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1. 发明申请

US20110230429A1 AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4"-OR 4'-POSITION 有权
标题翻译：在4“-OR 4'-位置具有烷氧基取代基的AVERMECTIN B1和AVERMECTIN B1单糖衍生物
公开(公告)号：US20110230429A1
公开(公告)日：2011-09-22
申请号：US13117292
申请日：2011-05-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jérôme Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jérôme Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A01N43/22 , C07H17/08 , A01P7/00
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

2. 发明授权

US07737261B2 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″ -or 4′-position 有权
标题翻译：在4“ - 或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物
公开(公告)号：US07737261B2
公开(公告)日：2010-06-15
申请号：US10539274
申请日：2003-12-19
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jérôme Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jérôme Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： C07H17/04
CPC分类号： C07H17/08 , A61K31/7042
摘要： Avermectin B1 and avermectin B1 monosaccharide derivative compounds having an alkoxymethyl substituent in the 4″- or 4′-position; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions are provided.
摘要翻译：在4“或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物化合物; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 并提供了这些化合物和组合物的制备方法。

3. 发明授权

US07704961B2 Avermectins and avermectin monosacharides substituted in the 4′-and 4″ position having pesticidal properties 有权
标题翻译：在具有杀虫性的4'和4“位置取代的阿维菌素和阿维菌素单糖苷
公开(公告)号：US07704961B2
公开(公告)日：2010-04-27
申请号：US10568715
申请日：2004-08-27
申请人： Fiona Murphy Kessabi , Thomas Pitterna , Peter Maienfisch , Jérôme Cassayre , Laura Quaranta , Pierre Jung , Ottmar Franz Hueter
发明人： Fiona Murphy Kessabi , Thomas Pitterna , Peter Maienfisch , Jérôme Cassayre , Laura Quaranta , Pierre Jung , Ottmar Franz Hueter
IPC分类号： A61K31/70 , A61K31/7028 , C07H17/08
CPC分类号： A01N43/90 , C07H19/01
摘要： Described is a compound of the formula (I) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.
摘要翻译：描述了式（I）的化合物，其中碳原子22和23之间的键是单键或双键; m为0或1; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; （A）R 2是-N（R 3）R 4，和（1）X是0，其中R 3是例如氢，未被取代的或单取代到五取代的C 1 -C 12烷基，R 4是例如，至五取代的C 1 -C 12烷基，未取代的或一至五取代的C 3 -C 12环烷基; 或（2）X为S，其中R 3为例如氢，未取代或单价至五价取代的C 1 -C 12烷基，R 4为例如氢，未取代或单价至五价取代的C 1 -C 12烷基; 或（3）X为0或S，其中R3和R4一起为例如三至七元亚烷基或四至七元亚烯基桥; 或（B）R 2是OR 5，X是0或S，其中R 5是例如C 1 -C 12烷基，一至五取代的C 1 -C 12烷基; 或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下都是游离形式或盐形式; 这种化合物显示出杀虫活性。

4. 发明授权

US08017589B2 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position 有权
标题翻译：在4“ - 或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物
公开(公告)号：US08017589B2
公开(公告)日：2011-09-13
申请号：US12768280
申请日：2010-04-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A61K31/70 , C07H17/04
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

5. 发明申请

US20100210574A1 AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4"-OR 4'-POSITION 有权
标题翻译：在4“-OR 4'-位置具有烷氧基取代基的AVERMECTIN B1和AVERMECTIN B1单糖衍生物
公开(公告)号：US20100210574A1
公开(公告)日：2010-08-19
申请号：US12768280
申请日：2010-04-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A01N43/16 , C07H17/08 , A01P17/00
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

