ring system is optionally substituted with 1 to 4 R5; K is, together with the two contiguous linking carbon atoms, a 5- or 6-membered heteroaromatic ring optionally substituted with 1 to 3 R4; and R1 R2, R3, R4, R5 and n are as defined in the disclosure. Also disclosed are methods for controlling an invertebrate pest comprising contacting the invertebrate pest or its environment with a biologically effective amount of a compound of Formula (I), an N-oxide thereof or a suitable salt of the compound (e.g., as a composition described herein). This invention also pertains to a composition for controlling an invertebrate pest comprising a biologically effective amount of a compound of Formula (I), an N-oxide thereof or a suitable salt of the compound and at least one additional component selected from the group consisting of surfactants, solid diluents and liquid diluents.
摘要翻译：本发明提供式（I）的化合物，其N-氧化物及其合适的盐，其中A和B独立地为O或S; 每个J独立地是苯基环，萘基环系，5或6元杂芳环或芳族8-，9-或10-元稠合杂双环系统，其中每个环或环系统任选被1至 4 R 5; K与两个相邻的连接碳原子连在一起，任选被1至3个R 4取代的5或6元杂芳环; 和R 1，R 2，R 3，R 4，R 5和R 5， n如本公开中所定义。还公开了用于控制无脊椎害虫的方法，包括使无脊椎害虫或其环境与生物有效量的式（I）化合物，其N-氧化物或该化合物的合适盐（例如，作为所述的组合物）接触这里）。本发明还涉及用于控制无脊椎害虫的组合物，其包含生物有效量的式（I）化合物，其N-氧化物或该化合物的合适的盐和至少一种选自以下的另外的组分：表面活性剂，固体稀释剂和液体稀释剂。

3. 发明申请

US20080108821A1 Method for preparing 3-halo-4,5-dihydro-1H-pyrazoles 有权
标题翻译：制备3-卤代-4,5-二氢-1H-吡唑的方法
公开(公告)号：US20080108821A1
公开(公告)日：2008-05-08
申请号：US12004902
申请日：2007-12-21
申请人： Gary Annis
发明人： Gary Annis
IPC分类号： C07D231/06 , C07D401/04
CPC分类号： C07D231/08 , C07D231/06 , C07D401/04
摘要： This invention relates to a method for preparing a 3-halo-4,5-dihydro-1H-pyrazole compound of Formula I comprising contacting with HX1 a different 4,5-dihydro-1H-pyrazole compound of Formula II wherein X1 is halogen and L, R, k and X2 are as defined in the disclosure. This invention also discloses preparation of compounds of Formula III wherein X1, R3, R6, R7, R8a, R8b and n are as defined in the disclosure.
摘要翻译：本发明涉及制备式I的3-卤代-4,5-二氢-1H-吡唑化合物的方法，包括与HX 1不同的4,5-二氢-1H-吡唑化合物其中X 1是卤素且L，R，k和X 2如本公开所定义。本发明还公开了式III化合物的制备，其中X 1，R 3，R 6，R 7， R 8a，R 8b和n如本公开所定义。

4. 发明申请

US20070021468A1 Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates 有权
公开(公告)号：US20070021468A1
公开(公告)日：2007-01-25
申请号：US10546165
申请日：2004-03-25
申请人： Gary Annis
发明人： Gary Annis
IPC分类号： A61K31/4439 , A61K31/4152 , C07D231/18 , C07D403/04
CPC分类号： C07D231/06 , C07D409/04
摘要： A method is disclosed for preparing a 2-substituted-5-oxo-3-pyrazolidinecarboxylate compound of Formula I. The method comprises contacting a succinic acid derivative of the formula R1OC(O)C(H)(X)C(R2a)(R2b)C(O)Y (i.e. Formula II) wherein X and Y are leaving groups and L, R1, R2a and R2b are as defined in the disclosure, with a substituted hydrazine of the formula LNHNH2 (i.e. Formula III) in the presence of a suitable acid scavenger and solvent. Also disclosed is the preparation of compounds of Formula IV wherein X1, R6, R7, R8a, R8b, R9, and n are as defined in the disclosure. Also disclosed is a composition comprising on a weight basis about 20 to 99% of the compound of Formula II wherein R1, R2a, R2b, R3, R4 and R5 are as defined in the disclosure; X is Cl, Br or I; and Y is F, Cl, Br or I; provided that when R2a and R2b are each H, and X and Y are each Cl then R1 is other than benzyl and when R2a and R2b are each phenyl, and X and Y are each Cl, then R1 is other than methyl or ethyl. Also disclosed is a crystalline composition comprising at least about 90% by weight of the compound of the formula R1OC(O)C(H)(X)C(R2a)(R2b)CO2H (i.e. Formula VI) wherein R2a and R2b are H, X is Br and R1 is methyl.

5. 发明申请

US20050215798A1 Method for preparing 3-halo-4,5-dihydro-1h-pyrazoles 有权
标题翻译： 3-卤代-4,5-二氢-1H-吡唑的制备方法
公开(公告)号：US20050215798A1
公开(公告)日：2005-09-29
申请号：US10518325
申请日：2003-07-29
申请人： Gary Annis
发明人： Gary Annis
IPC分类号： C07D231/06 , C07D231/08 , C07D401/04
CPC分类号： C07D231/08 , C07D231/06 , C07D401/04
摘要： This invention relates to a method for preparing 3-halo-4,5-dihydro-1H-pyrazole compound of Formula (I), comprising contacting with HX1 a different 4,5-dihydro-1H-pyrazole compound of Formula (II), wherein X1 is halogen and L, R, k and X2 are as defined in the disclosure. This invention also discloses preparation of compounds of Formula (III) wherein X1, R3, R6, R7, R8a, R8b, and n are as defined in the disclosure.
摘要翻译：本发明涉及制备式（I）的3-卤代-4,5-二氢-1H-吡唑化合物的方法，包括与HX 1不同的4,5-二氢-1H- （II）的吡唑化合物，其中X 1是卤素，L，R 1，k和X 2如本公开所定义。本发明还公开了制备式（III）的化合物，其中X 1，R 3，R 6，R 7， R 8，R 8b，R 8b和n如本公开所定义。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式