6. 发明申请

US20080194498A1 Avermectins and Avermectin Monosacharides Substituted in the 4'-and 4" Position Having Pesticidal Properties 有权
标题翻译：在4'和4“位置具有农药性质的阿维菌素和阿维菌素单糖
公开(公告)号：US20080194498A1
公开(公告)日：2008-08-14
申请号：US10568715
申请日：2004-08-27
申请人： Fiona Murphy Kessabi , Thomas Pitterna , Peter Maienfisch , Jerome Cassayre , Laura Quaranta , Pierre Jung , Ottmar Franz Hueter
发明人： Fiona Murphy Kessabi , Thomas Pitterna , Peter Maienfisch , Jerome Cassayre , Laura Quaranta , Pierre Jung , Ottmar Franz Hueter
IPC分类号： A01N43/90 , C07H17/08 , A01P17/00
CPC分类号： A01N43/90 , C07H19/01
摘要： Described is a compound of the formula (1) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.
摘要翻译：描述了式（1）的化合物，其中碳原子22和23之间的键是单键或双键; m为0或1; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 3 -C 12烷基，C 3 -C 12烷基，C 3 -C 12烷基， >环烷基或C 2 -C 12 - 烯基; （A）R 2是-N（R 3）R 4，和（1）X是0，其中R _{3是例如氢，未取代的或一至五取代的C 1 -C 12烷基，R 4是氢，是例如一至五取代的C 1 -C 12烷基，未取代或单取代或五取代的C 3 -C 12烷基， 12环烷基; 或（2）X是S，其中R 3是例如氢，未取代的或一至五取代的C 1 -C 12 - 烷基和R 4是例如氢，未取代的或一至五取代的C 1 -C 12烷基; 或（3）X为0或S，其中R 3和R 4一起为例如三至七元亚烷基或四至七元亚烷基，多元亚烯基桥; 或（B）R 2是OR 5，X是0或S，其中R 5是例如C 1 C 1 -C 12烷基，一至五取代C 1 -C 12烷基; 或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下都是游离形式或盐形式; 这种化合物显示出杀虫活性。}

7. 发明授权

US08263566B2 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position 有权
标题翻译：在4“ - 或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物
公开(公告)号：US08263566B2
公开(公告)日：2012-09-11
申请号：US13117292
申请日：2011-05-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A61K31/70 , C07H17/04
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

8. 发明授权

US07378399B2 Avermectins substituted in the 4″ and 4′-positions having pesticidal properties 有权
标题翻译：在4“和4”位取代的阿维菌素具有杀虫特性
公开(公告)号：US07378399B2
公开(公告)日：2008-05-27
申请号：US10544274
申请日：2004-02-03
申请人： Jerome Cassayre , Hans Tobler , Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Laura Quaranta , Ottmar Franz Hueter
发明人： Jerome Cassayre , Hans Tobler , Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Laura Quaranta , Ottmar Franz Hueter
IPC分类号： A01N43/04 , A01N43/00 , A01N43/40 , A01N43/02 , A01N43/16 , A61K31/40 , A61K31/38 , A61K31/335 , A61K31/35 , A61K31/70 , A61K31/397 , A61K31/445 , A61K31/44 , A01N43/38 , A01N31/40
CPC分类号： C07H17/08
摘要： What is described are a compound of the formula (I) Wherein A-B is —CH═CH— or —CH2—CH2—; n is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 for instance are either, (i) independently from each other for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; or (ii) together form with the nitrogen atom to which they are bound a three- to seven-membered ring, (iii) together are ═C(R4)R5; R4 and R5 are, independently from each other, for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; Y is O or S; Q is for instance H or unsubstituted or mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions
摘要翻译：描述的是式（I）的化合物，其中A-B是-CH-CH-或-CH 2 -CH 2 - 。 n为0或1; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 3 -C 12烷基，C 3 -C 12烷基，C 3 -C 12烷基， >环烷基或C 2 -C 12 - 烯基; 例如，R 2和R 3是（i）彼此独立地例如-Q，-C（-Y）-Q或-C（ - Y）-OQ; 或（ii）与其结合的氮原子一起形成三至七元环，（iii）一起为-C（R 4）R 5 >; R 4和R 5各自独立地为例如-Q，-C（-Y）-Q或-C（-Y）-O-Q; Y为O或S; Q是例如H或未被取代或单取代或未取代的C 1 -C 12烷基; 或者，如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体; 制备这些化合物，其异构体和互变异构体的方法以及这些化合物，其异构体和互变异构体的用途; 活性化合物选自这些化合物及其互变异构体的杀虫组合物; 用于制备所述式（I）化合物的中间体，式（I）化合物的制备方法和使用这些组合物来控制害虫的方法

9. 发明申请

US20080300134A1 Derivatives of Avermectin, Avermectin Monosaccharide and Avermectin Aglycone 有权
标题翻译：阿维菌素，阿维菌素单糖和阿维菌素糖苷配基的衍生物
公开(公告)号：US20080300134A1
公开(公告)日：2008-12-04
申请号：US11574588
申请日：2005-08-19
申请人： Ottmar Franz Hueter , Thomas Pitterna , Pierre Jung , Fiona Murphy Kessabi , Laura Quaranta
发明人： Ottmar Franz Hueter , Thomas Pitterna , Pierre Jung , Fiona Murphy Kessabi , Laura Quaranta
IPC分类号： C07H17/08 , A01N43/90 , C07D313/00
CPC分类号： C07H17/08 , A01N43/90
摘要： A compound of the formula (I) wherein the bond between carbon atoms 22 and 23 indicated with a broken line is a single or double bond, n is 0, 1 or 2, R1 represents, for instance, a C1-C12alkyl group, R2 represents, for instance, R15 group, R3 represents, for instance, R2 group, R4 represents, for instance, a chemical constituent, R5 represents, for instance, hydrogen, and R6 represents, for instance, R16 group; wherein R15 represents, for instance, unsubstituted or mono- to pentasubstituted C1-C6alkyl group, and R16 represent, for instance, hydrogen, or R15; and if appropriate, an E/Z isomer and/or diastereoisomer and/or tautomer of the compound of formula (I), in each case in free form or in salt form. Such compounds have been found to have pesticidal properties.
摘要翻译：式（I）的化合物，其中用虚线表示的碳原子22和23之间的键是单键或双键，n是0,1或2，R1表示例如C1-C12烷基，R2 表示例如R 15基，R 3表示例如R 2基，R 4表示例如化学成分，R 5表示例如氢，R 6表示例如R 16基; 其中R 15表示例如未取代或单价至五价取代的C 1 -C 6烷基，R 16表示例如氢或R 15; 并且如果合适的话，式（I）化合物的E / Z异构体和/或非对映异构体和/或互变异构体在各种情况下均为游离形式或盐形式。已经发现这些化合物具有杀虫性质。

10. 发明授权

US07521429B2 Avermectin B1 monosaccharide derivatives 有权
标题翻译：阿维菌素B1单糖衍生物
公开(公告)号：US07521429B2
公开(公告)日：2009-04-21
申请号：US10560390
申请日：2004-06-15
申请人： Thomas Pitterna , Pierre Jung , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Ottmar Franz Hueter
发明人： Thomas Pitterna , Pierre Jung , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Ottmar Franz Hueter
IPC分类号： A61K31/70 , C07H17/08
CPC分类号： C07H19/01 , C07H17/08
摘要： A compound of formula (I) wherein the bond between carbon atoms 22 and 23 may be a single or a double bond; R1 is C1-C12alkyl, C3-C8cycloalkyl, or C2-C12alkenyl; R2 and R3 are, for example, independently of each other hydrogen, C1-C12alkyl, C3-C12cycloalkyl, C2-C12alkenyl, C2-C12alkynyl, aryl or heteroaryl; and, where applicable, to E/Z isomers, mixtures of E/Z isomers, diastereomers and/or tautomers, in each case in free form or in salt form; pesticidal compositions in which the active ingredient has been selected from those compounds and their tautomers; and a method of controlling pests using those compositions are described.
摘要翻译：式（I）的化合物，其中碳原子22和23之间的键可以是单键或双键; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R 2和R 3例如彼此独立地为氢，C 1 -C 12烷基，C 3 -C 12环烷基，C 2 -C 12烯基，C 2 -C 12炔基，芳基或杂芳基; 在适用的情况下，E / Z异构体，E / Z异构体，非对映异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 其中活性成分选自那些化合物及其互变异构体的杀虫组合物; 并描述了使用这些组合物来控制害虫的方法。

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